CZ64598A3 - Phenylacetic acid derivative, process of its preparation, intermediate of such process and preparation containing the derivative - Google Patents

Abstract

The invention concerns phenylacetic acids of formula (I) in which the substituents and the index have the following meanings: X is NOCH3, CHOCH3, CHCH3 and CHCH2CH3; Y = O and NR (R = hydrogen and alkyl); Z is an optionally substituted nitrogen atom-bonded heterocyclyl or heteroaryl; R<1> = hydrogen and alkyl; R<2> = cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m = 0, 1 or 2; R<3> = hydrogen, cyano, nitro, hydroxy, amino, cyclopropyl, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylamino and dialkylamino; R<4> = hydrogen, optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkylsulphonyl, cycloalkyl, aryl, arylcarbonyl, arylsulphonyl, hetaryl, hetarylcarbonyl and hetarylsulphonyl. The invention further concerns salts thereof, processes for their preparation and agents containing them.

Description

Technical field

The present invention relates to the phenylacetic acetates of the formula I

where it means

X NOCH ₃ , CHOCHO ₃ , CHCH ₃ and CHCH ₂ CH _{3 <}

Y 0 and NR,

And R is hydrogen of C ₁ -C ₄ -alkyl,

Z is an optionally substituted saturated or partially or fully unsaturated cyclic radical which, in addition to the nitrogen atom through which it is bound, may contain, in addition to the carbon ring members, one to four nitrogen, oxygen and sulfur heteroatoms,

R ^{1 is} hydrogen and C ₁ -C ₄ -alkyl;

R ² cyano, nitro, trifluoromethyl, halogen, C, _T and --C ₄ -alkyl.

C ₁ -C ₄ -alkoxy, m 0, 1 or 2, wherein the radicals R ¹ may be different if m is 2

R ³ is hydrogen, cyano, nitro, hydroxy, amino, cyclopropyl, halogen, C ₃ -C ₄ -alkyl, C ₁ -C ₄ -haloalkyl, C ₁ -C ₄ -alkoxy, C _x - C ₄ - and ii. 1 ogen alkoxy, C _; - C ₄ - ai quatio, C ₃ - C ₄ - ayl amineo D 1 - C ₃ - C ₄ - a 1 cy 1 amine,

R ⁴ is hydrogen, α, -Ο, η and θ-i alkyl, C ₂ -C ₁₀ -alkenyl, C ₂ -C ₁₀ -alkynyl, C ₁ -C ₁₀ -a.lkylkarbonyl, C ₂ -C ₁₀ 1-a keny 1 ka rbony 1, C ₂ - C _x0 a1k and ny1karbony1 11 ebo C _x - C _{x 0} - a 1ky1s u. l · f ony1 par routine or tyt the radicals may be partially or fully halogenated or may carry one to three of the following groups:

- cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarboriyl,

- halogen, C _x -C ₆ -haloalkyl, C ₁ -C ₆ -alky.lsulfonyl, C ₁ -C ₆ -alkylsulfoxyl, C _x -C ₆ -alkoxy, C _x --C ₆ -haloalkoxy, C-Cg- alkoxycarbonyl, C _x -C ~ ₆ alkylthio, C ₆ -C _x 1 -a 1 alkyl amino, di-C _x -C ₆ -alkylamino, C -Cg _{x-alkylaminocarbonyl,} di-C-Cg-alkyl aminocarbonyl al! , C ₁ -C ₆ -alkylated not iocarbonyl, C ₁ -C ₆ -alkylaminothiocarbonyl, C ₂ -C ₆ -alkenyloxy

C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -cycloalkyl; And oxy, heterocyclyl, heterocyclyoxy, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy and hetarythio, wherein the cyclic groups may be partially or fully halogenated or may carry one to three of the following: cyano, nitro, hydroxy , mercapto, amino, •

- 3-carboxyl, aminocarbonyl, amines. not iocarbonyl, halogen,

C ₁ -C ₆ -alkyl, C ₃ -C ₆ -cycloalkyl, C 1 -C ₆ -haloalkyl, C ₁ -C ₆ -alkylsulfonyl, C ₁ -C ₆ -alkylsulfoxyl, C ₁ -C ₆ -alkoxy, C _and -C ₆ -haloalkoxy, C ₁ -C ₆ -alkoxycarbonyl, C ^ -Cg-alkylthio, C-C ₆ -alkylamino, di-C ₁ -C ₆ -alkylamino, _C-C6 alkylaminocarbonyl, di-C ^ -Cg-alkylaminocarbonyl, C j C ₆ - allyl notiocarbonyl, Di-C 1 -C ₆ -alkylaminothiocarbonyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio and C (= NOR ^a ) -Yy-lV ⁵ ,

C ₃ -C ₆ cycloalkyl, aryl, and ry 1 ka rboriy 1 arylsuif onyl, hetaryl, hetarylcarbonyl and hetaryIsulfonyl, where these radicals may be partially or fully halogenated or may carry one to three of the following groups:

- cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl,

- halogen, C ₁ -C ₆ -alkyl, C ₃ -C ₆ -cycloalkyl, C ₁ -C ₆ -haloalkyl, C j-Cg-alkylcarbonyl, _C-C6 alkylsulfonyl -al.kylsulf, C-C ₆ - alkylsul-, foxyl, C ₁ -C ₆ -alkoxy, C ₁ -C ₆ -haloalkoxy, C ₁ -C ₆ -alkoxycarbonyl C ₁ -C ₆ -alkyloxy, C 1 -C ₆ -alkylamino, Di-C ₁ -C ₆ -alkylamino, C ₁ -C ₆ -alkylaminocarbonyl, Di-C ₁ -C ₆ -alkylaminocarbonyl, C ₁ -C ₆ -alkylaminocarbonyl, Di-C ₁ -C ₆ -alkylaminocarbonyl C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkenes. loxy, benzyl, benzyloxy, aryl, aryloxy, hetaryl, hetaryloxy and C (NOR ' ¹ ) -A. _rl -R ^b where • · · · · ·

-4Λ means oxygen, sulfur and nitrogen and nitrogen carries hydrogen or

C ₁ -C ₆ -alkyl, n is 0 or 1 a

R ^a , R ^b are hydrogen or C 1 -C ₆ -alkyl, as well as 1 salts thereof.

In addition, the present invention relates to processes and intermediates for the preparation of these compounds, as well as compositions containing them, suitable for combating animal pests and harmful fungi and fungi.

Do the state of the technique

We know from the literature that phenylacetic acid derivatives are used for controlling animal pests and harmful fungi and fungi (EP-A 422 597, EP-A 463 488, EP-A 370 629, EP-A 460 575, EP-A 472 300, WO- No. A 90/70, 493, WO-A 92/13, 830, WO-A

92 / 18,487). In addition, the earlier German patent applications P 44 03 447.4 and P 44 03 448.2 disclose phenylacetic acid derivatives having bis-oxime side-effects with action against, pests and harmful fungi and fungi.

However, it is an object of the present invention to provide improved performance compounds.

Thus, the above-defined phenylacetic acid acetates I have been found. In addition, processes and Λ have also been developed

We have found intermediates in their production and compositions containing them which are suitable for combating animal pests and harmful fungi and fungi.

Compounds 1 as such can, however, be obtained by the use of pervases known in the art. In principle the synthesis of compounds I unimportant if first creating an array of -C (= X) -COYR ¹ or -CH ₂ 0N ^ CR ³ -C (Z) = ^ NOR ^fourth Various methods of forming a -C (-X) -COYR ^{3 group} (in the following, the samples are sometimes used to abbreviate the representation of the mark 7) are known from the above-mentioned literature.

Process for side chain synthesis _; ON CR ^{f -} C (Z) · NOR ⁴ is essentially governed by the type of substituent R ³ .

1. In the case where R ^{3 is} not halogen, the general procedure is to form -CH ₂ N = CR ³ -C (Z) = NOR ⁴ by reacting the benzyl derivative of formula II with a hydroxyimine of formula III.

HON = CR ³ -NOR ⁴

From ^C -z

O = ^C-YR1

I • ·

-6L ¹ in formula 11 means a nukloot j. an example of a halogen or a suliona love group, mostly chlorine, bromine, iodine, mesylate, tosylate and a.

The reaction proceeds in a manner known per se in an inert organic solvent in the presence of a base (for example sodium hydride, potassium hydroxide, potassium carbonate and triethylamine) according to the methods described in Houben-Wey 1, Vol. E lib, p. 3 701 and Houben-Weyl, vol. 10/1, pp. 11891.

The desired hydroxy imiri III is obtained, for example, by reacting the corresponding dihydroxy indole III with a nucleophilically substituted reagent V.

R ⁴ --- L ²

H0N = CR ³ -

lila

H0N ³ = CR ⁴ -nor

OF

III

In formula V, L ² is a nucleophilically replaceable group, such as halogen or sulfonate groups, in particular chlorine, bromine, iodine, mesylate, tosylate and triflate. The reaction proceeds in a manner known per se, in an inert organic solvent in the presence of a base (eg potassium carbonate, potassium hydroxide, sodium hydride, pyridine and triethylamine) according to the methods described in Houben-Weyl, Vol. E 14 b, S-30'7f, p. 3 / 0f and p.35f, Houben-Weyl, vol.10 / 4, p. 55f, p. 1.80I and p. 217f, Houben-Weyl, vol. . E 5, pp. 780f.

• ·

Alternatively, the compounds 111 obtained with the first carbonylated hydroxylimine 11b together with facilitating the introduction of sulfur into the compound corresponding to the thiocarbonylhydroxyrminine 111c may subsequently be converted either by t and k, z and the reagent may also be

(a) does not exist with hydroxylamine or a salt thereof, and then with a compound of formula V; or

b) with a hydroxy] amine or a hydroxylammonium salt of the formula

Villa resp. VIIb to formula III.

HON = CR ³ -

HON = CR ³ -

lílb

IIIc

NOR <

HON = ^CR3 --C

III

Q 'in formula VIIb means an anion of an inorganic acid (especially a halide such as chloride).

In addition, compounds III can be obtained as outlined in Example 1 and at Synthesis Nos 9 and 10.

The conversion from Blb to 111c takes place in a manner known per se (see Bull. Soc. Chirn. Belg. 87, 293 (1978) at a temperature of 10 ° C.

From about 20 ° C to about 120 ° C, in an inert organic solvent.

• ·

-δ

Suitable solvents are aliphatic hydrocarbons such as pentane, hexane, cyclohexane and petroleum ether, aromatic hydrocarbons such as toluene, o-, m- and p-xylene, halogenated hydrocarbons such as methylene chloride, chloroform. and chlorobenzole, an ether such as diethyl ether, diisopropyl ether, tert-butyl methyl ether, dioxane, anisole and tetahydrofuran, nitriles such as acetonitrile and propionitrile, in particular dioxane, toluene and xylene.

Mixtures of the solvents mentioned may also be used.

For example, P ₄ S ₁₀ or Lawesson's reagent (2,4-bis (4-methoxyphenyl) -1,3-dithia-2,4-diphosphetan-2,4-disulfide) is used as a sulfur facilitator to the compounds. .

Oximation of lile formulas in a known manner (cf.

Houben-Weyl with v.VI11, solvent.

V i i o.

J. iieterocycl.

694f) v

VI Ib in progress

Chem 17, inert per se

819 (1980), organic

1.1 Alternatively, compounds 1 can also be obtained by first converting the benzyl derivative II with the dihydroxyimine IIIa to the corresponding benzyloxime IVa and IVa, followed by the nucleophin-substituted reagent V

IVa

O == C - YR ¹

- q-

The reaction proceeds in a manner known per se in an inert solvent in the presence of a base (11a. Example potassium carbonate, potassium hydroxide, sodium hydride, pyridine and triethylamine) according to the methods described in Houben-Weyl, Vol. 10/1, pp. 11891, Houben-Weyl, vol. E 14b, pp. 3071, 3701 and 3851, Houben-Weyl, vol. 10/4, pp. 551, 1801 and 2171, Houben-Weyl, vol. E 5, pp. 7801.

2 Correspondingly, compounds 1 can also be obtained by first converting the benzyl derivative II with carbonylhydroxyimine IIIb to the corresponding benzyloxyimine VIa, then converting VIa together with the sulfur-facilitating agent into the compound to the thio compound VIb and VIb either

(a) first with hydroxylamine or a salt thereof, and then with a compound of formula V; or

b) with a hydroxylamine or a hydroxylammonium salt according to formula VIIa and III, respectively; VIIb converts 11a I.

H0N = CR ³ -II

Illb • ·

0 = ^C-YR1

Via

NOR ⁴

OF

O = ^C-YR1

The reaction of the benzyl derivative II with carbonylhydroxyimirium 11 Ib proceeds as described generally and specifically for the reaction of II with III. The sulfur and oximation reactions to I proceed generally and specifically under the conditions described above.

The compounds VIa can also be obtained, for example, by reacting the carboxylic acid More in a manner known per se (Houben-Weyi, vol. E5, p. 9411) with a nitrogen-containing heterocycle IX.

+

HZ

More

IX

Via

The reaction generally takes place at room temperature. from -20 ° C to 100 ° C, mostly from -10 ° C to 50 ° C, in an inert organic solvent, usually in the presence of an activating agent (e.g. phosgene, i.e., chloride, oxalyichi ori.d,

N, N-carbonyldiimidazole and triphenylphosphine / CCl ₄ ).

1.3 A further possibility of obtaining compounds I consists in reacting the benzyl derivative II with N-hydroxyphthalimide followed by hydrazinolysis to benzylhydroxylamine IIa and in a further reaction. IIIa with carbonyl compound VIIIa.

0 = ^C-YR1

O • ·

- At. -

H2NNH2

Ha ^ NOR ⁴ to + 0 == CR ³ - (f —► ¹ ^ z)

Vlila

The reaction proceeds in a manner known per se in a free-standing organic solvent according to the methods described in EP-A 463 488 and EP-A 585 751.

The necessary carbonyl compounds VIIIa are obtained by cross-reacting the corresponding hydroxyiminocarbonyl compounds IIIb with nucleophilically substituted reagent V.

^ NOH

0 = CR ³ - + +

VlIIb

R ⁴

IN

Vlila

The compounds IIIb can also be obtained by introducing the hydroxamic acid chloride VIJd in a manner known per se. (See J. Heterocycl. Chem. 21, 1029 (1984), Coll, Czech. Chem. Comm. 41, 3085 (39'6) to react with a nitrogen containing heterocycle (IX).

^ NOH

0 = CR ³ - C 1 Cl

VII Id

IX

VlIIb

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·· · · · ···

1.4 Accordingly, the compounds 1 can also be obtained by first converting the benzylhydroxylamine IIIa with the hydroxyimino derivative V1 'and 1b to the first benzyloxyiminoderivative of formula IVa and IVa then subsequently converting it with a nucloilyl substituted reagent. V, as described above, at. AND.

CH ₂ ONH ₂

Π-

0 = ^C-YR1

ΝΟΗ

OF

R ⁴ --- L ²

ch ₂ on = cr ³ -C-YR ¹

AND

• φ φ • φ φ φ φ φ • φ φ φ φ φ φ φ Logically, the compounds i can also be obtained by converting the benzyl hydroxylamine according to formula 11a first with α-dicarbonyl VIIlc to the benzyloxyiminoderivative Via and then converting it later to I as described above.

CH ₂ ONH ₂

O— CR ³ -

O = C-YR ¹ lbs

VIIlc

Via

^ NOR ⁴

O = ^C-YR1

AND

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

According to another method, compounds I can also be obtained by first converting the benzylhydroxylamine 11a with the hydroxamic acid chloride VIIId to the corresponding compound IVb and then converting IVb first to iq. IVa and IVa. then on I.

CH ₂ ONH ₂

0 = CR ³ -

O — C — YR1

NOH

Cl

IVb

0 = C-YR 1

-46 -

1.7. A further possibility for the preparation of the compounds I consists in converting the benzylhydroxylamine IIa with the alpha-oxocarboxylic acid VHIe into the corresponding oximinocarboxylic acid More, more by reacting with VIIa and VIIb, respectively. corresponding hydroxamic acid. IVc, IVc are then halogenated to the hydroxamic acid halide

IVd and IVd then convert the reaction with IX to I.

Ha

0 = CR ^{3 -} CO ₂ H

VHIe

More

IVc

0 = ^C-YR1

0 = C-YR ¹

• • • • •

1.8 Compounds in which R ³ represents a halogen atom are obtained from the corresponding precursors in which the corresponding radical is a hydroxy group according to methods known per se (see Houben-Wey1, vol. E5, p. 631,

J. Org. Chem. 36, 233 (1971); J. Org. Chem. 57, 3245 (1992). Preferably, the corresponding reactions to the helogen derivative are carried out on steps I and VIa.

1.9 Compounds in which R 'is through an atom. O, S or N bonded to the molecular backbone are obtained from the corresponding precursors where the corresponding residue is a halogen atom by methods known per se (see Houben-Weyl, vol. E5, p. 8261. and 12801, J. Org. Chem. 36, 233 (1971), J. Org Chem 46 4623 (1981) Preferably, the corresponding reactions to the halogen derivative are carried out on Stages I and VIa.

2. Compounds 1, where 1 'is attached via an oxygen atom, to the molecule, are also obtained from the corresponding precursors, where the residue in question is a hydroxy group, according to known methods (see Houben-Weyl, vol. E5, p. 8261). Chem., 1974, 27, 1341. Preferably, the corresponding conversions to alkoxy derivatives are carried out on Steps I and VIa.

3. Compounds I, where R ^{3 is} not halogen, are obtained mostly by converting a compound of formula III according to the methods described in EP-A 493 711 with Lacton X first to the corresponding benzoic acid XTa and Xla then subsequently over the corresponding halide (X1b, hal halogen.) Is converted to cyanocarboxylic acid XIc, which is then converted to the so-called Pinner reaction (Angew. Chem. 94, 1 (1982) to the α-keto ester X1.1 and (see EP-A 348 766, EP). DE-A 37 05 389, DE-A 36 23 921).

NOR ⁴

OF

Xlb

CO2R ¹

Xlla

NOR ⁴

Z (R ¹ * H)

• · • ·· ·· • · ·· • ·· • · ·· • • • · • • · ··· • · • · • · • * · · • · • ··· • • • · • • · • · • • • ·· ··· ·· ·· ·· ··

α-ketoester XIaa. where appropriate, the corresponding acetates and -ketokarboxylové acid (R ¹ = hydrogen, obtainable by known per se, hydrolysis of esters) are the central intermediates for preparing various groupings - C (= X) COYR ^first

For example, the corresponding .alpha.-ketocarboxylic acid amides XTIc can be obtained by reacting the .alpha.-ketocarboxylic acid acetates XI Ib and IIc, respectively. esters of XIa (see Uouben-WevI, Vol. E5, p. 941f).

4. In contrast to the procedure described above, α-ketocarboxylic acid amides XIIc, where R is hydrogen, can also be obtained directly from carboxylic acid halides XIIb by reaction with isocyanides XIII (R'-NC) (see EP-A 547 825).

NOR ⁴

OF

Xlb

+

R1-NC

XIIc (R = H)

5. In another variant, compounds XIIc are obtained by first substituting hydrogen for the ortho-halobenzyl derivatives Xld with metal and converting the organo-metal compound obtained with oxal chloride to the corresponding chloride. acid

- ketocarboxylic XIII, which is then converted with the amine to the corresponding amide XIIc (see J. Org. Chem. 46, 212-1 1981),

DE-A 40 42 280

Houben-Weyl, Vol.

9721).

NOR ⁴ , Z ch ₂ on = cr ³ -

Xld

NOR ⁴ , Z ch ₂ on = cr ³ - c.

Xlld

0 = CNRR ¹

NOR ⁴ ch ₂ on = cr ³ - c.

XIIc

Conversion of the acid derivatives of the corresponding compound I as described in the above-mentioned expert 585 751, EP-A 513 580, EP-A 477 389, EP-A 348 766, EP-A. No. 251 082, DE-A 36 23 921.

Compounds T can be formed at a C = N-double bonds as a mixture of:

α-ketocarboxylic XII on.

the production of the compounds T1 is in the literature as well as in EP-A

631, EP-A-400 417, DE 37 05

EP-A 398 692, EP-A 178 826 and production based on their C = Czomer E / Z, which, for example,

Crystallization or chromatography may be conveniently separated into the individual compounds.

With respect to the C = X double bond, the E-isomers of compounds 1 are preferred due to their activity (the arrangement relates to the CH ₃ , CH ₂ CH ₃ and OCH groups, respectively, relative to the COYR ¹ group).

In view of the CH ₂ ON = CR ³ -d 2 bond and the cis-isomers of compounds I are preferred for their activity (the arrangement refers to thia residues R ³ relative to the OCH ₂ moiety).

The double bond arrangement of C (Z) NOR ⁴ insignificant effect on biological.

generally has only the effect of 11 osts 1 lessons η I. In cases where the subcatching is calm a certain influence, we attribute the most significant and not related to the residues OR ⁴ in proportion to group Z).

Once a mixture of isomers is formed in the synthesis, separation into individual compounds is generally not absolutely necessary, since the individual isomers may be reciprocally transformed in part during processing for use or during their own use (for example under the influence of light, acid or base). Corresponding transformations can also take place after use, for example in the treatment of plants, molds, and animal pests, in the treated organism.

In the above definition of Compounds (I), collective terms are used that are representative of the following groups:

Halogen y fluorine, chlorine, bromine and iodine

Alkyl: straight or branched chain alkyl groups having 1 to 4, 6 or 10 carbon atoms, for example 0 _τ- O- _6- alkyl such as methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl,

2-methylpropyl, 1,1-dimethylethyl, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl, 1 -methylpentyl,

2-methylpentyl,

1.1-dimethylbutyl,

2.2-dimethylbutyl,

1-ethylbutyl,

3-Methylpentyl,

1,2-dimethylbutyl,

2.3- dimethylbutyl,

2-ethylbutyl,

4-methylpenty.1.,

1,3-dimethylbutyl,

3.3- dimethylbutyl,

1,1,2-trimethylpropyl,

1,2,2-trimethylpropyl,

1-ethyl-1-methylpropyl

- e t y 1 - 2 - m y t 1 p o r 1,

Alkylamino: an amino group which may carry a straight or branched chain alkyl group having 1 to 4 or 6 carbon atoms, as described above,

Dialkylamino: an amino group which carries two independent straight or branched chain alkyl groups having from 1 to 4 or 6 carbon atoms, as indicated in the preceding cases,

Alkylcarbonyl: straight or branched chain alkyl groups having 1 to 6 or 10 carbon atoms which are bonded to the backbone via a carbonyl group (-CO-),

Alkylsulfonyl: straight or branched chain alkyl groups having 1 to 6 or 10 carbon atoms, which are attached to the backbone via a sulfonyl (-SO ₂ -) group,

-

Alkylsulfoxyl: a. Straight or branched alkyl groups chain with 1 to 6 carbon atoms that are through sulfoxyl group (-S (== 0) -) tied to the skeleton, Alky 1 arn i n o c a r b o n y 1 : alkylamino groups having 1 to 6 atoms carbon that are bonded via a carbonyl group (-CO-) skeleton, ri yl: dialkylamino groups each having 1 to 6

carbon atoms per alkyl moiety that are attached to the backbone via a carbonyl (-CO-) group,

Alkylaminothiocarbonyl: a (C1 -C6) alkyl group which is bonded to the backbone via a thiocarbonyl (-CS-) group,

Dialkylaminothiocarbonyl: dialkylamino groups of 1 to 6 carbon atoms per alkyl moiety that are attached to the backbone via a thiocarbonyl (-CS-) group,

Haloalkyl: straight-chain or branched alkyl groups having 1 to 4 or 6 carbon atoms, in which groups the hydrogen atoms may be partially or fully replaced by halogen atoms, for example C 1 -C 6 -haloalkyl such as chloromethyl, dichloromethyl, tritium Methyl 1, fluoromethyl 1, difluoromethyl, trifluoromethyl, chlorofluoromethyl, difluoromethyl 1, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-dufluoroethyl, 2,2,2-trifluoroethyl i. nonethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl,

2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl and pentafluoroethyl, · · · · · · · · · · · · · ·

Alkoxy: alkyl groups having straight or branched chain with 1 to 4 or 6 carbon atoms, which are connected via an oxygen atom (-0-) bonded to the backbone, for example C ₁ -C ₆ -alkoxy such as methyloxy, ethyloxy, propyloxy, 1- methyletyloxy, butyloxy, 1-methylpropyloxy, 2-methylpropyloxy, 1,1-dimethyletyloxy, pentyloxy, 1-methylbutyloxy, 2-methylbutyloxy, 3-methylbutyloxy,

2,2-dimethylpropyloxy, 1,1-dimethylpropyloxy, 2-methylthioxy, 1.1- dime tylb u tyoxox y, 1,3-dimethylbutyloxy, 2,3-dimethylbutyloxy, 2-ethylbenzyloxy, 1 - e t y 1 r o py 1 o x y, h e x y .1. oxy, 1,2-dimethylpropyloxy, 1-methylptytyloxy, 3-methylpolyoxy, 4-methylpolyloxy, 1,2-dime tylbutyloxy, 2.2-dimethylbutyloxy, 3,3-dimethylbutyloxy, 1-ethylbutyloxy, 1,1,2-trimethylpropyloxy, 1,2,2-Trimethylpropyl χ; y, 1 - e t y 1 -1-met ip oil i oxy a

1-Ethyl-2-methylpolyoxy,

Alkoxycarbonyl: straight or branched chain alkyl groups having 1 to 6 carbon atoms, which are bonded to the backbone via an oxycarbonyl group (-00 (= 0) -),

Haloadkoxy: straight or branched chain alkyl groups having 1 to 4 or 6 carbon atoms, in which groups the hydrogen atoms may be partially or fully replaced by halogen atoms, which groups are attached to the skeleton via an oxygen atom,

Alkylthio: alkyl groups straight or branched chain with 1 to 4 or 6 carbon atoms, which are connected via a sulfur atom (-S-) bonded to the backbone, for example C ₁ -C ₆ alkylthio such as methylthio, ethylthio, propylthio, 1 -methylethylthio, butylthio,

1-methylpropylthio, 2-methylpropylthio, 1,1-dimethylethylthio, pentylthio, 1-methylbutylthio, 2-methylbutylthio, 3-methylbutylthio,

2,2-dimethylpropylthio, 1-ethylpropylthio, hexylthio,

1,1-dimethylpropylthio, 1,2-dimethylpropylthio, 1-methylpentylthio,

2 - m e t y 1 p e n t y .11 i o, 1,1-dimethylbutylthio, 1, 3 - dime t y 1. b u t y 11 i o, 2,3-dimethylbutylthio, 2-ethylbutylthio, 3 - meters 1. p e n t 11 i, 4 - meters 1 p e n t 11 i, 1,2-dimethylbutylthio, 2.2-dimethylbutylthio, 3,3-dimethylbutylthio, 1-ethylbutylthio, 1,1,2-trimethylpropylthio,

-e ty 1 -1 -me tylpr opy 11 i o a.

1,2,2-trimethylpropylthio,

1-ethyl-2-methylpropyl i,

Cycloalkyl: monocyclic alkyl groups having 3 to 6 ring carbon members, for example cyclopropyl, cycloalkyl, cycloalkyl and cycloalkyl,

Alkenyl is alkenyl straight or branched chain having 2 to 6 or 10 carbon atoms and a double bond in any position, for example C ₂ -C ₆ -a1keny1 as ethenyl, 1-propeny1, 2-propenyl, 1-methylethenyl, 1 -butenyl, 2-butenyl,

3-Butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl,

1-methyl-2-propenyl,

2-methyl-2-propenyl,

1-pentenyl,

- p e n t e n y 1, 3 - p e n t e n y 1,

4-pentenyl,

2-methyl-1-butenyl,

2-Methyl-2-butenyl,

3-methyl-1-butenyl,

-me ty .1 - 2 - b u tenyl,

1-methyl-1-butenyl,

1-methyl-2-butenyl,

1-Methylen-3-butenes 1,

-methyl. - 3-butenyl,

3-methyl-3-butenyl,

1,1-dimethyl-2-propenyl,

1,2-Dimethyl-1-propenyl,

1,2-dimethyl-2-propenyl,

-ethyl-1-propenyl 1,1-ethyl-2-propenyl, 1-hexenyl, 2-hexenyl,

3-hexenyl,

4-hexenyl,

5-hexenyls,

1-Methyl-1-pentenyl,

2-Methyl-1-pentenyl

- methods .1 - 2 - foams 1,

4-Methyl-2-pentenyl

3-Methyl-3-pentenyl

2-methyl-4-pentenyl,

3-Methyl-1-pentenyl

2-Methyl-2-pentenyl

1-methyl-3-pentenyl,

4-Methyl-3-pentenyl

3-Methyl-4-pentenyl

4-methyl-1-pentenyl,

3-Methyl-2-pentenyl

2-methyl-3-pentenyl,

1-methyl-4-pentenyl,

4-Methyl-4-pentenyl

1,1-dimethyl-2-butenyl,

1,2-dimethyl-1-butenyl,

1,2-dimethyl-3-butenyl,

1,3-dimethyl-2-butenyl,

1,1-dimethyl-3-butenyl,

1,2-dimethyl-2-butenyl,

1,3-dimethyl-1-butenyl,

1,3-dimethyl-3-butenyl,

2,2-dimethyl-3-butenyl,

2,3-dimethyl-2-butenyl,

3,3-dimethyl-1-butenyl,

2,3-dimethyl-1-butenyl.,

2,3-dimethyl-3-butenyl,

3,3-dimethyl-2-butenyl

1-ethyl-1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl,

2-ethyl-1-butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl,

1,1,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl,

-ethyl-2-methyl-1-propenyl and 1-ethyl, 2-methyl-2-propenyl,

Alkenyloxy: straight or branched chain alkylene groups of 2 to 6 carbon atoms and a double bond at any position, which are bonded to the backbone via an oxygen (-O-) atom,

Alkenyl carborryl: straight or branched chain alkenyl groups having 2 to 10 carbon atoms and a double bond at any position, which are bonded to the backbone via a carbonyl group (—CO—),

Alkynyl: alkynyl groups having straight or branched chain having 2 to 10 carbon atoms and a triple bond in any position, for example C ₂ -C ₆ -alkynyl such as ethynyl, 2-propynyl,

2-butynyl, 3-butynyl, 1-methyl-2-propynyl, 2-pentynyl,

3-pentynyl, 4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl,

2-methyl-3-butynyl, 1,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl,

1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1-methyl-4-pentynyl,

2-methyl-3-pentynyl, 2-methyl-4-pentynyl, 3-methyl-4-pentynyl,

4-methyl-2-pentynyl, 1,1-dimethyl-2-butynyl,

1,1-dimethyl-3-butynyl, 1,2-dimethyl-3-butynyl,

2,2-dimethyl-3-butynyl, 1-ethyl-2-butynyl, 1-ethyl-3-butynyl,

2-ethyl-3-butynyl and 1-ethyl-1-methyl-2-propynyl;

-2.7Alkynylcarbonyl ________: straight or branched chain alkynyl groups having 3 to 10 carbon atoms and a triple bond at any position, which are bonded to the backbone via a carbonyl group (-CO--),

Cycloalkoxy: monocyclic alkenyl groups of 3 to 6 carbon atoms which are bonded to the backbone via an oxygen atom, for example cyclopropyl, cyclopentyl or cyclohexyl,

He t e r o c y k .1. y 1 r e s p. heterocyclyloxy: Lr 1- to 6-member, saturated or partially monounsaturated mono- or polycyclic he terocy tusks that contain one to t are heteroaternized from group consisting of > e from oxygen, nitrogen <·. and which are sulfur directly resp. (hetero cycles and oxy) through the atom oxygen bound to skeleton, for example k 1 and d 2 -1 e t r a hv d r o f u iranyl, oxiranyl, 3-1 e t: raby dr of uranyl 2-1 E t rahydrothienyl, 3-1 et rahydro thiene1, 2-pyrrolidinyl, 3-pyrrole di. ny 1, 3-isoxazoldinyl, 4 - also from ox and from .1 diy 1, 5-i from ox and from oldi ny1, 3 - i o o t i a o o 1 d 1 4-isothiazole1, 5 - i z o t i and z o 1 d i ny 1, 3 - p y r a z o 1 i. 4-paryzolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-ox a z i i d i 1, 2-thiazolidinyl, 4 -1 i and z oli di ny 1, 5-1 i and o1i di ny1, 2-imidazolidinyl, 4-imi da from oli di ny1 1,2,4- -oxadiazoiidin-3.yl,

1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazidin-3-yl,

1,2,4-thiadiazolidin-5-yl, 1,2,4-triazolidin-3-yl

1,3,4-oxadiazol-2-yl-1,3,4-thiadiazolidin-2-yl;

1,3,4'-triazolidin-2-yl, 2,3-dihydrofur-2-yl,

2,3-dihydrofur-3-yl

2,3-dihydro-fur-5-yl,

2,5-dihydro-fur-3-yl,

2,3-dihydrothien-3-yl,

2,3-dihydro-fur-4-yl,

2,5-dihydro-fur-2-yl,

2,3-dihydrothien-2-yl,

2,3-dihydrothien-4-yl,

2,3-dihydrothien-5-yl,

2, 5 - d i h y d r o t - 3 - y 1,

2,3-dihydropyrrol-3-yl,

2,3-dihydropyrrole-5-yl,

2,5-dihydroparrol-3-yl,

2,3-dihydroisoxazol-4-yl,

4,5-dihydroisoxazol-3-yl,

4,5-dihydroisoxazol-5-yl,

2,5-dihydroisothiazol-4-yl;

2,3-di.hydropyrazol-3-yl,

2,3-dihydroparyzol-5-yl,

4,5-dihydropyrazol-1-yl,

2,5-dihydropyrazol-3-yl,

2,5-dihydropyrazol-5-yl;

2,3-dihydrooxazol-4-yl,

4,5-dihydrooxazol-2-yl, 4,5-dihydrooxazo-5-yl-2,5,5-dihydrooxazol-4-yl;

2,3-dihydrothiazol-2-yl,

2,3-dihydrothiazol-5-yl,

4,5-dihydropyrido-4-yl,

2,5-dihydrothiazol-2-yl,

2,5-dihydrothiazol-5-yl,

2,3-dihydroimidazol-4-yl

4,5-dihydroimidazol-2-yl

4,5-dihydroimidazo 1-5-yl 1,2,3

2,5-dihydrothien-2-yl,

2.3-dihydropyrrole-2-y1,

2,3-dihydropyrrole-4-yl,

2,5-dihydropyrrol-2-yl,

2,3-dihydroisoxazol-3-yl,

2,3-dihydroisoxazol-5-yl,

4,5-dihydroisoxazol-4-yl,

2,5-dihydroisothiazol-3-yl,

2,5-dihydroisothiazol-5-yl,

2,3-dihydropyrazol-4-yl,

4.5- dihydro-pyrazol-3-yl, _R 5 dlhydropyrazol.-5-yl,

2,5-dihydropyrazol-4-yl,

2.3- drooxa z o1-2-v 1,

2,3-dihydrooxazol-5-yl,

4,5-dihydrooxazol-4-yl,

2,5-dihydrohydroazol-2-yl;

2,5-dihydrooxazol-5-yl;

2,3-dihydrothiazol-4-yl,

4.5- di hy dro t i z1-2-y1,

4,5-dihydrothiazol-5-yl,

2,5 - d i hy d r o t 1 - 4 - y 1,

2,3-dihydroimidazol-2-yl,

2,3-dihydroimidazol-5-yl,

4,5-dihydroimidazol-4-yl,

-di hydroimidazol-2-yl,

2,5-dihydroimidazol-4-yl, 2,5-dihydroimidazol-5-yl,

2-morpholinyl, 3-morpholinyl, 2-piperidinyl, 3-piperidinyl,

4-piperidinyl, 3-hexahydropyridazine, 4-hexahydropyridazinyl,

2-hexahydropyrimidinyl, 4-hexahydropyrimidinyl,

5-hexahydropyrimidinyl, 2-hexahydropyrazinyl,

• · ···· · · ··· · · · · · ·

1,3,5-hexahydrotriazin-2-yl, 1,2,4-hexahydrotriazin-3-yl,

1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, 2-tetrahydropyran,

1,3-dioxolan-2-yl, 3,4,5,6-tetrrahydropyridin-2-yl,

4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl,

1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl

2H-1,4-benzothiazin-3-yl 2H-1,4-benzoxazin-3-yl

1,3-dihydrooxazin-2-yl 1,1,3-di-thian-2-yl, optionally substituted via a nitrogen atom, bound saturated or partially or totally unsaturated cycles, ______ which ________ be purged ____ of the atom

nitrogen through which they are vases except for ring members The carbon may contain one up to five heteroatoms from the group

nitrogen, oxygen and sulfur: three to twelve-membered saturated or partially or fully senasycled mono- or polycyclic systems containing, in addition to the nitrogen atom through which they are bound and annular members, one to five additional heteroatoms from the group consisting of nitrogen, oxygen and sulfur, and in the event that the cycle contains more than one annular oxygen and / or sulfur member, the oxygen and / or sulfur atoms are not, respectively. sulfur adjacent to one another, for example: 1-aziridinyl, 1-diaziridinyl, 1-acetidinyl, 1-pyrrolidinyl,

- i from oxazole i di 1, 2 - i z o t i and from ol i di. ny 1, 1 - py r z z i i ny ny 1,

- oxa z o i i di 1 i 3 -1 i and z o i i di i i, 1 - imi z z i i d i n i 1,

1,2,4-oxadiazolidin-2-yl, 1,2,4-oxadiazolidin-4-yl,

1,2,4-thiadiazolidin-2-yl 1,1,2,4-thiadiazolidin-4-yl,

-tr i.azolidines 1,

1,3,4-thiadiazolidin-3-yl,

2,5-dihydropyrrol-1-yl

2,5-dihydroisoxazol-2-yl

2,5-dihydroisothiazol-2-yl

2,3-dihydropyrazol-2-yl

1,3,4-oxadiazolidin-3-yl,

2,3-dihydropyrrol-1-yl,

2,3-dihydroisoxazol-2-yl,

2,3-dihydroisothiazol-2-yl,

2,3-dihydropyrazol-1-yl,

4,5-dihydropyrazol-1-yl,

2,3-dihydrooxazol-3-yl,

2,3-dihydroimidazol-1-yl

2,5-dihydroimidazol-1-yl, 1-piperazinyl,

1-hexahydropyrimidinyl,

4-thiomorpholinyl,

2,3-dihydroisoindol-2-yl, 1-pyrazolyl, 1-triazoles

-1 valleys 1, 1. - i ndaz o 1 y 1 pyrrolopyridi di-1-y1, pyrrolopyrimidin-1-yl, pyrrole-thiazin-1-yl, with name from py ri da zlu-1-yl, imidazopyrazin-1-yl, pyrazolopyridine iodo-1-ylpyrazolopyrazine-2,3-dihydrothiazol-3-yl, 4,5-dihydroimidazol-1-yl yl, 1-piperidinyl-4-morpholinyl,

- hexahy dr opyr i da z i riy 1,

2,3-dihydroindol-1-yl,

1,2,4-hexahydrotriazin-1-yl, 1-pyrrolyl, 1-imidazolyl,

1-tetrazolyl, 2-tetrazolyl, yl, benztriazol-1-yl, pyrrolidinopyrid-1-yl, pyrrolidopyridin-1-yl, iodine and pyridyl-1-yl. - y 1, imi d and z opy r imi di-1-y 1, pyrazopyridin-1-yl, pyr and z 1 opy r imi di n-i-y 1, f

benzimidazole-1r

1-yl and parazolotriazin-1-yl,

Aryl resp. Aryloxy, Aryl, Arylcarbonyl and Arylsulfonyl: aromatic mono- or polycyclic hydrocarbon radicals which are directly or substantially free of carboxylic acid; (aryloxy) via an oxygen atom (-O-) or (arylthio) via a sulfur atom (-S-), (arylcarbonyl) via a carbonyl group (-CO-) or (arylsulfonyl) via a sulfonyl group (-SO ₂ -) linked to a skeleton such as phenyl, naphthyl and phenanthrenes; phenyloxy, naphthyloxy and phenanthrenyloxy and the corresponding carbonyl or sulfonyl binders,

Hetary1 resp. Hetaryloxy, Hetarylthio, Hetarylcarbonyl and Hetarylsulfonyl: aromatic mono- or polycyclic radicals which, in addition to the ring carbon members, may additionally contain one to four nitrogen atoms or one to three nitrogen atoms and one oxygen or sulfur atom or an oxygen or sulfur atom, and which are directly resp. (hetaryloxy) through an oxygen atom (-0-) or (hetarythio) sulfur atom (-S-),

··

· (Hetarylcarbonyl) via a carbonyl group (-CO-) or (hetarylsulfonyl) via a sulfonyl group (-SO ₂ -) attached to the backbone, for example

a five-membered heteroaryl containing one to three nitrogen atoms of a five-ring heteroaryl group which, in addition to the carbon atoms, may contain one to three nitrogen atoms as ring members, for example 2-pyrrolyl, 3-pyrrolyl, 3-pyrazo. lyl,

4-pyrazolyl, 5-pyrazolyl, 2-imidazolyl-1,4-imidazolyl,

1,2,4-triazol-3-yl and 1,3,4-triazol-2-yl,

a five-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and is sulfur or oxygen or one oxygen atom or one sulfur atom of a five-ring heteroaryl group which, in addition to carbon atoms, may contain one to four nitrogen atoms or one to three atoms nitrogen and one atom, sulfur or oxygen, or one oxygen atom, or sulfur as ring members, for example

2-furyl, 3-furyl, 2-thienyl, 3-thienyl, 2-pyrrolyl, 3-pyrrolyl,

3-isoxazolyl, 4-isoxazolyl, 5-isoxazolyl, 3-isothiazolyl,

4-isothiazolyl, 5-isothiazolyl, 3-pyrazolyl, 4-pyrazolyl,

5-pyrazolyl, 2-oxazolyl, 4-oxazolyl, 5-oxazolyl, 2-thiazolyl, 4-thiazolyl, 5-thiazolyl, 2-imidazolyl, 4-imidazolyl,

1,2,4-oxadiazol-3-yl, 1,2,4-oxadiazol-5-yl

1,2,4-thiadiazol-3-yl, 1,2,4-triazol-5-yl,

1,2,4-tri-o-3-yl-1,3,4-oxadiazol-2-yl,

1,3,4-thiadiazol-2-yl, 1,3,4-triazol-2-yl, fused five-membered heteroaryl containing one to four, nitrogen or one to three, nitrogen atoms and / or

-52One oxygen or sulfur atom: five-ring heteroaryl groups which, in addition to carbon atoms, may contain one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom or one oxygen or sulfur atom as ring members and carbon members or adjacent in which two adjacent. an annular one annular nitrogen and one carbon member may be linked to an aromatic or heteroaromatic bi- or polycycle, for example: benzoluranyl, isobenzofuranyl, benzolienyl, 1 zobenzothiyl, 1. valley 1, isool 1, benziz ox and oly 1, benzoxazolyl, benzoisothiazolyl, benzol azoyl, 1, indazolyl, benzimidazolyl 1, pyrrolidinylpyrrolidine 1, fu roprldilnyl, f uropyridyl zine 1, thiopyrrolidine ziyl, thiotrophiazine, imidium from opyridium 1., pyrazo-1-opyri-diyl, pyrazolopyrazinyl, is ox azo-1-opiated zisonyisoxazo 1 otriaziny 1., rrolopyridinyl , pyrro 1 opyraziiiy 1, fucopyridiazininyl, iuro L riaz .iiiyi, thienopyrimidyl, opyri dinyl imide, opyr aziyl imide, propylene pyridine ny1, pyrazolot riazine ny1,

L, i z oxazolopyrimidyl, oxazolopyridinyl, pyrrolidinyl zinyl, pyrrolidinyl and zinc, uropyrimides1, thiopyrrolidine. nyl, thiopyrazinyl 1, imidazopyridazinyl, imidazotriazine 1, pyra z olopyrimidyl1, isox azzo pyrrolidinyl1, isoxazolopyrazinyl, oxazolopridazinyl, oxazo 1 opyrimides 1, oxazo 1 opy Razyl, oxazo 1 otriazi ny .1., isothiazolopyridinyl, isothiazolopyrimides1, isothiazolothiazinyl, thiazolopyridinyl 1, triazolopyridinyl, triazolopyrazinyl ai, thiazolopyridinyl 1, thiazole 1, thiazolopyridinyl 1, thiazolopyridine zi ny1, triazolotriazinyl, o azopyri da zi ny1, isotiazo 1 opy raziny 1, thiazo.1 opyridazinyl, thiazo 1 oti a. zines 1, triazolopyrimidyl,

-33 ·· ♦ a · • · · 33 33 33 33 33 33 ♦

- a nitrogen-bonded five-membered heteroaryl containing one to four nitrogen atoms or a nitrogen-bonded fused 1-membered heteroaryl containing from one to five African nitrogen atoms:

five-ring heteroaryl groups which, in addition to the carbon atoms, may contain one to four nitrogen atoms respectively. one to three nitrogen atoms as ring members a. in which two adjacent ring carbon members can be linked to aromatic or heteroaromatic

Py-pyrazoles i,

1-indolyl, on a bl- or polycycle, from ring members, example 1-pyrrolyl,

-1 y i a z o 1. y 1., 1 -1 e t y a z o 1. y 1,

- in da z 1 y 1, benzi da da 1 -1-y .1., benzotriazo 1 -1-y 1., py.rrol.opyri.mid i. η-1-yl, py rol thre az R-1-yl, imidazopyridin-1-yl, imidazopyrimidin-1-yl, the rings being bonded through one nitrogen

1- imidazolyl,

2-tetrazolyl, pyro 1 opy ri di n -1-y 1, pyiro 1 opyri da zi 11 -1-y 1, py iro 1 opy razi η -1-y 1, i rn i da opy ri da zi η -1-γ 1, imidazopyrazin-1-yl, pyrazolopyridin-1-yl, pyrazol. opyrid z 1 n -1 -y 1, py r a z 1 op r imidin-1-y 1, py r a z oopyr z i η-1-y1 and py r a z o 1 o t r i and z i η -1-y 1,

- a six-membered heteroaryl containing one to three and three, respectively. one to four du atoms. with heteroaryl carbon atoms of four atoms

2-pyridinyl; one to members, for example

3-pyridazinyl-1,4-pyridazinyl, 2-pyrimidinyl 5-pyrimidinyl, 2-pyrazinyl,

1,2,4-triazin-3-yl and 1,2,4,5-tetrazin-3-yl, which may contain one to nitrogen as annular 3-pyridinyl, 4-pyridinyl, 4-pyrimidinyl,

1,3,5-triazin-2-yl, b is not fused six i, heteroaryl containing one

-36 nitrogen atoms of up to four nitrogen atoms: six-ring groups in which two adjacent annular groups can be joined by a buta-1,3-diene-1,4-diyl group 1 ad c h. I η o 1 lnem, isochi η o 1 i π em, quinoxaline, iieteroaryl carbon members, quinazoline at resp. the corresponding oxy-, thio-, carbonyl- or sulfonyl groups.

The indication optionally substituted in relation to group Z indicates that the groups concerned may be partially or wholly halogenated and / or that they may carry one to three of the following groups:

- cyano, nitro, hydroxy, mercapto, amino, carboxy,

a.not a. r b o ny 1, am i n o th th o. a r b o ny 1,

C 1 -C ₆ -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylcarbonyl, C ₁ -C ₆ -alkylsulfonyl, C ₃ -C ₆ -alkylsulfoxyl, C ₁ -C ₆ -alkoxy,

Ci-Cg-haloalkoxy, C ₁ -C ₆ -alkoxycarbonyl, _C-C6 alkylthio, Cj-C ₆ -alkylamino, di-C Cg-alkyamino, C ₁ -C ₆ alkylaminocarbonyl, the di-Cg -alkylaminocarbonyl, C1- _C6- alkylaminothiocarbonyl,

Di-C 1 -C 8 -alkyl aminothiocarbonyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkenyloxy or C (= NOR ^a ) -, - R ^b ,

C ₃ -C ₆ -cycloalkoxy, C ₃ -C ₆ -cycloalkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy and hetarythio, wherein the cyclic groups may be partially or fully halogenated or can carry

-35 * one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, h and 10g, C 1 -C 6 -alkyl,

C 1 -C 6 -haloalkyl,

C 1 -C ₆ -alkyl is If 1,

C j - C ₆ - alkyl 1 foxy 1,

C 6 -C 7 -alkoxycarbonyl,

C ₁ -C ₆ -alkoxy,

C 1 -C 8 -alkylthio,

C ₁ - C yha 1 ogena 1 ko xy,

Cj-Cg-al hernia well,

Di-Cy-Cy-allyl amino,

C ₁ -C ₆ alkylaminocarbonyl,

Di-C ₆ -C 8 -alkylaminocarbonyl, C ₁ -C ₆ -al. kyl aminothiocarbonyl,

Di-C ₁ -C ₆ -alkylainiriothiocarbonyl, C ₂ -C ₆ -alkenyl,

C ₂ -C ₆ -alkenyloxy, C (= NOR ^a ) -Ay-R ^b , or benzyl, benzyloxy, aryl, aryloxy, aryloxy, arylthio, hetaryl, hetaryloxy and hetarythio substituted with non-conventional groups, and / or that these groups may be one of these residues are linked by: Cy-Cy-alkylene, oxy-C ₁ C ₄ -alkyl only and oxy-C ₁ -C ₄ alkyleneoxy, wherein the alkylene chain may be partially or fully halogenated and / or may carry one to three C ₊ - C ₃ -alkyl.

Indication substituted by customary groups indicates that the radicals in question can be partially or fully halogenated and / or may carry one to three of the following substituents: cyano, nitro, C -C ₄ -a I ky I CyCyhalogenalkyl, C ₁ -C ₄ ~ al koxy,

C _x -C ₄ -haloalkoxy, C ₁ -C ₄ alkylthio, C ₁ -C ₄ -haloalkylthio, C j - C ₄ - alkyl and 1 to 1 and. Rbony 1, L-Y- .; 1. carbonyloxy, 1, phenyl, phenoxy, benzyl and benzyloxy and / or C (= NOR ^a ) -Ay-R ^b .

Partially or wholly halogenated ”indicates that in the groups so characterized, the hydrogen atoms may be partially or fully replaced by the same or different halogen atoms.

»- - -

In view of their biological activity, compounds of formula I in which m is 0 are preferred.

Equally preferred are compounds of formula I wherein R ¹ is methyl.

Further preferred are compounds I wherein R ³ is hydrogen, hydroxy, cyano, cyclopropyl, chloro, methyl, ethyl, 1-methylethyl, methoxy, methylthio or phenyl.

In addition, also they preferred compounds I in which R ³ is methyl.

Also preferred are compounds I wherein R ³ is methoxy.

Also preferred are compounds I wherein R ³ is cyano.

Also preferred are compounds I wherein R ³ is trifluoromethyl.

Also preferred are compounds I wherein R ³ is hydroxy.

Preference is also given to compounds I in which R ³ represents chlorine.

• ·· ·· ·· • 4 ·· • · • • · • • • • · ··· • · 4 · • ♦ · · • 4 • ··· • • • 9 · • · • • • ··· ·· ·· 44

-34Upřednostňovány are compounds I in which R ³ znameriří methylthio.

Also preferred are compounds I wherein R ⁴ is hydrogen, C ₁ -C ₆ -alkyl, arylalkyl, hetarylalkyl, aryloxyalkyl, hetaryloxyalkyl, aryl, hetaryl, C ₂ -C ₆ -alkenyl or C ₂ -C ₆ -a 1 to aryl .

Further preferred are compounds 1 wherein R ⁴ is C 1 -C 8 -alkyl.

Preference is also given to compounds I in which. R ⁴ represents methyl or ety1.

Also preferred are compounds I wherein R ⁴ is aryloxyalkyl or hetaryloxyalkyl.

Further preferred are compounds I wherein R ⁴ is arylalkyl or heteroarylalkyl.

Also preferred are compounds I , in which R ⁴ means aryl or hetaryl. Further preferred are compounds I, in which R ⁴ means C ₂ -C ₆ -alkenyl. Preference is also given to compounds I, in which R ⁴ means

C ₂ -C ₆ -alkynyl.

Further preferred are compounds of formula I wherein X is NOCH ₃ .

• ·

-38 - means choch ₃ .

It also means

in which compounds of the formula I are preferred

CHCH ₃ or CHCH ₂ CH ₃ .

Also preferred are compounds of the formula

I in which is 0.

Further preferred are compounds of formula I, in which is

NH or N-CH ₃ .

in which

Particularly preferred are compounds of formula is NH and R ¹ then methyl.

.1.

which

Up of dn e os tnovány is NH and R ¹ are also compounds of formula

I, in which

Also preferred are compounds of formula T wherein Y is O and R ¹ is methyl.

Also preferred are compounds of formula I wherein Z is optionally substituted, nitrogen-bonded heterocyclyl.

Further preferred are also compounds of formula I in which

Z is optionally substituted, nitrogen-bonded heteroaryl.

• · • ·

Particularly preferred are compounds of formula 1 wherein Z is optionally substituted 1-pyrrolyl, 1-pyrazolyl, 1-imidazolyl, 1-triazolyl or 1-tetrazolyl.

Particularly preferred for use are the compounds 1 listed and described in the following tables. In addition, independently of the combination in which they are listed, the groups listed as substituents in these tables represent a particularly preferred form of the substrate.

Table 1

S1o is a general formula

J>

in which R ³ represents a moiety Z with apprentices 11 in each case corresponding to one of the residues listed in Table A.

CO2CH3

NOR ⁴

OF

1.1

Table 2

Compounds of the general formula 1.2, in which R ³ denotes hydrogen, R ⁴ is methyl and the group Z corresponds for each compound 0-4k one of the radicals mentioned in Table Ά.

NOR ⁴

OF

CO ₂ CH ₃

1.2

Table 3

Compounds of the general formula 1.3, in which R denotes hydrogen, R ⁴ is methyl and the group Z corresponds for each compound is m uz θ from the de tkuuve n 1 characterized chvtabu CE A.

, NOR ⁴

OF

1.3 CONH ₂

Table. 4

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

CO ₂ CH ₃

1.4

Table 5

Compounds of the general formula 1.5, in which R denotes hydrogen, R ⁴ is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

1.5 _CONHCH3

Table 6

Compounds of formula (1.1) in which R @ ³ is hydrogen, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

The Bulk '7

Compounds of formula (1.2) in which R @ ³ is hydrogen, R ^{@ 4} ethyl after Z are each one corresponding to one of the radicals listed in Table A.

Table 8

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table.

Table 9

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 10

Compounds of formula (1.5) in which R @ ³ is hydrogen, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 11

Compounds of formula (1.1) in which R @ ³ is hydrogen, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 12

Compounds of formula (1.2) in which R @ ³ is hydrogen, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 13

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 14

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 15

Compounds of formula (1.5) in which R @ ³ is hydrogen, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 16

Compounds of general formula 1.1 in which:. R ³ is hydrogen, R ⁴ isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 17

Compounds of formula (1.2) wherein R ³ is hydrogen, R ⁴ isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 18

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 19

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4} isopropyl and Z is each one corresponding to one of the radicals listed in Table A.

Table 20

Compounds of the general formula 1.5, in which R ³ is hydrogen, R ⁴ and iso-propyl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 21

Compounds of formula (1.1) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 22

Compounds of formula (1.2) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 23

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propenyl and in which L @ 1 is a compound corresponding to one of the radicals listed in Table A.

Table 24

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals. listed in Table A.

Table 25

Compounds of formula (1.5) in which:. R ³ is hydrogen, R ^{4 is} 2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 26

Compounds of formula (1.1) in which R @ ³ is hydrogen, R ^{@ 4} E-3-chloro-2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 27

Compounds of formula (1.2) wherein R ³ is hydrogen, R ^{4 is} E-3-chloro-2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 28

Compounds of formula (1.3) wherein R ³ is hydrogen, R ^{4 is} E-3-chloro-2-propenyl, and Z is then. a compound corresponding to one of the residues listed in Table A.

• ·

-4fTTable 29

Compounds of the general formula 1.4, in which R ^J is hydrogen, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 30

Compounds of the general formula 1.5, in which R ³ is hydrogen, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 31

Compounds of formula 1.1 wherein R ³ is hydrogen, R ⁴ n-butyl and a group. Z then. a compound corresponding to one of the residues listed in Table A.

Table 32

Compounds of formula (1.2) in which R @ ³ is hydrogen, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 33

Compounds of the general formula 1.3, in which R ³ is hydrogen, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 34

Compounds of the general formula 1.4, in which R ³ is hydrogen, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

Λ *

Table 35

Compounds of the general formula 1.5, in which R ³ is hydrogen, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 36

Compounds of the general formula 1.1, in which R ³ denotes hydrogen, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 37

Compounds of formula (1.2) wherein R ³ is hydrogen, R ⁴ CH ³ . and Z is a compound corresponding to one of the radicals listed in Table A.

Table 38

Compounds of the general formula 1.3, in which R ³ denotes hydrogen, R ⁴ CH ₂ F and R 7 corresponds for each compound to one of the radicals mentioned in Table A.

Table 39

Compounds of the general formula 1.4, in which R ³ denotes hydrogen, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 40

Compounds of the general formula 1.5, in which R ³ denotes hydrogen, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-41Table 41

Compounds of the general formula 1.1, in which R ^J is hydrogen, R ⁴ CHF ₂ and -S to a compound of the levers, each corresponding to one of the radicals mentioned in Table A.

Table 42

Compounds of the general formula 1.2, in which R ³ means hydrogen, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 43

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4} CH.F @ ₂ and Z are each corresponding to one of the radicals listed in Table A.

Table 44

Compounds of the general formula 1.4, in which R ³ is hydrogen, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 45

Compounds of the general formula 1.5, in which R ³ is hydrogen, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 46

Compounds of formula (i). 1, in which. R ³ means hydrogen, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

Table. 4'7

Compounds of the general formula 1.2, in which R ³ is hydrogen, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 48

Compounds of formula (1.3) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 49

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 50

Compounds of formula (1.5) wherein R ³ is hydrogen, R ^{4 is} 2-propynyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 51

Compounds of general formula 1.1 in which:. R ³ represents hydrogen, R ⁴ CH ₂ CF ₃ and a group. Z then each corresponds to one of the radicals listed in Table A.

Table 52

Compounds of the general formula 1.2, in which R ³ denotes hydrogen, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ········································ · ·· ·· · · · ·

Table 53 The compounds of general formula 1.3, in which R ³ is hydrogen., R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 54

Compounds of formula (1.4) in which R @ ³ is hydrogen, R ^{@ 4} and Z are each corresponding to one of the radicals listed in Table A.

Table 55

Compounds of the general formula 1.5, in which R ³ denotes hydrogen, R ⁴ CH ₂ CF ₃ and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 56

Compounds of formula 1.1 wherein R ³ is hydrogen, R ⁴ CH ₂ CH ₂ OCH ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 57

Compounds of the general formula 1.2, in which R ³ denotes hydrogen, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 58

Compounds of the general formula 1.3, in which R ³ denotes hydrogen, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

99 9

999

-ΓΟTable 59

Compounds of the general formula 1.4, in which R ³ denotes hydrogen, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 60

Compounds of formula (1.5) in which R ³ is hydrogen, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each one corresponding to one of the radicals listed in Table A.

Table 61

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 62

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 63

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 64

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• ·

-5Γ4Table 65

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 66

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 67

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 68

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4} ethyl and Z are the elephants of the value corresponding to one of the radicals listed in Table A.

Table 69

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 70

Compounds of the general formula 1.5, in which R ³ is cyano, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-2 Table 71

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 72

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table 5.

Table 73

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 74

Compounds of formula (1.4) in which R ^{@ 3} is cyano, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 75

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 76

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

-Γ3Table 77

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 78

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 79

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table.

Table 80

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 81

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 82

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 83

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 84

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 85

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 86

Compounds of formula (1.1) wherein R @ ³ is cyano, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 87

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} E-3-chloro-2-propropenyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 88

Compounds of the general formula 1.3, in which R ³ is cyano, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· A a a a a a a a a a a a a a a a a a a a a a a a a a a a a a aaa ·· aaa ·· ·· ··· *

Table 89

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 90

Compounds of the general formula 1.5, in which R ³ is cyano, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 91

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4} n -butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 92

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4} n -butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 93

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 94

Compounds of formula (1.4) in which R @ ³ is cyano, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·······················

Table 95

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4 is} n-butyl and Z is each one of the radicals listed in Table A.

Table 96

Compounds of formula (1.1) in which R @ ³ is cyano, R @ ⁴ CH3 F and Z are each one corresponding to one of the radicals listed in Table A.

Table 97

Compounds of formula (1.2) in which R ³ denotes cyano, R ⁴ CH ₂ F and Z each represent a compound corresponding to one of the radicals listed in Table A.

Table 98

Compounds of the general formula 1.3, in which R ³ is cyano, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 99

Compounds of formula (1.4) in which R @ ³ is cyano, R @ ⁴ CP @ ⁴ F and Z are each one corresponding to one of the radicals listed in Table A.

Table 100

Compounds of vzrce 5.1, in which R ³ is cyano, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ················································· · ·· ·· · »··

Table 101

Compounds of formula Ι.Ί in which R ^J is cyano, R ⁴ C; and Z is a compound corresponding to one of the radicals listed in Table A.

Table 102

Compounds of the general formula 1.2, in which R ³ is cyano, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 103

Compounds of vzrce 1.3, in which R ³ is cyano, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 104

Compounds of formula (1.4) wherein:. R ³ is cyano, R ^{4 is} C 1-6 and Z is a compound corresponding to one of the radicals listed in Table A.

Table 105

Compounds of formula (1.5) wherein R ³ is cyano, R ⁴ CHF ₂ and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 106

Compounds of formula (1.1) in which R @ ³ is cyano, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

• • •

-nTable 107

Compounds of formula (1.2) in which R @ ³ is cyano, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 108

Compounds of formula (1.3) in which R @ ³ is cyano, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in the table. AND.

Table 109

Compounds of the general formula 1.4, in which R ³ is cyano, R ⁴ 2-propynyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 110 '

Compounds of formula (1.5) in which R @ ³ is cyano, R ^{@ 4 is} 2-propynyl and Z is each corresponding to one of the radicals listed in Table A.

Table 111

Compounds of formula 1.1 wherein R ³ is cyano, R ⁴ CH ₂ CF ₃ and Z then. a compound corresponding to one of the residues listed in Table A.

Table 112

Compounds of formula (1.2) in which R ³ is cyano, R ⁴ CH ₂ CF ₃ and Z are each one corresponding to one of the radicals listed in Table A.

• · • ·

-5 ^ Table 113

Compounds of the general formula 1.3, in which R ³ is cyano, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 114

Compounds of the general formula 1.4, in which R ³ is cyano, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 115

Compounds of the general formula 1.5, in which R ³ is cyano, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 116

Compounds of the formula 1,1 in which R ³ is cyano, R ⁴ CH ₂ CH ₂ OCH ₃ and Z each represent a compound corresponding to one of the radicals listed in Table A.

Table 117

Compounds of the general formula 1.2, in which R ³ is cyano, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 118

Compounds of the general formula 1.3, in which R ³ is cyano, R ⁴ CH ₂ CH ₂ 0CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• • •

- € 0Table 119

Compounds of the general formula 1.4, in which R ³ is cyano, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 120

Compounds of the general formula 1.5, in which R ³ is cyano, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 121

Compounds of formula (1.1) in which R @ ³ is nitro, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 122

Compounds of the general formula 1.2, in which R ³ is nitro, R ⁴ is methyl and the group Z compound corresponding to each one of the radicals mentioned in Table A.

Table 123

Compounds of formula (1.3) in which R @ ³ is nitro, R ^{@ 4} methyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 124

Compounds of formula (1.4) in which R @ ³ is nitro, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 125

Compounds of formula (1.5) in which R @ ³ is nitro, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 126

Compounds of the general formula 1.1, in which R ³ is nitro, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 12.7

Compounds of formula (1.2) in which R @ ^{3 is} a! nitro, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 128

Compounds of formula (1.3) in which R @ ³ is nitro, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 12.9

Compounds of formula (1.4) in which R @ ³ is nitro, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 130

Compounds of formula (1.5) in which R @ ³ is nitro, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

• · • ·

-62.Table 131

Compounds of formula (1.1) in which R @ ³ is nitro, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 132

Compounds of formula (1.2) in which R @ ³ is nitro, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 133

Compounds of formula (1.3) in which R @ ³ is nitro, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 134

Compounds of formula (1.4) in which R @ ³ is nitro, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 135

Compounds of formula (1.5) in which R @ ³ is nitro, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 136

Compounds of formula (1.1) in which R @ ³ is nitro, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

• · • ·

-63Table '137

Compounds of formula (1.2) in which R @ ³ is nitro, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 138

Compounds of formula (1.3) in which R @ ³ is nitro, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 139

Compounds of formula (1.4) wherein:. R ³ is nitro, R ⁴ and iso-propyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 140

Compounds of formula (Ib) wherein R ³ is nitro, R ⁴ isopropyl. and group Z then. a compound corresponding to one of the residues listed in Table A.

Table 141

Compounds of the formula 1.1 in which R @ ³ is nitro, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 142

Compounds of formula (1.2) in which R @ ³ is nitro, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

• «« β β β β β β β β β β β β β β β β β β β β β β

Table. 14 3

Compounds of formula (1.3) wherein R ³ is nitro, R ^{4 is} 2-propenyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 144

Compounds of formula (1.4) in which R @ ³ is nitro, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 145

Compounds of formula (1.5) in which R @ ³ is nitro, R ^{@ 4 is} 2-propenyl, and Z is one in each case. from residues listed in Table Leo A.

Table 146

Compounds of the general formula 1.1, in which R ³ is nitro, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 147

Compounds of the general formula 1.2, in which R ³ is nitro, R ⁴ E-3-chl.or-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 148

Compounds of formula (1.3) in which:. R ³ represents, nitro, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• • • •

-65 * - Table 149 Compounds of general formula 1.4, in which nitro, R ⁴ E-3-chloro-2-propenyl and skupina wherein R ³ is L then the compound

corresponding to one of the residues listed in Table A.

Table 150

Compounds of the general formula 1.5, in which R ³ is nitro, R ⁴ E-3-chloro-2-propeny1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 151

Compounds of formula (1.1) in which R @ ³ is nitro, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 152

Compounds of the general formula 1.2, in which R ³ is nitro, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 153

Compounds of the general formula 1.3, in which R ³ is nitro, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 154

Compounds of formula (1.4) in which R @ ³ is nitro, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

·· ·· · · · · · · · · · · · · · · · · · · · · · · · · · · ·

66Compounds of the general formula nitro, R ⁴ n-butyl and a group. . one of the residues mentioned

1.5 wherein R ³ represents a corresponding compound

Wherein R ³ represents the corresponding compound in each case

1.1, ve

The compounds of the general formula nitro, R ⁴ CH ₂ F and Z are then one of the radicals listed in Table A.

Table 157 means

Table 158

Compounds of the general formula 1.3, in which R ³ is nitro, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 159

Nitro compounds, R ⁴ to one of the groups

ClTF and Z are each a compound corresponding to the residues listed in Table A.

Table 160

Compounds according to

CH ₂ F and a group of radicals of formula 1.5 wherein R ³ is nitro, R ⁴ Z is a compound corresponding to one of Table A.

• · • ·

€ Ί- -

Table 16'1

Compounds of the general formula 1.1, in which R ³ is nitro, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 162

Compounds of the general formula 1.2, in which R ³ is nitro, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 163

Compounds of the general formula 1.3, in which R ³ is nitro, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 164

Compounds of formula (1.4) in which R @ ^{3 is} a! nitro, R ⁴ CHF ₂ and Z then each corresponding to one of the radicals listed in Table A.

Table 165

Compounds of the general formula 1.5, in which R ³ is nitro, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 166

Compounds of formula (1.1) in which R @ ³ is nitro, R ^{@ 4 is} 2-propynyl and Z is each corresponding to one of the radicals listed in Table A.

Table 167

Compounds of the general formula 1.2, in which R ³ is nitro, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 168

Compounds of formula (1.3) in which R @ ³ is nitro, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 169

Compounds of the general formula 1.4, in which R ³ is nitro, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 170

Compounds of formula (1.5) in which R @ 1 is nitro, R ^{@ 4 is} 2-propynyl and Z then each corresponds to one of the radicals listed in Table A.

Table 171

Compounds of formula (1.1) wherein R ³ is nitro, R ^{4 is} CllyCl ² ; and Z is a compound corresponding to one of the radicals listed in Table A.

Table 172

Compounds of formula (1.2) in which R ³ is nitro, R ⁴ αΐχΓ ₃ and Z are each one corresponding to one of the radicals listed in Table A.

• ·

-69Table. 1'7 3

Compounds of the general formula 1.3, in which R ^J is nitro, R ⁴ CH ₂ CF ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 174

Compounds of the general formula 1.4, in which R ³ is nitro, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 175

Compounds of the general formula 1.5, in which R ³ is nitro, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 176

Compounds of the general formula 1.1, in which R ³ represents, nitro, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1.77

Compounds of the general formula 1.2, in which R ³ is nitro, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 178

Compounds of the general formula 1.3, in which R ³ is nitro, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

A AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA AAA

Table 179

Compounds of the general formula 1.4, in which R ³ is nitro, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 180

Compounds of the general formula 1.5, in which R ³ is nitro, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 181

Compounds of formula (1.1) in which R @ ³ is hydroxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 182

Compounds of formula (1.2) in which R @ ³ is hydroxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 183

Compounds of formula (1.3) in which R @ ³ is hydroxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1.8 4

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• · · • · «4 4 4 4 4 4 4 4« »·

-ΉTable 185

Compounds of formula (1.5) in which R @ ³ is hydroxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 186

Compounds of formula (1.1) in which R @ ³ is hydroxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 187

Compounds of the general formula 1.2, in which R ³ is hydroxy, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 188

Compounds of formula (1.3) in which R @ ³ is hydroxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 189

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 190

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Φ · «· · · · · · · · · · · · · · · · φ φ φ φ φ φ φ φ φ · φ 9 99

999 99 99 9999

Table 191 of the formula

Compounds of general hydroxy, R ⁴ propyl and the group L are each one of the radicals mentioned

1.1 wherein R ³ is; 1 instructed in u. Corresponding in Table A.

Table 192

Compounds of the formula hydroxy, R ⁴ propyl and a group, each of which is mentioned above

1.2, wherein R ³ is the compound corresponding to Table A.

Table 193

1.3, wherein R ³ is the compound corresponding to Table A.

Table 194

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 195

Compounds of formula (1.5) in which R @ ³ is hydroxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 196

Compounds of formula 1.1 wherein R ³ is hydroxy, R ⁴ isopropyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

• · · · ·

-73Table 197

Compounds of formula (1.2) wherein R 1 is ^: sign! hydroxy, R ⁴ isopropyl and Z then a compound corresponding to one of the radicals listed in Table A.

Table 198

Compounds of formula (1.3) in which R @ ³ is hydroxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 199

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 200

Compounds of formula (1.5) in which R @ ³ is hydroxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 201.

Compounds of formula (1.1) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 202

Compounds of formula (1.2) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 203

Compounds of formula (1.3) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 204

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 205

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 206

Compounds of the general formula 1.1, in which R ³ is hydroxy, R ⁴ E-3-chl.or-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 207

Compounds of the general formula 1.2, in which R ³ is hydroxy, R @ ⁴ -3-E-2-ch1or propeny1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 208

Compounds of the general formula 1.3, in which R ³ is hydroxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- Ί-ϋΓTable 209

Compounds of formula 1.4 , in who R ³ represents hydroxy, R ⁴ E-3-chloro-2-propenyl a group Z then the compound corresponding always one of the leftovers listed in Table A. Table 210 Compounds 1.5 , in who R ³ represents hydroxy, R ⁴ E - 3 - c h 1 o r - 2 ~ p: fo es 1 a group Z then the compound corresponding always one of the leftovers. listed in Table A.

Table 211

Compounds of formula (1.1) in which R @ ³ is hydroxy, R ^{@ 4} n -butyl and Z is a compound corresponding to one of the radicals listed in Table.

Table 212

Compounds of formula (1.2) wherein R ³ is hydroxy, R ^{4 is} n-butyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 213

Compounds of the general formula 1.3, in which R ³ is hydroxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 214

Compounds of formula 1.4 wherein R ³ is hydroxy, R ^{4 is} n-butyl. and Z is a compound corresponding to one of the residues listed in Table A.

• · • ·

-? 6 ~

Table 215

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ n buty.1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 216

Compounds of the general formula 1.1, in which R ³ is hydroxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 217

Compounds of the general formula 1.2, in which R ³ is hydroxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 218

Compounds of the general formula 1.3, in which R ³ is hydroxy, R ⁴ CH ₂ F and the group Z corresponds for each compound pa.k one of the radicals mentioned in Table A

Table 219

Compounds of the general formula 1.4, in which R ³ is hydroxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 220

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

- -

Table 221

Compounds of the general formula 1.1, in which R ³ is hydroxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 222

Compounds of the general formula 1.2, in which R ³ is hydroxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 223

Compounds of the general formula 1.3, in which R ³ is hydroxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals listed in the above table.

Table 224

Compounds of the general formula 1.4, in which R ³ is hydroxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 225

Compounds of the general formula 1.5, in which R ³ is hydroxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 226

Compounds of the general formula 1.1, in which R ³ is hydroxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-78Table 227

Compounds of formula (1.2) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding only to the moieties listed in Table A.

Table 228

Compounds of the general formula 1.3, in which R ³ znameriíá hydroxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 229

Compounds of formula (1.4) in which R @ ³ is hydroxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 230

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 231

Compounds of formula 1.1 wherein R ³ is hydroxy, R ^{4 is} CH ² Cl 2 and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 232

Compounds of the general formula 1.2, in which R ³ is hydroxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 233

Compounds of the formula hydroxy, R ⁴ CH ₂ CF ₃ and Z each represent one of the radicals mentioned

Table 234

Compounds of the formula hydroxy, R ⁴ CH ₂ CF ₃ and Z each represent one of the radicals mentioned

Table 235

A hydroxy compound of general formula R ⁴ _CH? CF ₃ and Z each represent one of the radicals mentioned

1.3, wherein R ³ is the compound corresponding to Table 71.

1.4, wherein R ³ is the compound corresponding to Table A.

1.5, in which R ³ represents a compound corresponding to Table A.

Table 236

Compounds of the general formula 1.1, in which R ³ is hydroxy, R ⁴ CH ₂ CH ₂ OCH ₃ and skupirna Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 237

Compounds of formula (1.2) in which R ³ is hydroxy, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each a compound corresponding to the nucleus of the radicals listed in Table A.

Table 238

Compounds of the general formula 1.3, in which R ³ is hydroxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

- Table 239

Compounds of the general formula 1.4, in which R ³ is hydroxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 240

Compounds of the general formula 1.5, in which R ³ is hydroxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 241

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 242

Compounds of the general formula 1.2, in which R ³ is amino, R ⁴ is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 243

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 244

Compounds of formula (1.4) in which R @ ³ is amino, R ^{@ 4} methyl and Z is a compound corresponding to one of the radicals listed in Table A.

-81Table 245

Compounds of formula (1.5) in which R @ ³ is amino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 246

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table. 247

Compounds of formula 1.2 wherein R ³ is amino, R ^{4 is} ethyl. a. Z is a compound corresponding to one of the radicals listed in Table A.

Table 248

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 249

Compounds of formula (1,4) in which R @ ³ is amino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 250

Compounds of the general formula 1.5, in which R ³ is amino, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

··· • ·

44 4

4 44

Table 251

Compounds of the general formula 1.1, in which R ³ is amino, R ⁴ propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 252

Compounds of formula (1.2) in which R @ ³ is amino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 253

Compounds of the general formula 1.3, in which R ³ is amino, R ^4, and propyl group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 254

Compounds of formula (1.4) in which R @ ³ is amino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 255

Compounds of formula (1.5) in which R @ ³ is amino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 256

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

-831'abulka 2 57

Compounds of formula (1.2) in which R @ ³ is amino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 258

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 259

Compounds of formula (1.4) in which R @ ³ is amino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table.

Table 260

Compounds of formula (1.5) in which R @ ³ is amino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 261

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 262

Compounds of formula (1.2) in which R @ ³ is amino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Tables 2 63

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 264

Compounds of formula (1.4) in which R @ ³ is amino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 265

Compounds of formula (1.5) in which R @ ³ is amino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 266

Compounds of the general formula 1.1, in which R ³ is amino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 267

Compounds of the general formula 1.2, in which R ³ is amino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 268

Compounds of the general formula 1.3, in which R ³ is amino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-arTable 269

Compounds of formula 1.4 wherein R ³ is amino, R ^{4 is} E-3-chloro-2-propenyl; and Z is a compound corresponding to one of the radicals listed in Table A.

Table 270

Compounds of the general formula 1.5, in which R ³ is amino, R @ ⁴ -3-E-2-ch1oi propenyJ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 271

Compounds of the general formula .1.1 wherein R ³ is amino, R ⁴ and n-butyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 272

Compounds of the general formula 1.2, in which R ³ is amino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 273

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 274

Compounds of formula (1.4) in which R @ ³ is amino, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 275

Compounds of the general formula 1.5, in which R ³ is amino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 276

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4} CHg F and Z are each one corresponding to one of the radicals listed in Table A.

Table 277

Compounds of formula (1.2) wherein:. R ³ is amino, R ^{4 is} CH ₂ F and Z is then. the corresponding compound. one of the residues listed in Table A.

Table 278

Compounds of the general formula 1.3, in which R ³ is amino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 279

Compounds of the general formula 1.4, in which R ³ is amino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 280

Compounds of formula (1.5) wherein R ³ is amino, R ^{4 is} CH ₂ F and Z is then. a compound corresponding to one of the residues listed in Table A.

• ·

Table 281

Compounds of the general formula 1.1, in which R ³ is amino, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 282

Compounds of the general formula 1.2, in which R ³ is amino, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 283

Compounds of the general formula 1.3, in which R ³ znzimená amino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 284

Compounds of the general formula 1.4, in which R ³ is amino, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 285

Compounds of the general formula I.5 where ^R3 is amino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 286

Compounds of formula (1.1) in which R @ ³ is amino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

-83Table 287

Compounds of vzorxe 1.2, in which R ³ is amino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 288 Compounds general formulas 1.3 in which R ³ means amino, R ⁴ 2- propynyl and the group Z then a compound odpo \ Jew always one l of residues. listed in Table A. Table 289 Compounds general formula 1.4 in which R ³ z namená amino, R ⁴ 2- propi. ny 1. a. group. Z then the compound corresponding. always one i. from residues listed in Table A.

Table ^ 290

Compounds of formula (1.5) wherein R ³ is amino, R ^{4 is} 2-propynyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 2.

Compounds of the general formula I .1, in which R ³ is amino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 292

Compounds of formula (1.2) in which R @ ³ is amino, R ^{@ 4} and Z are each corresponding to one of the radicals listed in Table A.

Table 293

Compounds of formula (1.3) in which R @ ³ is amino, R ^{@ 4 is} C1LCr @ ₃ and group 7 are each one corresponding to one of the radicals listed in Table.

Table 294

Compounds of formula (1.4) in which R @ ³ is amino, R @ ⁴ Cl2 CF3 and Z are each one corresponding to one of the radicals listed in Table A.

Table 295

Compounds of the general formula 1.5, in which R ³ is amino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 296

Compounds of the general formula 1.1, in which R ³ is amino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 297

Compounds of the general formula 1.2, in which R ³ is amino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 298

Compounds of the general formula 1.3, in which R ³ is amino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• • •

-qoTable 299

Compounds of the general formula 1.4, in which R ³ is amino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 300

Compounds of the general formula 1.5, in which R ³ is amino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 301

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 302

Compounds of the general formula 1.2, in which R ³ is chlorine, R ⁴ is methyl and the group Z correspond to the compound no. one of the residues listed in Table A.

Table 303

Compounds of the general formula 1.3, in which R ³ is chlorine, R ⁴ is methyl and the group Z. a compound corresponding to one of the residues listed in Table A.

Table 304

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• · ·

Table 305 General apprenticeships formulas 1.5, in which R ’ means

chlorine, R ⁴ methyl and Z then each corresponding to one of the radicals listed in Table A.

Table 306

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 307

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 308

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 309

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 310

Compounds of formula (1.5) in which R @ ³ is chlorine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

- «92

Table 311 Compounds of general use formulas 1.1 in which] R ^{J is} known

chlorine, R ⁴ propyl and Z then each corresponding to one of the radicals listed in Table A.

Table 312

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 313

Compounds of formula ³ wherein R ³ is chlorine, R ⁴ propyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 314

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 315

Compounds of formula (1.5) in which R @ ³ is chlorine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 316

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

- ^ 3Table. 317

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 318

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 319

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 320

Compounds of formula (1.5) in which R @ ³ is chlorine, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 321

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 322

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

• • •

Tabulkři 323

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 324

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 325

Compounds of formula (1.5) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 326

Compounds of general formula 1.1 in which:. R ³ is chlorine, R ^{4 is} E-3-chloro-2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 327

Compounds of formula (1.2) in which R ³ is chlorine, R ^{4 is} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 328

Compounds of the general formula 1.3, in which R ³ is chlorine, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 329

Compounds of the general formula 1.4, in which R ³ is chlorine, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 330

Compounds of the general formula 1.5, in which R ³ is chlorine, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 331

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 332

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 333

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 334

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

«· • ·

00 00 00 00 0 0 0 0 0 0 0 0 · 40

Table 335

Compounds of the general formula 1.5, in which R ³ is chlorine, R ⁴ and n-butyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 336

Compounds of vzrce 1.1, in which R ³ is chlorine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 337

Compounds of the general formula 1.2, in which R ³ is chlorine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 338

Compounds of the general formula 1.3, in which R ³ is chlorine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 339

Compounds of the general formula 1.4, in which R ³ is chlorine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 340

Compounds of the general formula 1.5, in which R ³ is chlorine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- <ΎΤ ~

Table 341

Compounds of formula (i) in which R ³ is chlorine, R ⁴ CHF ₂ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 342

Compounds of the general formula 1.2, in which R ³ is chlorine, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 343

Compounds of the general formula 1.3, in which R ₃ is chlorine, _{R4, CHF2} and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 344

Compounds of the general formula 1.4, in which R ³ is chlorine, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 345

Compounds of the general formula 1.5, in which R ³ is chlorine, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 346

Compounds of formula (1.1) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Table 347

Compounds of formula (1.2) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 348

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 349

Compounds of formula (1.4) in which R @ ³ is chlorine, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 350

Compounds of formula (1.5) wherein R ³ is chloro, R ^{4 is} 2-propynyl. a. Z is a compound corresponding to one of the radicals listed in Table A.

Table 351

Compounds of formula (1.1) in which R @ ³ is chlorine, R @ ⁴ CH3 CF3 and Z are each corresponding to one of the radicals listed in Table A.

Table 352

Compounds of formula (1.2) wherein R ³ is chlorine, R ⁴ CH ₂ CF ₃ and Z then. a compound corresponding to one of the residues listed in Table A.

• ·

Table 353

Compounds of formula (1.3) in which R @ ³ is chlorine, R ^{@ 4 is} Cl2 CF3 and Z are each one corresponding to one of the radicals listed in Table A.

Table 354

Compounds of the general formula 1.4, in which R ³ is chlorine, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 355

Compounds of formula (1.5) in which:. R ³ represents chlorine, R ⁴ CrL ₂ CF ₃ and the group Z in each case corresponds to one of the radicals listed in Table A.

Table 356

Compounds of the general formula 1.1, in which R ³ is chlorine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 357

Compounds of the general formula 1.2, in which R ³ is chlorine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 358

Compounds of the general formula 1.3, in which R ³ is chlorine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-ΛΰΟ

Table 359

Compounds of the general formula 1.4, in which R ³ is chlorine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 360

Compounds of the general formula 1.5, in which R ³ is chlorine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 361

Compounds of formula (1.1) in which R @ ³ is bromine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 362

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 363

Compounds of formula (1.3) in which R @ ³ is bromine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 364

Compounds of formula (1.4) in which R @ ³ is bromine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

- / foj -

Table 1 and 365

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 366

Compounds of formula (I) in which R @ ³ is bromine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 367

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 368

Compounds of formula (1.3) in which R @ ³ is bromo, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 369

Compounds of formula (1.4) in which R @ ³ is bromine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 370

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

- ANL Table 371

Compounds of formula (1.1) in which R @ ³ is bromine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 372

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 373

Compounds of formula (1.3) in which R @ ³ is bromine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 374

Compounds of formula (1.4) in which R @ ³ is bromine, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 375

Compounds of the general formula 1.5, in which R ³ is bromine. R ⁴ propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 376

Compounds of formula (1.1) in which R @ ³ is bromine, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 377

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} isopropyl and Z are each one of the radicals listed in Table A.

Table 378 General Purposes formulas 1.3 in which. R ³ means bromo, R ⁴ isopropyl. and group. OF then the compound odpov idající always one of the leftovers listed in Table A. Table 379 General compounds formulas 1.4 in which R ³ means bromo., R ⁴ iso-propyl a group Z then the compound responds always one of the leftovers listed in Table A. Table. 380 S1 o u e u i n y generalized o formulas 1.5 in which R ³ means bromo, R ⁴ isopropyl and group Z then the compound odpov driving always one of the leftovers listed in Table A. Table 381 General compounds formulas 1.1. In which R ³ z namená bromo, R ⁴ 2-propenyl and group Z then the compound odpov driving always one of the leftovers listed in Table A. Table 382 General compounds formulas 1.2 in which R ³ means bromo, R ⁴ 2-propenyl and group Z then the compound odpov additional always one of the leftovers listed in Table A.

• ·

-AOh

Table 383

Compounds of formula (1.3) in which R @ ³ is bromo, R ^{@ 4 is} 2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 384

Compounds of formula (1.4) in which R @ ³ is bromo, R ^{@ 4 is} 2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 385

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4 is} 2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 386

Compounds of the general formula 1.1, in which R ³ is bromine, R ⁴ E-3-chloro-2-propenyl · and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 387

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} E-3-chloro-2-propylene and Z is a compound corresponding to one of the radicals listed in Table A.

Table 388

Compounds of formula (1.3) in which R @ ³ is bromine, R ^{@ 4} E-3-chloro-2-prenyl and Z are each one corresponding to one of the radicals listed in Table A.

- 4Off -

Table 389

Compounds of formula (1.4) in which R @ ^{3 is} a! bromine, R ⁴ E-3-chloro-2-propenyl and Z then each corresponding to one of the radicals listed in Table A.

Table 390

Merge Clay in general 1.5 in which R ³ z] namená bromine, R ⁴ E- 3-chloro-2-propenyl and a group. Z then compound corresponds to that to one of the residues. listed in the table AND. Table 391 Compounds in all cases 1.1 in which R ³ zi namená

bromine, R ⁴ n-butyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 392

Compounds of formula (1.2) in which R @ ^{3 is} a! bromo, R ⁴ n-butyl and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 393

Compounds of formula (1.3) in which R @ ³ is bromine, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 394

Compounds of formula (1.4) wherein R @ ³ is bromo, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 395

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4} n -butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 396

Compounds of the general formula 1.1, in which R ³ is bromine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 397

Compounds of the general formula 1.2, in which R ³ is bromine, R ⁴ CH ₂ F and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 398

Compounds of formula (1.3) wherein R ³ is bromo, R ⁴ CH ₂ F and the Z group then. a compound corresponding to one of the residues listed in Table A.

Table 399

Compounds of the general formula 1.4, in which R ³ is bromine, R ⁴ CH ₂ F e and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 400

Compounds of the general formula 1.5, in which R ³ is bromine, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · ·

-, ΛΟ £ ~

Table 401

Compounds of the general formula 1.1, in which R ³ is bromine, ^R4, _CHF2 and the group Z corresponds for each compound -jednomu of the radicals mentioned in Table A.

Table 402

Compounds of the general formula 1.2, in which R ³ is bromine, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 403

Compounds of formula (1.3) in which R @ ³ is bromine, R ^{@ 4} CHF, and Z are each one of the radicals listed in Table A.

Table 404

Compounds of formula (1.4) in which R is bromine, R ⁴ CHF ₂ and Z are each corresponding to one of the radicals listed in Table A.

Table 405

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4} Ciii ·, and Z are each corresponding to one of the radicals listed in Table A.

Table 406

Compounds of formula (1.1) in which R @ ³ is bromine, R ^{@ 4 is} 2-propynyl and Z is each one corresponding to one of the radicals listed in Table A.

-Λ06

Table 407

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4 is} 2-propynyl and Z is each one corresponding to one of the radicals listed in Table A.

Table 408

Compounds of formula (1.3) wherein R ³ is bromo, R ^{4 is} 2-propynyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 409

Compounds of formula (1.4) in which R @ ³ is bromine, R ^{@ 4 is} 2-propynyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 410

Compounds of formula (1.5) in which R @ ³ is bromine, R ^{@ 4 is} 2-propynyl and Z is each one corresponding to one of the radicals listed in Table A.

Table 411

Compounds of formula (1.1) in which R @ ³ is bromine, R ^{@ 4} Cl @ ¹ CF3 and Z are each one corresponding to one of the radicals listed in Table A.

Table 412

Compounds of formula (1.2) in which R @ ³ is bromine, R ^{@ 4} CH3 CF3 and Z are each one corresponding to one of the radicals listed in Table A.

• · • ·

- / 103Table. 413

Compounds of formula 1.3 wherein R ³ is bromo, R ⁴ CH ₂ CF _3, and Z is a compound corresponding to one of the residues listed in Table A.

Table 414

Compounds of the general formula 1.4, in which R ³ is bromine, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 415

Compounds of the general formula 1.5, in which R ³ is bromine, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 416

Compounds of the general formula 1.1, in which R ³ is bromine, R ⁴ CH ₂ CH ₂ OCH ₃ as the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 417

Compounds of the general formula 1.2, in which R ³ is bromine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 418

Compounds of the general formula 1.3, in which R ³ is bromine, R ⁴ CH ₂ CH ₂ 0CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

- 440 Table 419

Compounds of the general formula 1.4, in which R ³ is bromine, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 420

Compounds of the general formula 1.5, in which R ³ is bromine, R ⁴ CH ₂ CH ₂ 0CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 421

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 422

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 423

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 424

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• ··· 9J 99 ·· ·· · «9 9 9 9 9

9 9 999

9 9 9 9 9 9 999 9 9

9 9 9 9 9

9 99 99 99 99

- 444 _

Table 425

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 426

Compounds of formula (i). 1, in which R ³ is methyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 427

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 428

Compounds of formula (1.3) in which R ³ is methyl, R ^{4 is} ethyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 429

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 430

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

99 · ·· «· ·· ·· • • ·· • • • • · • • • • * • • ··· • · ·· • • • «· • • · • ··· • • • • • • • • · • • • ·· ··· ·· 99 ··

Table 431

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 432

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 433

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 434

Compounds of the general formula 1.4, in which R ³ represents methyl, R ⁴ propyl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 435

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 436

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

• • •

- / 143 Table 437

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 438

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 439

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4} isopropyl and Z is each one of the radicals listed in Table A.

Table 440

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 441

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1 42

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 443

Compounds of formula 1.3 in which R ³ is methyl, R ^{4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 444

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 445

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 446

Compounds of vziorce 1.1, in which R ³ is methyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 447

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 448

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- AIS '-

Table 44 9 and Compounds of the general formula 1.4, in which > rapid R ³ means methyl, R ⁴ E-3 - c .1. o r - 2 - fo rs .1 and Z group then the compound

corresponding to one of the residues listed in Table A.

Table 450

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-3 - chloro, or 2-propeny1 and the group Z corresponds for each compound jenodmu of the radicals mentioned in Table A.

Table 451

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 452

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 453

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 454

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 4 5.5

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 456

Compounds of the general formula 1.1, in which R ³ represents methyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 457

Compounds of the general formula 1.2, in which R ³ represents methyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 458

Compounds of the general formula 1.3, in which R ³ represents methyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 459

Compounds of the general formula 1.4, in which R ³ represents methyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 460

Compounds of the general formula 1.5, in which R ³ represents methyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

--mTable 461

Compounds of the general formula 1.1, in which R ³ is methyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 462

Compounds of the general formula 1.2, in which R ³ is methyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 463

Compounds of the general formula 1.3, in which R ³ is methyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 464

Compounds of formula 1.4 wherein R ³ is methyl, R ⁴ CHF ₂ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table. 4 65

Compounds of the general formula 1.5, in which R ³ represents methyl, R ⁴ CHF _2. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 466

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

-448Table 467

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 468

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 469

Compounds of the general formula 1.4, in kt.crých R ³ is methyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 470

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 471

Compounds of the general formula 1.1, in which R ³ represents methyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 472

Compounds of the general formula 1.2, in which R ³ represents methyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

-44 ^ Table 473

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ CIL ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 474

Compounds of the general formula 1.4, in which R ³ represents methyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 475

Compounds of the general formula 1.5, in which R ³ represents methyl, R ⁴ CH ₂ CF ₃ and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 476

Compounds in general! O formulas [.1 in which R ³ 7. riamená methyl, R ⁴ CH ₂ CH ₂ OCH ₃ a group Z pa k s 1. o u e n i n u odpo seeing always one of the leftovers listed in Table A. Table 477 Compounds of general formula formulas 1.2 in which R ³ means methyl, R ⁴ CH ₂ CH ₂ OCH ₃ a group Z then the compound corresponding always one of the leftovers listed in Table A. Table 478 General compounds formulas 1.3 in which R ³ means methyl, R ⁴ CH ₂ CH ₂ OCH ₃ a group Z then the compound odpovedájlei always one of the leftovers listed in Table A.

• · · · · · · · · · · · · · · ·

-42.0Table 47 9

Compounds of the general formula 1.4, in which R ³ represents methyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 480

Compounds of the general formula 1.5, in which R ³ mean methyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 481

Compounds of the general formula 1.1, in which R ³ is ethyl, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 482

Compounds of the general formula 1.2, in which R ³ is ethyl, R @ ⁴ methyl, and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 483

Compounds of formula (1.3) in which R @ ³ is ethyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 484

Compounds of the general formula 1.4, in which R ³ is ethyl, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

«*

Table 485

Compounds of formula (1.5) in which R @ ³ is ethyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 486

Compounds of the general formula 1.1, in which R ³ is ethyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 487

Compounds of the general formula 1.2, in which R ³ is ethyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 488

Compounds of the general formula 1.3, in which R ³ is ethyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 48 9

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 490

Compounds of the general formula 1.5, in which R ³ is ethyl, R ⁴ ethyl and the group Z compound amended always one of the radicals mentioned in Table A

-.411Table 491

Compounds of general formula (1.1) in which R @ ³ is ethyl, R ^{@ 4} propyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 492

Compounds of the general formula 1.2, in which R ³ represents ethyl, propyl, R ⁴ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 493

Compounds of the general formula 1.3, in which R ³ represents ethyl, propyl, R ⁴ and the group Z compound corresponding to each one of the radicals mentioned in Table A

Taboo 4 94

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ propyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 495

Compounds of the general formula 1.5, in which R ³ represents ethyl, propyl, R ⁴ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 496

Compounds of formula (1.1) in which R @ ³ is ethyl, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

· · · * * * * *

-413Table 497

Compounds of the general formula 1.2, in which ^R} = ethyl, R ⁴ iso-propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 498

Compounds of formula (1.3) wherein R ³ is ethyl, R ⁴ isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 499

Compounds of formula (1.4) in which R @ ³ is ethyl, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 500

Compounds of formula (1.5) wherein R ³ is ethyl, R ⁴ isopropyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 501

Compounds of formula 1.1 wherein R ³ is ethyl, R ^{4 is} 2-propenyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 502

Compounds of formula (1.2) in which R @ ³ is ethyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

-Table 503

Compounds of the general formula 1.3, in which R ³ is ethyl, R ^r 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 504

Compounds of formula (1.4) in which R @ ³ is ethyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 505

Compounds of the general formula 1.5, in which R ³ is ethyl, R 2 ^4-p.ropenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 506

Compounds of the general formula I.1, in which R ³ is ethyl, R ⁴ E-3-chloro-1 or 2-propenyl and 1. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 507

Compounds of the general formula 1.2, in which R ³ is ethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 508

Compounds of the general formula 1.3, in which R ³ is ethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · - -

Table 509

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 510

Compounds of the general formula 1.5, in which R ³ is ethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 511

Compounds of the general formula 1.1, in which R ³ is ethyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 512

Compounds of the general formula 1.2, in which R ³ is ethyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 513

Compounds of the general formula 1.3, in which R ³ is ethyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 514

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 515

Compounds of formula (I) in which R @ ³ is ethyl, R ^{@ 4} n-butyl and Z are each one of the radicals listed in Table A.

Table 516

Compounds of general formula 1.1 in which:. R ³ is ethyl, R ^{4 is} CH ₂ F and Z is each one corresponding to the radicals listed in Table A.

Table 517

Compounds of the general formula 1.2, in which R ³ is ethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 518

Compounds of the general formula 1.3, in which R ³ is ethyl, R ⁴ CH ₂ F and Z Peak compounds corresponding to each one of the radicals mentioned in Table A

Table 519

Compounds of formula (1.4), ethyl, R ⁴ CH ₂ F, and Z are then one of the residues listed in Table A.

of which R ³ corresponds always

Table 520

Compounds of the general formula 1.5, in which R ³ is ethyl. R ⁴ CH ₂ F and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 521

Compounds of the general formula I .1, wherein R ³ is ethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 522

Compounds of the general formula 1.2, in which R ³ is ethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 523

Compounds of the general formula 1.3, in which R ³ is ethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 524

Compounds of the general formula 1.4, in which R ³ is ethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 525

Compounds of the general formula 1.5, in which R ³ is ethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 526

Compounds of the general formula 1.1, in which R ³ is ethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

··

-42.3Table. 527

Compounds of formula (1.2) in which R @ ^{3 is} a! ethyl, R ⁴ 2-propynyl and Z then each corresponding to one of the radicals listed in Table A.

Table 528

Compounds of formula (1.3) in which R @ ³ is ethyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 529

Compounds of the general formula .1.4 wherein R ³ is ethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 530

Compounds of the general formula 1.5, in which R ³ is ethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 531

Compounds of formula 1.1 wherein R ³ is ethyl, R ^{4 is} C ¹ -CF 3 and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 532

Compounds of formula (1.2) in which R @ ³ represents ethyl, R ^{@ 4} Cl @ ³ CF @ ³ and Z are each one corresponding to one of the radicals listed in Table A.

- 41 «) ~

Taboo i 533

Compounds of formula (1.3) in which:. ! <'Means ethyl, Et ⁴ CELjCEý and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 534

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals uveddených in Table A.

Table 53.5

Compounds of the general formula 1.5, in kterýcii R ³ is ethyl, R ⁴ CH ₂ CF ₃ and the group Z. a compound corresponding to one of the residues given in Table A.

Table 536

Compounds of the general formula 1.1, in which R ³ is ethyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 537

Compounds of formula (1.2) in which R @ ³ is ethyl, R @ ⁴ C (CH3) OCH3 and Z are each one corresponding to one of the radicals listed in Table A.

Table 538

Compounds of formula (1.3) in which R @ ³ is ethyl, R @ ⁴ CH3 ClphyOCH3 and Z are each one corresponding to one of the radicals listed in Table A.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

53 \ Ο Table 539

Compounds of the general formula 1.4, in which R ³ is ethyl, R ⁴ Objective ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 540

Compounds of the general formula 1.5, in which R ³ friend ethyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 541

Compounds of formula (1.1) in which R @ ³ is propyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table.

Table 542

Compounds of formula (1.2) in which R @ ³ is propyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 543

Compounds of formula (1.3) in which R @ ³ is propyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 544

Compounds of formula (1.4) in which R @ ³ is propyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• · · · · · · · ·

Table 545

Compounds of formula (1.5) in which:. R ³ is propyl, R ^{4 is} methyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 546

Compounds of formula (1.1) wherein R ³ is propyl, R ^{4 is} ethyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 547

Compounds of the general formula 1.2, in which R ³ is propyl, and R ⁴ ety.1. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 548

Compounds of formula (1.3) in which R @ ³ is propyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 549

Compounds of formula (1.4) in which R @ ³ is propyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 550

Compounds of the general formula 1.5, in which R ³ is propyl, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

-32-Table 551

Compounds of formula (1.1) in which R ³ is propyl, R ^{4 is} propyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 552

Compounds of formula (1.2) in which R @ ³ is propyl, R ^{@ 4 is} propyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 553

Compounds of formula (1.3) in which R @ ³ is propyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 554

Compounds of formula (1.4) in which R @ ³ is propyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 555

Compounds of formula (1.5) in which R @ ³ is propyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 556

Compounds of formula (1.1) in which R @ ³ is propyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

·· • ·· ·· ·· 99 • • ·· • · • • · 9 • • • • 9 · ··· • 9 99 • · • • · · • · · 99 9 9 • • · • • · • · 9 9 • ·· ··· ·· · « 99 99

- 432 Table 557

Compounds of formula (1.2) in which R @ ³ is propyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 558

Compounds of formula (1.3) in which R @ ³ is proply, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 559

Compounds of formula 1.4 wherein R ³ is propyl, R ⁴ isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 560

Compounds of formula (1.5) wherein R ³ is propyl, R ⁴ isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 561

Compounds of formula (1.1) in which R @ ³ is propyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 562

Compounds of formula (1.2) in which R @ ³ is propyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

-434Table 563

Compounds of formula (1.3) in which R @ ³ is propyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 564

Compounds of formula (1.4) in which R @ ³ is propyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 565

Compounds of formula (1.5) in which R @ ³ is propyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 566

Compounds of the general formula 1.1, in which R ³ is propyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 567

Compounds of formula (1.2) in which R ³ is propyl, R ^{4 is} E-3-chloro-2-propenyl and Z is each a compound corresponding to one of the radicals listed in Table A.

Table 568

Compounds of formula (1.3) in which R ³ is propyl, R ^{4 is} E-3-chloro-2-propenyl and Z is each a compound corresponding to one of the radicals listed in Table A.

Table 569

Compounds of the general formula 1.4, in which R ³ is propyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 570

Compounds of the general formula 1.5, in which R ³ is propyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 571 Compounds of general formula 1.1 in which R ³ represents propyl, R ⁴ n-butyl and Z then the compound odpo v1da j1c1 one of the residues mentioned in Table A. Table 572 Compounds of general formula 1.2 in which R ³ represents propyl, R ⁴ n-butyl and Z p a k s 1 o u e n i n u corresponding one of the residues mentioned in Table A. Table 573 Compounds of general formula 1.3 in which R ³ represents propyl, R ⁴ n-butyl and Z then the compound corresponding one of the residues mentioned in Table A. Table 574 Compounds of general formula 1.4 in which R ³ represents propyl, R ⁴ n-butyl and Z then the compound corresponding one of the residues mentioned in Table A.

• · • ·

-436T bulb 57 5

Compounds of the general formula 1.5, in which R ³ is propyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 576

Compounds of the general formula 1.1, in which R ³ is propyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 577

Compounds of the general formula 1.2, in which R ³ is propyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 578

Compounds of the general formula 1.3, in which R ³ is propyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 579

Compounds of the general formula 1.4, in which R ³ is propyl, R ⁴ _CH? F and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 580

Compounds of the general formula 1.5, in which R ³ means interlocks, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 581

Compounds of the general formula 1.1, in which R ³ is propyl, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 582

Compounds of the general formula 1.2, in which R ³ is propyl, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 583

Compounds of the general formula 1.3, in which R ³ is propyl, ^R4, _CHF2 and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 584

Compounds of the general formula 1.4, in which R ³ is propyl, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 585

Compounds of the general formula 1.5, in which R ³ is propyl, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 586

Compounds of the general formula 1.1, in which R ³ is propyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 587

Compounds of formula (1.2) in which R @ ³ is propyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 588

Compounds of the general formula 1.3, in which R ³ is propyl, R ⁴ 2-propynyl. and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 589

Compounds of formula (1.4) in which R @ ³ is propyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Tab. 1 A. 590

Compounds of the general formula 1.5, in which R ³ is propyl, R ^4, and 2-propynyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 591

Compounds of general formula 1.1 wherein R ³ is propyl, R ⁴ CH ₂ CF ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 592

Compounds of formula (1.2) in which R @ ³ is propyl, R @ ^{4 is} C1-4 alkyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Table 593 S1 o u n e n i n e n e n e n e n e n e 1.3, ve of which R ³ means propyl, R ⁴ CH ₂ CF ₃ and a group. Z then compounds here cl always one of the residues listed in Table A. Table 594 Compounds of general formula 1.4, ve of which R ³ means propyl, R ⁴ CH ₂ CF ₃ and the group Z then compounds i.u answer cl always one of the residues listed in Table A. Table 595 Compounds of general formula 1.5, ve of which R ³ means propyl, R ⁴ CH ₂ CF ₃ and the group Z then s1o u u n n u u o n d i j1 cl always one of the residues listed in La; bulce A. Table 596 Compounds of general formula I .. 1, p of which R ³ z narnená propyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z i then serve .ceninu odpov Idajicl

one of the residues listed in Table A.

Table 597

Compounds of formula (1.2) in which R ³ is propyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z then each corresponds to one of the radicals listed in Table A.

Table 598

Compounds of the general formula 1.3, in which R ³ is propyl, R ⁴ C1T ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

• 9 · 9 · 999 · · Λ <ιθTable 599

Compounds of the general formula 1.4, in which R ³ is propyl, R ⁴ CH ₂ CH ₂ OC.H ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 600

Compounds of formula (1.5) in which:. R ³ represents propyl, R ⁴ ClýCIýOCIL and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 601

Compounds of formula (1.1) wherein R ³ is isopropyl, R ^{4 is} methyl, and R ^{3 is} methyl. 'L then. a compound corresponding to one of the residues listed in Table A.

Table 602

Compounds of formula (1.2) in which R @ ³ is isopropyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 603

Compounds of formula (1.3) in which:. ^R3 is iso-propyl and R ⁴ is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A:

Table 604

Compounds of formula (1.4) wherein R ³ is isopropyl, R ⁴ methyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

• ·

Table 605 Compounds' general of formula 1 [.5 in which R ³ means iso-propyl, R ⁴ methyl a group Z then the compound odpo ’ seeing always one of residues listed in Table A. Table 606 Compounds ’ general formulas 1.1 in which R ³ means iso-propyl, R ⁴ ethyl a group Z then the compound corresponding always one of residues listed in Table A. Table 607 Compounds general formulas 1.2 in which R ³ means. iso-propyl, R ⁴ ethyl a group Z then the compound odpo seeing always one of residues listed in Table A.

Table 608

Compounds of formula (1.3) in which R ³ is isopropyl, R ⁴ ethyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 609

Compounds of formula (1.4) in which R @ ³ is isopropyl, R ^{@ 4} ethyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 610

Compounds of formula (1.5) in which R @ ³ is isopropyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

• ·

Table 611

Compounds of the formula 1.1 in which R ^{3 is} injured with isopropyl, R ^{4 with} propyl and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 612

Compounds of formula (1.2) wherein:. R 1 is isopropyl, R ^{4 is} propyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 613

Compounds of the general formula I.3 where ^R3 is iso-propyl, propyl and R ⁴ group Z compound corresponding to each one of the radicals mentioned in Table A

Table 614

Compounds of formula (1.4) in which R @ ³ is isopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 615

Compounds of formula (1.5) in which R @ ³ is isopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table. 616

Compounds of formula (1.1) in which R @ ³ is isopropyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 617

Compounds of the general formula 1.2, in iso-propyl, R ⁴ and iso-propyl group and wherein R ³ is Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 618

Compounds of formula (1.3) in which R @ ³ is isopropyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 619

Compounds of formula (1.4) in which R @ ³ is isopropyl, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 620

Compounds of formula (1.5) in which R @ ³ is isopropyl, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 621

Compounds of formula (1.1) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 622

Compounds of formula (1.2) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 623

Compounds of formula (1.3) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 624

Compounds of formula (1.4) in which R @ ³ is isopropyl, R ^{@ 4} 2-propenyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 625

Compounds of formula (1.5) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 626

Compounds of the general formula 1.1, in which R ³ represents isopropyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 627

Compounds of formula (1.2) in which R @ ³ is isopropyl, R ^{@ 4} E -3-chloro-2-propenyl and Z are each corresponding to one of the radicals listed in Table A.

Table 628

Compounds of formula (1.3) in which R ³ is isopropyl, R ⁴ E-3-chloro-2-propenyl and Z is then

a compound corresponding to one of the residues listed in Table A.

Table 629

Compounds 1.4 which R ³ represents iso-propyl, R ⁴ E-3-chloro-2 -propenyl and group Z then compound always corresponding one of them residues referred to in Table A. Table 630 Compounds general in zorc: : e 1.5, ve which R ³ represents iso-propyl, R ⁴ E-3-chloro-2 -propenyl and group Z then compound corresponding always one of them residues referred to in Table A. Table 631 Compounds general pattern e 1.1, ve which. R ³ represents iso-propyl, R ⁴ n-butyl a group Z then compound corresponding to one of residues listed in Table A.

Table 632

Compounds of formula (1.2) in which R ³ is isopropyl, R ⁴ n-butyl and. Z then a compound corresponding to one of the radicals listed in Table A.

Table 633

Compounds of formula (1.3) in which R @ ³ is isopropyl, R ^{@ 4} n -butyl and Z are each one corresponding to one of the radicals listed in Table A.

····················································· · ···· ···

Table 634

Compounds of formula (1.4) in which R @ ³ is isopropyl, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 635

Compounds of formula (1.5) in which R @ ³ is isopropyl, R ^{@ 4} n -butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 636

Compounds of the general formula 1.1, in which R ³ represents isopropyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 63'7

Compounds of the general formula 1.2, in which R ³ represents isopropyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 638

Compounds of formula (1.3) wherein R ³ is isopropyl, R ⁴ CH ₂ F and Z then. a compound corresponding to one of the residues listed in Table A.

Table 639

Compounds of the general formula 1.4, in which R ³ represents isopropyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

Tcibulka 640

Compounds of the general formula 1.5, in which R ³ represents isopropyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 641

Compounds of the general formula 1.1, in which R ³ is iso-propyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 642

Compounds of general formula 1.2 wherein R ³ represents

isopropyl, one for each R. ⁴ CHF _{2 a} .: From residues group Z in the management p and k součoni nu in Table A. the responder replies Table 643 Compounds / general of formula i 1.3 in which R ³ represents iso-propyl, R ⁴ CHF _2a ; group Z then the compound corresponding always one of residues listed in Table A. Table 644 General compounds formulas 1.4 in which R ³ represents iso-propyl, R ⁴ CHF ₂ a group Z then. compound corresponding always one of residues listed in Table A. Table. 64 5 General compounds formulas I.5 R ³ represents iso-propyl, R ⁴ CHF ₂ a group Z then the compound corresponding always one of residues listed in Table A.

Table 646

Compounds of formula (1.1) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 647

Compounds of formula (1.2) in which R ³ is isopropyl, R ^{4 is} 2-propynyl and a group. Z then each corresponds to one of the radicals listed in Table A.

Table 648

Compounds of formula (1.3) in which R @ ³ is isopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 649

Compounds of formula (1.4) wherein R ³ is isopropyl, R ^{4 is} 2-propynyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 650

Compounds of formula (1.5) wherein R ³ is isopropyl, R ^{4 is} 2-propynyl and Z is then. a compound corresponding to one of the radicals listed in Table A.

Table 651

Compounds of the general formula 1.1, in which R ³ represents isopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· ·

· «« · »0 • · · · 0 · 0

0000 R 0 00 0 0 0 000 0 0 0 0 0 0 0 0

Table 652

Compounds of formula (1.2) wherein R ³ is isopropyl 1, R ⁴ CH ₂ CF ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 653

Compounds of the general formula 1.3, in which R ³ represents isopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 654

Compounds of the general formula 1.4, in the terých R ³ is iso-propyl and R ⁴ -CH ₂ CF ₃ and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 655

Compounds of the general formula 1.5, in which R ³ represents isopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 656

Compounds of general formula 1.1 wherein R ³ is isopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 657

Compounds of formula (1.2) in which R ³ is isopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each a compound corresponding to one of the radicals listed in Table A.

φφ

Table 658

Compounds of formula (1.3) in which R ³ is isopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and group 7 are each one corresponding to one of the radicals listed in Table A.

Table 659

Compounds of formula (1.4) in which R ³ is isopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 660

Compounds of the general formula 1.5, in which R ³ represents isopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 66'1

Compounds of formula (1.1) in which R @ ³ is trifluoromethyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 662

Compounds of the general formula T.2 wherein R ³ is trifluoromethyl, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 663

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4} meyl and Z are each corresponding to one of the radicals listed in Table A.

-λΖΛTable 664

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 665

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 666

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ ethyl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 667

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ ethyl and the group Z corresponds for each Compound of one of the radicals mentioned in Table A

Table 668

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 669

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

φ φ φ φ φ φ φ * * * φ φ φ φ φ φ φ φ φ φ · · · *

-45 * 2-- Table 670 Compounds of general formula 1.5, ve which R ³ represents trifluoromethyl, R ⁴ ethyl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 671

Compounds of formula (1.1) in which R @ ³ is trifluoromethyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 672

Compounds of formula (1.2) in which R @ ³ is trifluoromethyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 673

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 674

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 675

Compounds of formula (1.5) in which R @ ³ is trifluoromethyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

• • •

-45-3Table 676

Compounds of formula (1.1) in which R @ ³ is trifluoromethyl, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 677

Compounds of formula (1.2) in which R @ ³ is trifluoromethyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 678

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 679

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 680

Compounds of formula (1.5) in which R @ ³ is trifluoromethyl, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 681

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ 2-propenyl and the group Z corresponds for each compound to one for the radicals mentioned in Table A.

• · · · · · · · · · · · · · · · · · ·

Table 682

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 683

Compounds of formula (1.3) wherein R ³ is trifluoromethyl, R ^{4 is} 2-propenyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 684

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 685

Compounds of formula (1.5) in which R @ ³ is trifluoromethyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 686

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 687

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 455—

Table 688

Compounds of formula (1.3), in trifluoromethyl, R ⁴ E-3-chloro-2-propenyl wherein R ³ represents and Z is a compound corresponding to one of the radicals listed in Table A.

Table 689

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 690

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 691

Compounds of formula (1.1) in which R @ ³ is trifluoromethyl, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 692

Compounds of formula (1.2) in which R @ ³ is trifluoromethyl, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

• ······························

Table 693

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 694

Compounds of formula (1.4) in which R @ ³ is trifluoromethyl, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 695

Compounds of formula (1.5) in which R @ ³ is trifluoromethyl, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 696

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 697

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 698

Compounds of the general formula 1.3, in which R ³ is trifluoromethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 699

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 700

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 701

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 702

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 703

Compounds of the general formula 1.3, in which R ³ is trifluoromethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 704

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in the sheet A.

• · ~ Λ5 ~ β ~

Table 705

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 706

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 707

Compounds of formula (1.2) in which R @ ³ is trifluoromethyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 708

Compounds of formula (1.3) in which R @ ³ is trifluoromethyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 709

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 710

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 711

Compounds of formula (1.1), in trifluoromethyl, R ⁴ CH ₂ CF ₃ and a group in which R ³ represents Z then a compound corresponding to one of the radicals listed in Table A.

Table 712

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 713

Compounds of the general formula 1.3, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 714

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 715

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 716

Compounds of the general formula 1.1, in which R ³ is trifluoromethyl, R ⁴ CH ^ C ^ OCH and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 717

Compounds of the general formula 1.2, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 718

Compounds of the general formula 1.3, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 719

Compounds of the general formula 1.4, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CH ₂ OCH _3, and. The group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 720

Compounds of the general formula 1.5, in which R ³ is trifluoromethyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 721

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 722

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

-464Table 723

Compounds of formula (1.3) in which R @ ³ is cyclopropyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 724

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 725

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 72 6

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table. 727

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 728

Compounds of the general formula 1.3, in which R ³ is cyclopropyl, ^R4 ethyl and the group Z corresponds for each compound Paks one of the radicals mentioned in Table A

9 99

9 9

9 9 9 9 9

9 9 9 9 9 9 9 9 9 9 9

-Ί62Table 729

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 730

Compounds of formula (1.5) in which R @ ³ is cyclopropyl, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 731

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 732

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 733

Compounds of formula (1.3) in which R @ ³ is cyclopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 734

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 735

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, ^R4 propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 736

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 737

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 738

Compounds of formula (1.3) in which R @ ³ is cyclopropyl, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 739

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4} isopropyl and Z are each one of the radicals listed in Table A.

Table 740

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, ^R4 iso-propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-4G <1 Table 741

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 742

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 743

Compounds of formula (1.3) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 744

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 745

Compounds of formula (1.5) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 746

Compounds of the general formula 1.1, in which R ³ is cyclopropyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-.465Table. 747

Compounds of the general formula 1.2, in which R ³ is cyclopropyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 748

Compounds of the general formula 1.3, in which R ³ is cyclopropyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 74 9

Compounds of the general formula 1.4, in which R ³ is cyclopropyl, R ⁴ E-3-chloro-2-propenyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 750

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 751

Compounds of the general formula 1.1, in which R ³ is cyclopropyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 752

Compounds of general formula 1.2, in cyclopropyl, R ⁴ n-butyl and the group R ³ being

Z then a compound corresponding to one of the radicals listed in Table A.

Table 753

Compounds of formula (1.3) in which R @ ³ is cyclopropyl, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 754

Compounds of the general formula 1.4, in which R ³ is cyclopropyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 755

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 756

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4} CIL ^@ ₂ F and Z are each corresponding to one of the radicals listed in Table A.

Table 757

Compounds of formula (1.2) in which R @ ³ is cyclopropyl, R @ ⁴ CH3 F and Z are each one corresponding to one of the radicals listed in Table A.

Table 758

Compounds of formula (1.3) in which R ³ is cyclopropyl, R ⁴ CH ₂ F and Z are each one corresponding to one of the radicals listed in Table A.

Table 759

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R @ ⁴ CF3 F and Z are each one corresponding to one of the radicals listed in Table A.

Table 760

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of ZE) ytků listed in Table A.

Table 761

Compounds of formula (1.1). wherein R ³ is cyclopropyl, R ⁴ CHF ₂ and Z is a compound corresponding to one of the radicals listed in Table A.

Table 762

Compounds of the general formula 1.2, in which R ³ is cyclopropyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 763

Compounds of the general formula 1.3, in which R ³ is cyclopropyl, ^R4 _CHF2 and the group Z corresponds for each compound to one for the radicals mentioned in Table A.

· · · · · · · · · ··· · ♦ ·· ·· ··

- 44βTable 764

Compounds of the general formula 1.4, in which R ³ is cyclopropyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 765

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 766

Compounds of formula (1.1) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 767

Compounds of formula (1.2) wherein R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 768

Compounds of formula (1.3) wherein R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 769

Compounds of formula (1.4) in which R @ ³ is cyclopropyl, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

· A • A

A A

A

Table 770

Compounds of general formula cyclopropyl, R ' ² 2-propynyl and

5, ve which R ^J is kupína Z then compound

corresponding to one of the residues listed in Table A.

Table 771

Compounds of the general formula 1.1, in which R ³ represents cyclopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table Ά.

Table 772

Compounds of the general formula 1.2, in which R ³ represents cyclopropyl, R ⁴ CH ₂ CF _'3 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 773

Compounds of the general formula 1.3, in which R ³ represents cyclopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 774

Compounds of the general formula 1.4, in which R ³ is cyclopropyl, ^R4 C1L ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 775

Compounds of the general formula 1.5, in which v is cyclopropyl, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 776

Compounds of general formula 1.1, cyclopropyl,, · · · · · · • • • • φ φ φ φ · · · · · kterých kterých kterých R ³ represents

R ⁴ CH ₂ CH ₂ OCH ₃ and a group

Z then a compound corresponding to one of the radicals listed in Table A.

Table 777

Compounds of formula (1.2) in which R ³ is cyclopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each one corresponding to one of the radicals listed in Table A.

Table 778

Compounds of the general formula 1.3, in which R ³ is cyclopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 779

Compounds of the general formula 1.4, in which R ³ is cyclopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 780

Compounds of the general formula 1.5, in which R ³ is cyclopropyl, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A:

Table 781

Compounds of the general formula 1.1, in which R ³ is methoxy, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-4 * 4Table 782

Compounds of formula (1.2) in which R @ ³ is methoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 783

Compounds of the general formula 1.3, in which R ³ is methoxy, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 784

Compounds of the general formula 1.4, in which R ³ is methoxy, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 785

Compounds of formula (1.5) in which R @ ³ is methoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 786

Compounds of the general formula 1.1, in which R ³ is methoxy, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 787

Compounds of the general formula 1.2, in which R ³ is methoxy, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · • ·

-432Table 788

Compounds of formula (1.3) in which R @ ³ is methoxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 789

Compounds of formula (1.4) in which R @ ³ is methoxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 790

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 791

Compounds of formula (1.1) in which R @ ³ is methoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 792

Compounds of formula (1.2) in which R @ ³ is methoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 793

Compounds of formula (1.3) in which R @ ³ is methoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

· · · · · ·

> φ · ♦ · · · • • •

Table 794

Compounds of formula (1.4) in which R @ ³ is methoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 795

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 796

Compounds of formula (1.1) in which R @ ³ is methoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 797

Compounds of formula (1.2) in which R @ ³ is methoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 798

Compounds of formula (1.3) in which R @ ³ is methoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 799

Compounds of formula (1.4) in which R @ ³ is methoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

······································································ I · · · · ··················

Table 800 Compounds of general formula of formula i : .5, in which R ³ stands for methoxy, R ⁴ isopropyl and group Z then compound corresponding always one of the leftovers listed in Table A. Table. 801 S L o u e η 1 n y generic of formula I :.and, in which R ³ represents methoxy, R ⁴ 2-propenyl and group Z then compound corresponding always one of the leftovers listed in Table A. Table 802 General compounds of formula I in which R ³ represents methoxy, R ⁴ 2-propenyl and group Z then compound. corresponds to it always one of the leftovers listed in Table A. Table 803 General training of formula I .3, in which R ³ represents methoxy, R ⁴ 2-propenyl and group Z then compound corresponding always one of the leftovers listed in Table A. Table 804 S1. o u e n e n g e n e n e n e n e of formula I - 4 _y in which R ³ represents methoxy, R ⁴ 2-propenyl and. group Z then compound odpo v1da j i c1 always one of the leftovers listed in Table A. Table 805 Merging General of formula I '. 5, in which R ³ represents methoxy, R ⁴ 2-propenyl and group Z then. compound corresponding always one of the leftovers listed in Table A.

• ·

-.4-ψϊΓ

Table 806

Compounds of general formula 1.1 in which:. R ³ is methoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 807

Compounds of formula (1.2) wherein R ³ is methoxy, R ⁴ E-3-chloro-2-propenyl. and Z is a compound corresponding to one. the residues listed in Table A.

Table 808

Compounds of the general formula 1.3, in which R ³ znrimená. methoxy, R ⁴ E-3-chloro-2-propenyl Z then a compound corresponding to one of the radicals listed in Table A.

Table 809

Compounds of the general formula 1.4, in which R ³ is methoxy, R ⁴ E-3-chloro-2-propenyl and the group Z, a compound corresponding, in each case one of the radicals uvedsených in Table A.

Table 810

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 811

Compounds of the general formula 1.1, in which R ³ is methoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

_λϊ £>

Table 812

Compounds of formula (1.2) in which R @ ³ is methoxy, R ^{@ 4 is} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 813

Compounds of the general formula 1.3, in which R ³ is methoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 814

Compounds of the general formula 1.4, in which R ³ znameriíl methoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 815

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 816

Compounds of the general formula 1.1, in which R ³ is methoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 81.7

Compounds of the general formula 1.2, in which R ³ is methoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 818

Compounds of formula (1.3) wherein R ³ is

methoxy, R ⁴ CH ₂ F and Z then the corresponding compound always one of them residues in Table A. Table 819 Compounds of the general formula 1.4 wherein R ³ is methoxy, R ⁴ CH ₂ F and Z then the corresponding compound always one of them residues 11 in Table A. Table 820 Compounds the general model rce 1.5 wherein R ³ is methoxy, R ⁴ CH ₂ F and Z then the corresponding compound always one of them z c t u e d e c h v t a bulce A. Table 821 Compounds the general model rce 1.1 wherein R ³ is methoxy, R ⁴ CHF ₂ and Group Z then the corresponding compound always one of them residues in Table A. Table 822 Compounds of the general formula 1.2 wherein R ³ is methoxy, R ⁴ CHF ₂ and Group Z then the corresponding compound always one of them residues in Table A. Table 823 Compounds of the general formula 1.3, in which R ³ represents methoxy, R ⁴ CHF ₂ and Group Z then always the corresponding compound one of them residues in Table A.

• 9 9 9999 9999 * 9 9 9 9 9 9 9 9 9 99

9 9 9 9 9 9999

- ίιβTab 1 Cr 824

Compounds of the general formula 1.4, in which R ³ is methoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 825

Compounds of the general formula 1.5, in which R ³ is methoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 826

Compounds of the general formula 1.1, in which R ³ is methoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 827

Compounds of the general formula 1.2, in which R ³ is methoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 828

Compounds of the general formula 1.3, in which R ³ is methoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 829

Compounds of formula (1.4) in which R @ ³ is methoxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 830

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ 2-propynyl. a. Z is a compound corresponding to one of the radicals listed in Table A.

Table. 831

Compounds of formula (1.1) in which R @ ³ is methoxy, R @ ⁴ CEL2 CF, and Z are each corresponding to one of the radicals listed in Table A.

Table 832

Compounds of formula (1.2) wherein R ³ is methoxy, R ⁴ CH ₂ CF ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 833

Compounds of formula (1.3) in which R ³ is methoxy, R ⁴ CH 2 CH 2 and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 834

Compounds of formula 1.4 wherein R ³ is methoxy, R ⁴ CH ₂ CF ₃ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 835

Compounds of the general formula 1.5, in which R ³ is methoxy, R @ ⁴ Objective Cey and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 836

Compounds of the general formula 1.1, in which R ³ is methoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 837

Compounds of formula (1.2) in which R ³ is methoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each one corresponding to one of the radicals listed in Table A.

Table 838

Compounds of the general formula 1.3, in which R ³ is methoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 839

Compounds of the general formula 1.4, in which R ³ is methoxy, R ⁴ CH 2 CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 840

Compounds of the general formula 1.5, in which R ³ is methoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 841

Compounds of formula (1.1) in which R @ ³ is ethoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

• ·

484 Table 842

Compounds of VORC 1.2, in which R ³ is ethoxy, ^R4 is methyl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 843

Compounds of formula (1.3) in which R @ ³ is ethoxy, R ^{@ 4} methyl and Z are each one of the radicals listed in Table A.

Table 844

Compounds of the general formula 1.4, in which R ³ is ethoxy, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 8455

Compounds of formula (1.5) in which R @ ³ is ethoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 846

Compounds of the general formula 1.1, in which R ³ is ethoxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 847

Compounds of the general formula 1.2, in which R ³ is ethoxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

* · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

Table 048

Compounds of the general formula 1.3, in which R ³ is ethoxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 849

Compounds of formula (1.4) in which R @ ³ is ethoxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table. 850

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ and ethyl groups. Z then a compound corresponding to one of the radicals listed in Table A.

Table. 851

Compounds of the general formula 1.1, in which R ³ is ethoxy, ^R4, propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 852

Compounds of formula (1.2) in which R @ ³ is ethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 853

Compounds of formula (1.3) in which R @ ³ is ethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

• * 9 · · · · · · · • • · • · • · «« 9 9 9 9 · ···· · · · ···············

Table 854

Compounds of formula (1.4) in which R @ ³ is ethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 855

Compounds of the general formula 1.5, in which R ³ is ethoxy, ^R4, propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 856

Compounds of formula (1.1) in which R @ ³ is ethoxy, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 857

Compounds of formula (1.2) in which R @ ³ is ethoxy, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 858

Compounds of formula (1.3) in which R @ ³ is ethoxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 859

Compounds of formula (1.4) in which R @ ³ is ethoxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 860

Compounds of the general formula 1.5, in which R ³ is ethoxy, ^R4 iso-propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 861

Compounds of formula (1.1) in which R @ ³ is ethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 862

Compounds of formula (1.2) in which R @ ³ is ethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 863

Compounds of formula (1.3) in which R @ ³ is ethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 864

Compounds of the general vzrce 1.4, in which R ³ is ethoxy, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 865

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 4B5 * Table. 866

Compounds of the general formula 1.1, in which R ³ is ethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 867

Compounds of the general formula 1.2, in which R ³ is ethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 868

Compounds of the general formula 1.3, in which R ³ is ethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 869

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 870

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 871

Compounds of the general formula 1.1, in which R ³ is ethoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· · · · · · · · • · · · · · · · · · · · · · · · · · · · · · ·

-4SCT table 872

Compounds of formula (1.2) in which R ³ is ethoxy, R ⁴ n-butyl and. Z then a compound corresponding to one of the radicals listed in Table A.

Table 873

Compounds of the general formula 1.3, in which R ³ is ethoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 874

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 875

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ^c, n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 876

Compounds of vzrce 1.1, in which R ³ is ethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 877

Compounds of the general formula 1.2, in which R ³ is ethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 878

Compounds of the general formula 1.3, in which R ³ is ethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 879

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 880

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 881

Compounds of general formula 1.1 in which R ³ is ethoxy, R ⁴ CHF ₂ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 882

Compounds of the general formula 1.2, in which R ³ is ethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 883

Compounds of the general formula 1.3, in which R ³ is ethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

Table. 884

Compounds of the general formula 1.4, in which R ³ is ethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 885

Compounds of the general formula 1.5, in which R ³ is ethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 886

Compounds of the general formula 1.1, in which R ³ is ethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 887

Compounds of the general formula 1.2, in which R ³ is ethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 88’8

Compounds of the general formula 1.3, in which R ³ is ethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 889

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 890

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 891

Compounds of the general formula 1.1, in which R ³ is ethoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 892

Compounds of the general formula 1.2, in which R ³ is ethoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 893

Compounds of formula (1.3) in which R @ ³ is ethoxy, R @ ⁴ CH3 CF6 and Z are each one corresponding to one of the radicals listed in Table A.

Table 894

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 895

Compounds of formula (1.5) in which R @ ³ is ethoxy, R @ ⁴ C @ ⁴ CF3 and Z are each one corresponding to one of the radicals listed in Table A.

- jqo -

Table 896

Compounds of the general formula 1.1, in which R ³ is ethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 897

Compounds of the general formula 1.2, in which R ³ is ethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 898

Compounds of the general formula 1.3, in which R ³ is ethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 899

Compounds of the general formula 1.4, in which R ³ is ethoxy, R ⁴ CH ₂ CH ₂ OCH _3, and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 900

Compounds of the general formula 1.5, in which R ³ is ethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 901

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

-4 ^ 4Table 902

Compounds of formula (1.2) wherein R ³ is propyloxy, R ⁴ methyl and a group. Z then a compound corresponding to one of the radicals listed in Table vždy.

Table 903

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 904

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 905

Compounds of the general formula 1.5, in which R ³ is propyloxy, ^R4 is methyl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 906

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 907

Compounds of formula (1.2) in which R @ ³ is propyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 908

Compounds of the general formula 1.3, in which R ³ represents propyloxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 909

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 910

Compounds of formula (1.5) in which R @ ³ is propyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 911

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 912

Compounds of formula (1.2) in which R @ ³ is propyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 913

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

··· · v · v · v · v

• · • · ···

Table 914

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 915

Compounds of formula (1.5) in which R @ ³ is propyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 916

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 917

Compounds of formula (1.2) in which R @ ³ is propyloxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 918

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

Table 919

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4} isopropyl and Z are each corresponding to one of the radicals listed in Table A.

- 4 ^ * 1 - Table 920 Compounds 1.5 which R ³ represents propyloxy, R ⁴ isopropyl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 921

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4} '- 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 922

Compounds of formula (1.2) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 923

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 924

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 925

Compounds of formula (1.5) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

9 9 9 9 9 9 9 9 9 9 10 11 12 13 14 15 16 17 18 19 20 • · · · · · · · · · · · · · · · ·

Table. 92 6

Compounds of the general formula 1.1, in which R ³ represents propoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 927

Compounds of formula (1.2) in which R @ ³ is propyloxy, R ^{@ 4} E-3-chloro-2-propenyl and Z are each one corresponding to one of the radicals listed in Table.

Table 928

Compounds of the general formula 1.3, in which R ³ represents propoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 929

Compounds of formula 1.4 wherein R ³ is propyloxy, R ⁴ E-3-chloro-2-propenyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 930

Compounds of the general formula 1.5, in which R ³ represents propoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 931

Compounds of the general formula 1.1, in which R ³ represents propoxy, R ⁴ n-butyl and the group Z. a compound corresponding to one of the residues listed in Table A.

Table 932

Compounds of the general formula 1.2, in which R ³ represents propoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 933

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 934

Compounds of formula 1.4 wherein R ³ is propyloxy, R ^{4 is} n-butyl and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 935

Compounds of the general formula 1.5, in which R ³ represents propoxy, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Tabulkři 936

Compounds of the general formula 1.1, in which R ³ represents propoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 937

Compounds of formula (1.2) wherein R ³ is propyloxy, R ⁴ CH ₂ F and. Z then a compound corresponding to one of the radicals listed in Table A.

• ·

-Wt · Table 938

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4} CELJ 'and Z are each corresponding to one of the radicals listed in Table A.

Table 939

Compounds of the general formula 1.4, in which R ³ represents propoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 940

Compounds of formula (1.5) in which R @ ³ is propyloxy, R @ ⁴ CE @ F and Z are each one corresponding to one of the radicals listed in Table A.

Table 941

Compounds of the general formula 1.1, in which R ³ represents propyloxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 942

Compounds of the general formula 1.2, in which R ³ represents propyloxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 943

Compounds of the general formula 1.3, in which R ³ represents propyloxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 944

Compounds of the general formula 1.4, in which R ₃ represents propyloxy, _{R4, CHF2} and the group Z corresponds for each paksloučeninu one of the radicals mentioned in Table A

Table 945

Compounds of the general formula 1.5, in which R ³ represents propyloxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 946

Compounds of formula (1.1) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 947

Compounds of the general formula 1.2, in which R ³ represents proplyoxy R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 948

Compounds of formula (1.3) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 949

Compounds of formula (1.4) in which R @ ³ is propyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Table 950

Compounds of general formula 1.5, in propyloxy, R ⁴ 2-propynyl and the group wherein R ³ represents Z then a compound corresponding to one of the radicals listed in Table A.

Table 951

Compounds of the general formula 1.1, in which R ³ represents proplyoxy R ⁴ -CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 952

Compounds of the general formula 1.2, in which R ³ represents propoxy, R ⁴ CH ₂ and CF _3. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 953

Compounds of vzrce 1.3, in which R ³ represents propoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 954

Compounds of the general formula 1.4, in which R ³ represents propoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 955

Compounds of the general formula 1.5, in which R ³ represents propoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · • ·

- zoo - Table 956 Compounds of the general public e 1.1, ve which R ³ represents propyloxy, R ⁴ CH ₂ CH ₂ OCH ₃ a group Z then compound

corresponding to one of the residues listed in Table A.

Table 957

Compounds of formula (1.2) in which R ³ is propyloxy, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 958

Compounds of the general formula 1.3, in which R ³ represents propoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 959

Compounds of the general formula 1.4, in which R ³ represents propoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 960

Compounds of the general formula 1.5, in which R ³ represents propoxy, R ⁴ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 961

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 962

- from-t

Compounds of formula (1.2), iso-propyloxy,

in which R ³ represents

R ^{4 is} methyl and

Z then a compound corresponding to one of the radicals listed in Table A.

Table 963

Compounds of formula (1.3) in which R @ ³ is isopropyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 964

Compounds of formula (1.4) in which R @ ³ is isopropyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 965

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 966

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 967

Compounds of formula (1.2) in which R @ ³ is isopropyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 968

Compounds of formula (1.3) in which R @ ³ is isopropyloxy, R ^{@ 4} ethyl and a group corresponding to one of the radicals listed in Table A.

Table 969

Compounds of formula (1.4) in which R @ ³ is isopropyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 970

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 971

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 972

Compounds of formula (1.2) in which R @ ³ is isopropyloxy, R ^{@ 4} propyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 973

Compounds of the general formula 1.3, in which R ³ represents iso proplyoxy, ^R4 propyl and the group Z corresponds for each paksloučeninu one of the radicals mentioned in Table A

Table 974

Compounds of the general formula 1.4, in iso-propyloxy, ^R4 propyl group and wherein

R ³ represents

Z then a compound corresponding to one of the residues listed in Table A.

Table 975

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 976

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 977

Compounds of the general formula 1.2, in which R ³ is iso-propyloxy, ^R4 isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 978

Compounds of formula (1.3) in which R @ ³ is isoproplyoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 979

Compounds of formula (1.4) in which R @ ³ is isopropyloxy, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

- 10¼ -

Table 980

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 981

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 982

Compounds of formula (1.2) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 983

Compounds of formula (1.3) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 984

Compounds of formula (1.4) in which R @ ³ is isoproplyoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 985

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

- 2OS ~ Table 986

Compounds of the general formula 1.1, in which R ³ is iso-propyloxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 987

Compounds of the general formula 1.2, in which R ³ is iso-propyloxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 988

Compounds of formula (1.3) in which R @ ³ is isopropyloxy, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 989

Compounds of the general formula 1.4, in which R ³ is iso-propyloxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 990

Compounds of the general formula 1.5, in which R ³ is iso-propyloxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-2OGTable 991

Compounds of formula (1.1) in which R @ ³ is iso-propyloxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 992

Compounds of formula (1.2) in which R @ ³ is iso-propyloxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 993

Compounds of formula (1.3) in which R @ ³ is iso-propyloxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 994

Compounds of formula (1.4) in which R @ ³ is isopropyloxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 995

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 996

Compounds of the general formula 1.1, in which R ³ is iso-propyloxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 997

Compounds of the general formula 1.2, in which R ³ is iso-propyloxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 998

Compounds of the general formula 1.3, in which R ³ is iso-propyloxy, R ⁴ _Z F CH and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 999

Compounds of the general formula 1.4, in which R ³ is iso-propyloxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1000

Compounds of the general formula 1.5, in which R ³ is iso-propyloxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1001

Compounds of the general formula 1.1, in which R ³ is iso-propyloxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1002

Compounds of the general formula 1.2, in which R ³ is iso-propyloxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 208 -

Table 1003

Compounds of the general formula 1.3, in which R ³ is iso-propyloxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1004

Compounds of the general formula 1.4, in which R ³ is iso-propyloxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1005

Compounds of the general formula 1.5, in which R ³ is iso-propyloxy, ^R4 _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1006

Compounds of formula (1.1) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1007

Compounds of formula (1.2) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1008

Compounds of formula (1.3) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

·· · · · · φ φ φ φ φφ

- ΖΟ <) Table 1009

Compounds of formula (1.4) in which R @ ³ is isopropyloxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1010

Compounds of the general formula 1.5, in which R ³ is iso-propyloxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1011

Compounds of the general formula 1.1, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1012

Compounds of the general formula 1.2, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1.013

Compounds of the general formula 1.3, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1014

Compounds of the general formula 1.4, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- Evil -

Table 1015

Compounds of the general formula 1.5, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1016

Compounds of the general formula 1.1, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1017

Compounds of formula (1.2) in which R @ ³ is isopropyloxy, R @ ⁴ CH3 CH2 Cl2 and Z are each one corresponding to one of the radicals listed in Table A.

Table 1018

Compounds of the general formula 1.3, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 101.9

Compounds of the general formula 1.4, in which R ³ is iso-propyloxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1020

Compounds of formula (1.5) in which R @ ³ is isopropyloxy, R @ ⁴ CH3 CH3 OCH3 and Z are each corresponding to one of the radicals listed in Table A.

-2.ΊΑTable. 1021

Compounds of the general formula 1.1, in trifluoromethoxy, methyl, and R ⁴ group wherein R ³ is Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1022

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1023

Compounds of the general formula 1.3, in which R ³ is trifluoromethoxy, ^R4 is methyl. and Z is a compound corresponding to one of the residues listed in Table A.

Table 1024

Compounds of the general formula 1.4, in which R ³ is trifluoromethoxy, ^R4 is methyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1025

Compounds of formula (1.5) in which R @ ³ is trifluoromethoxy, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1026

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

* ·

• ♦ · ····· · · • in ···. ··. .... • · · · · · · · · · · • 9 · · · · ··· -.141 -

Table. 1.027 Compounds of general formula 1.2, ve which R ³ represents trifluoromethoxy, R ⁴ ethyl and a group Z then compound.

corresponding to one of the residues listed in Table A.

Table 1028

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1029

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1030

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1031

Compounds of formula (1.1) in which R @ ³ is trifluoromethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1032

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R ^{@ 4} propyl and, in turn, a compound corresponding to one of the radicals listed in Table A.

-H3Table. 1033

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1034

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1035

Compounds of formula (1.5) in which R @ ³ is trifluoromethoxy, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1036

Compounds of general formula 1.1 in which R ³ is trifluoromethoxy, R ⁴ isopropyl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1037

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1038

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1039

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1040

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, ^R4 and isopropyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1041

Compounds of formula (1.1) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1042

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1.043

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1044

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

-Ϊ4 * Γ—

Table 1045

Compounds of formula (1.5) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1046

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, R ⁴ E-3-chloro-2-propeny1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1047

Compounds of the general formula 1.2, in which R ³ is trifluoromethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1048

Compounds of the general formula 1.3, in which R ³ is trifluoromethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1049

Compounds of the general formula 1.4, in which R ³ is trifluoromethoxy, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

«Φ φ I I I I I I I I I I I I I I I

-146Table 1050

Compounds of formula (1.5) in which R @ ³ is trifluoromethoxy, R ^{@ 4} E-3-chloro-2-propenyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1051

Compounds of formula (1.1) in which R @ ³ is trifluoromethoxy, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1052

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1053

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1054

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1055

Compounds of formula (1.5) in which R @ ³ is trifluoromethoxy, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

• ·

-2.0 - Table 1056 Compounds of formula 1.1, in trifluoromethoxy, R ⁴ CE ⁴ F and a group kterýcli Z then R ³ means a compound

corresponding to one of the residues listed in Table A.

Table 1057

Compounds of formula (1.2) in which R @ ³ is trifluoromethoxy, R @ ⁴ CE @ F and Z are each one corresponding to one of the radicals listed in Table A.

Table 1058

Compounds of the general formula 1.3, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1059

Compounds of the general formula 1.4, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ F and skupirma Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1060

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1061.

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1062

Compounds of the general formula 1.2, in which R ³ is trifluoromethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1063

Compounds of the general formula 1.3, in which R ³ is trifluoromethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1064

Compounds of the general formula 1.4, in which R ³ is trifluoromethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1065

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1066

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1067

Compounds of the general formula 1.2, in which R ³ is trifluoromethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• «•»

-24 ^ Table 1068

Compounds of formula (1.3) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1069

Compounds of formula (1.4) in which R @ ³ is trifluoromethoxy, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1070

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1071.

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1072

Compounds of formula (1.2) wherein R ³ is trifluoromethoxy, R ⁴ CH ₂ CF ₃ and a. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1073

Compounds of the general formula 1.3, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ and CF _3. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

• »

94 • · 94 • 94 - ttoTable 1074

Compounds of the general formula 1.4, in which R ³ is, trifluoromethoxy, R ⁴ CH ₂ CT _'3 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1075

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1076

Compounds of the general formula 1.1, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A.

Table 1.077

Compounds of the general formula 1.2, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1078

Compounds of formula (1.3) wherein R ³ is trifluoromethoxy, R ⁴ CF ³ C 2 OCH 8 and a group. Z then a compound corresponding to one of the residues listed in Table A.

Table 1079

Compounds of the general formula 1.4, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-2 2- / Table 1080

Compounds of the general formula 1.5, in which R ³ is trifluoromethoxy, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1081

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1082

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1083

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1084

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4} methyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1085

Compounds of formula (1.5) in which R @ ³ is methylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

2.21

Table 1086

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1087

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1088

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1089

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1090

Compounds of formula (1.5) in which R @ ³ is methylthio, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A:

Table 1091

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

·· ·

- 113Table 1092

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1093

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1094

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4} propyl and Z are each one of the radicals listed in Table A.

Table 1095

Compounds of formula (1.5) in which R @ ⁵ is methylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1096

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1097

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table '1098 Compounds of formula (1.3), in kt erých R ³ represents methylthio, R ⁴ isopropyl and Z then compound

corresponding to one of the residues listed in Table A.

Table 1099

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1100

Compounds of formula (1.5) in which R @ ³ is methylthio, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1101

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1102

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1103

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

-2t5 * Table 1104

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1105

Compounds of formula (1.5) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the groups listed in Table A.

Table 1106

Merging the general formula 1.1, in which R ³ represents methylthio, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1107

Compounds of the general formula 1.2, in which R ³ represents methylthio, R ⁴ E-3 "Chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1108

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1109

Compounds of the general formula 1.4, in which R ³ represents methylthio, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-2.16 Table 1110

Compounds of formula (1.5) in which R @ ³ is methylthio, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1111

Compounds of formula (1.1) in which R @ ³² is methylthio, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1112

Compounds of the general formula 1.2, in which R ³ represents methylthio, R ⁴ n-butyl and the group Z corresponds for each compound to one of the ytků listed in Table A.

Table 1113

Compounds of formula (1.3) in which R @ ³ is methylthio, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1114

Compounds of formula (1.4) in which R @ ³ is methylthio, R ^{@ 4} n-butyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1115

Compounds of the general formula 1.5, in which R ³ represents methylthio, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1116

Compounds of the general formula 1.1, in which R ³ represents methylthio, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1117

Compounds of the general formula 1.2, in which R ³ represents methylthio, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1118

Compounds of formula (1.3) wherein R ³ is methylthio, R ^{4 is} CH 2 _; F and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 1119

Compounds of the general formula 1.4, in which R ³ represents methylthio, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table Λ.

Table. 1120

Compounds of the general formula 1.5, in which R ³ represents methylthio, R ⁴ CH ₂ E, and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1121

Compounds of the general formula 1.1, in which R ³ represents methylthio, ^R4, _CHF2 and the group Z compound corresponding to each one of the radicals mentioned in Table A

- 2.2.8 -

Table 1122

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4} CHF .. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1123

Compounds of the general formula 1.3, in which R ³ represents methylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1124

Compounds of the general formula 1.4, in which R ³ represents methylthio, ^R4, _CHF2 and the group Z sloučeninuodpovídající always one of the radicals mentioned in Table A

Table 1125

Compounds of the general formula 1.5, in which R ³ represents methylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1126

Compounds of formula (1.1) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1127

Compounds of formula (1.2) in which R @ ³ is methylthio, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1128

Compounds of formula (1.3), in methylthio, R ⁴ 2-propynyl and a group wherein R ³ is

Z then a compound corresponding to one of the radicals listed in Table A.

Table 1129

Compounds of the general formula 1.4, in which R ³ represents methylthio, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1130

Compounds of formula (1.5) in which:. R ³ represents methylthio, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1131

Compounds of the general formula 1.1, in which R ³ represents methylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1132

Compounds of the general formula 1.2, in which R ³ represents methylthio, R ⁴ CH ₂ CF ₃ and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 1133

Compounds of the general formula 1.3, in which R ³ represents methylthio, R ⁴ CH ₂ CF _3, and Zpak corresponds for each compound to one of the radicals mentioned in Table A.

A · ··

A A ««

230

Table 1134

Compounds of the general formula 1.4, in which R ³ represents methylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table Ά.

Table 1135

Compounds of the general formula 1.5, in which R ³ represents methylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1136

Compounds of the general formula 1.1, in which R ³ represents methylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1137

Compounds of the general formula 1.2, in which R ³ represents methylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each slouičeninu one of the radicals mentioned in Table A

Table 1138

Compounds of the general formula 1.3, in which R ³ represents methylthio, R ⁴ CH 2 CH ₂ 0CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1139

Compounds of formula (1.4) in which R @ ³ is methylthio, R @ ⁴ ClCl2 OCH3 and Z are each one corresponding to one of the radicals listed in Table A.

• · ·

-111Table 1140

Compounds of the general formula 1.5, in which R ³ represents metylLio, R ⁴ CH ₂ CH ₂ CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1141

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4 is methyl and the group Z corresponds for each compound to one of the residuals indicated in Table A.

Table 1142

Compounds of formula (1.2) in which R @ ³ is ethylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1143

Compounds of formula (1.3) in which R @ ³ is ethylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1144

Compounds of formula (1.4) in which R @ ³ is ethylthio, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1145

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 232.Table 1146

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1147

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1148

Compounds of formula (1.3) wherein R ³ is ethylthio, R ⁴ ethyl, and Z is a compound of formula (I). one of the residues listed in Table A.

Table 1149

Compounds of the general formula 1.4, in which R ³ is ethylthio, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A:

Table 1150

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4 ethyl and the group Z corresponds for each compound one of the radicals mentioned in Table A.

Table 1151

Compounds of formula (1.1) in which R @ ³ is ethylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

- 23¾ Table 1152

Compounds of formula (1.2) in which R ^{3 is} O, O, R ^4, propyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1153

Compounds of formula (1.3) in which R @ ³ is ethylthio, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1154

Compounds of formula (1.4) in which R @ ³ is ethylthio, R ^{@ 4} propyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1155

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4, propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1156

Compounds of the general formula 1.1, in which R ³ represents ethylthio, R ^R iso-propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A:

Table 1157

Compounds of formula (1.2) in which R @ ³ is ethylthio, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

· 99 999 99 9 9 99

9

9 9 9 9 9

99 9 9 · »

-Ί36 - Table. 11.58 Compounds of general formula 1.3, ve which R ³ represents ethylthio, R ⁴ isopropyl and a group Z then. compound

corresponding to one of the residues listed in Table A.

Table 1159

Compounds of formula (1.4) in which R @ ³ is ethylthio, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A:

Table 1160

Compounds of formula (1.5) in which R @ ³ is ethylthio, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1161

Compounds of formula (1.1) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1162

Compounds of formula (1.2) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1163

Compounds of formula (1.3) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

······················································. • · · · · · ·

-235 *

Table 1164

Compounds of formula (1.4) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1165

Compounds of formula (1.5) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 1166

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4, E-3-chl.or-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1167

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4, E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1168

Compounds of the general formula 1.3, in which R ³ is ethylthio, ^R4, E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1169

Compounds of the general formula 1.4, in which R ³ is ethylthio, ^R4, E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 236Table '1170

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4, E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1171

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4, n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1172

Compounds of formula (1.2) in which R @ ³ is ethylthio, R ^{@ 4} n-butyl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1173

Compounds of the general formula 1.3, in which R ³ is ethylthio, ^R4, n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1174

Compounds of the general formula 1.4, in which R ³ is ethylthio, ^R4, n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1175

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4, n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• φ

-131Table '117 6

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4 _CH2 F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1177

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4 _CH2 F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1178

Compounds of formula (1.3) wherein R ³ is ethylthio, R ⁴ CH ₂ F and. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1.1.7 9

Compounds of the general formula 1.4, in which R ³ is ethylthio, ^R4 _CH2 F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1180

Compounds of formula (1.5) in which R ³ is ethylthio, R ⁴ CH ₂ F and Z are each one corresponding to one of the radicals listed in Table A.

Table 1181

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• »

-L38Table 1182

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1183

Compounds of the general formula 1.3, in which R ³ is ethylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1184

Compounds of the general formula 1.4, in which R ³ is ethylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table Λ.

Table 1185

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1186

Compounds of the general formula 1.1, in which R ³ is ethylthio, ^R4, 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1187

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4, 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1188

Compounds of formula (1.3) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1189

Compounds of formula (1.4) in which R @ ³ is ethylthio, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1190

Compounds of the general formula 1.5, in which R ³ is ethylthio, ^R4, 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1191

Compounds of the general formula 1.1, in which R ³ represents ethylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1192

Compounds of the general formula 1.2, in which R ³ is ethylthio, ^R4 CII ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1193

Compounds of formula (1.3) in which R @ ³ is ethylthio, R @ ⁴ Cl2 CF, and Z are each one corresponding to one of the radicals listed in Table A.

• • •

-1 ^ 0 Table 1194

Compounds of the general formula 1.4, in which R ³ represents ethylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1195

Compounds of the general formula 1.5, in which R ³ represents ethylthio, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1196

Compounds of the general formula 1.1, in which R ³ represents ethylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 11.97

Compounds of the general formula 1.2, in which R ³ represents ethylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1198

Compounds of the general formula 1.3, in which R ³ represents ethylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1199

Compounds of the general formula 1.4, in which R ³ represents ethylthio, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

·

-264Tabuika 1200

Compounds of formula (1.5) in which R ³ is octyl, R ⁴ CH ₂ CH ₂ OCH ₃ and Z is the corresponding compound. one of the residues listed in Table A.

Table 1201

Compounds of the general formula 1.1, in which R ³ is methylamino, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1202

Compounds of formula (1.2) wherein R ³ is methylamino, R ^{4 is} methyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1.203

Compounds of the general formula 1.3, in which R ³ is methylamino, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1204

Compounds of the general formula 1.4, in which R ³ is methylamino, ^R4 is methyl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1205

Compounds of formula (1.5) wherein R ³ is methylamino, R ⁴ methyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

9

Table 1206

Compounds of formula (1.1) in which R @ ³ is methylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1207

Compounds of formula (1.2) in which R @ ³ is methylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1208

Compounds of formula (1.3) in which R @ ³ is methylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1209

Compounds of formula (1.4) in which R @ ³ is methylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1210

Compounds of formula (1.5) in which R @ ³ is methylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1211

Compounds of formula (1.1) in which R @ ³ is methylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

• to • to • to

- 1 * i 3—

Table 1212

Compounds of formula (1.2) in which R @ ³ is methylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1213

Compounds of formula (1.3) in which R @ ³ is methylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1214

Compounds of the general formula 1.4, in which R ³ is methylamino, ^R4, propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1215

Compounds of formula (1.5) in which R @ ³ is methylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1216

Compounds of formula (1.1) in which R @ ³ is methylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1217

Compounds of formula (1.2) in which R @ ³ is methylamino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1218

Compounds of formula (1.3) in which R @ ³ is methylamino, R ^{@ 4} isopropyl and Z are each one corresponding to one of the radicals listed in Table.

Table 1219

Compounds of formula (1.4) in which R @ ³ is methylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1220

Compounds of formula (1.5) in which R @ ³ is methylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1221

Compounds of the formula I.1 in which R @ ³ is methylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A:

Table 1222

Compounds of formula (1.2) in which R @ ³ is methylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1223

Compounds of formula (1.3) in which R @ ³ is methylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Table 1.224

Compounds of formula (1.4) in which R @ ³ is methylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1225

Compounds of formula (1.5) in which R @ ³ is methylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1226

Compounds of the general formula 1.1, in which R ³ is methylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1227

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1228

Compounds of the general formula 1.3, in which R ³ is methylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 2 ^ 6

Table 1229

Compounds of the general formula 1.4, in which R ³ is methylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1230

Compounds of the general formula 1.5, in which R ³ represents metfylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1.23.1

Compounds of the general formula 1.1, in which R ³ is methylamino, R ⁴ n-butyl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1232

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1233

Compounds of the general formula 1.3, in which R ³ is methylamino, R ⁴ n-butyl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

• ·

- Z.Table 1234

Compounds of the general formula 1.4, in which R ³ is methylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1235

Compounds of the general formula 1.5, in which R ³ is methylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1236

Compounds of the general formula 1.1, in which R ³ is methylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1237

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1238

Compounds of the general formula 1.3, in which R ³ is methylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1239

Compounds of the general formula 1.4, in which R ³ is methylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · · · · · · · · · · · · · ·

_ 2- <rg Table 1240

Compounds of the general formula 1.5, in which R ³ represents mety1arn and amino, R ⁴ CH ₂ F and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1241

Compounds of the general formula 1.1, in which R ³ is methylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1242

Compounds of the general formula 1.2, in which R ³ is methylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1243

Compounds of the general formula 1.3, in which R ³ is methylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1244

Compounds of the general formula 1.4, in which R ³ is methylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1245

Compounds of the general formula 1.5, in which R ³ is methylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

Table 1246 Compounds of formula 1.1, ve which R ³ represents methylamino, R ⁴ 2-propynyl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 1247

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1248

Compounds of the general formula 1.3, in which R ³ is methylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound jedomu of the radicals mentioned in Table A.

Table 1249

Compounds of the general formula 1.4, in which R ³ is methylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1250

Compounds of the general formula 1.5, in which R ³ is methylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1251

Compounds of formula (1.1) in which R @ ³ is methylamino, R @ ⁴ CH3 CF6 and Z are each corresponding to one of the radicals listed in Table A.

-1SO Table 1252

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1253

Compounds of the general formula 1.3, in which R ³ is methylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1254

Compounds of the general formula 1.4, in which R ³ is methylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table Λ.

Table 1255

Compounds of the general formula 1.5, in which R ³ is methylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

1256

Compounds of the general formula 1.1, in which R ³ is methylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1257

Compounds of the general formula 1.2, in which R ³ is methylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · • ·

Table 1258 Compounds of general formula 1.3, ve which R ³ represents methylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and a group Z then compound corresponding to one of residues listed in Table A. Table 1259 Compounds of general formula 1.4, ve which R ³ represents methylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and a group Z then compound corresponding to one of residues listed in Table A. Table 1260 Compounds of general formula 1.5, ve which R ³ represents methylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and a group Z then compound corresponding to one of residues listed in Table A. Table 1261 Compounds of formula 1.1, ve which R ³ represents dimethylamino, R ⁴ methyl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 1262

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1263

Compounds of formula (1.3) in which R @ ³ is dimethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1264

Compounds of the general formula 1.4, in dimethylamino, ^R4 is methyl and the group Z which then each corresponding to one of the radicals mentioned in Table A.

R ³ means a compound

Table 1265

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1266

Compounds of the general formula 1.1, in which R ³ is dimethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

1267

Compounds of the general formula 1.2, in which R ³ is dimethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1268

Compounds of formula (1.3) in which R @ ³ is dimethylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1269

Compounds of the general formula 1.4, in which R ³ is dimethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · ·

-ira -

Table 1270

Compounds of the general formula 1.5, in which R ³ is dimethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1271

Compounds of formula (1.1) in which R @ ³ is dimethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1272

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1273

Compounds of formula (1.3) in which R @ ³ is dimethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1274

Compounds of formula (1.4) in which R @ ³ is dimethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1275

Compounds of the general formula 1.5, in which R ³ is dimethylamino, ^R4 propyl. and Z is a compound corresponding to one of the radicals listed in Table A.

-2-n - Table 1276 Compounds of formula (I) . 1, ve which R ³ represents dimethylamino, R ⁴ isopropyl and group Z then compound

corresponding to one of the residues listed in Table A.

Table 1277

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4} isopropyl and Z [kappa] is a compound corresponding to one of the radicals listed in Table A.

Table 1278

Compounds of formula (1.3) in which R @ ³ is dimethylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1279

Compounds of formula (1.4) in which R @ ³ is dimethylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1280

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R ^{@ 4} isopropyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1281

Compounds of formula (1.1) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

·· ·· 99 ··

9 9 9 9 9 9 * 4 ·· 9 9 99

9 9 9 9 · «·· ·

9 9 9 9 9

99 99 99

· ♦ ·

Table 1282

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1283

Compounds of formula (1.3) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1284

Compounds of formula (1.4) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1285

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1286

Compounds of formula (1.1) in which R @ ³ is dimethylamino, R ^{@ 4} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1287

Compounds of the general formula 1.2, in which R ³ is dimethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1288

SLoučenirry general formula 1.3, in which R ³ is dimethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1289

Compounds of the general formula 1.4, in which R ³ is dimethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1290

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R ^{@ 4} -3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1291

Compounds of the general formula 1.1, in which R ³ is dimethylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1292

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

·· • ·· ·· ·· ·· • · ·· • · • • · • • • · • • · ··· • · ·· • · • · • · • · • ··· • • • · • • · • · • • • ·· ··· O ·· ·· ··

Table 1293 Compounds of general formula 1.3, ve which R ³ represents dimethylamino, R ⁴ n-butyl and a group Z then compound corresponding to one of residues listed in Table A. Table 1294 Compounds of general formula 1.4, ve which R ³ represents dimethylamino, R ⁴ n-butyl and a group Z then compound corresponding to one of residues listed in Table A. Table 1295 Compounds of general formula 1.5, ve which R ³ represents dimethylamino, R ⁴ n-butyl and a group Z then. compound

corresponding to one of the residues listed in Table A.

Table 1296

Compounds of the general formula 1.1, in which R ³ is dimethylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of zbytlů listed in Table A.

Table 1297

Compounds of the general formula 1.2, in which R ³ is dimethylamino, R ⁴ CH ₂ F and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 1298

Compounds of the general formula 1.3, in which R ³ is dimethylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-253Table 1299

Compounds of the general formula 1.4, in which R ³ is dimethylamino, R ⁴ CH ₂ F askupina Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1300

Compounds of the general formula 1.5, in which R ³ is dimethylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1301

Compounds of the general formula 1.1, in which R ³ is dimethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1302

Compounds of formula (1.2) wherein:. ^R3 is dimethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1303

Compounds of the general formula 1.3, in which R ³ represents, dimethylamino, ^R4, _CHF2 and the group Z corresponds for each sloučeinu one of the radicals mentioned in Table A

Table 1304

Compounds of the general formula 1.4, in which R ³ is dimethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

·· _ 2.Γ <? Table 1305

Compounds of the general formula 1.5, in which R ³ is dimethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1306

Compounds of the general formula 1.1, in which R ³ is dimethylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1307

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1308

Compounds of formula (1.3) wherein R @ ³ is dimethylamino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1309

Compounds of formula (1.4) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1310

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

· · · · · · · · · · · · · · · · · · · · · ·

- 260Table 1311

Compounds of the general formula 1.1, in which R ³ is dimethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1312

Compounds of formula (1.2) in which R @ ³ is dimethylamino, R ^{@ 4} CH3 CF3 and Z are each corresponding to one of the radicals listed in Table A.

Table 1313

Compounds of the general formula 1.3, in which R ³ is dimethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1314

Compounds of the general formula 1.4, in which R ³ is dimethylamino, R ⁴ CH ₂ CF ₃ group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1315

Compounds of formula (1.5) in which R @ ³ is dimethylamino, R @ ⁴ CH3 CF3 and Z are each corresponding to one of the radicals listed in Table A.

Table 1316

Compounds of the general formula 1.1, in which R ³ is dimethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 2X-Table 1317

Compounds of formula 1.2, in dimethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and a group wherein R ³ is

Z then a compound corresponding to one of the radicals listed in Table A.

Table 1318

Compounds of the general formula 1.3, in which R ³ is dimethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1319

Compounds of the general formula 1.4, in which R ³ is dimethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1320

Compounds of the general formula 1.5, in which R ³ is dimethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1321

Compounds of formula (1.1) in which R @ ³ is ethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1322

Compounds of formula (1.2) in which R @ ³ is ethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

- 262 Table 1323

Compounds of formula (1.3) in which R @ ³ is ethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1324

Compounds of the general formula 1.4, in which R ³ is ethylamino, ^R4 is methyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1325

Compounds of formula (1.5) in which R @ ³ is ethylamino, R ^{@ 4} methyl and Z are each corresponding to one of the radicals listed in Table A below.

Table 1326

Compounds of the general formula 1.1, in which R ³ is ethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1327

Compounds of formula (1.2) in which R @ ³ is ethylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1328

Compounds of the general formula 1.3, in which R ³ is ethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

2.G3Table 1.32 9

Compounds of formula (1.4) in which R @ ³ is ethylamino, R ^{@ 4} ethyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1330

Compounds of the general formula 1.5, in which R ^J is ethylamino, ^R4 ethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1331

Compounds of formula (1.1) wherein R ³ is ethylamino, R ^{4 is} propyl, and the like. Z then a compound corresponding to one of the radicals listed in Table A.

Table. 1.332

Compounds of the general formula 1.2, in which R ³ represents ethylamino, propyl, and R ^4. Group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1333

Compounds of formula (1.3) in which R @ ³ is ethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

Table 1334

Compounds of formula (1.4) in which R @ ³ is ethylamino, R ^{@ 4} propyl and Z are each corresponding to one of the radicals listed in Table A.

«· • ·

- tch Table 1335

Compounds of formula (1.5) in which R @ ³ is ethylamino, R ^{@ 4} propyl and Z are each one of the radicals listed in Table A.

Table 1336

The compounds of geneal formula 1.1 wherein ^R3 is ethylamino, ^R4 iso-propyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1337

Compounds of formula (1.2) in which R @ ³ is ethylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1338

The compounds of the general formula # ³ in which R @ ³ is ethylamino, R ^{@ 4} isopropyl and Z is each a compound corresponding to one of the radicals listed in Table A.

Table 1339

Compounds of formula (1.4) in which R @ ³ is ethylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1340

Compounds of formula (1.5) in which R @ ³ is ethylamino, R ^{@ 4} isopropyl, and Z is a compound corresponding to one of the radicals listed in Table A.

• · · • · · · • · · • · · • · · · · • · · · · · • · · · • · · · · · • · · · • · · · · · - 26Γ * - Table 1341 Compounds of formula 1.1, ve which R ³ represents ethylamino, R ⁴ 2-propenyl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 1342

Compounds of formula (1.2) in which R @ ³ is ethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1343

Compounds of the general formula 1.3, in which R ³ represents ethylamino, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1344

Compounds of formula (1.4) in which R @ ³ is ethylamino, R ^{@ 4 is} 2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1345

Compounds of the general formula 1.5, in which R ³ represents ethylamino, R ⁴ 2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1346

Compounds of the general formula 1.1, in which R ³ represents ethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 2 € GTtable 1347

Compounds of formula (1.2) in which R @ ³ is ethylamino, R @ ^{c is} E-3-chloro-2-propenyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1348

Compounds of the general formula 1.3, in which R ³ represents ethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1349

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ E-3-chloro-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1350

Compounds of the general formula 1.5, in which R ³ represents ethylamino, R ⁴ E-3-chl.or-2-propenyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1351

Compounds of formula (1.1) in which R @ ³ is ethylamino, R ^{@ 4} n-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1352

Compounds of the general formula 1.2, in which R ³ represents ethylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1353

Compounds of formula (1.3), in ethylamino, R ⁴ n-butyl and a group in which R ³ is Z then a compound corresponding to one of the radicals listed in Table A.

Table 1354

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1355

Compounds of the general formula 1.5, in which R ³ represents ethylamino, R ⁴ n-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1356

Compounds of the general formula 1.1, in which R ³ represents ethylamino, R ⁴ CH ₂ F and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1357

Compounds of formula (1.2) in which R @ ³ is ethylamino, R ^{@ 4} CT @ ¹ and Z are each corresponding to one of the radicals listed in Table A.

Table 1358

Compounds of formula (1.3) wherein R ³ is ethylamino, R ⁴ CH ₂ F and. Z then a compound corresponding to one of the radicals listed in Table A.

- 268 -

Table 1359

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ CH ₂ F and benzylthio Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1360

Compounds of formula (1.5) in which R @ ³ is ethylamino, R @ ⁴ Cl @ ⁴ F and Z are each corresponding to one of the radicals listed in Table A.

Table 1361

Compounds of formula (1.1) in which R ³ is ethylamino, R ⁴ CHF ₂ and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1362

Compounds of the general formula 1.2, in which R ³ is ethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1363

Compounds of the general formula 1.3, in which R ³ is ethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1364

Compounds of the general formula 1.4, in which R ³ is ethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · · ·

Table 1365

Compounds of the general formula 1.5, in which R ³ is ethylamino, ^R4, _CHF2 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1366

Compounds of formula (1.1) in which R @ ³ is ethylamino, R ^{@ 4 is} 2-propynyl and Z is each one corresponding to the radicals listed in Table A.

Table 136'7

Compounds of the general formula 1.2, in which R ³ represents ethylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1368

Compounds of formula (1.3) in which R @ ³ is ethylamino, R ^{@ 4 is} 2-propynyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1369

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1370

Compounds of the general formula 1.5, in which R ³ represents ethylamino, R ⁴ 2-propynyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· · • • · · · · · · · · · · · · · · · · · · · ·

- ί 'ί -

Table 1371

Compounds of the general formula 1.1, in which R ³ represents ethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1372

Compounds of the general formula 1.2, in which R ³ represents ethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1373

Compounds of the general formula 1.3, in which R ³ represents ethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1374

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1375

Compounds of the general formula 1.5, in which R ³ represents ethylamino, R ⁴ CH ₂ CF ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1376

Compounds of the general formula 1.1, in which R ³ represents ethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 24-1 Table 1377

Compounds of the general formula 1.2, in which R ³ represents ethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1378

Compounds of the general formula 1.3, in which R ³ represents ethylamino, R ⁴ CH ₂ CH ₂ 0CH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1379

Compounds of the general formula 1.4, in which R ³ represents ethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1380

Compounds of formula (1.5) in which R ³ is ethylamino, R ⁴ CH ₂ CH ₂ OCH ₃ and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 1381

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 2-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1382

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-Lit Table 1383

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 2-butyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1384

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1385

Compounds of the general formula 1.5, in which R ³ is methyl, R 2 ^r-butyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1386

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 2-methylprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1387

Compounds of the general formula 1.2, in which R ³ is methyl, ^R4 is 2-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1388

Compounds of the general formula 1.3, in which R ³ is methyl, ^R4 is 2-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-215Table 1389

Compounds of formula (1.4) in which methyl,

R ^{4 is} 2-methylprop-1-yl and a group

Z then

R 'means a compound corresponding to one of the residues listed in Table A.

Table 1390

Compounds of formula (1.5) wherein R ³ is methyl, R ^{4 is} 2-methylprop-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1391

Compounds of vzrce 1.1, in which R ³ is methyl, R ⁴ 1,1-Dimethylethyl-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1392

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} 1,1-dimethylet-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1393

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 1,1-dimethylethyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1394

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 1,1-Dimethylethyl-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

· · · · · <<<<<• • • • · • • · • • · • • • • • • • • • • · · · · · · · · · · · · · · · · · · · · · · · · ·

- 2-MTable 1395

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 1,1-Dimethylethyl-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1396

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 1-pentyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1397

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 1-pentyl and Z is a compound corresponding to one of the radicals listed in the table. AND.

Table 1398

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 1-pentyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1399

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 1-pentyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1400

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 1-pentyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-23-5 *

Table 1401

Compounds of the general formula 1.1, in methyl, R ⁴ 3-methylbut-l-yl and the group wherein R ³ represents

Z then a compound corresponding to one of the radicals listed in Table A.

Table 1402

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-methylbut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1403

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 3-methylbut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1404

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-methylbut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1405

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-methylbut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1406

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 2,2-dimethylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 246

Table 1407

Compounds of formula 1.2 wherein R ³ is methyl, R ^{4 is} 2,2-dimethylprop-1-yl and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 1408

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2,2-dimethylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1409

Compounds of formula (1.4) wherein R @ ³ is methyl, R ^{@ 4 is} 2,2-dimethylprop-1p-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1410

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2,2-dimethylprop-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1411

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} 2-methylbut-1-yl and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 1412

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-methylbut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · · · · · · · · · · · ·

Table 1413

Compounds of the general formula 1.3, in which R ^j is methyl, R ⁴ 2-Methyl IBU T-1. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1414

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2-methylbut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1415

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-methylbut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1416

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ methylbut-1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1417

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 1-methylbut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1418

Compounds of formula 1.3 wherein R ³ is methyl, R ^{4 is} 1-methylbut-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1419

In general, 2-methyl-methyl, R ^4, 11-methyl-but-1-yl and corresponding to one of the following in Table A.

: .4, ve which R ³ represents group Z then net compound pentyl? i group From 4 residues

Table 1420

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ methylbut-1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1421

Compounds of general formula 1.1 wherein R ³ is methyl, R ^{4 is} 3-pentyl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1422

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-pentyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1.42 3

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 3-pentyl and Z is each corresponding to one of the radicals listed in Table A.

Table 1424

Compounds of the general formula 1.4, in which R ³ is methyl, R ³ 3-pentyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1425

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 3-pentyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1426

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 3-methylbutan-2-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1427

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-methylbutan-2-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1428

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 3-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1429

Compounds of formula (1.4) wherein R ³ is methyl, R ^{4 is} 3-methylbutan-2-yl and Z is the corresponding compound. one of the residues listed in Table A.

Table 1430

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1431

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ mety1 2-butan-2-yl, and the first group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1432

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1433

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1434

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1435

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-methylbutan-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1436

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 1-hexyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-2.31

Table. 1437

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 1-hexyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1438

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 1-hexyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1439

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 1-hexyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1440

Compounds of formula (1.5) in which:. R ³ is methyl, R ^{4 is} 1-hexyl and Z is then. a compound corresponding to one of the residues listed in Table A.

Table 1441

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3,3-dimethyl-butan-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1442

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3,3-dimethylbutan-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

- 2.81 -

Table 1443

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 3,3-dimethyl-butan-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1444

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3,3-dimethyl-butan-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1445

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3,3-dimethyl-butan-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1446

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ et.ylbut-2-yl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 1447

Compounds of formula (1.2) wherein R ³ is methyl, R ^{4 is} 2-ethyl-but-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1448

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

···············································

Table 1449

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1450

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1451

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 1-methylprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1452

Compounds of czorc EL.2 wherein R ³ is methyl, R ⁴ 1-methylprop-l-yl, and. Sloučninu group Z corresponds for each one of the radicals mentioned in Table A

Table 1453

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 1-ethylbut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

1454

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 1-methylprop-l-yl, and scales from corresponds for each compound to one of the radicals mentioned in Table A.

Table 1455

Compounds of formula (1.5) wherein R ³ is methyl, R ^{4 is} 1-ethylbut-1-yl and Z is a compound corresponding to any one of the radicals listed in Table A.

Table 1456

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 4-methylpent-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1457

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 4-methylpent-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1458

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-methylpent-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1459

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 4-methylpent-1-yl and the group Z @ a is a compound corresponding to one of the radicals listed in Table A.

Table 1460

Compounds of the general formula 1.5, in which R ^j is methyl. R ⁴ 4-methylpent-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · · · · · · · · · ·

Table 1461

Compounds of formula Ι.Ι in which methyl, R ⁴ cyclopropylmethyl and Z are then

R ³ means corresponds for each compound to one of the radicals mentioned in Table A.

Table 1462

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ cyclopropylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1463

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} cyclopropylmethyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1464

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyclopropylmethyl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1465

Compounds of formula (1.5) in which:. R ³ represents methyl, R ⁴ and cyclopropylmethyl. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1466

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ cyclopentylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

18GTable 1467

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ cyclopentylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1468

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ cyclopentylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1469

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyclopentylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1470

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ cyclopentylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1471

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ cyclohexylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1472

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ cyclohexylmethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 14'73

Compounds of the general formula 1.3, where methyl, cyclohexylmethyl and R ⁴ group wherein R ³ is Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1474

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyclohexylmethyl and the group Z corresponds for each compound to one of the radicals mentioned .in Table A.

Table 1475

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ cyclohexylmethyl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table 1476

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ cyklopropylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1477

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ cyklopropylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1478

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ cyklopropylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• 4 • 4

··· · · · · ·

Table 1479

it always corresponds to one of the residues listed in Table Lee Λ

Table 1480

corresponding to one of the./.yts listed in i..aLuK, Table 1481

Table 1482

Compounds of ecobecnério formula 1.2, in which R ³ is methyl, R ⁴ cyklopentylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1483

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 2-cyclopentylet-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1484

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyklopentylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 148 5

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ cykLopentylet-2-yl and the group Z corresponds for each compound to one zezbytků listed in Table A.

Table 1486

Compounds of formula (I.1) wherein R ³ is methyl, R ^{4 is} 2-cyclohexylet-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1487

Všebecného Compounds of formula 1.2 wherein R ³ is methyl, R ⁴ 1ohexylet 2-cyclohexyl-1-one and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1488

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is 2-} cyclohexyl-ethyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1489

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyklohexylet-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1490

Compounds of formula (1.5) wherein R ³ is methyl, R ^{4 is} 2-cyclohexylet-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 14 91

Compounds of formula (1.1), in methyl, R ⁴ 2-fluoro-1-yl and a group wherein R ³ is Z then a compound corresponding to one of the radicals listed in Table A.

Table 1492

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ fluoret-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1493

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ fluoret-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1494

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 2-fluoroethyl _and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1495

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 2-fluoro-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1.4 9 6

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-fluoroprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · · • · · · • · · • · · • · · • · · · · • · · · · • · · · • · · · · · • · · · · · · · • · · · • · · · zw / Z - Table. 14 97 Compounds of general formula 1.2, ve which R ³ represents methyl, R ⁴ 3-fluoroprop-1-yl and a group Z then compound

corresponding to one of the residues listed in Table A.

Table 1498

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 3-fluoroprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1499

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ .3 luorprop-f-1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1500

Compounds of the general formula 1.5, in which R ^j is methyl, R ⁴ 3-fluoroprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1501

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} 2,2-difluoro-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1502

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 2,2-difluoro-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

• ·

Table 1503

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 2,2-difluoroethyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1504

Compounds of formula (1.4) wherein R ³ is methyl, R ^{4 is} 2,2-difluoro-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table. 1505

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2,2-difluoret 1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1506

Compounds of the general formula 1.1, in which R ³ is methyl, R 2 ^{4-Bromet-l-y1,} and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1507

Compounds of the general formula 1.2, in which R ³ is methyl, R 2 ^{4-Bromet-l-y1,} and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1508

Compounds of the general formula 1.3, in which R ³ is methyl, R 2 ^{4-Bromet-l-y1,} and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1509

Compounds of formula (1.4), methyl, (1), (1), (1), (1), (1), (1), (1) • ···· · · · · φ φ φ φ φφφ φφ φφ φφ ··· · · φ φ in which R ³ represents

R ^{4 is 2-} bromoethyl group

Z then. a compound corresponding to one of the residues listed in Table A.

Table 1510

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Bromet-2-L-Y1. Group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1.511

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} 3-bromopropan-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 1512

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-bromopropinyl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 15.13

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 3-bromopropan-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1514

Compounds of formula (1.4) in which R ³ is methyl, R ^{4 is} 3-bromopropan-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · Table 1515

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 3-bromopropanols L and / or a group corresponding to one of the radicals listed in Table A.

Table 1516

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 4-bromobutan-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1517

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 4-bromobutane-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1518

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-bromobutane-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1519

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-bromobutane-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1520

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 4-bromobutane-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1.521

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} 2-iodo-1-yl. a group corresponding to one of the residues listed in Table A.

Table 1522

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 2-iodo-1-yl and Z is a compound corresponding to one of the radicals. listed in Table A.

Table 1523

Compounds of formula (1.3) wherein R ³ is methyl, R ⁴ 2-iodo-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1524

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 2-iodo-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1525

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4} 2-iodo-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1526

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 2-chloroethyl-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · • ·

Table 1527

Compounds of formula wherein R ³ is methyl, R ^{4 is} 2-chloro-1-yl and the group is one corresponding to one of the radicals listed in Table A.

Table 1528

Compounds of formula 1.3 wherein R ³ is methyl, R ^{4 is} 2-chloro-1-yl and. Z is a compound corresponding to one of the radicals listed in Table A.

Table 1529

Compounds of formula (1.4) wherein R ³ is

methyl.R ⁴ 2-chloro-1-yl and Z then. compound corresponding in each case one of the residues listed in Table A.

Table 1530

Compounds \ wherein R ³ is methyl, R ⁴ 2-chloro-1-yl and Z then the compound corresponds to that in each case one of the residues listed in Table A.

Table 1531

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1532

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ··· · · · · · · · · · · ·

Table 1533

The general formula (1.3) in which R @ ³ is methyl, R @ 3 - chlorpropen-1-yl and the group each corresponds to one of the radicals listed in Table A.

Table 1534

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

- Z & 9Table 1535

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-ch1orprop-1 -Y 1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1536

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 4-chlo'rbut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1537

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 4-chlorobut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1538

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-chloro-but-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1539

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-chloro-but-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1540

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 4-chloro-but-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• it

- 2.40 Table 1541

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ kyanomety.I and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1542

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ cyanomethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1543

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ cyanomethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1544

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ cyanomethyl and the group Z. a compound corresponding to one of the residues listed in Table A.

Table 1545

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ cyanomethyl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1546

Compounds of the general formula 1.1, in which R ³ is methyl, R ^4-cyano-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1547

Compounds of formula (1.2), in methyl, R ⁴ 2-cyanoet-1-yl and a group wherein R ³ is

Z then a compound corresponding to one of the radicals listed in Table A.

Table 1548

Compounds of the general formula 1.3, in which R ³ is methyl, R ^4-cyano-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1549

Compounds of the general formula 1.4, in which R ³ is methyl, R ^4-cyano-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1550

Compounds of the general formula 1.5, in which R ³ is methyl, R ^4-cyano-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1551

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-cyanobut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1552

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-cyanoprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

• 9

- 2. Table 1553

Compounds of formula (1.3) wherein methyl, R ⁴ 3-cyanoprop-1-yl and Z then

R ³ means corresponds for each compound to one of the radicals mentioned in Table A.

Table 1554

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-cyanobut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1555

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-cyanobut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1556

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 4-cyanobut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1557

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 4-cyanobut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1558

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-cyanobut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

ΦΦ ΦΦ • Φ Φ

Φ Φ Φ · *

Φ Φ · Φ Φ

Φ Φ · ·· · · * »

9Φ

Φ · Φ

Φ <

Φ ·

Φ4

ΦΦ 99 • 9 · Φ · 9 99 · ΦΦ

Φ Φ · ·· ··

Table 1559

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-cyanobut-yl, and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1560

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 4-cyanobut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1561

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 2-methoxyethyl-1-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1562

Compounds of the general formula 1.2, in which R ^j is methyl, R ⁴ 2methoxyeth-yl and the group Z. a compound corresponding to one of the residues listed in Table A.

Table 1563

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2methoxyeth-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1564

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2methoxyeth-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A

Table 1565

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 2-methoxyet-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1566

Compounds of formula (1.1) wherein R @ ³ is methyl, R ^{@ 4 is} 2-ethoxyet-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1567

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 2-ethoxyet-1-yl and Z is a compound corresponding to one of the radicals listed in Table.

Table 1568

Compounds of the general formula 1.3, in which R ³ is methyl, R 2-ethoxyethyl ^4-yl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A.

Table 1569

Compounds of the general formula 1.4, in which R ³ is methyl, R 2-ethoxyethyl ^4-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1570

Compounds of the general formula 1.5, in which R ³ is methyl, R 2-ethoxyethyl ^4-yl, and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

-29 5 * Table I ka. 1571

Compounds of general formula 1.1. wherein R ³ is methyl, R ^{4 is} 2-isopropoxyet-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1572

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 2-isopropoxyethyl-yl skupian and Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1573

Compounds of formula 1.3 wherein R ³ is methyl, R ^{4 is} 2-isopropoxyet-1-yl and a group. Z then a compound corresponding to one of the residues listed in Table Λ.

Table 1574

Compounds of formula (1.4) wherein R ³ is methyl, R ^{4 is} 2-isopropoxyet-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1575

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-isopropoxyethyl-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1576

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-methoxyprop-l-yl and skupian Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1577

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-methoxyprop-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1578

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 3-methylprop-l-y1, and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1579

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-methoxyprop-l-yl and the group Z corresponds for each compound to one of the radicals vuedených in Table A.

Table 1580

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-methoxyprop-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1581

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} 3-ethoxy-oxo-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1582

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} 3-ethoxyprop-1-yl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1583

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 3-ethoxyprop-1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1584

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-ethoxyprop-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1585

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-ethoxyprop-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1586

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-izopropoxyprop-1-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1587

Compounds of general formula. 1.2, in which R ³ is methyl, R ⁴ izopropoxyprop 3-yl and the group Z corresponds for each compound to one of the radicals vuedených in Table A.

Table 1588

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 3-izopropoxyprop-yl skupian and Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1589

Compounds of vzrce 1.4, in which R ³ is methyl, R ⁴ izopropoxyprop 3-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1590

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ izopropoxyprop-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1591

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 4-methoxybut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1592

Compounds of general formula 1.2 wherein R ³ is methyl, R ^{4 is} 4-methoxybut-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1593

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-methoxybut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1594

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-methoxybut-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

-WTable 1595

Compounds of the general formula 1.5, in which R ^'! is methyl, R &lt; ⁴ &gt; -methoxybutyl and Z is a compound corresponding to one of the radicals listed in Table Λ.

Table 1596

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 4-ethoxybut-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1597

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 4-ethoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1598

Compounds of the general formula 1.3, in which R ³ represents methyl,! <'Ethoxybut-4-yl and skupian Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1599

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-ethoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1600

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 4-ethoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1601

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 4-izopropoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1602

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 4-izopropoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1603

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 4-izopropoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1604

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 4-izopropoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1605

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 4-izopropoxybut-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1606

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ E-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 3ΟΊTable 1607

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ E-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1608

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ E-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1609

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ E-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1610

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1611

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ Z-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1612

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ Z-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• · 30l Table 1613

Compounds of formula (1.3) in which R ³ is methyl, R ^{4 is} Z-but-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1614

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ Z-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1615

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1616

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-methylbut-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1617

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-methylbut-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1618

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ metyl.but 3-en-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• • •

-303Table 1619

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-methylbut-2-en-1-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1620

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-methylbut-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in A. tabulcea

Table 1621

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} 2-methylprop-2-en-1-yl and a group. Z then the compound corresponds to one of the radicals listed in Table A.

Table 1622

Compounds of the general formula 1.2, in which R ³ is methyl, ^R4 is 2-methylprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1623

Compounds of the general formula 1.3, in which R ³ is methyl, ^R4 is 2-methylprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1624

Compounds of the general formula 1.4, in which R ³ is methyl, ^R4 is 2-methylprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-3θ6

Table 1625

Compounds of the general formula 1.5, in which R ³ is methyl, ^R4 is 2-methylprop-2-en ~ -l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1626

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ but-3-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1627

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ but-3-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1628

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} but-3-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1629

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} but-3-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1630

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ but-3-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-3Ο5ΓTable 1631

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} Z-3-chloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1632

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-3-chloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1633

Compounds of formula (1.3) in which R @ ³ is methyl, R @ ^{1 is} Z-3-chloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1634

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} Z-3-chloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1635

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z-3-chloro-prop-2-en-l-yl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1636

Compounds of formula (I) in which R ³ is methyl, R ^{4 is} 2-chloroprop-2-en-1-yl and Z is each a compound corresponding to one of the radicals listed in Table A.

• ·

-306 -

Table 1637

Compounds of the general formula 1.2, in which R ³ is methyl, R 2 ^{4-ch1orprop-2-en-l-y1,} and the group Z corresponds for each compound to one zezbytků listed in Table A.

Table 1638

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ 2-chloro-prop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1639

Compounds of the general formula 1.4, in which R ³ is methyl, R 2 ^{4-ch1orprop-2-en-l-yl} and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1640

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2-chloro-prop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1641

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3,3-dichloropropene-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1642

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ 3,3-dichloropropene-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1643

Methyl compounds, R ^{4 a} compound of general formula 1.3,

3,3-dichloroprop-2-en-1-yl corresponding to one in which R @ ³ and a group of the radicals listed in Table A then represent Table A.

Table 1644

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3,3-dichloropropene-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1645

Methyl compounds, R ⁴ compound of general formula 1.5,

3,3-dichloropropene-2-en-yl .1 each corresponding to one in which R ³ represents a group. Z then the residues listed in ze

Table 1646

Methyl compounds, R ⁴ compound of formula 1.1, ve

2,3,3-trichloroprop-2-en-1-yl corresponding in each case to R ³ and Z to the radicals listed in Table A.

Table 1647

Compounds methyl, R ⁴ compound of formula 1.2, ve

2,3,3-trichloroprop-2-en-1-yl corresponding in each case to R ³ and Z to the radicals listed in Table A.

· «·· · · · · · · · · · ·

«

-308

Table 1648

Compounds of formula (1.3) in which R ³ is methyl, R ^{4 is} 2,3,3-trichloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1649

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 2,3,3-trichloroprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1650

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 2,3,3-trichloroprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1651

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} Z-2,3-dichloroprop-2-en-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1652

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-2,3-dichloroprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

·· ··· · · · · · · · · · ·

B · ··· · · · · · · · · * ·· · · ··

309-

Table 1653 S ubling th e all th e s 1.3 which R ³ represents methyl, R ⁴ Z-2,3-dichloro i r p r o p — 2 — e n-1-y 1 and group i on Z then s1ou c eη i η 1i response in ida ji c i always one of them residues referred to in Table A.

Table 1654 Compounds of the general formula 1.4, ve which R ³ represents methyl, R ⁴ Z-2,3-dichloroprop-2 1-en-1-yl and groups to Z then compound always matching j ednomu ze residues referred to in Table A.

Table 1655 Compounds all general o c c ’1.5, ve of which R ^J is methyl., R. ' Z-2,3-dichloroprop- 2-en-1-yl and group Z then compound always corresponds one of them ; residues referred to in table Λ.

Table 16.56

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} E-2,3-chloro-prop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1657

Compounds methyl, R. ^{4 a} compound of formula 1.2, ve

E-2,3-dichloroprop-2-en-1-yl corresponding in each case to R ³ and Z to the radicals listed in Table A.

• · • ·

4

4

-34ο Compounds methyl, R ⁴ compound of general formula 1.3, ve

E-2,3-dichloro-prop-2-en-1-yl corresponding in each case to R ³ and Z to the radicals listed in Table A.

Table 1659

Compounds r.ei.yi, R ^{4 a} compound of general formula 1.4, ve

E-2,3-dichloroprop-2-en-1-yl corresponding in each case to R ³ and Z to the radicals listed in Table A.

Compounds methyl, R ^{4 a} compound of general formula 1.5, in?

The E-2,3-dichloroprop-2-enyl 1 is in each case one of which R ³ is and the group Z is the radicals listed in Table A.

Table 1661

Compounds of formula (1.1) in methyl, R ^{@ 4} Z-3-bromoprop-2-en-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

wherein R ³ represents

Table. 1662

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-3-bromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

• • •

-344 Table 1663

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} Z-3-bromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1664

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ Z-3-bromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1665

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z-3-bromoprop-2-en-l-y1, and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1666

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} E-3-bromoprop-2-en-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1667

Compounds of formula (1.2) wherein R ³ is methyl, R ^{4 is} E-3-bromoprop-2-en-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1668

Compounds of formula (1.3) in which R ³ is methyl, R ^{4 is} E-3-bromoprop-2-en-1-yl and Z is each a compound corresponding to one of the radicals listed in Table A.

-3H1Table 1669

Compounds of formula (1.4) wherein R @ ³ is methyl, R ^{@ 4} E-3-bromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1670

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-3-bromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1671

Compounds of formula 1.1 wherein R ³ is methyl, R ^{4 is} 2-bromoprop-2-en-1-yl. and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1672

Compounds of formula (T.2) in which R @ ³ is methyl, R ^{@ 4 is} 2-bromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1673

Compounds of formula (1.3) wherein R ³ is methyl, R ^{4 is} 2-bromo-prop-2-en-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table. 167 4

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 2-bromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 16'7 5

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ brom.prop-2-en-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1676

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 3,3-dibromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1677

Compounds of general formula 1.2 in which R ³ is methyl, R ^{4 is} 3,3-dibromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1678

Compounds of the general formula 1.3, in which R ^j is methyl, R ⁴ 3,3-dibromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1679

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4} 3,3-dibromoprop-2-en-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1680

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3,3-dibromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

99 99 99 • • • • • •

Table 1681

Compounds of the general formula II, in which R ³ represents methyl,

R ⁴ 2,3,3-tribromoprop-2-en-1-yl and a group.

a compound corresponding to one of the residues listed in Table A.

Table 1682

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ tribromprop 2,3,3-2-en-l-yl and the group Z, a compound corresponding, in each case one of the radicals mentioned in Table A

Table. 168 3 S .1. o u e n i n y all general of formula 1.3, '' which Rt stands for methyl, R ⁴ 2,3,3-1 ni p r p-2-e n-1-y 1 and group Z then s 1 o u e n i n u u d d o i d i j i c always one from residues mentioned in

Table A.

Table 1684

Compounds general formula 1.4, ve which R ³ means methyl, R ⁴ 2,3,3-Tribromoprop-2-en-1-yl and a group Z then compound corresponding always one that residues uve děných v Table A. Table. 168 5 Compounds general formula 1.5, ve which R ³ means methyl, R ⁴ 2,3,3-1: ribromprop-2-ene-1 yl a skup i na Z then compound corresponding always one that residues referred to in Table A.

Table 1 and 1686

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} Z-2,3-dibromoprop-2-en-1-yl and Z is each one of the radicals listed in Table A.

Table 1687

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-2,3-dibromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1688

Compounds of formula (1.3) in which R ³ is methyl, R ^{4 is} Z-2,3-dibromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1689

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ Z-2,3-dibromoprop-2-en-l_yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1.690

Compounds of formula (1.5) in which:. R ³ is methyl, R ^{4 is} Z-2,3-dibromoprop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

-546 -

Table 1691

Methyl compounds, R ⁴ compound of formula 1.1, ve

E-2,3-dibromoprop-2-en-1-yl corresponding in each case to which R @ ³ and the radical group shown in Table A.

Table 1692

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} E-2,3-dibromo-prop-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1693

Compounds of the general formula 1.3, in which R ³ znamenej methyl, R ⁴ E-2,3-dibromoprop-2-en-1-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1694

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ E-2,3-dibromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1695

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-2,3-dibromoprop-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-s-ti '

Tab.1. ka 1696

Compounds of formula (1.1) in which R ³ is methyl, R ⁴ E-2-chloro-but-2-en-1-yl and Z are each a compound corresponding to one of the radicals listed in Table A.

Table 1697

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ E-2-chloro-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table. 1698

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4} E-2-chlorobut-2-en-1-yl or Z are each one corresponding to one of the groups listed in Table A.

Table 1699

Compounds of formula (1.4) in which R @ ^{3 is} a! methyl, R ⁴ E-2-chlorobut-2-en-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1700

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-2-chloro-but-2-en-l-yl and the group Z compound corresponding to each one of the radicals mentioned in Table A

Table 1701

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ Z-2-chloro-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ♦ · ♦ · ♦ ·

Table 1702 S .1. oučenlny general vz : orce 1.2, in which : R ^J means. methyl, R ⁴ Z-2-chlorobut-2-e n-1-yl and Z p and k s i o č '. n i n u. corresponding to one: from the flats listed in Table A.

Table 1703

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ ZZ-chloro-but-Z-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1704

General compounds formula 1.4 in which. R ³ represents methyl, R ⁴ Z-2-chlorobut-2 -en-1-yl a group Z then compound corresponding to one u from residues listed in Table A. Table 17 05 General compounds formulas 1.5 , in which R ³ represents methyl, R ⁴ Z-2-chlorobut-2 -en-1-yl. and group. Z then compound corresponding to one of the residues listed in tal bulce A. Table. 1706 General compounds of formula I.1 , in which R ³ represents methyl, R ⁴ E-3-chlorobut-2 -en-1-yl a group Z then compound corresponding to one of the residues listed in Table A. Table 1707 General training formulas 1.2 , in which R. ³ stands for methyl, R ⁴ E-3-chlorobut-2 -en-1-yl a group Z then merged, nu corresponding to one the residues listed in Table A.

Table 1708

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ E-3-chiorbut-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1709

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ E-3-chloro-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1710

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-3-chloro-but-2-en-l - yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1711

Compounds of formula (1.1) in which R ³ is methyl, R ^{4 is} Z-3-chlorobut-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1712

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} Z-3-chloro, t-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1713

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ Z-3-chloro-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

• ·

- 3ZO Table 1714

Compounds of formula (1.4) in which R ³ is methyl, R ^{4 is} Z-3-chlorobut-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1715

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z-3-chloro-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1716

Compounds of general formula 1.1 in which:. R ³ represents methyl, R ⁴ E-2-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1717

Compounds of general formula 1.2 in which:. R ³ represents methyl, R ⁴ E-2-brom.but-2-en-1-one and the group Z corresponds for each compound then with one of the radicals mentioned in Table A

Table 1718

Compounds of formula 1.3 wherein R ³ is methyl, R ⁴ E-2-bromobut-2-en-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1719

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ E-2-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A

• ·

-324Table 1. ka 1720

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-2-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1721

Compounds of formula 1.1 wherein R ³ is methyl, R ⁴ Z-2-bromo-but-2-en-l-yl and the group Z compound corresponding to one zezbytků always listed in Table A.

Table 1722

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-2-bromobut-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1.723

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ Z-2-bromo-but-2-en-yl and the group Z and the first compound to the corresponding, in each case one of the radicals mentioned in Table A

Table 1724

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ Z-2-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1.725

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z-2-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-522.Tabulka 1726 The compounds of general formula 1.1, in which R ^j is methyl, 1 <^'E - 3-b Rombo t-2-en - 1 -yia group Z corresponding compound. one of the residues listed in Table A.

Table 1727

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} E-3-bromobut-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1728

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ E-3-bromo-but-2-en-1-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1729

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4} E-3-oxo-but-2-en-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table .1730

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ E-3-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1731

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} Z-3-bromobut-2-en-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · • · · · · · · · · · · · · · ·

Table 1732

Compounds of formula (1.2) in which R ³ is methyl, R ^{4 is} Z-3-bromobut-2-en-1-yl and Z is each a compound corresponding to one of the radicals listed in Table A.

Table 1733

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ Z 3-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1734

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ Z-3-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A

Table 1735

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ Z 3-bromo-but-2-en-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1736

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1737

The compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-2-yn - + - yl and Z is a compound corresponding to one of the radicals listed in Table A.

• • • •

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ··

Table '17 38

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4} 3-chloro-prop-2-yl-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1739

Compounds of formula (1.4) in which R @ ³ is methyl, R @ ^13, 3-chloroprop-2-yn-1-yl, and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1740

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} 3-chloroprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1741

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} 3-bromoprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1742

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} 3-bromoprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table. 174 3

Sloučeiny general formula 1.3, in which R ³ is methyl, R ⁴ 3-bromoprop-2-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

V · 4 · 0 · 4 ···· · ··

0 0 4 4 00 0 0440

-32.5-The bullet 1'744

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ 3-bromoprop-2-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1745

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ 3-bromoprop-2-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1746

Compounds of formula 1.1 wherein R ³ is methyl, R 4 is 3-iodoprop-2-yn-1-yl and a group. Z then a compound corresponding to one of the radicals listed in Table A.

Table 1747

Compounds of the general formula 1.2, in which R ³ is methyl, R @ ^4, 3-iodo-2-.in-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1.748

Compounds of formula (1.3) in which R @ ³ is methyl, R ^{@ 4 is} 3-iodoprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1749

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} 3-iodoprop-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

• * ·

Table k < 1750

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4} 3-iodoprop-2-yn-1-yl and Z are each one corresponding to one of the radicals listed in Table A.

Table 1751

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4 is} but-2-i-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1.752

Compounds of formula (1.2) wherein:. R ³ represents methyl, R ⁴ but-2-.in-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1753

Compounds of formula 1.3 wherein R ³ is methyl, R ⁴ but-2-yn-1-yl and Z then. a compound corresponding to one of the radicals listed in Table A.

Table 1754

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ But-2 - .. yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1755

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} but-2-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1756

Compounds of the general formula 1.1, in which methyl, R ⁴ but-3-yn-l-yl and the group Z

R ³ means corresponds for each compound to one of the radicals mentioned in Table A.

Table 1757

Compounds of formula (1.2) in which R @ ³ is methyl, R ^{@ 4 is} but-3-yn-1-yl and Z is each corresponding to one of the radicals listed in Table A.

Table 1758

Compounds of formula 1.3 wherein R ³ is methyl, R ⁴ but-3-yn-1-yl. and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1759

Compounds of formula (1.4) in which R @ ³ is methyl, R ^{@ 4 is} but-3-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1760

Compounds of formula (1.5) in which R @ ³ is methyl, R ^{@ 4 is} but-3-yn-1-yl and Z is a compound corresponding to one of the radicals listed in Table A.

Table 1761

Compounds of formula (1.1) in which R @ ³ is methyl, R ^{@ 4} but-3-yn-2-yl and Z are each corresponding to one of the radicals listed in Table A.

♦ · • • 9 99 99 ·· • · • · • · • 9 9 • · • · • • · 999 9 · ·· • · • • · · 9 9 • ··· • · 9 · • • · 9 9 • • · ·· «·· 99 99 ·· ··

-32 <£ Table 1762

Compounds 1.2 which R is methyl, R ⁴ but-3-yn-2-yl. and a group Z then compound corresponding always one of them residues listed in Table A. Table 1763 Compounds 1.3 which R ³ represents methyl, R ⁴ b for t - 3 - i n - 2 - y 1 and a group Z then compound corresponding always one of them residues listed in Table A. Table. 17 64 Compounds 1.4 which R ³ represents methyl, R ⁴ b ut-3-yn-2-yl and a group Z then compound da answers. . always one of them residues mentioned in t. abulce A. Table 1765 Compounds 1.5 which R ³ represents methyl, R ⁴ but-3-yn-2-yl and a group Z then compound corresponding always one of them residues listed in Table A. Table 1766 Compounds 1.1 which R ³ represents methyl, R ⁴ p e n t - 3 - i η - '1 - y 1 and a group. Z then merged, nu corresponding. in all cases residues listed in Table A. Table 1767 Compounds 1.2 which R ³ represents methyl, R ⁴ pent-3-yn-1-yl and a group Z then compound

corresponding to one of the residues listed in Table A.

· · · · · · * *

Table 17 68

Compounds of the general formula 1.3, in which ^R is methyl, R ⁴ pent-3-yn-ly.L. Groups 7 corresponds for each compound to one of the radicals mentioned in Table A.

Table 1769

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ pent-3-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1'770

Compounds of formula (1.5). in which R ^j is methyl, R ⁴ pent-3-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1771

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ pent-4 - yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1772

Compounds of the general formula 1.2, in which R ^j is methyl, R ⁴ pent-4-yn-l-yl, and. The group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1773

Compounds of the general formula 1.3, in which R ³ is methyl, R ⁴ pent-4-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

- 330Ta Bulk 17 '/ 4

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ pent-4-iη 1-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1775

Compounds of the general formula 1.5, in which R ³ is methyl, R ⁴ pent-4-yn-l-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1776

Compounds of the general formula 1.1, in which R ³ is methyl, R ⁴ 3-pentenoate, and η - 2-γ1 and skupirmi Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1777

Compounds of the general formula 1.2, in which R ³ is methyl, R ⁴ pent-3-yn-2-y1 and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1778

Všeoobecného Compounds of formula 1.3 wherein R ³ is methyl, R ⁴ pent-3-yn-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

Table 1779

Compounds of the general formula 1.4, in which R ³ is methyl, R ⁴ pent-3-yn-2-yl and the group Z corresponds for each compound to one of the radicals mentioned in Table A.

-334-

Table 178 0 S1 o u n e n i n e n e n e n e n e n e 1.5, ve which R ³ represents methyl, R ⁴ pent-3-yn-2-yl and group Z then compound

corresponding to one of the residues listed in Table A.

-332Table A

Nr. OF 1 pyrrol-1-yl 2 2 -CH ₃ -pyrr 1 -1 -y 1 3 3 -CH ₃ -pyrr 1 -1 -y 1 4 3,4- _(CH3) 2-pyrrol-l-yl 5 2,5- (CH ₃ ) 2 -pyrrol-1-yl 6 2,3- (CH ₃ ) 2 -pyrrol-1-yl 7 2,4- (CH ₃ ) 2 -pyrrol-1-yl 8 2-CH ₂ CH ₃ -pyrrol-1-yl 9 3-CH ₂ CH ₃ -pyrrol-1-yl 10 3,4- (CH ₂ CH ₃ ) 2 -pyrrol-1-yl 11 2,5- (CH ₂ CH ₃ ) 2 -pyrrol-1-yl 12 2,3- (CH ₂ CH ₃ ) 2 -pyrrol-1-yl 13 2,4- (CH ₂ CH ₃ ) 2 -pyrrol-1-yl 14 2-CH (CH ₃ ) 2 -pyrrol-1-yl 15 Dec 3-CH (CH ₃ ) 2 -pyrrole-1-yl 16 2,5- [CH _{(CH3) 2]} 2-pyrrol-l-yl 17 2,4 - [CH (CH ₃₎ 2] 2-pyrrol-l-yl 18 2-C (CH ₃ ) ₃ -pyrrol-1-yl 19 Dec 3-C (CH ₃ ) ₃ -pyrrol-1-yl 20 May 2,5- [C (CH ₃ ) ₃ ] 2-pyrrol-1-yl 21 2,4- [C (CH3) ₃₎ 2 ^_ pyrrol-yl 22nd 3-C6H5-pyrrol-1-yl 23 2-F-pyrrol-1-yl 24 3-F-pyrrole-1-yl 25 2,3-F 2 -pyrrol-1-yl 26 2,4-F 2 -pyrrol-1-yl 27 Mar: 2,5-F 2 -pyrrol-1-yl 28 3,4-F 2 -pyrrol-1-yl 29 2,3,4-F ₃ -pyrrol-1-yl 30 2,3,5-F ₃ -pyrrol-1-yl

-333 -

Nr. OF 31 2,3,4,5-F4-pyrrol-1-yl 32 2-C1-pyrrolidin-1-yl 33 3-Cl-pyrrol-1-yl 34 2,3-Cl ₂ -pyrrol-1-yl 35 2,4-C12-pyrrol-1-yl 36 2,5-C12-pyrrol-1-yl 37 3,4-C12-pyrrol-1-yl 38 2,3,4-C13-pyrrol-1-yl 39 2,3,5-C13-pyrrol-1-yl 40 2,3,4,5-C14-pyrrol-1-yl 41 2-Br-pyrrol-1-yl 42 3-Br-pyrrol-1-yl 43 2,3-Br 2 -pyrrol-1-yl 44 2,4-Br 2 -pyrrol-1-yl 45 2,5-Br ₂ -pyrrol-1-yl 46 3,4-Br 2 -pyrrol-1-yl 47 2,3,4-Br- ₃ -pyrrol-1-yl 48 2,3,5-Br 3 -pyrrol-1-yl 49 2,3,4,5-Br 4 -pyrrol-1-yl 50 2-CN-pyrrol-1-yl 51 3-CN-pyrrol-1-yl 52 2,3-CN 2 -pyrrol-1-yl 53 2,4-CN 2 -pyrrol-1-yl 54 2,5-CN ₂ -pyrrol-1-yl 55 3,4-CN 2 -pyrrol-1-yl 56 2 -NO2-pyrrole-1-y1 57 3-NO 2 -pyrrol-1-yl 58 2,3- (NO ₂ ) 2 -pyrrol-1-yl 59 2,4- (NO 2) 2 -pyrrol-1-yl 60 2,5- (NO 2) 2 -pyrrol-1-yl 61 3,4 - (NO2) ₂ ^_ pyrrol-yl 62 2 -CF 3 -pyrr 1 -1 -y 1

-33 ^ -

1 ^Nr · OF 63 3-CF ₃ -pyrrol-1-yl 64 2,3- (CF ₃ ) 2 -pyrrol-1-yl 65 2,4- (CF ₃ ) 2 -pyrrol-1-yl 66 2,5- (CF ₃ ) 2 -pyrrol-1-yl 67 3,4- (CF ₃ ) 2 -pyrrol-1-yl 68 2-OCH ₃ -pyrrol-1-yl 69 3-OCH ₃ -pyrrol-1-yl 70 2,3- (OCH ₃ ) 2 -pyrrol-1-yl 71 2,4- (OCH ₃ ) 2 -pyrrol-1-yl 72 2,5- (OCH ₃ ) 2 -pyrrol-1-yl 73 3,4- (OCH ₃ ) 2 -pyrrol-1-yl 74 2-OC 6 H 5 -pyrrol-1-yl 75 3 -OCgH5 -pyrrole-1-y1 76 2-OCH ₂ C 6 H 5 -pyrrol-1-yl 77 OCH2CeH _{3-pyrrol-5-yl} 78 2-COCH ₃ -pyrrol-1-yl 79 3 -COCH ₃ -pyrrol-1-yl 80 2-n (ch ₃ ) 2 * ργχ · χ · οΐ * ι · γΐ 81 3 -N (CH ₃ ) 2 -pyrrol-1-yl 82 3,4- (CO ₂ CH ₂ CH ₃ ) 2 -pyrrol-1-yl 83 3,4- (COCH ₃₎ 2 ^_ pyrrol-l-yl 84 2-C (CH ₃ ) = NOCH ₃ -pyrrol-1-yl 85 3-C (CH ₃ ) = NOCH ₃ -pyrrol-1-yl 86 2-C (CH ₃ ) ^s = NOCH ₂ CH ₃ -pyrrol-1-yl 87 3-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -pyrrol-1-yl 88 2-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -pyrrol-1-yl 89 3-C (CH ₃ ) -NOCH ₂ CH ₃ -pyrrol-1-yl 90 2-C (CH ₃ ) = NOCH (CH ₃ ) 2 -pyrrol-1-yl 91 3-C (CH ₃ ) = NOCH (CH ₃ ) 2 -pyrrol-1-yl 92 2-CO 2 CH ₃ -pyrrol-1-yl 93 3-CO ₂ CH ₃ -pyrrol-1-yl 94 2 -CONH 2 -Pyrrol-1-yl

Nr. OF 95 3-CONH2-pyrrolidin-1-yl 96 2-CONHCH 3 -pyrrol-1-yl 97 3 -CONHCH 3 -pyrrol-1-yl 98 2-CON (CH ₃ ) 2 -pyrrol-1-yl 99 3-CON (CH 3) 2 "Pyrrol-1-yl 100 ALIGN! 2-SCH3-pyrrole-1-y 1 101 3-SCH 3 -pyrrol-1-yl 102 2-SO 2 CH 3 -pyrrol-1-yl 103 3-SO 2 CH 3 -pyrrol-1-yl 104 indol-1-yl 105 3-F-indol-1-yl 106 4-F-indol-1-yl 107 5-F-indol-1-yl 108 6-F-indol-1-yl 109 7-F-indol-1-yl 110 3-Cl-indol-1-yl 111 4-Cl-indol-1-yl 112 5-Cl-indol-1-yl 113 6-Cl-indol-1-yl 114 7-Cl-indol-1-yl 115 3-Br-indol-1-yl 116 4-Br-indol-1-yl 117 5-Br-indol-1-yl 118 6-Br-indol-1-yl; 119 7-Br-indol-1-yl 120 3-CN-indol-1-yl 121 4-CN-indol-1-yl 122 5-CN-indol-1-yl 123 6-CN-indol-1-yl 124 7-CN-indol-1-yl 125 3-NO 2 -indol-1-yl 126 4-NO 2 -indol-1-yl

• • •

- 336 -

Nr. OF 127 5-N02 ^_ indol-l-yl 128 6 -NO2 ^- i ndo 1 -1 -y 1 129 7 -NO2 'indol -1 -y 1 130 2-CH 3 -indol-1-yl 131 3 -CH 3 -indol-1-yl 132 4-CH 3 -indol-1-yl 133 5-CH 3 -indol-1-yl 134 6-CH 3 -indol-1-yl 135 7-CH 3 -indol-1-yl 136 2,3- (CH ₃ ) 2 * indol-1-yl 137 2,5- (CH 3) 2 -indol-1-yl 138 3-OCH 3 -indol-1-yl 139 4-OCH 3 -indol-1-yl 140 5-OCH ₃ -indol-1-yl 141 6-OCH 3 -indol-1-yl 142 7-OCH 3 -indol-1-yl 143 5- (CO 2 CH 3) -indol-1-yl 144 5-OH-indol-1-yl 145 carbazol-1-yl 146 4-Aza-indol-1-yl 147 pyrazol-1-yl 148 3-CN-pyrazol-1-yl 149 4-CN-pyrazol-1-yl 150 5-CN-pyrazol-1-yl 151 3.4 _{2-CN-pyrazol-yl} 152 3,5-CN 2 -pyrazol-1-yl 153 4,5-CN 2 -pyrazol-1-yl 154 3-NO 2 -pyrazol-1-yl 155 4-NO 2 -pyrazol-1-yl 156 5-NO ₂ -pyrazol-1-yl 157 3,4- (NO 2) 2 ^- Pyrazol-1-yl 158 3,5- (NO2) ₂ -Pyrazol-1-yl

Nr. OF 159 4,5- _(NO2) 2-pyrazol-l-yl 160 3-F-pyrazol-1-yl 161 4-F-pyrazol-1-yl 162 5-F-pyrazol-1-yl 163 3,4-F- _2- pyrazol-1-yl 164 3,5-F- _2- pyrazol-1-yl 165 4,5-F- _2- pyrazol-1-yl 166 3,4,5-F 3 -pyrazol-1-yl 167 3-Cl-pyrazol-1-yl 168 4-Cl-pyrazol-1-yl 169 5-Cl-pyrazol-1-yl 170 3,4-Cl ₂ -pyrazol-1-yl 171 3,5-Cl ₂ -pyrazol-1-yl 172 4,5-Cl ₂ -pyrazol-1-yl 173 3,4,5-C13-pyrazol-1-yl 174 3-Br-pyrazol-1-yl 1 ¹⁷⁵ 4-Br-pyrazol-1-yl 1 ¹⁷⁶ 5-Br-pyrazol-1-yl 1 ¹⁷⁷ 3,4-Br- _2- pyrazol-1-yl 178 3,5-Br- _2- pyrazol-1-yl 179 4,5-Br. _2- pyrazol-1-yl 180 3,4,5-Br 3 -pyrazol-1-yl 181 3-CH 3 -pyrazol-1-yl 182 4-CH 3 -pyrazol-1-yl 183 5 -CH 3 -pyrazol-1-yl 184 3,4- (CH 3) ₂ -pyrazol-1-yl 185 3,5- (CH 3) 2 -pyrazol-1-yl 186 4,5- (CH 3) 2 -pyrazol-1-yl 187 3,4,5- (CH 3) 3 -pyrazol-1-yl 188 3 -CH 2 CH 3 -pyrazol-1-yl 189 4-CH 2 CH 3 -pyrazol-1-yl 190 5-CH ₂ CH 3 -pyrazol-1-yl

Nr. 2 191 3,4- (CH 2 CH 3) 2 -pyrazol-1-yl 192 3,5- (CH 2 CH 3) 2 -pyrazol-1-yl 193 4,5- (CH 2 CH 3) 2 -pyrazol-1-yl 194 3-CH ₂ CH ₂ CH ₃ -pyrazol-1-yl 195 4-CH ₂ CH ₂ CH ₃ -pyrazol-1-yl 196 5 -CH 2 CH 2 CH 3 -pyrazo 1 -1 -y 1 197 3,4- (CH 2 CH 2 CH 3) 2 -pyrazol-1-yl 19 8 3,5- (CH 2 CH 2 CH 3) 2 -pyrazol-1-yl 199 4,5- (CH 2 CH 2 CH 3) 2 -pyrazol-1-yl 200 3-CH (CH ₃ ) 2 -pyrazol-1-yl 201 4-CH (CH 3) 2 -pyrazol-1-yl 202 5-CH (CH 3) 2 -pyrazol-1-yl 203 3,4 - [CH (CH ₃ ) 2] 2 "Pyrazol-1-yl 204 3,5- [CH (CH 3) ₂ ] 2 "Pyrazol-1-yl 205 4,5- [CH _{(CH3) 2]} 2-pyrazol-l-yl 206 3-C (CH 3) 3 -pyrazol-1-yl 207 4-C (CH 3) 3 -pyrazol-1-yl 208 5-C (CH 3) 3 -pyrazol-1-yl 209 3,4- [C (CH 3) 3] 2 "Pyrazol-1-yl 210 3,5- [C (CH ₃ ) 3] 2-pyrazol-1-yl 211 4,5- [C (CH ₃ ) 3] 2-pyrazol-1-yl 212 3,4,5- [C (CH ₃ ) 3] 3-pyrazol-1-yl 213 3-CF 3 -pyrazol-1-yl 214 4-CF 3 -pyrazol-1-yl 215 5-CF 3 -pyrazol-1-yl 216 3,4- (CF 3) 2 -pyrazol-1-yl 217 3,5- (CF 3) 2 -pyrazol-1-yl 218 4,5- (CF 3) 2 -pyrazol-1-yl 219 3-OCH 3 -pyrazol-1-yl 220 4-OCH ₃ -pyrazol-1-yl 221 5-OCH ₃ -pyrazol-1-yl 222 3,4- (OCH ₃ ) 2 -pyrazol-1-yl

-33q -

Nr. OF 223 3,5- (OCH ₃ ) 2 -pyrazol-1-yl 224 4,5- (OCH 3) 2 -pyrazol-1-yl 225 3-C 6 H 5 -pyrazol-1-yl 226 4-C ₆ H ₅ -pyrazol-1-yl 227 5 -C 8 H 5 -pyrazol-1-yl 228 3,4- (C6H5) 2-pyrazol-1-yl 229 3- (2'-CH 3 -C 6 H 4) -pyrazol-1-yl 230 3- (3'-CH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 231 3- (4'-CH 3 -C 6 H 4) -pyrazol-1-yl 232 3- [2 ', 3' - (CH ₃ ) 2 -C 6 H ₃ ] -pyrazol-1-yl 233 3- [2 ', 4' - (CH 3) 2 -C 8 H ₃ ) -pyrazol-1-yl 234 3- (2 ', 5' - (CH ₃ ) 2 -C ₆ H ₃ ] -pyrazol-1-yl 235 3- [2 ', 6' - (CH ₃ ) 2 * C ₈ H ₃ ] -pyrazol-1-yl 236 3- [3 ', 4' - (CH 3) 2-06 '] pyrazol-1-yl 237 3- [3 ', 5' - (CH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 3- (2'-F-C 6 H 4) -pyrazol-1-yl 239 3- (3'-F-C 6 H 4) -pyrazol-1-yl 240 3- (4'-F-C 6 H 4) -pyrazol-1-yl 241 3- (2 ', 3'-F 2 -C 6 H 3) -pyrazol-1-yl 242 3- (2 ', 4'-F 2 -C 6 H 3) -pyrazol-1-yl 243 3- (2 ', 5'-F 2 -C 6 H 3) -pyrazol-1-yl 1 ²⁴⁴ 3- (2 ', 6'-F 2 -C 6 H 3) -pyrazol-1-yl 1 ²⁴⁵ 3- (3 ', 4'-F ₂ -C ₆ H ₃ ) -pyrazol-1-yl 246 3- (3 ', 5'-F 2 -C 6 H 3) -pyrazol-1-yl 247 3- (2'-01-06 ') -pyrazol-1-yl 248 3- (3 * -C1-C6H4) -pyrazol-1-yl 249 3- (4'-C 1 -C 6 H 4) -pyrazol-1-yl η 250 3- (2 ', 3' -C 12 -C 6 H 3) -pyrazol-1-yl 251 3- (2 ', 4'-C 12 -C 6 H 3) -pyrazol-1-yl 252 3- (2 ', 5'-C 12 -C 6 H 3) -pyrazol-1-yl 253 3- (2 ', 6'-C 12 -C 6 H 3) -pyrazol-1-yl 254 3- (3 ', 4'-C 12 -C 6 H 3) -pyrazol-1-yl

- 340-

Nr. OF 255 3- (3 ', 5'-C 12 -C 6 H 3) -pyrazol-1-yl 256 3- (2'-Br-CgHi) -pyrazol-1-yl 257 3- (3'-Br-C8Hi) -pyrazol-1-yl 258 3- (4'-ΒΓ-β-β) -pyrazol-1-yl 259 3- (2 ', 3'-Br 2 -C ₆ H 3) -pyrazol-1-yl 260 3- (2 ', 4'-Br 2 * C ₈ H ₃ ) -pyrazol-1-yl 261. 3- (2 ', 5'-Br 2 -C 8 H 3) -pyrazol-1-yl 262 3- (2 ', 6' -Br2-CgH3) -pyrazol-1-yl 263 3- (3 ', 4'-Br 2 -C 8 H 3) -pyrazol-1-yl 264 3- (3 ', 5'-Br 2 -C 8 H 3) -pyrazol-1-yl 265 3- (2 '-CF 3 -C 6 H 4) -pyrazol-1-yl 266 3- (3 '-CF 3 -C 6 H 4) -pyrazol-1-yl 267 3- (4'-CF 3 -C 6 H 4) -pyrazol-1-yl 268 3- [2 ', 3' - (CF ₃ ) 2 -C ₆ H ₃ ] -pyrazol-1-yl 269 3- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ) -pyrazol-1-yl 270 3- (2 ', 5' - (CF ₃ ) ₂ * _{C 6} H ₃ ] -pyrazol-1-yl 271 3- [2 '. 6 '- (CF ₃ ) ₂ -C ₆ H ₃ ) -pyrazol-1-yl 272 3- [3 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ) -pyrazol-1-yl 273 3- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ) -pyrazol-1-yl 274 3- (2'-OCH ₃ -C ₆ H 4) -pyrazol-1-yl 275 3- (3'-OCH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 276 3- (4'-OCH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 277 3- [2 ', 3' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -pyrazol-1-yl 278 3- [2 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 279 3- [2 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 280 3- [2 ', 6' - (OCH ₃ ) 2 * C ₆ H ₃ ] -pyrazol-1-yl 281 3- [3 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 282 3- [3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 283 3- (2'-NO 2 -C 6 H 4) -pyrazol-1-yl 284 3- (3'-NO 2 -C 6 H 4) -pyrazol-1-yl 285 3- (4'-NO 2 -C 6 H 4) -pyrazol-1-yl 286 3- (2'-CN-C6H4) -pyrazol-1-yl

-344-

Nr. OF 287 3- (3 ' -CN-C6H4) -pyrazol-1-yl 288 3- (4 ' -CN-C6H4) -pyrazol-1-yl 289 4- (2'-CH 3 -C 6 H 4) -pyrazol-1-yl 290 4- (3'-CH 3 -C 6 H 4) -pyrazol-1-yl 291 4- (4'-CH 3 -C 6 H 4) -pyrazol-1-yl 292 4- (2 ', 3' - (CH ₃ ) 2 -C 6 H ₃ ] -pyrazol-1-yl) 293 4- [2 ', 4' - (CH 3) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 294 4- [2 ', 5' - (CH 3) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 295 4- [2 ', 6' - (CH 3) ₂ -C ₆ H 3) -pyrazol-1-yl 296 4- [3 ', 4' - (CH 3) ₂ -CeH 3] pyrazol-1-yl 297 4- [3 ', 5' - (CH ₃ ) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 298 4- (2'-F-C 6 H 4) -pyrazol-1-yl 299 4- (3'-F-C 6 H 4) -pyrazol-1-yl 300 4- (4'-F-C 6 H 4) -pyrazol-1-yl 301 4- (2 ', 3'-F ₂ -C ₆ H 3) -pyrazol-1-yl 302 4- (2 ', 4'-F ₂ -C ₈ H 3) -pyrazol-1-yl 303 4- (2 ', 5'-F 2 -C 6 H 3) -pyrazol-1-yl 304 4- (2 *, 6'-F 2 -C 6 H 3) -pyrazol-1-yl 305 4- (3 ', 4'-F 2 -C 6 H 3) -pyrazol-1-yl 306 4- (3 ', 5'-F 2 -C 6 H 3) -pyrazol-1-yl 307 4- (2'-C 1 -C 6 H 4) -pyrazol-1-yl 308 4- (3'-C 1 -C 6 H 4) -pyrazol-1-yl 309 4- (4'-C 1 -C 6 H 4) -pyrazol-1-yl 310 4- (2 ', 3'-C 12 -C 6 H 3) -pyrazol-1-yl 311 4- (2 ', 4'-C 12 -C 6 H 3) -pyrazol-1-yl 312 4- (2 ', 5'-C 12 -C 6 H 3) -pyrazol-1-yl 313 4- (2 ', 6'-C 12 -C 6 H 3) -pyrazol-1-yl 314 4- (3 ', 4'-C 12 -C 6 H 3) -pyrazol-1-yl 315 4- (3 ', 5'-C 12 -C 6 H 3) -pyrazol-1-yl 316 4- (2'-Br-C 8 H 4) -pyrazol-1-yl 317 4- (3'-Br-C 6 H 4) -pyrazol-1-yl 318 4- (4'-Br-C 6 H 4) -pyrazol-1-yl

• 4 4 4 44 44 4 - 3 S 2- *

Nr. OF 319 4- (2 ', 3'-Br 2 -C 6 H 3) -pyrazol-1-yl 320 4- (2 ', 4'-Br 2 -C 6 H 3) -pyrazol-1-yl 321 4- (2 ', 5'-Br2-C8H3) -pyrazol-1-yl 322 4- (2 ', 6'-Br 2 -C 8 H 3) -pyrazol-1-yl 323 4- (3 ', 4'-Br ₂ -C ₆ H ₃ ) -pyrazol-1-yl 324 4- (3 ', 5'-Br ₂ -C ₆ H ₃ ) -pyrazol-1-yl 325 4- (2'-CF 3 -C 6 H 4) -pyrazol-1-yl 326 4- (3'-CF 3 -C 6 H 4) -pyrazol-1-yl 327 4- (4'-CF 3 -C 6 H 4) -pyrazol-1-yl 328 4- [2 ', 3' - (CF ₃ ) 2 -C ₆ H 3] -pyrazol-1-yl 329 4- [2 ', 4' - (CF ₃ ) 2 -C ₆ H 3] -pyrazol-1-yl 330 4- [2 ', 5' - (CF 3) 2 -C 6 H 3] -pyrazol-1-yl 331 4- [2 ', 6' - (CF 3) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 332 4- [3 ', 4' - (CF 3) 2 -C ₆ H ₃ ) -pyrazol-1-yl 333 4- [3 ', 5' - (CF ₃ ) 2 -C 6 H ₃ ] -pyrazol-1-yl 334 4- (2'-OCH 3 -C 6 H 4) -pyrazol-1-yl 335 4- (3'-OCH 3 -C 6 H 4) -pyrazol-1-yl 336 4- (4'-OCH 3 -C ₆ H ₄ ) -pyrazol-1-yl 337 4- [2 ', 3' - (OCH 3) 2 * _{C 6} H ₃ -pyrazol-1-yl 338 4- [2 ', 4' - (OCH 3) 2 -C ₆ H ₃ ] -pyrazol-1-yl 339 4- [2 ', 5' - (OCH ₃ ) 2 -C ₆ H ₃ ] -pyrazol-1-yl 340 4- [2 ', 6' * (OCH 3) 2-06 '] -pyrazol-1-yl 341 4- [3 ', 4' - (OCH 3) 2 -C 6 H 3) -pyrazol-1-yl 342 4- [3 ', 5' - (OCH 3) ₂ -C ₆ H ₃ ] -pyrazol-1-yl 343 4- (2'-NO 2 -C 6 H 4) -pyrazol-1-yl 344 4- (3'-NO 2 -C 6 H 4) -pyrazol-1-yl 345 4- (4'-NO 2 -C 6 H 4) -pyrazol-1-yl 346 4- _{(2'-CN-C6 H4)} -pyrazol-l-yl 347 4- _{(3'-CN-C6 H4)} -pyrazol-l-yl 348 4- (4'-CN-C 6 H 4) -pyrazol-1-yl 349 3-CH 3 -4- (2'-C 1 -C 6 H 4) -pyrazol-1-yl 350 3-CH 3,4 - (3 '- C 1 -C ₆ H ₄ ) -pyrazol-1-yl

-3U «· • ·

Nr. Z ~ ' 351 3-CH ₃ , 4- (4'-C 1 -C 6 H 4) -pyrazol-1-yl 352 3-CH ₃ , 4- (2 ', 4'-Cl ₂ -C ₆ H ₃ ) -pyrazol-1-yl 353 3-CH ₃ , 4- (2'-OCH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 354 3-CH ₃ , 4- (3'-OCH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 355 3-CH ₃ , 4- (4'-OCH ₃ -C ₆ H ₄ ) -pyrazol-1-yl 356 3-CH ₃ , 4- [3'4 '- (OCH ₃ ) ₂ -C ₆ H ₃ -pyrazol-1-yl 357 3-CO ₂ CH ₃ , 4- (2 ', 4'-C ₂ -C ₆ H ₃ ) -pyrazol-1-yl 358 3-CO ₂ CH ₂ CH ₃ , 4- (2 ', 4'-C ₂ -C ₆ H ₃ ) -pyrazol-1-yl 359 3- (3'-NO ₂ -C ₆ H ₄ ), 4-NO ₂ -pyrazol-1-yl 360 3- (3'-NO ₂ -C ₆ H ₄ ), 4-Br-pyrazol-1-yl 361 3- (2 ', 6'-F ₂ -C ₆ H ₃ ), 4-CH ₂ CH ₃ -pyrazol-1-yl 362 3-l-pyrazol-1-yl 363 4-1-Pyrazol-1-yl 364 5-1-Pyrazol-1-yl 365 3,4-1 _2- pyrazol-1-yl 366 3,5-1 _{2-pyrazol-1-yl} 367 4.5 ₂ -1 H -pyrazol-1-yl 368 3,4,5 ₃ -1 H -pyrazol-1-yl at 369 3-OCH ₂ CH ₃ -pyrazol-1-yl 370 4-OCH ₂ CH ₃ -pyrazol-1-yl ³⁷¹ 5-OCH ₂ CH ₃ -pyrazol-1-yl ³⁷² 3,4- (OCH ₂ CH ₃ ) ₂ -pyrazol-1-yl ³⁷³ 3,5- (OCH ₂ CH ₃ ) ₂ -pyrazol-1-yl ³⁷⁴ 4,5- (OCH ₂ CH ₃ ) 2 -pyrazol-1-yl 375 3-OCH _(CH3) 2-pyrazol-1-yl 376 4-OCH (CH ₃ ) 2 -pyrazol-1-yl 377 5 - OCH (CH ₃₎ 2 - pyrazol-1-yl 378 3,4- [OCH (CH ₃ ) ₂ 12-pyrazol-1-yl 379 3,5- [OCH _{(CH3) 2]} 2-pyrazol-1-yl 380 4,5- [OCH (CH _{3) 2} 2 J pyrazol-1-yl 381 3 -OC 6 H 5 -pyrazol-1-yl 382 4 -OC6H5-pyrazol-1-yl

·························································

Nr. OF 383 5-OC 6 H 5 -pyrazol-1-yl 384 3-OCH 2 C 6 H 5 -pyrazol-1-yl 385 4-OCH 2 C 6 H 5 -pyrazol-1-yl 386 5-OCH 2 C 6 H 5 -pyrazol-1-yl 387 3 -COCH 3 -pyrazol-1-yl 388 4-COCH 3 -pyrazol-1-yl 389 5-COCH 3 -pyrazol-1-yl 390 3 -C (CH ₃ ) = NOCH ₃ -pyrazol-1-yl 391 4-C (CH ₃ ) = NOCH ₃ -pyrazol-1-yl 392 5 -C (CH ₃ ) = NOCH ₃ -pyrazol-1-yl 393 3 -C (CH ₃ ) = NOCH ₂ CH ₃ -pyrazol-1-yl 394 4-C (CH ₃ ) = NOCH ₂ CH ₃ -pyrazol-1-yl 395 5-C (CH ₃ ) = NOCH ₂ CH ₃ -pyrazol-1-yl 396 3 -C (CH ₃ ) = NOCH ₂ CH ₂ CH 3 -pyrazol-1-yl 397 4-C (CH ₃ ) = NOCH ₂ CH ₂ CH 3 -pyrazol-1-yl 398 5-C (CH ₃ ) = NOCH ₂ CH ₂ CH 3 - pyrazol-1-yl 399 3-C (CH ₃ ) = NOCH (CH ₃ ) 2 -pyrazol-1-yl 400 4 -C (CH ₃ ) = NOCH (CH 3) 2 -pyrazol-1-yl 401 5-C (CH ₃ ) = NOCH (CH ₃ ) 2 -pyrazol-1-yl 402 3-CO 2 CH 3 -pyrazol-1-yl 403 4-CO 2 CH 3 -pyrazol-1-yl 404 5-CO 2 CH 3 - pyrazol-1-yl 405 3 -CO 2 CH 2 CH 3 -pyrazol-1-yl 406 4-CO 2 CH 2 CH 3 -pyrazol-1-yl 407 5-CO 2 CH 2 CH 3 - pyrazol-1-yl 408 3 -CO 2 CH 2 CH 2 CH 3 -pyrazol -1-yl 409 4-CO ₂ CH ₂ CH ₂ CH 3 - pyrazol-1-yl 410 5-CO 2 CH 2 CH 2 CH 3 -pyrazol-1-yl 411 3-CO ₂ CH (CH ₃ ) 2 -pyrazol-1-yl 412 4-CO 2 CH (CH ₃ ) 2 -pyrazol-1-yl 413 5-CO ₂ CH (CH ₃ ) 2 -pyrazol-1-yl 414 3 -SCH 3 -pyrazol-1-yl

- 3sr-

Nr. OF 415 4-SCH 3 -pyrazol-1-yl 416 5-SCH 3 -pyrazol-1-yl 417 3-SO 2 CH 3 -pyrazol-1-yl 418 4-SO 2 CH 3 -pyrazol-1-yl 419 5-SO 2 CH 3 -pyrazol-1-yl 420 3,4,5- (CF ₃ ) 3 -pyrazol-1-yl 421 3-Cl, 4-Br-pyrazol-1-yl 422 3-Cl, 4-l-pyrazol-1-yl 423 3-Cl, 4-CH 3 -pyrazol-1-yl 424 3-Cl, 5-CH 3 -pyrazol-1-yl 425 3-Cl, 5-CH (CH ₃ ) 2 -pyrazol-1-yl 426 3-Cl, 5-C (CH 3) 3 -pyrazol-1-yl 427 3-Cl, _5-CF3 -pyrazol-1-yl 428 3-Br, 4-Cl-pyrazol-1-yl 429 3-Br, 4-l-pyrazol-1-yl 430 3-Br, 4-CH 3 -pyrazol-1-yl 431 3-Br, 5-CH 3 -pyrazol-1-yl 432 3-Br, 5-CF 3 -pyrazol-1-yl 433 3-1,4-Cl-pyrazol-1-yl 434 3-1,4-Br-pyrazol-1-yl 435 3-1,4 -CH 3 -pyrazol-1-yl 436 3-1,5 -CH 3 -pyrazol-1-yl 437 3 -CH 3, 4-F-pyrazol-1-yl 438 3-CH 3, 4-Cl-pyrazol-1-yl 439 3-CH3,4-Br-pyrazol-1-yl 440 3-CH 3, 4-I-pyrazol-1-yl 441 3 -CH ₃ 4 -CH (CH ₃₎ 2 - pyrazol-1-yl 442 3-CH 3, 5-Br-pyrazol-1-yl 443 3 -CH 3, 5-CH (CH 3) 2 -pyrazol-1-yl 444 3 -CH 3, -CF 3 -pyrazol-1-yl 445 3-CH (CH 3) 2,4-Br-pyrazol-1-yl 446 3-CH (CH 3) 2,5-CH ₃ -pyrazol-1-yl

-

Nr. OF 447 3-CH _{(CH3) 2,} 5-C (CH3) _{3-pyrazol-1-yl} 448 3-CH (CH 3) 2,5-CF 3 -pyrazol-1-yl 449 3 - C (CH ₃₎ 3.4 - Br-pyrazol-1-yl 450 3-C (CH ₃ ) 3,5-CH 3 -pyrazol-1-yl 451 3-C (CH ₃ ) 3,5-CF 3 -pyrazol-1-yl 452 3-CF ₃ , 4-Br-pyrazol-1-yl 453 3-CF 3, 4-CH 3 -pyrazol-1-yl 454 3-CF 3, 5-Br-pyrazol-1-yl 455 3,5- _(CH3) 2> 4-Cl-pyrazol-1-yl 456 3,5-12,4-Br-pyrazol-1-yl 457 3,5-Br _2, 4-Cl-pyrazol-1-yl 458 3-Br, 4,5 -Cl ₂ -pyrazol-1-yl 459 3-CH ₃ , 4,5- (CF ₃ ) 2 -pyrazol-1-yl 460 3,5- _(CH3) 2,4-F-pyrazol-l-yl 461 3,5-Br _2, 4-CH3-pyrazol-1-yl 462 3,4 -Br ₂ 5 CH _(CH3) 2-pyrazol-1-yl 463 3,4-Br _2, 5-C (CH3) _{3-pyrazol-1-yl} 464 3-CH 3, 4-Br, 5-CF 3 -pyrazol-1-yl 465 3-CH 3, 4-Br, 5-CH (CH 3) ₂ -pyrazol-1-yl 466 3-Cl, 4-Br, 5-CH 3 -pyrazol-1-yl 467 3,4-C12,5-CF 3 -pyrazol-1-yl 468 3-F, 4,5- _(CH3) 2-pyrazol-1-yl 469 3,4-Br _2, 5-CF 3 H -pyrazol-1-yl 470 3,5- _(CH3) 2,4-C (CH3) _{3-pyrazol-1-yl} 471 3,5 - [C (CH ₃ ) 3] 2,4-CH ₃ -pyrazol-1-yl 472 3-CH 3, 4-Br, 5-Cl-pyrazol-1-yl 473 3,5- (CH 3) 2,4-1-pyrazol-1-yl 474 3,5- (CH 3) 2,4-Br-pyrazol-1-yl 475 3,4 -Br _2, 5-CH3-pyrazol - 1-yl 476 3,4-12,5-CH ₃ -pyrazol-1-yl 477 3,5- _(CH3) 2,4-CH _(CH3) 2-pyrazol-1-yl 478 3-CH ₃ , 4,5-Cl 2 -pyrazol-1-yl

- 35? -

Nr. OF 479 3,4-C12,5-CH3-pyrazol-1-yl 480 3,5-C12, 4-CH3-pyrazol-1-yl 481 3-CH3,5-C6H5-pyrazol-1-yl; 482 3-CF 3, 4 -CO 2 CH 3 -pyrazol-1-yl 483 3 -CF 3,4 -CO 2 CH 2 CH ₃ -pyrazol-1-yl 484 3,5- (CH 3) 2,4-OCH 3 -pyrazol-1-yl 485 3,5- (CH 3) 2,4-NO 2 -pyrazol-1-yl 486 3-CH 3, 5-CO 2 CH 3 -pyrazol-1-yl 487 3-CH ₃ , 5-CO 2 CH ₂ CH ₃ - pyrazol-1-yl 488 3-CF 3, 4 -C 6 H 5 -pyrazol-1-yl 489 3-CO 2 CH 3, 4-CH 3 -pyrazol-1-yl 490 4-Br, 5-Cl-pyrazol-1-yl 491 4-1,5-Cl-pyrazol-1-yl 492 4-CH 3, 5-Cl-pyrazol-1-yl 493 3-CH 3, 5-Cl-pyrazol-1-yl 494 3-CH (CH 3) 2,5-Cl-pyrazol-1-yl 495 3-C (CH 3) 3,5-Cl-pyrazol-1-yl 496 3-CF 3, 5-Cl-pyrazol-1-yl 497 4-Cl, 5-Br-pyrazol-1-yl 498 4-1,5-Br-pyrazol-1-yl 499 4-CH 3, 5-Br-pyrazol-1-yl 500 4-Cl, 5-1-pyrazol-1-yl 501 4-Br, 5-1-pyrazol-1-yl 502 4-CH3,5-1-pyrazol-1-yl; 503 3-CH 3, 5-I-pyrazol-1-yl 504 4-F, 5-CH 3 -pyrazol-1-yl 505 4-Cl, 5-CH 3 -pyrazol-1-yl 506 4-Br, 5-CH 3 -pyrazol-1-yl 507 4-1,5-CH 3 -pyrazol-1-yl 508 4-CH (CH 3) 2,5-CH 3 -pyrazol-1-yl 509 3-CF 3, 5-CH 3 -pyrazol-1-yl 510 4-Br, 5-CH (CH ₃ ) ₂ -pyrazol-1-yl

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·

Nr. OF 511 3, -C (CH _{3) 3,} 5 - CH _{(CH3) 2-pyrazol-1-yl} 512 3 -CF _3, 5-CH _(CH3) 2-pyrazol-1-yl 513 4-Br, 5-C (CH ₃ ) ₃ -pyrazol-1-yl 514 _3-CH3, 5-C (CH3) _{3-pyrazol-1-yl} 515 _3-CF3, 5-C (CH3) _{3-pyrazol-1-yl} 516 4-Br, 5-CF 3 -pyrazol-1-yl 517 4-CH3,5-CF3-pyrazol-1-yl 518 3,4 ₂ -Cl, -Br, 5-pyrazol-1-yl 519 3,4- (CF 3) 2,5-CH 3 -pyrazol-1-yl 520 3-CH (CH 3) 2,4,5 -Br 2 -pyrazol-1-yl 521 3-C (CH 3) 3,4,5-Br 2 -pyrazol-1-yl 522 3-CF 3, 4-Br, 5-CH 3 -pyrazol-1-yl 523 3-CH _(CH3) 2,4-Br, _5-CH3 -pyrazol-1-yl 524 3-CF 3, 4, 5-Cl 2 -pyrazol-1-yl 525 3,4- _{(CH3) 2,} 5-F-pyrazol-l-yl 526 3-CF 3, 4, 5-Br 2 -pyrazol-1-yl 527 3-CH 3, 4, 5-Br 2 -pyrazol-1-yl 528 3-CH3,4,5-12-pyrazol-1-yl 529 3-C6H5,5-CH3-pyrazol-1-yl; 530 4-NO ₂ , 5-CH ₃ -pyrazol-1-yl 531 _{4-C6H5,5-CH3-pyrazol-1-yl} 532 4-CO 2 CH 3, 5-CF 3 -pyrazol-1-yl 533 4-CO ₂ CH ₂ CH ₃ , 5 -CF ₃ -pyrazol-1-yl 534 3-CO 2 CH _3, 5-CH ₃ -pyrazol-1-yl 535 3-CO ₂ CH ₂ CH ₃ , 5-CH ₃ -pyrazol-1-yl 536 4-Cl, 5-CN-pyrazol-1-yl 537 4-C 6 H 5, 5-CF 3 -pyrazol-1-yl 538 4-CH3,5-CO2CH3-pyrazol-1-yl 539 4 -CH _3, 5 - CO ₂ CH ₂ CH ₂ H -pyrazol-1-yl 540 3-Cl, 4-CH ₂ CH ₃ -pyrazol-1-yl 541 3-Cl, 5-CH ₂ CH 3 -pyrazol-1-yl 542 3-Br, 4-CH ₂ CH ₃ -pyrazol-1-yl

• ·

-3 ^ 9 "

Nr. OF 543 3-Br, 5-CH 2 CH 3 -pyrazol-1-yl 544 3-1,4-CH 2 CH 3 -pyrazol-1-yl 545 3-1,5-CH 2 CH 3 -pyrazol-1-yl 546 3-CH2CH3-4-F-pyrazol-1-yl 547 3-CH 2 CH 3 -4 -Cl-pyrazol-1-yl 548 3 -CH 2 CH 3 -4 -Br-pyrazol-1-yl 549 3 -CH 2 CH 3 -4-1-pyrazol-1-yl 550 3-CH 2 CH 3 -5-Br-pyrazol-1-yl 551 3 -CH 2 CH 3 -5 -CF ₃ -pyrazol-1-yl 552 3 _-CF3, -CH2CH3 4-pyrazol-1-yl 553 4-CH2CH3,5-C1-pyrazol-1-yl 554 3 -CH 2 CH 3, 5-Cl-pyrazol-1-yl 555 4-CH 2 CH 3, 5-Br-pyrazol-1-yl 556 4-CH 2 CH 3, 5-I-pyrazol-1-yl 557 3-CH 2 CH 3,5 -pyrazol-1-yl 558 4-F, 5 -CH 2 CH 3 -pyrazol-1-yl 559 4-Cl, 5-CH 2 CH 3 -pyrazol-1-yl 560 4-Br, 5-CH 2 CH 3 -pyrazol-1-yl 561 4 -1,5 -CH 2 CH 3 -pyrazol-1-yl 562 3 -CF 3,5 -CH 2 CH 3 -pyrazol-1-yl 563 -CH2CH3,5 4 - _CF3 - pyrazol-1-yl ~ 564 3-C 6 H 5, 5-CH 3 CH 3 -pyrazol-1-yl 565 4 -NO2.5 -CH2CH3-pyrazol-1-yl 566 4-C ₆ H ₅ , 5 -CH 2 CH 3 -pyrazol-1-yl 567 3-CO 2 CH 3, 4-NO 2 -pyrazol-1-yl 568 4-NO 2, 5-CO 2 CH 3 -pyrazol-1-yl 569 3-CO 2 CH 2 CH 3, 4-NO 2 -pyrazol-1-yl 570 4-NO2,5 -CO2CH2CH3-pyrazol-1-yl 571 3-CO 2 CH 2 CH 2 CH 3, 4-NO 2 -pyrazol-1-yl 572 4-NO2,5 -CO2CH2CH2CH3-pyrazol-1-yl 573 3-CO 2 CH (CH 3) 2,4-NO 2 -pyrazol-1-yl 574 4-NO ₂ .5-CO ₂ CH (CH ₃ ) 2 -pyrazol-1-yl

• 0 •

-3Γ0

Nr. OF 575 3 -CH = NOCH 3,4 -Br-pyrazol-1-yl 576 3 -CH = NOCH ₂ CH ₃ , 4-Br-pyrazol-1-yl 577 3-NO ₂ , 4-CH ₃ -pyrazol-1-yl 578 3-NO ₂ , 4-CH ₂ CH ₃ -pyrazol-1-yl 579 3-NO ₂ , 4-CH (CH ₃ ) ₂ -pyrazol-1-yl 580 3-NO ₂ , 4-C (CH ₃ ) 3 -pyrazol-1-yl 581 3 -NO _2, 4-F-pyrazol-l-yl 582 3-NO ₂ -Cl 4-pyrazol-1-yl 583 3-NO _2, 4-Br-pyrazol-l-yl 584 -NO ₂ 3 4 -1 H -pyrazol-1-yl 585 3-NO ₂ , 4 -C 8 H 5 -pyrazol-1-yl 586 3-NO ₂ , 4 -CF ₃ -pyrazol-1-yl 587 3-NO ₂ , 4 -CN-pyrazol-1-yl 588 _{3-CH3, 4-NO2-pyrazol-1-yl} 589 3-CH ₃ CH ₃ , 4-NO ₂ -pyrazol-1-yl 590 3 -CH (CH _{3) 2, 4-NO2-pyrazol-1-yl} 591 3-C (CH3) _{3, 4-NO2-pyrazol-1-yl} 592 3-F, 4-NO ₂ -pyrazol-1-yl 593 3-Cl, 4-NO ₂ -pyrazol-1-yl 594 3-Br, 4-NO ₂ -pyrazol-1-yl 595 3 -1,4-NO ₂ -pyrazol-1-yl 596 3 - CgHs 4 -NO _{2-pyrazol-1-yl} 597 3-CF ₃ , 4-NO ₂ -pyrazol-1-yl 598 3-CN, 4-NO ₂ -pyrazol-1-yl 599 3-CN, 4-CH 3 -pyrazol-1-yl 600 3 - CN, 4 - CH ₂ CH 3-pyrazol-1-yl 601 3 -CN, 4-CH (CH ₃ ) 2 -pyrazol-1-yl 602 3 -CN, 4-C (CH 3) 3 -pyrazol-1-yl 603 3-CN, 4-F-pyrazol-1-yl 604 3-CN, 4-Cl-pyrazol-1-yl 605 3-CN, 4-Br-pyrazol-1-yl 606 3-CN, 4-I-pyrazol-1-yl

-3Γ4-

Nr. OF 607 3 -CN, 4 -C 8 H 8 -pyrazol-1-yl 608 3 - CN, 4 - _CF3 - pyrazol-1-yl 609 3-CH 3, 4 -CN-pyrazol-1-yl 610 3-CH ₂ CH ₃ , 4 -CN-pyrazol-1-yl 611 3 -CH (CH _{3) 2,} 4-CN-pyrazol-1-yl 612 3-C (CH3) _3, 4-CN-pyrazol-1-yl 613 3 -C 8 H 4, 4 -CN-pyrazol-1-yl 614 3-CF 3, 4 -CN-pyrazol-1-yl 615 3-CN, 4- (CH 2) 3 CH 3 -pyrazol-1-yl 616 3-C8H4, 4-CH3-pyrazol-1-yl 617 CGH-3 ₅ 4 -CH2CH3 - pyrazol - 1-yl 618 3-C 8 H 8, 4-CH (CH 3) 2 -pyrazol-1-yl 619 3 -C 8 H 4, 4-C (CH 3) 3 -pyrazol-1-yl 620 3-C 8 H 5, 4-F-pyrazol-1-yl 621 3-C8H4,4-Cl-pyrazol-1-yl 622 3-C6H5,4-Br-pyrazol-1-yl 623 3 -C 8 H 4, 4-1-pyrazol-1-yl 624 4-C 8 H 5, 5- (CH 2) 3 CH 3 -pyrazol-1-yl 625 3-C 8 H 8, 4-CF ₃ -pyrazol-1-yl 626 3-CH ₃ , 4-C ₈ H ₈ -pyrazol-1-yl 627 3 -CH 2 CH 3, 4 -C 8 H 5 -pyrazol -1-yl 628 3 - CH _(CH3) 2 »4 - ₅ CGH-pyrazol-1-yl 629 3-C (CH ₃ ) 3,4-C 6 H 5 -pyrazol-1-yl 630 3-F, 4-C8H5-pyrazol-1-yl 631 3-Cl, 4 -C ₈ H ₅ -pyrazol-1-yl 632 3-Br, 4-C8H5-pyrazol-1-yl 633 3-1,4-C6H5-pyrazol-1-yl 634 3-CF 3, 4-C 8 H 8 -pyrazol-1-yl 635 3 -CO 2 CH 2 CH 3, 4 -CH 3 -pyrazol-1-yl 636 Indazol-1-yl 637 3-F-indazol-1-yl 638 4-F-indazol-1-yl

• • • •

- 3Γ2- -

Nr. OF 639 5-F-indazol-1-yl 640 6-F-indazol-1-yl 641 7-F-indazol-1-yl 642 3,4-F _{2-indazol-1-yl} 643 3.5 - ₂ F-indazol-1-yl 644 3.6 - ₂ F-indazol-1-yl 645 3.7 - ₂ F-indazol-1-yl 646 4,5-F ₂ -indazol-1-yl 647 4,6-F _{2-indazol-1-yl} 648 4.7 - ₂ F-indazol-1-yl 649 5.6 - ₂ F-indazol-1-yl 650 5.7 * F ₂ -indazol-1-yl 651 6.7 - ₂ F-indazol-1-yl 652 3-Cl-indazol-1-yl 653 4-Cl-indazol-1-yl 654 5-Cl-indazol-1-yl 655 6-Cl-indazol-1-yl 656 7-Cl-indazol-1-yl 657 3,4-Cl ₂ -indazol-1-yl 658 3,5-Cl ₂ -indazol-1-yl 659 3,6-Cl ₂ -indazol-1-yl 660 3,7-Cl ₂ -indazol-1-yl 661 4,5-Cl ₂ -indazol-1-yl 662 4,6-Cl ₂ -indazol-1-yl 663 4,7-Cl ₂ -indazol-1-yl 664 5,6-Cl ₂ -indazol-1-yl 665 5,7-Cl ₂ -indazol-1-yl 666 6,7-Cl ₂ -indazol-1-yl 667 3-Br-indazol-1-yl 668 4-Br-indazol-1-yl 669 5-Br-indazol-1-yl 670 6-Br-indazol-1-yl

-353 "

Nr. OF 671 7-Br-indazol-1-yl 672 3,4-Br ₂ -indazol-1-yl 673 3,5-Br ₂ -indazol-1-yl 674 3,6-Br ₂ -indazol-1-yl 675 3,7-Br ₂ -indazol-1-yl 676 4,5-Br. ₂ -indazol-1-yl 677 4,6-Br ₂ -indazol-1-yl 678 4,7-Br ₂ -indazol-1-yl 679 5,6-Br ₂ -indazol-1-yl 680 5,7-Br ₂ -indazol-1-yl 681 6,7-Br ₂ -indazol-1-yl 682 3-l-indazol-1-yl 683 4-1-indazol-1-yl 684 5-1-indazol-1-yl 685 6-1-indazol-1-yl 686 7-I-indazol-1-yl 687 3-CH 3 -indazol-1-yl 688 4-CH 3 -indazol-1-yl 689 5-CH 3 -indazol-1-yl 690 6-CH 3 -indazol-1-yl 691 7-CH 3 -indazol-1-yl 692 3,4- (CH ₃ ) ₂ -indazol-1-yl 693 3,5- (CH 3) ₂ -indazol-1-yl 694 3,6- (CH 3) ₂ -indazol-1-yl 695 3,7- (CH 3) ₂ -indazol-1-yl 696 4,5- (CH ₃ ) ₂ -indazol-1-yl 697 4,6- (CH 3) ₂ -indazol-1-yl 698 4,7- (CH 3) ₂ -indazol-1-yl 699 5,6- (CH ₃ ) ₂ -indazol-1-yl 700 5,7- (CH ₃ ) ₂ -indazol-1-yl 701 6,7- (CH ₃ ) ₂ -indazol-1-yl 702 3-NO ₂ -indazol-1-yl

- 359 -

Nr. OF 703 4-NO 2 -indazol-1-yl 704 5-NO 2 -indazol-1-yl 705 6-NO 2 -indazol-1-yl 706 7-NO 2 -indazol-1-yl 707 3,4- (NO 2) 2 'indazol-1-yl 708 3,5- (NO2) 2'- ^indol -1-yl 709 3,6- (NO 2) 2 -indazol-1-yl 710 3,7- (NO 2) 2 -indazol-1-yl 711 4,5- (NO2) 2'indazol-1-yl 712 4,6- (NO 2) 2 -indazol-1-yl 713 4,7- (NO 2) 2 'indazol-1-yl 714 5,6- (NO 2) 2 -indazol-1-yl 715 5,7- (NO 2) 2 * indazol-1-yl 716 6,7- (NO 2) 2 -indazol-1-yl 717 3-CN-indazol-1-yl 718 4-CN-indazol-1-yl 719 5-CN-indazol-1-yl 720 6 -CN-indazol-1-yl 721 7-CN-indazol-1-yl 722 3-CF 3 -indazol-1-yl 723 4-CF 3 -indazol-1-yl 724 5 -CF 3 -indazol-1-yl 725 6 -CF 3 -indazol-1-yl 726 7 -CF 3 -indazol-1-yl 727 3-OCH 3 -indazol-1-yl 728 4-OCH 3 -indazol-1-yl 729 5-OCH 3 -indazol-1-yl 730 6-OCH 3 -indazol-1-yl 731 7-OCH 3 -indazol-1-yl 732 Imidazol-1-yl 733 2-CN-imidazol-1-yl 734 4-CN-imidazol-1-yl

- ^ 55--

Nr. OF 735 5-CN-imidazol-1-yl 736 2,4- (CN) 2-imidazol-1-yl 737 2-CN, 4- (CH ₂ ) 4 CH ₃ -imidazol-1-yl 738 2,5- (CN) 2-imidazol-1-yl 739 4,5- (CN) 2 -imidazol-1-yl 740 2,4,5- (CN) 3 -imidazol-1-yl 741 2-NO2-imidazol-1-yl 742 4-NO ₂ -imidazol-1-yl 743 5-NO2-imidazol-1-yl 744 2,4- (NO 2) 2 -imidazol-1-yl 745 2,5- (NO2) 2-imidazol-1-yl 746 4,5- (NO 2) 2 -imidazol-1-yl 747 2,4,5- (NO ₂ ) 3 -imidazol-1-yl 748 2-F-imidazol-1-yl 749 4-F-imidazol-1-yl 750 5-F-imidazol-1-yl 751 2,4-F- ₂ -imidazol-1-yl 752 2,5-F- _2- imidazol-1-yl 753 4,5-F- _2- imidazol-1-yl 754 2,4,5-F- _3- imidazol-1-yl 755 2-Cl-imidazol-1-yl 756 4-Cl-imidazol-1-yl 757 5-Cl-imidazol-1-yl 758 2,4-Cl ₂ -imidazol-1-yl 759 2,5-Cl ₂ -imidazol-1-yl 760 4,5-Cl ₂ -imidazol-1-yl 761 2,4,5-Cl- _3- imidazol-1-yl 762 2-Br-imidazol-1-yl 763 4-Br-Imidazol-1-yl 764 5-Br-imidazol-1-yl 765 2,4-Br- ₂ -imidazol-1-yl 766 2,5-Br 2 -imidazol-1-yl

• · • ·

Nr. OF 767 4,5-Br 2 -imidazol-1-yl 768 2,4,5-Br ₃ -Imidazol-1-yl 769 2-l-imidazol-1-yl 770 4-l-imidazol-1-yl 771 5-l-imidazol-1-yl 772 2,4-12 * imidazol-1-yl 773 2,5-12-imidazol-1-yl 774 4,5-12 * imidazol-1-yl 775 2,4,5-13-Imidazol-1-yl 776 2-CH 3 -imidazol-1-yl 777 4-CH 3 -imidazol-1-yl 778 5-CH ₃ -imidazol-1-yl 779 2,4- (CH ₃ ) 2 -imidazol-1-yl 780 2,5- (CH ₃ ) 2 -imidazol-1-yl 781 4,5- (CH ₃ ) 2 -imidazol-1-yl 782 2,4,5- (CH ₃ ) ₃ -imidazol-1-yl 783 2-CH2CU2-imidazol-1-yl 784 4-CH ₂ CH ₃ -imidazol-1-yl 785 5-CH ₂ CH ₃ -imidazol-1-yl 786 2,4- (CH ₂ CH ₃ ) 2 -imidazol-1-yl 787 2,5- (CH ₂ CH ₃ ) 2 -imidazol-1-yl 788 4,5- (CH ₂ CH ₃ ) 2 -imidazol-1-yl 789 2 - CH ₂ CH 2 CH ₃ - imidazol-1-yl 790 4-CH ₂ CH ₂ CH ₃ -imidazol-1-yl 791 5-CH ₂ CH ₂ CH ₃ -imidazol-1-yl 792 2,4- (CH ₂ CH ₂ CH ₃ ) 2 -imidazol-1-yl 793 2,5- (CH ₂ CH ₂ CH ₃ ) 2 -imidazol-1-yl 794 4,5- (CH ₂ CH ₂ CH ₃ ) 2 -imidazol-1-yl 795 2-CH (CH ₃ ) 2 * imidazol-1-yl 796 4-CH (CH ₃ ) ₂ -imidazol-1-yl 797 2,4- [CH (CH ₃ ) 2] 2 * imidazol-1-yl 798 2,5- (CH (CH ₃ ) ₂ ) 2'-imidazol-1-yl

• • • • • • • • • • • • • • • • • • • • • • • • • • · · · ·

.....

Nr. of 799 4,5- [CH (CH3) 2 * 2 * imidazol-1-yl 800 2 -C (CH 3) 3 -imidazol-1-yl 801 4-C (CH 3) 3 -imidazol-1-yl 802 5 -C (CH 3) 3 -imidazol-1-yl 803 2,4- [C (CH 3) 3] 2-imidazol-1-yl 804 2,5- [C (CH 3) 3] 2-imidazol-1-yl 805 4,5- [C (CH 3) 3] 2-imidazol-1-yl 806 2 -CF 3 -imidazol-1-yl 807 4-CF 3 -imidazol-1-yl 808 5-CF 3 -imidazol-1-yl 809 2,4- (CF 3) 2 -imidazol-1-yl 810 2,5- (CF 3) 2 -imidazol-1-yl 811 4,5- (CF 3) 2 -imidazol-1-yl 812 2,4,5- (CF 3) 3 -imidazol-1-yl 813 2-OCH 3 -imidazol-1-yl 814 4-OCH 3 -imidazol-1-yl 815 5-OCH 3 -imidazol-1-yl 816 2-C 6 H 5 -imidazol-1-yl 817 4-C6H5-imidazol-1-yl 818 5-C8H8-imidazol-1-yl 819 2-OCH 2 CH 3 -imidazol-1-yl 820 4-OCH 2 CH 3 -imidazol-1-yl 821 5-OCH 2 CH 3 -imidazol-1-yl 822 2-OCH (CH 3) 2 -imidazol-1-yl 823 4-OCH (CH ₃ ) 2 -imidazol-1-yl 824 5-OCH (CH 3) 2 -imidazol-1-yl 825 2-OC8H5-imidazol-1-yl 826 4-OCH5-imidazol-1-yl 827 5-OC8H5-imidazol-1-yl 828 2-OCH 2 C 6 H 5 -imidazol-1-yl 829 4-OCH ₂ C ₆ H ₅ -imidazol-1-yl 830 5-OCH 2 C 6 H 5 -imidazol-1-yl

- 3SM *

Nr. OF 831 2-COCH 3 -imidazol-1-yl 832 _{4-COCH3-imidazol-1-yl} 833 5-COCH 3 -imidazol-1-yl 834 2-C (CH ₃ ) = NOCH ₃ -imidazol-1-yl 835 4-C (CH ₃ ) = NOCH ₃ -imidazol-1-yl 836 5-C (CH ₃ ) = NOCH ₃ -imidazol-1-yl 837 2 -C (CH ₃ ) = NOCH ₂ CH ₃ -imidazol-1-yl 838 4 -C (CH ₃ ) = NOCH ₂ CH ₃ -imidazol-1-yl 839 5-C (CH ₃ ) = NOCH ₂ CH ₃ -imidazol-1-yl 840 2-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -imidazol-1-yl 841 4-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -imidazol-1-yl 842 5-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -imidazol-1-yl 843 2-C (CH ₃ ) = NOCH (CH ₃ ) ₂ -imidazol-1-yl 844 4 -C (CH ₃ ) = NOCH (CH ₃ ) 2 * imidazol-1-yl 845 5 -C (CH ₃ ) = NOCH (CH ₃ ) 2 * imidazol-1-yl 846 2-CO ₂ CH ₃ -imidazol-1-yl 847 4-CO ₂ CH ₃ -imidazol-1-yl 848 5-CO ₂ CH ₃ -imidazol-1-yl 849 2-CO ₂ CH ₂ CH ₃ -imidazol-1-yl 850 4-CO ₂ CH ₂ CH ₃ -imidazol-1-yl 851 5-CO 2 CH 2 CH 3 - imidazol-1-yl 852 2-CO ₂ CH ₂ CH ₂ CH ₃ -imidazol-1-yl 853 4-CO ₂ CH ₂ CH ₂ CH ₃ -imidazol-1-yl 854 5-CO ₂ CH ₂ CH ₂ CH ₃ -imidazol-1-yl 855 2-CO ₂ CH (CH ₃ ) ₂ -imidazol-1-yl 856 4-CO ₂ CH (CH ₃ ) ₂ -imidazol-1-yl 857 5-CO ₂ CH (CH ₃ ) ₂ -imidazol-1-yl 858 2-CH ₃ - imidazol-1-yl 859 4-CH ₃ -imidazol-1-yl 860 5-CH ₃ -imidazol-1-yl 861 2-SO ₂ CH ₃ -imidazol-1-yl 862 4-SO ₂ CH ₃ -imidazol-1-yl

- SS '9 -

Nr. OF .863 5-SO2CH3-imidazol-1-yl 864 2-CH 3, 5-F-imidazol-1-yl 865 2-CH _3,4 -F-imidazol-1-yl 866 2-CH _3, 5-Cl-imidazol-1-yl 867 2-CH ₃ 4-Cl-imidazol-1-yl 868 2-CH ₃ , 5-Br-imidazol-1-yl 869 2-CH _3, 4-Br imidazol-1-yl 870 2 -CH ₃ 5 -1 - imidazol-1-yl 871 2 -CH ₃ 4 -1-imidazol-1-yl 872 2 -CH ₃ 5 -CH (CH ₃₎ 2 - imidazol-1-yl 873 2-CH ₃ , 4-CH (CH ₃ ) 2 -imidazol-1-yl 874 2-CH ₃ , 5 -C (CH ₃ ) 3 -imidazol-1-yl 875 2-CH ₃ , 4-C (CH ₃ ) 3 -imidazol-1-yl 876 2-CH3,5-CF3-imidazol-1-yl 877 2 -CH _{3, 4} -CF ₃ -imidazol-1-yl 878 4-CH3,5 -CF ₃ - imidazol-1-yl 879 5-CH _{3, 4} -CF ₃ -imidazol-1-yl 880 4-CH ₃ , 5-CH (CH ₃ ) 2 -imidazol-1-yl 881 5 -CH ₃ 4 -CH (CH ₃₎ 2 -imidazol-1-yl 882 4-CH ₃ , 5-C (CH ₃ ) ₃ -imidazol-1-yl 883 5-CH _3,4 -C (CH ₃ ) ₃ -imidazol-1-yl 884 2-F, _{5-CH3-imidazol-1-yl} 885 2-F, 4-CH ₃ - imidazol-1-yl 886 2-F, 5-l-imidazol-1-yl 887 2-F, 4-l-imidazol-1-yl 888 2 -1,5-Cl-imidazol-1-yl 889 2 -1,4-Cl-Imidazol-1-yl 890 2 -1,5 -CH ₃ -imidazol-1-yl 891 _2-CH3 -1,4 - imidazol-1-yl 892 4-1,5-Br-imidazol-1-yl 893 4-Br, 5-l-imidazol-1-yl 894 4 -Cl. 5-CH ₃ -imidazol-1-yl

- 360 -

Nr. 2 895 4-CH 3, 5-Cl-imidazol-1-yl 896 _{2-CF3, 5-CH3-imidazol-1-yl} 897 2-CF 3, 4-CH 3 -imidazol-1-yl 898 2 -CF ₃ , 4,5 -C 12 -imidazol-1-yl 899 2-CH3,4,5-12-Imidazol-1-yl 900 2-F, 4,5-12 * imidazol-1-yl 901 2-CH (CH 3) 2,4,5- (CH 3) 2 -imidazol-1-yl 902 2,5- (CH 2 CH 3) 2,4 -CH ₃ -imidazol-1-yl 903 2,4- (CH 2 CH ₃ ) 2,5 -CH ₃ -imidazol-1-yl 904 2,4- (CH ₃ ) 2,5 -CH ₂ CH ₃ -imidazol-1-yl 905 2,5- _(CH3) 2> 4-CH2CH3-imidazol-1-yl 906 2-CH 2 CH _{3, 4} -CH ₃ -imidazol-1-yl 907 -CH2CH3,5 2 -CH ₃ - imidazol-1-yl 908 2 -CH _3, 5 -NO2- imidazol-1-yl 909 2-CH ₃ , 5- (CH ₂ ) 4 CH ₃ -imidazol-1-yl 910 2-CH2CH3,5-F-imidazol-1-yl 911 2-CH2CH3,4-F-imidazol-1-yl 912 2-CH 2 CH 3, 5-Cl-imidazol-1-yl 913 2-CH 2 CH 3,4 -Cl-imidazol-1-yl 914 2-CH 2 CH 3, 5-Br-imidazol-1-yl 915 2-CH 2 CH 3, 4-Br-imidazol-1-yl 916 2 -CH2CH3,5 -1-imidazol-1-yl 917 2-CH 2 CH 3 - 4-I-imidazol-1-yl 918 2-CH ₃ , 4-CH 2 CH ₃ -imidazol-1-yl 919 2-CH 3, 5-CH 2 CH 3 -imidazol-1-yl 920 2-CH 2 CH _3, 5-CF ₃ -imidazol-1-yl 921 2-CH 2 CH _{3, 4} -CF ₃ -imidazol-1-yl 922 4-CH 2 CH _3, 5-CF ₃ -imidazol-1-yl 923 5-CH 2 CH _{3, 4} -CF ₃ -imidazol-1-yl 924 2-F, 5-CH 2 CH 3 -imidazol-1-yl 925 2-F, 4-CH ₂ CH ₃ -imidazol-1-yl 926 2 -1,5-CH 2 CH 3 -imidazol-1-yl

• ·

Nr. OF 927 2-1,4-CH 2 CH 3 -imidazol-1-yl 928 4 - Cl, 5 - CH ₃ CH ₂ - imidazol-1 - yl 929 4-CH2CH3,5-Cl-imidazol-1-yl 930 2 -CF 3,5 -CH 2 CH 3 -imidazol-1-yl 931 2 -CF 3,4 - CH 2 CH 3 - imidazol-1-yl 932 2 - CH2CH3,4 - CH _(CH3) 2 - imidazol-1 - yl 933 2-CH2CH3,4-C (CH3) 3-imidazol-1-yl 934 4-CH (CH ₃ ) 2,5 -CH 2 CH 3 -imidazol-1-yl 935 4-C _(CH3) 3,5-CH2CH3-imidazol-1-yl 936 2-CH 3 -4,5-Cl 2 -imidazol-1-yl 937 2-CH 3 -4,5-Br 2 -imidazol-1-yl 938 2-CH 3 -4,5- (CF 3) 2 -imidazol-1-yl 939 2-Br, 5-CH 3 -imidazol-1-yl 940 2-Br, 4-CH 3 -imidazol-1-yl 941 2-Br, 4,5-Cl 2 -imidazol-1-yl 942 2-Br, 4,5- (CH3) 2-imidazol-1-yl 943 2-CF3,4,5- (CH3) 2-imidazol-1-yl 944 2 - CH (CH ₃ ) 2,5 - CH ₃ - imidazol - 1 - y 1 945 2-CH (CH 3) 2 -4-CH 3 -imidazol-1-yl 946 2-CH (CH ₃ ) 2,4 -C (CH ₃ ) 3 -imidazol-1-yl 947 2-CH (CH ₃ ) 2.5 -CF ₃ -imidazol-1-yl 1 ⁹⁴⁸ 2-CH (CH ₃ ) 2.4 -CF ₃ -imidazol-1-yl 1 949 2-CF 3, 4, 5-Br 2 -imidazol-1-yl 950 2-C (CH 3) 3,4,5-Cl 2 -imidazol-1-yl 951 2 -1,4,5-Br 2 -imidazol-1-yl 952 4-Cl, 5-Br-imidazol-1-yl 953 4-Br, 5-Cl-imidazol-1-yl 954 4-CH 3, 5-Br-imidazol-1-yl 955 4-Br, 5-CH 3 -imidazol-1-yl ⁹⁵⁶ 4-1,5-CH 3 -imidazol-1-yl 957 4-CH3,5-1-Imidazol-1-yl 958 4-F, 5-CH 3 -imidazol-1-yl

- “• 4 · 9 9 9 9 · 9 B B B B B B B B B B B B B B B B B B B B ·· ·· ··

Nr. OF 959 4-CH 3, 5-F-imidazol-1-yl 960 2,5- (CH 3) 2,4-Cl-imidazol-1-yl 961 2,4- (CH 3) 2,5-Cl-imidazol-1-yl 962 2,5-B, 2,4-Cl-imidazol-1-yl 963 2,4-η 2,5 -Cl-imidazol-1-yl 964 2,5- _(CH3) 2,4-CH _(CH3) 2-imidazol-1-yl 965 2,4- (CH 3) 2,5 -CH (CH ₃ ) 2 -imidazol-1-yl 966 2,4-B1,5 -CF 3 -imidazol-1-yl 967 2,5-Br 2, 4-CF 3 -imidazol-1-yl 968 2,4- (CH3) 2 < 5-CF3-imidazol-1-yl 969 2,5- (CF 3) 2,4-CH 3 -imidazol-1-yl 970 2,4- (CF ₃ ) 2,5-CH 3 -imidazol-1-yl 971 2,4-12,5-CH3-imidazol-1-yl 972 2,5-12,4-CH3-imidazol-1-yl 973 2-Br, 5-CH 2 CH 3 -imidazol-1-yl 974 2-Br, 4 -CH 2 CH 3 -imidazol-1-yl 975 2 - CH (CH ₃₎ 2.4 - CH2CH3 - imidazol-1-yl 976 4-CH 2 CH 3, 5-Br-imidazol-1-yl 977 4-Br, 5-CH 2 CH 3 -imidazol-1-yl 978 4-1,5-CH 2 CH 3 -imidazol-1-yl 979 4-CH 2 CH 3,5-1-imidazol-1-yl 980 4-F, 5-CH 2 CH 3 -imidazol-1-yl 981 4-CH 2 CH 3, 5-F-imidazol-1-yl 982 2,5 -12,4 -CH 2 CH 3 -imidazol-1-yl 983 2-NO2,4-CH3-imidazol-1-yl 984 2-NO2,4 -CH2CH3-imidazol-1-yl 985 2-NO2,4 -CH (CH3) 2-imidazol-1-yl 986 2-NC &lt; 2,4 &gt; C (CH3) 3-imidazol-1-yl 987 2-NO2, 4-F-imidazol-1-yl 988 2-NO2, 4-Cl-imidazol-1-yl 989 2-NO2, 4-Br-imidazol-1-yl 990 2-NC-2,4-1-imidazol-1-yl

• 4 ·· ···· «· φ · 9 9 999

9 9 9 9 9 999 99

9

9999 9999 ···

Nr. OF 991 4-NO 2, 2-CH 3 -imidazol-1-yl 992 4-NO2,2 -CH2CH3-Imidazol-1-yl 993 4-NO2,2-F-imidazol-1-yl 994 4-NO 2, 2-Cl-imidazol-1-yl 995 4-NO 2, 2-Br-imidazol-1-yl 996 4-NO2,2-l-imidazol-1-yl 997 4-NO2,2 -CF3-imidazol-1-yl 998 4-NO2,2 -OCH3-imidazol-1-yl 999 4-NO2,5 -CH3-imidazol-1-yl 1000 4 - N0 ₂ .5 - CH2CH3 - imidazol-1-yl 1001 4-NO 2, 5-F-imidazol-1-yl 1002 4-NO 2/5-Cl-imidazol-1-yl 1003 4-NO 2, 5-Br-imidazol-1-yl 1004 4-NO2,5-1-imidazol-1-yl 1005 4-NO 2, 5-CF 3 -imidazol-1-yl 1006 4-NO2,5-OCH3-imidazol-1-yl 1007 5-NO2,4-CH3-imidazol-1-yl 1008 5-NO _2,4 - CH ₂ CH 3 - imidazol-1-yl 1009 5-NO ₂ , 4-CH (CH ₃ ) 2 -imidazol-1-yl 1010 5-NO 2, 4-C (CH 3) 3 -imidazol-1-yl 1011 5-NO2, 4-F-imidazol-1-yl 1012 5-NO2, 4-Cl-imidazol-1-yl 1013 5-NO2,4-Br-imidazol-1-yl 1014 5-NO2,4 -1-imidazol-1-yl 1015 5-η 2 -4-C 6 H 5 -imidazol-1-yl 1016 5-NO2,4 -CF3-imidazol-1-yl 1017 5 -NO ₂ . 4-OCH ₃ -imidazol-1-yl 1018 4-C 6 H 5,2 -CH 3 -imidazol-1-yl 1019 4-C8H5, 2-CH2CH3-imidazol-1-yl 1020 4-C 8 H 8, 2 -CF 3 -imidazol-1-yl 1021 4 -C 6 H 5,2 -CN- imidazol-1-yl 1022 4-C 6 H 5, 5-CH 3 -imidazol-1-yl

Nr. OF 1023 4-C6H5, 5-F-imidazol-1-yl 1024 4-C8H5,5-Cl-imidazol-1-yl 1025 4-C 6 H 5, 5-Br-imidazol-1-yl 1026 4 -C 6 H 5, 5-1-imidazol-1-yl 1027 4-C 6 H 5, 5-CF 3 -imidazol-1-yl 1028 4-C 6 H 5, 5-OCH 3 -imidazol-1-yl 1029 4-OCH 3,5 -CH 3 -imidazol-1-yl 1030 4-OCH 3, 5-CH 2 CH 3 -imidazol-1-yl 1031 5-OCH 3,4 -CH 3 -imidazol-1-yl 1032 5-OCH 3, 4-CH 2 CH 3 -imidazol-1-yl 1033 5 - OCH3,4 - CH _(CH3) 2 - imidazol-1-yl 1034 5-OCH 3, 4 -C (CH ₃ ) 3 -imidazol-1-yl 1035 2 -CN, 4-CH 3 -imidazol-1-yl 1036 2-CN, 4 -CH 2 CH 3 -imidazol-1-yl 1037 2-CN, 4-CH (CH 3) 2 * imidazol-1-yl 1038 2-CN, 4-C (CH 3) 3 -imidazol-1-yl 1039 2-CN, 4-F-imidazol-1-yl 1040 2 -CN, 4-Cl-imidazol-1-yl 1041 2-CN, 4-Br-imidazol-1-yl 1042 2-CN, 4-1-Imidazol-1-yl 1043 4-CN, 2-CH 3 -imidazol-1-yl 1044 4-CN, 2-CH 2 CH 3 -imidazol-1-yl 1045 4 -CN, 5-CH ₃ -imidazol-1-yl 1046 4 -CN, 5 -CH 2 CH 3 -imidazol-1-yl 1047 5 -CN, 4-CH 3 -imidazol-1-yl 1048 5-CN, 4-CH ₂ CH ₃ -imidazol-1-yl 1049 5 -CN, 4-CH (CH ₃ ) 2 -imidazol-1-yl 1050 5-CN, 4-C (CH 3) 3 -imidazol-1-yl 1051 4- (2'-CH ₃ -C ₆ H ₄ ) -imidazol-1-yl 1052 4- (3'-CH 3 -C 6 H 4) -imidazol-1-yl 1053 4- (4'-CH ₃ -C ₆ H ₄ ) -imidazol-1-yl 1054 4- [2 ', 3' - (CH 3) _{2 C 8} H ₃ ] imidazol-1-yl

9 · 99 · 9

9 99 ··· · · · 9

9 9 99 99 9 9 99

9 9 9 9 9 9 9 9 999 9 9

9 9 9 9 9

9 * 9 * 9

- 3 65

Nr. OF 1055 4- [2 ', 4' - (CH 3) 2 * C 6 H 3] -imidazol-1-yl 1056 4- [2 ', 5' - (CH 3) ₂ -C ₆ H ₃ J -imidazol-1-yl 1057 4- [2 ', 6' - (CH ₃ ) 2 -C ₆ H ₃ ] -imidazol-1-yl 1058 4- [3 ', 4' - (CH 3) 2 -C 6 H 3] -imidazol-1-yl 1059 4- [3 ', 5' - (CH ₃ ) ₂ -C ₆ H 3] imidazol-1-yl 1060 4- (2'-FC ₆ H ₄ ) -imidazol-1-yl 1061 4- (3'-F-C 6 H 4) -imidazol-1-yl 1062 4- (4'-F-C 6 H 4) -imidazol-1-yl 1063 4- (2 ', 3'-F ₂ -C ₆ H ₃ ) -imidazol-1-yl 1064 4- (2 ', 4'-F 2 -C 6 H 3) -imidazol-1-yl 1065 4- (2 ', 5'-F ₂ -C ₆ H ₃ ) -imidazol-1-yl 1066 4- (2 ', 6'-F 2 -C 6 H 3) -imidazol-1-yl 1067 4- (3 ', 4'-F 2 -C 6 H 3) -imidazol-1-yl 1068 4- (3 ', 5'-F 2 -C 6 H 3) -imidazol-1-yl 1069 4- (2'-Cl-C6H4) -imidazol-1-yl 1070 4- (3'-Cl-C6H4) -imidazol-1-yl 1071 4- (4'-Cl-C 8 H 4) -imidazol-1-yl 1072 4- (2 ', 3'-C ₁₂ -C ₆ H ₃ ) -imidazol-1-yl 1073 4- (2 ', 4'-C 12 -C 6 H 3) -imidazol-1-yl 1074 4- (2 ', 5'-C 12 -C 6 H 3) -imidazol-1-yl 1075 4- (2 ', 6'-C 12 -C 15 H 3) -imidazol-1-yl 1076 4- (3 ', 4'-C 12 -C 6 H 3) -imidazol-1-yl | 1077 4- (3 ', 5'-C 12 -C 6 H 3) -imidazol-1-yl | 1078 4- (2'-Br-C 8 H 4) -imidazol-1-yl I 1079 4- (3'-Br-C 6 H 4) -imidazol-1-yl I 1080 4- (4 ' -Br-C6gyl) -imidazol-1-yl 1081 4- (2 ', 3'-Br2-C8H3) -imidazol-1-yl 1082 4- (2 ', 4'-Br 2 -C 6 H 3) -imidazol-1-yl 1083 4- (2 ', 5'-Br 2 -C 8 H 3) -imidazol-1-yl 1084 4- (2 ', 6'-Br ₂ -C 6 H 3) -imidazol-1-yl 1085 4- (3 ', 4'-Br ₂ -C ₆ H 3) -imidazol-1-yl 1086 4- (3 ', 5'-Br 2 -C 6 H 3) -imidazol-1-yl

·· • ·· ·· ·· ·· • • ·· • · • • · • • • • • • • ··· • · ·· • • • • · • • · • ··· • • • • • • • • · • • · ·· ··· ·· * · ·· ··

- 366-

Nr. OF 1087 4- (2'-CF ₃ -C ₆ H 4) -imidazol-1-yl 1088 4- (3'-CF ₃ -C ₈ H ₄ ) -imidazol-1-yl 1089 4- (4'-CF ₃ -C ₈ H ₄ ) -imidazol-1-yl 1090 4- [2 ', 3' - (CF ₃ ) 2 * _{C 6} H ₃ ] -imidazol-1-yl 1091 4- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -imidazol-1-yl 1092 4- [2 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -imidazol-1-yl 1093 4- [2 ', 6' - (CF ₃ ) ₂ -C ₆ H ₃ ) -imidazol-1-yl 1094 4- (3 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ) -imidazol-1-yl 1095 4- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ) -imidazol-1-yl 1096 4- (2'-OCH ₃ -C ₆ H ₄ ) -imidazol-1-yl 1097 4- (3'-OCH ₃ -C ₈ H ₄ ) -imidazol-1-yl 1098 4- (4'-OCH ₃ -C ₆ H ₄ ) -imidazol-1-yl 1099 4- [2 ', 3' - (OCH ₃ ) 2 -C ₆ H ₃ -imidazol-1-yl 1100 4- [2 ', 4' - (OCH ₃ ) 2 * C ₆ H ₃ -imidazol-1-yl 1101 4- [2 ', 5' - (OCH ₃ ) 2 -C ₆ H ₃ -imidazol-1-yl 1102 4- [2 ', 6' - (OCH ₃ ) 2 -C 6 H ₃ -imidazol-1-yl 1103 4- [3 ', 4' - (OCH ₃ ) 2 -C ₆ H ₃ -imidazol-1-yl 1104 4- [3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ -imidazol-1-yl 1105 4- (2'-NO ₂ -C ₆ H ₄ ) -imidazol-1-yl 1106 4- (3'-NO ₂ -C ₆ H ₄ ) -imidazol-1-yl 1107 4- (4'-NO 2 -C 8 H ₄ ) -imidazol-1-yl 1108 4- (2'-CN-C ₆ H ₄₎ -imidazol-l-yl 1109 4- (3'-CN-C ₆ H ₄₎ -imidazol-l-yl 1110 4- (4'CN-C ₈ H ₄ ) -imidazol-1-yl 1111 Benzimidazol-1-yl 1112 2-F-Benzimidazol-1-yl 1113 4-F-Benzimidazol-1-yl 1114 5-F-Benzimidazol-1-yl 1115 6-F-Benzimidazol-1-yl 1116 7-F-Benzimidazol-1-yl 1117 _{2,4-F2-benzimidazol-1-yl} 1118 2,5-F ₂ -Benzimidazol-1-yl

Nr. OF 1119 _{2,6-F2-benzimidazol-1-yl} 1120 2,7- F _{2-benzimidazol-1-yl} 1121 4,5-F ₂ -Benzimidazol-1-yl 1122 _{4,6-F2-benzimidazol-1-yl} 1123 _{4,7-F2-benzimidazol-1-yl} 1124 _{5,6-F2-benzimidazol-1-yl} 1125 _{5,7-F2-benzimidazol-1-yl} 1126 _{6,7-F2-benzimidazol-1-yl} 1127 2-Cl-Benzimidazol-1-yl 1128 4-Cl-Benzimidazol-1-yl 1129 5-Cl-Benzimidazol-1-yl 1130 6-Cl-Benzimidazol-1-yl 1131 7-Cl-Benzimidazol-1-yl 1132 2,4-Cl 2 -Benzoimidazol-1-yl 1133 2,5-Cl 2 -Benzoimidazol-1-yl 1134 2,6-Cl ₂ -Benzimidazol-1-yl 1135 2,7-Cl ₂ -Benzimidazol-1-yl 1136 4,5-Cl 2 -Benzoimidazol-1-yl 1137 4,6-Cl 2 -Benzoimidazol-1-yl 1138 4,7-Cl 2 -benzimidazol-1-yl 1139 5,6-Cl 2 -Benzoimidazol-1-yl 1140 5,7-C12-Benzimidazol-1-yl 1141 6,7-Cl ₂ -Benzimidazol-1-yl 1142 2-Br-Benzoimidazol-1-yl 1143 4-Br-Benzoimidazol-1-yl 1144 5-Br-Benzimidazol-1-yl 1145 6-Br-Benzoimidazol-1-yl 1146 7-Br-Benzimidazol-1-yl 1147 2,4-Br ₂ -Benzimidazol-1-yl 1148 2,5-Br ₂ -Benzimidazol-1-yl 1149 2,6-Br ₂ -Benzimidazol-1-yl 1150 2,7-Br ₂ -Benzimidazol-1-yl

- 368

Nr. OF 1151 · 4,5-Br 2 * Benzimidazol-1-yl 1152 4,6-Br 2 -Benzoimidazol-1-yl 1153 4,7-Br 2 -Benzimidazol-1-yl 1154 5,6-Br 2 * Benzimidazol-1-yl 1155 5,7-Br 2 -Benzoimidazol-1-yl 1156 6,7-Br 2 -Benzoimidazol-1-yl 1157 2-I-Benzimidazol-1-yl 1158 4-I-Benzimidazol-1-yl 1159 5-1-Benzimidazol-1-yl 1160 6-1-Benzimidazol-1-yl 1161 7-1-Benzimidazol-1-yl 1162 2-CH 3 -Benzimidazol-1-yl 1163 4-CH 3 -Benzimidazol-1-yl 1164 5-CH 3 -Benzimidazol-1-yl 1165 6-CH 3 -Benzimidazol-1-yl 1166 7-CH 3 -Benzimidazol-1-yl 1167 2,4- (CH 3) 2-Benzimidazol-1-yl 1168 2,5- (CH 3) 2-Benzimidazol-1-yl 1169 2,6- (CH 3) 2-Benzimidazol-1-yl 1170 2,7- (CH 3) 2-Benzimidazol-1-yl 1171 4,5- (CH 3) 2-Benzimidazol-1-yl 1172 4,6- (CH 3) 2-Benzimidazol-1-yl 1173 4,7- (CH 3) 2-Benzimidazol-1-yl 1174 5,6- (CH 3) 2-Benzimidazol-1-yl 1175 5,7- (CH 3) 2-Benzimidazol * 1-yl 1176 6,7- (CH 3) 2-Benzimidazol-1-yl 1177 2-NO 2 -Benzimidazol-1-yl 1178 4-NO 2 -Benzimidazol-1-yl 1179 5-NO 2 - Benzimidazol-1-yl 1180 6-NO 2 -Benzimidazol-1-yl 1181 7-NO 2 -Benzimidazol-1-yl 1182 2,4- (NO 2) 2-Benzimidazol-1-yl

- 369-

Nr. OF 1183 2,5- (NO2) 2'-Benzimidazol-1-yl 1184 2,6- (NO 2) 2'-Benzimidazol-1-yl 1185 2,7- (NO2) 2'-Benzimidazol-1-yl 1186 4,5- (NO2) 2'-Benzimidazol-1-yl 1187 4,6- (NO2) 2'-Benzimidazol-1-yl 1188 4,7- (NO2) 2'-Benzimidazol-1-yl 1189 5,6- (NO2) 2'-Benzimidazol-1-yl 1190 5,7- (NO2) 2'-Benzimidazol-1-yl 1191 6,7- (NO2) 2'-Benzimidazol-1-yl 1192 2 -CN-Benzimidazol-1-yl 1193 4-CN-Benzimidazol-1-yl | 1194 5-CN-Benzimidazol-1-yl 1195 6 -CN-Benzimidazol-1-yl 1196 7 -CN-Benzimidazol-1-yl 1197 2 -CF 3 -Benzimidazol-1-yl 1198 4-CF 3 -Benzimidazol-1-yl 1199 5-CF 3 -Benzoimidazol-1-yl 1200 6-CF 3 -Benzimidazol-1-yl 1201 7 -CF 3 -Benzoimidazol-1-yl 1202 2-OCH 3 - Benzimidazol-1-yl 1203 4-OCH 3 -Benzimidazol-1-yl 1204 5-OCH 3 - Benzimidazol-1-yl 1205 6-OCH 3 - Benzimidazol-1-yl 1206 7-OCH 3 - Benzimidazol-1-yl 1207 4,7- (OCH 2 CH 3) 2-Benzimidazol-1-yl 1208 4-Cl, 6-CF 3 -Benzimidazol-1-yl 1209 4-Br, 6-CF 3 -Benzoimidazol-1-yl 1210 5-F, 6-Cl-benzoimidazol-1-yl 1211 1,2,4-Triazol-1-yl 1212 3-CN-1,2,4-Triazol-1-yl 1213 5-CN-1,2,4-Triazol-1-yl 1214 3-NO 2 -1,2,4-Triazol-1-yl

- 59-0 -

Nr. OF 1215 5-NO ₂ -1,2,4-Triazol-1-yl 1216 3-F-1,2,4-Triazol-1-yl 1217 5-F-1,2,4-Triazol-1-yl; 1218 3,5-F ₂ -1,2,4-Triazol-1-yl 1219 3-Cl-1,2,4-Triazol-1-yl 1220 5-Cl-1,2,4-Triazol-1-yl 1221 3,5-Cl ₂ -1,2,4-Triazol-1-yl 1222 3-Br-1,2,4-Triazol-1-yl 1223 5-Br-1,2,4-Triazol-1-yl; 1224 3,5-Br ₂ -1,2,4-Triazol-1-yl 1225 3-1-1,2,4-Triazol-1-yl 1226 5-1-1,2,4-Triazol-1-yl 1227 3,5-1 ₂ H -1,2,4-triazol-1-yl 1228 3 -CH 3 -1,2,4-Triazol-1-yl 1229 5-CH 3 -1,2,4-Triazol -1-yl 1230 3,5- _(CH3) 2 * 1 »2,4-triazol-1-yl 1231 3-CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1232 5-CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1233 3,5- (CH ₂ CH 3) ₂ -1,2,4-Triazol-1-yl 1234 3-CH ₂ CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1235 5-CH ₂ CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1236 3,5- (CH ₂ CH ₂ CH ₃ ) ₂ -1,2,4-Triazol -1-yl 1237 3-CH (CH ₃ ) 2-1,2,4-Triazol-1-yl 1238 5-CH _(CH3) 2-I, 2,4-triazol-1-yl 1239 3.5 - (CH _{(CH3) 2]} 2 -1,2,4- triazol-1-yl 1240 3-C (CH ₃ ) ₃ -1,2,4-Triazol-1-yl 1241 5-C (CH ₃ ) ₃ -1,2,4-Triazol-1-yl 1242 3,5 - [C (CH ₃ ) 3] 2-1,2,4-Triazol-1-yl 1243 3-CF 3 -1,2,4-Triazol-1-yl 1244 5-CF 3 - 1,2,4-Triazol-1-yl 1245 3,5- (CF 3) 2 * 1,2,4-Triazol-1-yl 1246 3-OCH 3 -1,2,4-Triazol-1-yl

- 3ΤΪ-

Nr. OF 1247 5-OCH 3 -1,2,4-Triazol-1-yl 1248 3,5- _(OCH3) 2-1,2,4-triazol-1-yl 1249 3-C 8 H 8 -1,2,4-Triazol-1-yl 1250 5-C 6 H 5 -1,2,4-Triazol-1-yl 1251 3,5- (C ₆ H ₅ ) 2-1,2,4-Triazol-1-yl 1252 3-OCH 2 CH 3 -1,2,4-Triazol-1-yl 1253 5-OCH 2 CH 3 -1,2,4-Triazol-1-yl 1254 3-OCH (CH ₃ ) ₂ -1,2,4-Triazol-1-yl 1255 5-OCH (CH ₃ ) 2 -1,2,4-Triazol-1-yl 1256 3-OC ₆ H ₅ -1,2,4-Triazol-1-yl 1257 5 -OC 6 H 5 -1,2,4-Triazol-1-yl 1258 3-OCH ₂ C ₆ H ₅ -1,2,4-Triazol -1-yl 1259 5-OCH ₂ C ₆ H ₅ -1,2,4-Triazol -1-yl 1 1260 3-COCH 3 -1,2,4-Triazol-1-yl 1 1261 5-COCH 3 -1,2,4-Triazol-1-yl 1262 3 -C (CH ₃ ) = NOCH ₃ -1,2,4-Triazol-1-yl 1263 5-C (CH ₃ ) = NOCH ₃ -1,2,4-Triazol-1-yl 1264 3 -C (CH ₃ ) = NOCH ₂ CH ₃ -1,2,4-Triazol -1-yl 1265 5-C (CH ₃ ) = NOCH ₂ CH ₃ -1,2,4-Triazol -1-yl 1266 3 -C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -1,2,4-Triazol -1-yl 1267 5-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1268 3 -C (CH ₃ ) = NOCH (CH ₃ ) 2-1,2,4 -Triazol -1-yl 1269 5 -C (CH ₃ ) = NOCH (CH ₃ ) ₂ -1,2,4-Triazol -1-yl 1270 3-CO ₂ CH ₃ -1,2,4-Triazol-1-yl 1271 5-CO ₂ CH ₃ -1,2,4-Triazol-1-yl 1272 3-CO ₂ -CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1273 5-CO ₂ -CH ₂ CH ₃ -1,2,4-Triazol -1-yl 1274 3-CO ₂ -CH ₂ CH ₂ CH ₃ -1,2,4-Triazol -1-yl 1275 5-CO ₂ -CH ₂ CH ₂ CH ₃ -1,2,4-Triazol -1-yl 1276 3-CO ₂ -CH (CH ₃ ) 2-1,2,4-Triazol-1-yl 1277 5-CO ₂ -CH (CH ₃ ) ₂ -1,2,4-Triazol-1-yl 1278 3 -SCH ₃ -1,2,4-Triazol-1-yl

Nr. of . 1279 5-SCH 3 -1,2,4-Triazol-1-yl 1280 3-SO 2 CH 3 -1,2,4-Triazol-1-yl 1281 5-SO ₂ CH ₃ -1,2,4-Triazol-1-yl 1282 3-Cl, 5-CH 3 -1,2,4-Triazol-1-yl 1283 _3-CH3, 5-Cl-1,2,4-triazol-1-yl 1284 3-Cl, 5-Br-1,2,4-Triazol-1-yl 1285 3-Br, 5-Cl-1,2,4-Triazol-1-yl 1286 3 -1,5-Br-1,2,4-Triazol-1-yl 1287 3-Br, 5-I-1,2,4-Triazol-1-yl 1288 3 -1,5 -CH ₃ -1,2,4-Triazol-1-yl 1289 _3-CH3, 5 -1-1,2,4-triazol-1-yl 1290 3-Br, 5-CH 3 -1,2,4-Triazol-1-yl 1291 3-CH3,5-Br-1,2,4-Triazol-1-yl 1292 3-Br, 5-F-1,2,4-Triazol-1-yl 1293 3-F, 5-Br-1,2,4-Triazol-1-yl 1294 -Cl 3 5 -CH (CH ₃₎ 2-1,2,4-triazol -1-yl 1295 3-CH (CH ₃ ) 2,5-Cl-1,2,4-Triazol-1-yl 1296 3-CH _3, 5-CH (CH3) 2 -1,2,4-triazol-1-yl 1297 3-CH (CH ₃ ) 2,5 -CH ₃ -1,2,4-Triazol-1-yl 1298 3-1,5-Cl-1,2,4-Triazol-1-yl 1299 3-Cl, 5-1-1,2,4-Triazol-1-yl 1300 3-Br, 5-CH (CH 3) ₂ -1,2,4-Triazol-1-yl 1301 3-CH (CH ₃ ) 2,5-Br-1,2,4-Triazol-1-yl 1302 3-Cl, 5-CH 2 CH 3 -1,2,4-Triazol-1-yl 1303 3-CH ₂ CH ₃ , 5 -Cl-1,2,4-Triazol-1-yl 1304 3-Br, 5 -CH ₂ CH ₃ -1,2,4-Triazol -1-yl 1305 3 -CH2CH3,5 -Br -1,2,4-Triazol-1-yl 1306 3-1,5-CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1307 3-CH ₂ CH ₃ , 5-1-1,2,4-Triazol-1-yl 1308 3 _-CH3, -CH2CH3 5 1,2,4 - triazol - 1-yl 1309 3-CH ₂ CH 3, 5-CH ₃ -1,2,4-Triazol-1-yl 1310 3-NO 2,5-CH 3 -1,2,4-Triazol-1-yl

• ·

Nr. OF 1311 3-NO ₂ , 5 -CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1312 3-ΝΟ2,5-F-1,2,4-Triazol-1-yl 1313 3-NO 2, 5-Cl-1,2,4-Triazol-1-yl 1314 3-NO 2, 5-Br-1,2,4-Triazol-1-yl 1315 3-NO2,5-1-1,2,4-Triazol-1-yl 1316 3 - NO _2, 5 -OCH 3 H -1,2,4-triazol-1-yl 1317 3-CH ₃ , 5-NO 2 -1,2,4-Triazol-1-yl 1318 3 -CH 2 CH 3, 5 -NO ₂ -1,2,4 -Triazol -1-yl 1319 3-CH (CH ₃ ) ₂ /5-NO ₂ -1,2,4-Triazol-1-yl 1320 3-C (CH ₃ ) 3,5-NO 2 -1,2,4-Triazol-1-yl 1321 3-F, 5-NO ₂ -1,2,4-Triazol-1-yl 1322 3-Cl, 5-NO2-1,2,4-Triazol-1-yl 1323 3-Br, 5-NO ₂ -1,2,4-Triazol-1-yl 1324 3-1,5-NO ₂ -1,2,4-Triazol-1-yl 1325 3-C ₆ H _S 5-NO2-1,2,4-triazol-1-yl 1326 3-OCH 3, 5-NO ₂ -1,2,4-Triazol-1-yl 1327 3-CN, 5-CH ₃ -1,2,4-Triazol-1-yl 1328 3 -CN, 5 -CH 2 CH 3 -1,2,4 -Triazol -1-yl 1329 3-CN, 5-F-1,2,4-Triazol-1-yl 1330 3-CN, 5-Cl-1,2,4-Triazol-1-yl 1331 3-CN, 5-Br-1,2,4-Triazol-1-yl ~ 1332 3-CN, 5-1-1,2,4-Triazol-1-yl 1333 _3-CH3, 5-CN-1,2,4-triazol-1-yl 1334 3 -CH2CH3,5 -CN-1,2,4-Triazol-1-yl 1335 3-CH (CH ₃ ) 2,5 -CN-1,2,4-Triazol-1-yl 1336 3-C (CH ₃ ) 3,5-CN-1,2,4-Triazol-1-yl 1337 3-F, 5-CN-1,2,4-Triazol-1-yl 1338 3-Cl, 5-CN-1,2,4-Triazol-1-yl 1339 3-Br, 5-CN-1,2,4-Triazol-1-yl 1340 3-1,5-CN-1,2,4-Triazol-1-yl 1341 3 -C ₆ H _5, -CN, 5-1,2,4-triazol-1-yl 1342 3 -C ₆ H _5, 5-CH ₃ -1,2,4-triazol-1-yl

Nr. 2 1343 3- C ₆ H ₅ .5 -CH ₂ CH ₃ -1,2,4-Triazol-1-yl 1344 3-C6H5,5-F -1,2,4-Triazol-1-yl 1345 3-C ₆ H _s , 5-Cl -1,2,4-Triazol -1-yl 1346 3-βββ, 5 -Br-1,2,4-Triazol-1-yl 1347 3-C8H5,5-1-1,2,4-Triazol-1-yl 1348 3 -C 6 H 5, 5-CF 3 -1,2,4-Triazol-1-yl 1349 3- C ₆ H ₅ , 5 -OCH 3 -1,2,4-Triazol-1-yl 1350 3 -OCH _3, -CH ₃ 5 1,2,4-triazol-1-yl 1351 3-OCH 3,5 -CH 2 CH 3 -1,2,4-Triazol-1-yl 1352 3-OCH 3,5 -F-1,2,4-Triazol-1-yl 1353 3-OCH 3, 5-Cl-1,2,4-Triazol-1-yl 1354 3-OCH3,5-Br-1,2,4-Triazol-1-yl 1355 3-OCH3,5-1-1,2,4-Triazol-1-yl 1356 _3-CH3, 5 -OCH ₃ H -1,2,4-triazol-1-yl 1357 3-CH 3 CH 3, 5-OCH 3 -1,2,4-Triazol-1-yl 1358 3-CH (CH ₃ ) 2,5-OCH ₃ -1,2,4-Triazol-1-yl 1359 3-C (CH ₃ ) 3,5-OCH ₃ -1,2,4-Triazol-1-yl 1360 3-F, 5-OCH ₃ -1,2,4-Triazol-1-yl 1361 3-Cl, 5-OCH 3 -1,2,4-Triazol-1-yl 1362 3-Br, 5-OCH 3 -1,2,4-Triazol-1-yl 1363 3-1,5-OCH 3 -1,2,4-Triazol-1-yl 1364 3- (2'-CH ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1365 3- (3'-CH ₃ -C ₆ H ₄ ) -1,2,4-Triazol- 1,1-yl 1366 3- (4'-CH ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1367 3- [2 ', 3'- (CH ₃ ) 2 -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1368 3- [2 ', 4'- (CH ₃ ) 2 -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1369 3- [2 ', 5' - (CH 3) 2 -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1370 3- [2 ', 6' - (CH 3) 2 -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1371 3- [3 ', 4'- (CH ₃ ) 2 -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1372 3- [3 ', 5'- (CH ₃ ) 2 -C 6 H ₃ ] -1,2,4-Triazol-1-yl 1373 3- (2'-FC ₆ H ₄ ) -1,2,4-Triazol-1-yl 1374 3- (3-FC ₆ H ₄₎ -1,2,4-triazol-yl

• • •

Nr. OF 1375 3- (4'-FC ₆ H ₄ ) -1,2,4-Triazol-1-yl 1376 3- (2 ', 3' - F ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1377 3- (2 ', 4'-F 2 -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1378 3- (2 ', 5'-F 2 -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1379 3- (2 ', 6'-F ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1380 3- (3 ', 4'-F ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1381 3- (3 ', 5'-F 2 -C 6 H 3) -1,2,4-Triazol-1-yl 1382 3- (2'-C ₁ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1383 3- (3'-C ₁ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl '1384 3- (4'-Cl-C ₈ H ₄ ) -1,2,4-Triazol-1-yl 1385 3- (2 ', 3'-C ₁₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1386 3- (2 ', 4'-C ₁₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1387 3- (2 ', 5'-Cl ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1388 3- (2 ', 6'-Cl ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1389 3- (3 ', 4'-Cl ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1390 3- (3 ', 5'-Cl ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1391 3- (2'-Br-C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1392 3- (3'-Br-C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1393 3- (4'-Br-C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1394 3- (2 ', 3'-Br ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1395 3- (2 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1396 3- (2 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1397 3- (2 ', 6'-Br 2 -C 6 H ₃ ) -1,2,4-Triazol-1-yl 1398 3- (3 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1399 3- (3 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1400 3- (2'-CF ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1401 3- (3'-CF ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1402 3- (4'-CF ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1403 3- [2 ', 3' - (CF ₃ ) ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1404 3- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1405 3- [2 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1406 3- [2 ', 6' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl

· ♦ «« «« «· · · · · · · · · · · · · · · · · · · · · ·· · ·

Nr. OF 1407 3- [3 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1408 3- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1409 3- (2'-OCH ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1410 3- (3'-OCH ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1411 3- (4'-OCH ₃ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1412 3- [2 ', 3' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1413 3- (2 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -1,2,4-Triazol-1-yl 1414 3- (2 ', 5' - (OCH ₃₎ 2 -C ₆ H _3] -1,2,4-triazole-l-yl 1415 3- [2 ', _6'<OCH3) 2 -C ₆ H _3] -1,2,4-triazole-l-yl 1416 3- [3 ', 4' - (OCH ₃₎ 2 -C ₆ H _3] -1,2,4-triazole-l-yl 1417 3- [3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,4-Triazol-1-yl 1418 3- (2'-NO ₂ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1419 3- (3'-NO ₂ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1420 3- (4 H -NO ₂ -C ₆ H ₄ ) -1,2,4-Triazol-1-yl 1421 3- _{(2'-CN-C6 H4)} -1,2,4-triazol-yl 1422 3- _{(3'-CN-C6 H4)} -1,2,4-triazol-yl 1423 3- _{(4'-CN-C6 H4)} -1,2,4-triazol-yl 1424 1,3,4-Triazol-1-yl 1425 2-F-1,3,4-Triazol-1-yl 1426 2,5-F ₂ -1,3,4-Triazol-1-yl 1427 2-Cl-1,3,4-Triazol-1-yl; 1428 2,5-Cl ₂ -1,3,4-Triazol-1-yl 1429 2-Br-1,3,4-Triazol-1-yl 1430 2,5-Br ₂ -1,3,4-Triazol-1-yl 1431 2-I-1,3,4-Triazol-1-yl 1432 2,5-I ₂ -l, 3,4-triazol-1-yl 1433 2-CH ₃ -1,3,4-Triazol-1-yl 1434 2,5- (CH ₃ ) 2 ', 1,3,4-Triazol-1-yl 1435 2 -CH _3, -F 5-1,3,4-triazol-1-yl 1436 2-CH ₃ , 5-Cl-1,3,4-Triazol-1-yl 1437 2-CH ₃ , 5-Br-1,3,4-Triazol-1-yl 1438 _2-CH3, 5-1-1,3,4-triazol-1-yl

·· ·· ·· ··

- rw • · · · · · · · · · · · ·

Nr. OF 1439 2-Cl, 5-F-1,3,4-Triazol-1-yl 1440 1,2,3-Triazol-1-yl 1441 4-CH 3 -1,2,3-Triazol-1-yl 1442 4,5- (CH3) 2-1,2,3-Triazol-1-yl 1443 4-CH 2 CH 3 -1,2,3-Triazol-1-yl 1444 4,5- (CH ₂ CH ₃ ) 2 -1 / 2,3-Triazol-1-yl 1445 4-CH (CH ₃ ) 2 -1,2,3-Triazol-1-yl 1446 4-C (CH ₃ ) 3 -1,2,3-Triazol-1-yl 1447 4-C ₆ H ₅ -1,2,3-Triazol-1-yl 1448 4,5- (CeHs) 2 &apos; / 2,3-Triazol-1-yl 1449 4-F-1,2,3-Triazol-1-yl 1450 4,5-F ₂ -1,2,3-Triazol-1-yl 1451 4-Cl-1,2,3-Triazol-1-yl 1452 4,5-Cl ₂ -1,2,3-Triazol-1-yl 1453 4-Br-1,2,3-Triazol-1-yl 1454 4,5-Br ₂ -1,2,3-Triazol-1-yl 1455 4,5-1-1,2,3-Triazol-1-yl 1456 4,5-12-1,2,3-Triazol-1-yl 1457 4-CN-1,2,3-Triazol-1-yl 1458 4,5- (CN) 2-1,2,3-Triazol-1-yl 1459 4-NO ₂ -1,2,3-Triazol-1-yl 1460 4,5- (NO ₂ ) _{2 ',} 1,2,3-Triazol-1-yl 1461 4-CF 3 -1,2,3-Triazol-1-yl 1462 4,5- (CF ₃ ) 2-1,2,3-Triazol-1-yl 1463 4-OCH 3 -1,2,3-Triazol-1-yl 1464 4-OCH ₂ CH ₃ -1,2,3-Triazol-1-yl 1465 4-OCH (CH ₃ ) ₂ -1,2,3-Triazol-1-yl 1466 4-OC 5 H -1,2,3-Triazol-1-yl 1467 4-COCH 3 -1,2,3-Triazol-1-yl 1468 4 -C (CH ₃ ) = NOCH ₃ -1,2,3-Triazol-1-yl 1469 4-C (CH ₃ ) = NOCH ₂ CH ₃ -1,2,3-Triazol -1-yl 1470 4-C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -1,2,3-Triazol -1-yl

-

Nr. OF 1471 4-C _(CH3) = NOCH _(CH3) 2 * r 1 2,3-triazol - 1-yl 1472 4-CO ₂ CH ₃ -1,2,3-Triazol-1-yl 1473 4,5- (CO ₂ CH ₃ ) ₂ -1,2,3-Triazol-1-yl 1474 4-CO ₂ CH ₂ CH ₃ -1,2,3-Triazol-1-yl 1475 4,5- (CO ₂ CH ₂ CH ₃ ) 2-1,2,3-Triazol-1-yl 1476 4-CO ₂ CH ₂ CH ₂ CH ₃ -1,2,3-Triazol -1-yl 1477 4,5 - (CO 2 CH 2 CH 2 CH 3) 2 * 1 »2,3 -Triazol -1-y 1 1478 4-CO ₂ CH (CH ₃ ) 2-1,2,3-Triazol-1-yl 1479 4,5- [CO ₂ CH (CH ₃ ) ₂ ] 2-1 / ² '3-Triazol-1-yl 1480 4-CH ₃ -1,2,3-Triazol-1-yl 1481 4-SO 2 CH 3 -1,2,3-Triazol-1-yl 1482 4- (2'-CH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1483 4- (3'-CH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1484 4- (4'-CH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1485 4- [2 ', 3' - (CH 3) 2 -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1486 4- [2 ', 4' - (CH 3) 2 -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1487 4- [2 ', 5' - (CH 3) 2 -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1488 4- [2 ', 6' - (CH ₃ ) 2 -C ₆ H 3] -1,2,3-Triazol-1-yl 1489 4- [3 ', 4' - (CH 3) 2 -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1490 4- [3 ', 5' - (CH 3) 2 -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1491 4- (2'-FC ₆ H ₄ ) -1,2,3-Triazol-1-yl 1492 4- (3'-FC ₆ H ₄₎ -1,2,3-triazol-yl 1493 4- (4'-FC ₆ H ₄ ) -1,2,3-Triazol-1-yl 1494 4- (2 ', 3'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1495 4- (2 ', 4'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1496 4- (2 ', 5'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1497 4- (2 ', 6'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1498 4- (3 ', 4'-F ₂ -C ₈ H ₃ ) -1,2,3-Triazol-1-yl 1499 4- (3 ', 5'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1500 4- (2'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1501 4- (3'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1502 4- (4'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-1-yl

♦ ·

-ago -

Nr. OF 1503. 4- (2 ', 3'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1504 4- (2 ', 4'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1505 4- (2 ', 5'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1506 4- (2 ', 6'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1507 4- (3 ', 4'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1508 4- (3 ', 5' -C 1 -C ₂ -C ₆ H ₃₎ -1,2,3-triazol-yl 1509 4- (2'-Br- _C6 H4) -1,2,3-Triazol-1-yl 1510 4- (3'-Br- _C6 H4) -1,2,3-Triazol-1-yl 1511 4- _(4'-Br-C6 H4) -1,2,3-triazol-yl 1512 4- (2 ', 3'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1513 4- (2 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1514 4- (2 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1515 4- (3 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1516 4- (3 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1517 4- (2'-CF ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1518 4- (3'-CF ₃ -C ₈ H 4) -1,2,3-Triazol-1-yl 1519 4- (4'-CF ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1520 4- [2 ', 3' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1521 4- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ J -1,2,3-Triazol-1-yl 1522 4- (2 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1523 4- (2 ', 6' - (CF ₃ ) 2 -C ₆ H ₃ J -1,2,3-Triazol-1-yl) 1524 4- [3 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1525 4- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1526 4- (2'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1527 4- (3'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1528 4- (4'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1529 4- (2 ', 3' - (OCH ₃ ) ₂ -C ₆ H ₃ J -1,2,3-Triazol-1-yl) 1530 4- [2 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1531 4- [2 ', 5' - (OCH ₃ ) 2-C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1532 4- [2 ', 6' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl 1533 4- [3 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-1-yl 1534 4- [3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-1-yl

• 9 9 9 9 9 9 9 9 9 9 9

999 99 99 99 99

Nr. OF 1535 4- (2'-NO ₂ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1536 4- (3'-NO ₂ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1537 4- (4'-NO ₂ -C ₆ H ₄ ) -1,2,3-Triazol-1-yl 1538 4- _{(2'-CN-C6 H4)} -1,2,3-triazol-1-yl 1539 4- _{(3'-CN-C6 H4)} -1,2,3-triazol-yl 1540 4- _{(4'-CN-C6 H4)} -1,2,3-triazol-yl 1541 1,2,3-Triazol-2-yl 1542 4-CH ₃ -1,2,3-Triazol-2-yl 1543 4,5- (CH ₃ ) 2 -1,2,3-Triazol-2-yl 1544 4-CH ₂ CH ₃ -1,2,3-Triazol-2-yl 1545 4,5- (CH ₂ CH ₃ ) ₂ -1,2,3 -Triazol -2-yl 1546 4-CH _(CH3) 2-1,2,3-triazol-2-yl 1547 4-C (CH 3) 3 -1,2,3-Triazol-2-yl 1548 4-C ₆ H ₅ -1,2,3-Triazol-2-yl 1549 4,5- (C ₆ H ₅ ) j -1,2,3-Triazol-2-yl 1550 4-F-1,2,3-Triazol-2-yl; 1551 4,5-F ₂ -1,2,3-Triazol-2-yl 1552 4-Cl-1,2,3-Triazol-2-yl 1553 4,5-Cl ₂ -1,2,3-Triazol-2-yl 1554 4-Br-1,2,3-Triazol-2-yl; 1555 4,5-Br ₂ -1,2,3-Triazol-2-yl 1556 4-1-1,2,3-Triazol-2-yl 1557 4,5-I _{2-1,2,3-triazol-2-yl} 1558 4-CN-1,2,3-Triazol-2-yl 1559 4,5- (CN) 2-1,2,3-Triazol-2-yl 1560 4-NO ₂ -1,2,3-Triazol-2-yl 1561 4,5- (NO) 2-1,2,3-Triazol-2-yl 1562 4-CF 3 -1,2,3-Triazol-2-yl 1563 4,5- (CF ₃ ) 2-1,2,3-Triazol-2-yl 1564 4-OCH 3 -1,2,3-Triazol-2-yl 1565 4-OCH 2 CH 3 -1,2,3-Triazol-2-yl 1566 4-OCH (CH ₃ ) ₂ -1,2,3-Triazol-2-yl

• 3 Oh 3 3 3 Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh Oh · ♦ · ♦ ··

Nr. OF 1567. 4-OC 6 H 5 -1,2,3-Triazol-2-yl 1568 4-COCH 3 -1,2,3-Triazol-2-yl 1569 4 -C (CH ₃ ) = NOCH ₃ -1,2,3-Triazol-2-yl 1570 4 -C (CH ₃ ) = NOCH ₂ CH ₃ -1,2,3-Triazol-2-yl 1571 4 -C (CH ₃ ) = NOCH ₂ CH ₂ CH ₃ -1,2,3-Triazol-2-yl 1572 4-C (CH ₃ ) = NOCH (CH ₃ ) ₂ -1,2,3-Triazol-2-yl 1573 4-CO 2 CH 3 -1,2,3-Triazol-2-yl 1574 4,5- (CO 2 CH 3) 2-1,2,3-Triazol-2-yl 1575 4-CO 2 CH 2 CH 3 -1,2,3-Triazol-2-yl 1576 4,5- (CO 2 CH 2 CH 3) 2 -1,2,3-Triazol-2-yl 1577 4-CO ₂ CH ₂ CH ₂ CH ₃ -1,2,3-Triazol -2-yl 1578 4,5- (CO 2 CH 2 CH 2 CH 3) 2-1,2,3-Triazol-2-yl 1579 4-CO ₂ CH (CH ₃ ) 2-1,2,3-Triazol-2-yl 1580 4,5- [CO ₂ CH (CH ₃ ) ₂ ] 2 -1,2,3-Triazol-2-yl 1581 4 -SCH 3 -1,2,3-Triazol-2-yl 1582 4 -SO 2 CH 3 -1,2,3-Triazol-2-yl 1583 4- (2'-CH 3 -C 6 H 4) -1,2,3-Triazol-2-yl 1584 4- (3'-CH 3 -C 6 H 4) -1,2,3-Triazol-2-yl 1585 4- (4'-CH 3 -C 6 H 4) -1,2,3-Triazol-2-yl 1586 4- [2 ', 3' - _{(CH3) 2} -C H _{3 e]} -l, 2,3-triazol-2-yl 1587 4- [2 ', 4' - (CH ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1588 4- [2 ', 5' - (CH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1589 4- [2 ', 6' - (CH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1590 4- [3 ', 4' - (CH ₃ ) ₂ -C ₆ H ₃ J -1,2,3-Triazol-2-yl 1591 4- [3 ', 5' - (CH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1592 4- (2'-FC ₆ H ₄ ) -1,2,3-Triazol-2-yl 1593 4- (3'-FC ₆ H ₄₎ -1,2,3-triazol-2-yl 1594 4- (4'-FC ₆ H ₄ ) -1,2,3-Triazol-2-yl 1595 4- (2 ', 3'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1596 4- (2 ', 4'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1597 4- (2 ', 5'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1598 4- (2 ', 6'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl

Φ · · · φ φ φ φ φ · · · · · · · · · · · · · · ΦΦΦ ΦΦΦ ΦΦΦ ΦΦΦ ΦΦΦ ΦΦΦ · - ·· ·

Nr. OF 1599 4- (3 ', 4'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1600 4- (3 ', 5'-F ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1601 4- (2'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1602 4- (3'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1603 4- (4'-C 1 -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1604 4- (2 ', 3'-Cl ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1605 4- (2 ', 4'-Cl ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1606 4- (2 ', 5'-Cl ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1607 4- (2 ', 6'-Cl ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1608 4- (3 ', 4'-C ₁₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1609 4- (3 ', 5'-Cl ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1610 4- (2'-Br-C ₈ H ₄ ) -1,2,3-Triazol-2-yl 1611 4- _{(3'-Br-C6 H4)} -1,2,3-triazol-2-yl 1612 4- _{(4'-Br-C6 H4)} -1,2,3-triazol-2-yl 1613 4- (2 ', 3'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1614 4- (2 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1615 4- (2 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1616 4- (2 ', 6'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1617 4- (3 ', 4'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1618 4- (3 ', 5'-Br ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1619 4- (2'-CF ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1620 4- (3'-CF ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1621 4- (4'-CF ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1622 4- [2 ', 3' - (CF ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1623 4- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1624 4- [2 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1625 4- [2 ', 6' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1626 4- [3 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1627 4- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1628 4- (2'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1629 4- (3'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1630 4- (4'-OCH ₃ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl

- 3SQ

Nr. OF 1631 4- [2 ', 3' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1632 4- [2 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1633 4- [2 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ J -1,2,3-Triazol-2-yl 1634 4- (2 ', 6' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1635 4- [3 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -1,2,3-Triazol-2-yl 1636 4- {3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -1,2,3-Triazol-2-yl 1637 4- (2'-NO ₂ -C ₆ H 4) -1,2,3-Triazol-2-yl 1638 4- (3'-NO ₂ -C ₆ H ₄ ) -1,2,3-Triazol-2-yl 1639 4- (4'-NO ₂ -C ₆ H 4) -1,2,3-Triazol-2-yl 1640 4- _{(2'-CN-C6 H4)} -1,2,3-triazol-2-yl 1641 4- _(3'-CN-C6 H4) -1,2,3-triazol-2-yl 1642 4- _{(4'-CN-C6 H4)} -1,2,3-triazol-2-yl 1643 Benzotriazol-1-yl 1644 4-F-Benzotriazol-1-yl 1645 5-F-Benzotriazol-1-yl 1646 6-F-Benzotriazol-1-yl 1647 7-F-Benzotriazol-1-yl 1648 4,5-F ₂ -Benzotriazol-1-yl 1649 _{4,6-F2-benzotriazol-1-yl} 1650 4,7-F ₂ -Benzotriazol-1-yl 1651 _{5,6-F2-benzotriazol-1-yl} 1652 5,7-F ₂ -Benzotriazol-1-yl 1653 6,7-F ₂ -Benzotriazol-1-yl 1654 4-Cl-Benzotriazol-1-yl 1655 5-Cl-Benzotriazol-1-yl 1656 6-Cl-Benzotriazol-1-yl 1657 7-Cl-Benzotriazol-1-yl 1658 4,5-Cl ₂ -Benzotriazol -1-yl 1659 4,6-Cl ₂ -Benzotriazol-1-yl 1660 4,7-Cl ₂ -Benzotriazol-1-yl 1661 5,6-Cl ₂ -Benzotriazol-1-yl 1662 5,7-Cl ₂ -Benzotriazol-1-yl

- 3SS-

Nr. 2 1663 6,7-Cl 2 -Benzotriazol-1-yl 1664 4-Br-Benzotriazol-1-yl 1665 5-Br-Benzotriazol-1-yl 1666 6-Br-Benzotriazol-1-yl 1667 7-Br-Benzotriazol-1-yl 1668 4,5-Br 2 -Benzotriazol-1-yl 1669 4,6-Br 2 * Benzotriazol-1-yl 1670 4,7-Br 2 -Benzotriazol-1-yl 1671 5,6-Br 2 -Benzotriazol-1-yl 1672 5,7-Br 2 -Benzotriazol-1-yl 1673 6,7-Br 2 -Benzotriazol-1-yl 1674 4-I-Benzotriazol-1-yl 1675 5-1-Benzotriazol-1-yl 1676 6-1-Benzotriazol-1-yl 1677 7-1-Benzotriazol-1-yl 1678 4-CH 3 -Benzotriazol-1-yl 1679 5-CH 3 -Benzotriazol-1-yl 1680 6-CH 3 -Benzotriazol-1-yl 1681 7 -CH 3 -Benzotriazol-1-yl 1682 4,5- (CH 3) 2-Benzotriazol-1-yl 1683 4,6- (013) 2-Benzotriazol-1-yl 1684 4,7- (CH 3) 2-Benzotriazol-1-yl 1685 5,6- (013) 2-Benzotriazol-1-yl 1686 5,7- (013) 2-Benzotriazol-1-yl 1687 6,7- (CH 3) 2-Benzotriazol-1-yl 1688 4-NO 2 * Benzotriazol-1-yl 1689 5-NO 2 -Benzotriazol-1-yl 1690 6-NO 2 -Benzotriazol-1-yl 1691 7-NO 2 -Benzotriazol-1-yl 1692 4,5- (NO 2) 2-Benzotriazol-1-yl 1693 4,6- (NO 2) 2-Benzotriazol-1-yl 1694 4,7- (NO 2) 2-Benzotriazol-1-yl

wc -

Nr. OF 1695 5,6- (NO 2) 2 Benzotriazol-1-yl 1696 5,7- (NC2) 2 * Benzotriazol-1-yl 1697 6,7- (NO2) 2 -Benzotriazol-1-yl 1698 4-CN-Benzotriazol-1-yl 1699 5-CN-Benzotriazol-1-yl 1700 6-CN-Benzotriazol-1-yl 1701 7-CN-Benzotriazol-1-yl 1702 4-CF ₃ -Benzotriazol-1-yl 1703 5-CF ₃ -Benzotriazol-1-yl 1704 6 -CF ₃ -Benzotriazol-1-yl 1705 7-CF ₃ -Benzotriazol-1-yl 1706 4-OCH ₃ -Benzotriazol-1-yl 1707 5 -OCH ₃ - Benzotriazole-1-yl 1708 6-OCH ₃ -Benzotriazol-1-yl 1709 7-OCH ₃ -Benzotriazol-1-yl 1710 5,6- (OCH ₃ ) 2-Benzotriazol-1-yl 1711 4-CO ₂ CH ₃ -Benzotriazol-1-yl 1712 5-CO ₂ CH ₃ -Benzotriazol-1-yl 1713 6 -CO2CH ₃ - Benzotriazole-1-yl 1714 ..... 5F-6-Cl-Benzotriazol-1-yl 1715 Tetrazol-1-yl 1716 Tetrazol-2-yl 1717 5-F-Tetrazol-2-yl 1718 5-Cl-Tetrazol-2-yl 1719 5-Br-Tetrazol-2-yl 1720 5-1-Tetrazol-2-yl 1721 5 -CN-Tetrazol-2-yl 1722 5-NO2-Tetrazol-2-yl 1723 _{5-CH3-tetrazol-2-yl} 1724 5-CH ₂ CH ₃ -Tetrazol-2-yl 1725 5-CH 2 CH 2 CH 3 -Tetrazol-2-yl 1726 5 - CH _(CH3) 2-tetrazol-2 - yl

• • • • • •

387 • 9 9

9 9 9

Nr. of 1727 5 -C (CH ₃ ) ₃ -Tetrazol-2-yl 1728 _{5-CF3-tetrazol-2-yl} 1729 5-OCH 3 - Tetrazol-2-yl 1730 5-OCH 2 CH 3 -Tetrazol-2-yl 1731 5 - OCH 2 CH 2 CH 3 - Tetrazol-2-y 1 1732 5 - OCH (CH ₃₎ 2 - tetrazole - 2 -y 1 1733 5-OC 6 H 5 -Tetrazol-2-yl 1734 5-OCH2C6H5-Tetrazol-2-yl 1735 5-C6H5-Tetrazol-2-yl; 1736 5-COCH 3 -Tetrazol-2-yl 1737 5-C (CH ₃ ) = NOCH ₃ -Tetrazol-2-yl 1738 5 -C (CH ₃ ) = NOCH ₂ CH ₃ - Tetrazol-2-yl 1739 5-C (CH ₃ ) = NOCH ₂ CH ₂ CH 3 -Tetrazol-2-yl 1740 5-C (CH ₃ ) = NOCH (CH ₃ ) 2 -Tetrazol-2-yl 1741 5 - CO2CH3 - Tetrazol - 2 - y 1 1742 5 -CO 2 CH 2 CH 3 - Tetrazol-2-yl 1743 5-CO 2 CH 2 CH 2 CH 3 - Tetrazol-2-yl 1744 5-CO ₂ CH (CH ₃ ) 2 -Tetrazol-2-yl 1745 5 -SCH 3 -Tetrazol-2-yl 1746 5-SO 2 CH 3 -Tetrazol-2-yl 1747 5- (2'-CH ₃ -C ₆ H ₄ ) -Tetrazol-2-yl 1748 5- (3'-CH ₃ -C ₆ H ₄ ) -Tetrazol-2-yl 1749 5- (4'-CH ₃ -C ₈ H ₄ ) -Tetrazol-2-yl 1750 5- [2 ', 3' - (CH ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1751 5- [2 ', 4' - (CH ₃ ) 2 -C ₆ H ₃ ] -Tetrazol-2-yl 1752 5- [2 ', 5' - (CH ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1753 5- [2 ', 6'- (CH ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1754 5- [3 ', 4' - (CH ₃ ) ₂ -C ₆ H ₃ J-Tetrazol-2-yl 1755 5- [3 ', 5' - _(CH3) 2-C H _{3 e]} -tetrazol-2-yl 1756 5- (2'-F-C6K4) -Tetrazol-2-yl 1757 5- (3'-FC ₆ H ₄ ) -Tetrazol-2-yl 1758 5- (4'-F-C ₈ H ₄ ) -Tetrazol-2-yl

- 588-

II ^Nr · OF 1759 5- (2 ', 3'-F ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1760 5- (2 ', 4'-C ₂ H _{3 e)} -tetrazol-2-yl 1761 5- (2 ', 5'-F ₂ -C ₈ H ₃ ) -Tetrazol-2-yl 1762 5- (2 ', 6'-F ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1763 5- (3 ', 4'-F ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1764 5- (3 ', 5'-F ₂ -C ₆ H ₃ ) -Tetrazol-2-yl' 1765 5- (2'-C 1 -C ₆ H ₄ ) -Tetrazol-2-yl 1766 5- (3'-C 1 -C ₆ H ₄ ) -Tetrazol-2-yl 1767 5- (4'-C 1 -C 6 H ₄ ) -Tetrazol-2-yl 1768 5 - (2 ', 3' -C 1 -C ₂ -C 6 H ₃₎ tetrazol-2-yl 1769 5- (2 ', 4'-Cl ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1770 5- (2 ', 5'-Cl ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1771 5- (2 ', 6'-Cl ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1772 5- (3 ', 4'-C ₁₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1773 5- (3 * 5 &apos; -C1 ₂ -C 6 H ₃₎ tetrazol-2-yl 1774 5- (2'-Br-C ₆ H ₄₎ -tetrazol-2-yl 1775 5- (3'-Br-C ₆ H ₄₎ -tetrazol-2-yl 1776 5- (4'-Br-C ₈ H ₄ ) -Tetrazol-2-yl 1777 5- (2 ', 3'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1778 5- (2 ', 4'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1779 5- (2 ', 5'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1780 5- (2 ', 6'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1781 5- (3 ', 4'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1782 5- (3 ', 5'-Br ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1783 5- (2'-CF 3 -C 6 H 4) -Tetrazol-2-yl 1784 5- (3'-CF 3 -C 6 H 4) -Tetrazol-2-yl 1785 5- (4'-CF 3 -C 6 H 4) -Tetrazol-2-yl 1786 5- [2 ', 3' - (CF ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1787 5- [2 ', 4' - (CF ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1788 5- [2 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1789 5- [2 ', 6' - (CF ₃ ) ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1790 5- [3 ', 4' - (CF ₃ ) ₂ C 8 H ₃ ] -Tetrazol -2-yl

···························································································

-

Nr. OF 1791 5- [3 ', 5' - (CF ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1792 5- (2'-OCH ₃ -C ₆ H ₄ ) -Tetrazol-2-yl 1793 5- (3'-OCH ₃ -C ₆ H ₄ ) -Tetrazol-2-yl 1794 5- (4'-OCH ₃ -C ₆ H ₄ ) -Tetrazol-2-yl 1795 5- [2 ', 3' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1796 5- [2 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ) -Tetrazol-2-yl 1797 5- [2 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ J-Tetrazol-2-yl 1798 5 - [2 ', 6' - (OCH ₃ ) ₂ -C ₆ H ₃ J-Tetrazol-2-yl 1799 5- [3 ', 4' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1800 5- [3 ', 5' - (OCH ₃ ) ₂ -C ₆ H ₃ ] -Tetrazol-2-yl 1801 5- (2'-NO ₂ -C ₆ H ₄ ) -Tetrazol-2-yl 1802 5- (3'-NO ₂ -C ₆ H ₄ ) -Tetrazol-2-yl 1803 5- (4'-NO ₂ -C ₆ H ₄ ) -Tetrazol-2-yl 1804 5- (2'-CN-C ₆ H ₄₎ -tetrazol-2-yl 1805 5- (3'-CN-C ₆ H ₄₎ -tetrazol-2-yl 1806 5- (4'-CN-C 6 H ₄ ) -Tetrazol-2-yl 1807 1-Aziridinyl 1808 1-Diaziridinyl 1809 1-Azetidinyl 1810 1-Pyrrolidinyl 1811 2-Isoxazolidinyl 1812 2 -Isothiazolidinyl 1813 1-Pyrazolidinyl 1814 3 · Oxazolidinyl 1815 3-Thiazolidinyl 1816 1-Imidazolidinyl 1817 1,2,4-Oxadiazolidin-2-yl 1818 1,2,4-Oxadiazolidin-4-yl 1819 1,2,4-Thiadiazolidin-2-yl 1820 1,2,4-Thiadiazolidin-4-yl 1821 1-Triazolidinyl 1822 1,3,4-Oxadiazolidin-3-yl

- 3 ^ 0

1 Nr. Z | 1823 1,3,4-Thiadiazolidin-3-yl 1824 2,3-Dihydropyrrol-1-yl 1825 2,5-Dihydropyrrol-1-yl 1826 2,3-Dihydroisoxazol-2-yl 1827 2,5-Dihydroisoxazol-2-yl 1828 2,3-Dihydroisothiazol-2-yl 1829 2,5-Dihydroisothiazol-2-yl 1830 2,3-Dihydropyrazol-1-yl 1831 2,3-Dihydropyrazol-2-yl 1832 4,5-Dihydropyrazol-1-yl 1833 2,3-Dihydrooxazol-3-yl 1834 2,3-Dihydrothiazol-3-yl 1835 2,3-Dihydroimidazol-1-yl 1836 4,5-Dihydroimidazol-1-yl 1837 2,5-Dihydroimidazol-1-yl 1838 1-Piperidinyl 1839 1-Piperazinyl 1840 4-Methylpiperazin-1-yl 1841 4 -Morpholinyl 1842 2,6- (CH 3) 2-morpholin-4-yl 1843 1-Hexahydropyridazinyl 1844 1-Hexahydropyrimidinyl 1845 2,3-Dihydroindol-1-yl 1846 4-Thiomorpholinyl 1847 1,2,4-Hexahydrotriazin-1-yl 1848 2,3-Dihydroisoindol-2-yl 1849 4-Cl, 2,3-dihydroisoindol-2-yl 1850 5-Cl, 2,3-dihydroisoindol-2-yl 1851 6-Cl, 2,3-dihydroisoindol-2-yl 1852 7 -C1,2,3-dihydroisoindol-2-yl 1853 1,4-Oxazin-4-yl 1854 2,5- (CH ₃ ) 2,4 -CF 3 -imidazol-1-yl

0 0 0 0 000 0 0 000 0 0 0 0 0 0

- -

Nr. OF 1855 5-CH (CH ₃ ) 2 -imidazol-1-yl 1856 4 - CgHs 5 -CH 2 CH ₃ - imidazol-1-yl

Industry_Elive Elno s t

The compounds I are useful as active fungicides. It is characterized by excellent activity against a broad spectrum of phytopathogenic fungi and fungi, in particular, from the class of ascomycetes and basidiomycetes. In part, they have systemic efficacy and can be used as fungicides applicable to soil or foliar.

Of particular importance are these compounds for combating a variety of fungi attacking various crop plants such as wheat, rye, barley, oats, rice, corn, grasses, cotton, soybeans, coffee, cane, wine, fruit crops and ornamental plants, and vegetables as cucumbers, beans and pumpkins, and against mildew and seeds, and the seeds of these plants.

appropriate

These compounds are particularly suitable for the following plant diseases: Erysiphe pa dlí), the fish are eaten, Erythis cichoracear um fuliginea pumpkin, Podosphaera leucotricha for combating graminis (true and Sphaerotheca apples, Uncinula necator vine, various species of Puccinia on cereals, various Rhizoctonia species on cotton and grass, Ustilago species on cereals and sugar cane, Venturia inaequalis (scab) on apples, Helmithosporium species on cereals, Septoria nodorum on wheat, Botrytis c.inerea (gray mold) on strawberries and vines , Cercospora arachidicola on peanuts, Pseudocercosporella, herpotrichoides on wheat and barley, Pyricularioa oryzae on rice, Phytophtora infestans on potatoes and tomatoes, different Fusarium and Verticillium species on different plant species.

· · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · 0000 00 00

Compounds (I) are used by treating fungi or plants, soil, seed, materials or seeds to be protected from fungal attack with a sufficient amount of fungicidal active ingredients. The application of these active substances is carried out before or after the infection of the materials, plants, seeds or seeds by the fungi.

These compounds can be converted into conventional formulations such as solutions, emulsions, suspensions, powders, pastes or granules. The form of application always depends on the intended use. In any case, they must ensure a uniform and fine distribution of these compounds. The compounds are converted into the individual formalities in a manner known per se into. for example, by saturating the active ingredient with solvents and / or carriers, optionally using emulsifying and dispersing agents, and may be used in the case of water as a diluent. and other organic solvents as co-solvents. Suitable excipients are, in particular: solvents such as aromatics (e.g. xylene), chlorinated aromatics (e.g. chlorobenzols), paraffins (e.g. petroleum fractions), alcohols (e.g. methane, butanol), ketones (e.g. cyclohexanone) ), anibs (e.g. ethanolamine, dimethylformamide) and water .. carriers such as natural stoneware meal (e.g. kaolin, clay, talc, chalk) and synthetic stoneware meal (e.g., highly disperse silicic acid, silicates), emulsifying agents such as nonionic and anionic emulsifiers (for example polyoxyethylene ether of fatty alcohols, alkylsulfonates and arylsulfonates) and dispersants such as lignin-sulfite lyes and methylcellulose.

• 9

-Mi - Fu n g i c i d n i p r c In general, curves contain taken 0,1 a ž 95,

mostly. 0.5 to 90% by weight of active ingredient.

The application rate varies from 0.01 to 2.0 kg of active ingredient per hectare depending on the type of effect desired.

Generally, 0.001 to 0.1 is used for seed treatment. g, generally 0.01 to 0.05 g of active ingredient per kg of seed.

The compositions of the present invention may also be applied in conjunction with other active ingredients, for example herbicides, insecticides, growth regulators, fungicides or fertilizers.

Combined with fungicides, in many cases, the broadening of the spectrum results in fungicidal activity.

The following list of fungicides with which the compositions of the present invention can be applied merely illustrates the combination possibilities, and in no way restricts them:

Sulfur, dithiocarbamates and derivatives thereof such as zinc ferridimethyldithiocarbamate, zinc dimethyldithiocarbamate, ethylenebisdithiocarbamate rn a n g a n e th e e n bis d thio a b b a.m. α, manganese-zinc-ethylenediamine-bis-dithiocarbamate, zinc; ammoniacal complex of zinc- (N, N-ethylene-bis-dithiocarbamate), ammoniacal complex of zinc- (N, N'-propylene-bis-dithiocarbamate), zinc- (N, N'-propylene-bis-dithiocarbamate) ,

N, N'-polypropylene-bis- (thiocarbamoyl) disulfide,

-3Α5Γ nitroderivatives such as dinitro- (1-methylhepty) phenylcrotonate,

2-sec.-Butyl-4,6-dinitrophenyl-3,3-dimethyl-ethyl,

2-sec-butyl-4,6-dinitrophonyl iso-propyl carbonate,

5-nitro-iso-phthalic acid-di-i-o-propyl ester, heterocyclic substances such as

2-Heptadecyl-2-imidazoline acetate

2,4-dichloro-6- (o-chloroanilino) -s-triazine,

0, 0- di e t y 1 - f t a. 1 .i.mi dof o s f on o t i o a t,

5-amino-1- (bis- (dimethylamino) phosphinyl) -3-phenyl-1,2,4-triazole,

2,3-dicyano-1,4-dithioanthraquinone,

2-thio-1,3-dithiolo- (4,5-b) -quinoxaline,

1- (butylcarbamoyl) -2-benzimidazole-methyl ester of k and rbamino, 2-methoxyl and rbonylaminamino-m and m-1 and m-1,

2- (furyl- (2) benzimidazole, 2- (thiazolyl- (4) benzimidazole),

N- (1,1,2,2-tetrachloroethylthio) tetrahydroftalimid,

N-1 r i c h 1 m o d 11 i. O-1 e t r and hy d r o f t a 1 i m i d,

N-1 ri-chloromethyl i oft a1imi d,

N-dichlorofluoromethylthio-N ', N'-dimethyl-N-phenyl-sulfuric acid, 5-ethoxy-3-trichloromethyl-1,2,4-thiadiazole,

2-rhodanomethylthiobenzothiazole, 1,4-dichloro-2,5-dimethoxybenzole,

4- (2-chlorophenylhydrazono) -3-methyl-5-isoxazolone, pyridine-2-thio-1-oxide, 8-hydroxyquinoline, respectively. its cupric salt, 2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiin,

2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiine-4,4-dioxide,

2-Methyl-5,6-dihydro-4H-pyran-3-anilide

2-Methyl-furan-3-anilide acid

2,5-dimethyl-furan-3-anilide

2,4.5-Trimethyl-furan-3-anilide

2,5-Dimethyl-furan-3-cyclohexylamide

N-cyclohexyl-N-methoxy-2,5-dimethyl-furan-3-carboxylic acid, 2-methyl-anilide benzoic, carboxylic, carboxylic, carboxylic, carboxylic, carboxylic, 2-iodo-anilide

• · acidic acid,

N-formyl-N-morpholine-2,2,2-trichloroethyl acetyl, piperazine-1,4-diylbis- (1- (2,2,2-trichloroethyl)) formamide,

1- (3,4-dichloroanilino) -1-formylamino-2,2,2-trichloroethane,

2,6-dimethyl-N-tridecyl-morpholine resp. its salts,

2,6-dimethyl-N-cyclododecyl-morphine, respectively; its salts,

N- (3- (p-tert-butylphenyl) -2-methylpropyl) -cis-2,6-dimethylmorpholine, N- (3- (p-tert-butylphenyl) -2-methylpropyl) -piperidine,

1- (2- (2,4-dichlorophenoyl) -4-ethyl-1,3-dioxolan-2-yl-ethyl) -1H-1,

2,4-triazole,

1- (2- (2,4-dichlorophenyl) -4-n-propyl-1,3-dioxolan-2-yl-ethyl) -1H-1,2-4-triazole,

N- (n-propyl) -N- (2,4,6-trichloro-phenoxyethyl) -N'-imidazol-yl-urea,

1- (4-chlorophenoxy) -3,3-dimethyl-1- (1H-1,2,4-triazol-1-yl) -2-butanone, (2-chlorophenyl) - (4-chlorophenyl) -5 -pyrimidine-methanol,

5-Butyl-2-dimethylamino-4-hydroxy-6-methyl-pyrimidine;

Bis- (p-chlorophenyl) -3-pyrimidinedimethanol,

1,2-Bis- (3-ethoxycarbonyl-2-thioureido) benzole,

1,2-Bis-3-methoxycarbonyl-2-thiureido) benzole, (2- (4-chlorophenyl) ethyl) - (1-1-dimethylethyl) -1H-1,2,4-triazole-l-ol tanol as well as various fungicides such as dodecylguanidine acetate,

3- (3- (3,5-dimethyl-2-oxycyclohexyl) -2-hydroxyethyl) glutarimide, hexachlorobenzol,

DL-methyl-N- (2,6-dimethylphenyl) -N-furoyl (2) alaninate,

DL-N- (2,6-dimethylphenyl) -N- (2'-methoxyacetyl) alanine methyl ester N- (2,6-dimethylphenyl) -N-chloroacetyl-D, L-2-aminobutyroacetone, DL -N- (2,6-dimethylphenyl) -N- (phenylacetyl) alanine methyl ester,

5-Methyl-5-vinyl-3- (3,5-dichlorophenyl) -2,4-dioxo-1,3-oxazolidine

3- (3,5-dichlorophenyl) -5-methyl-5-methoxymethyl-1,3-oxazolidin-2,4-dione, 3- (3,5-dichlorophenyl) -1-isopropylcarbamoylhydantoin,

N- (3,5-dichlorophenyl) -1,2-dimethylcyclopropane-1,2-dicarboxylic acid imide,

2-cyano- (N- (ethylaminocarbonyl) -2-methoxyimino) acetamide, 1- (2- (2,4-dichlorophenyl) pentyl) -1H-1,2,4-triazole, 2,4-difluoro (X - (1H-1,2,4-triazolyl-1-methyl) benzhydryl alcohol,

N- (3-chloro-2,6-dinitro-4-trifluoromethyl-phenyl) -5-trifluoromethyl

-3-chloro-2-aminopyridine,

1 - ((bis- (4-fluorophenyl) methylsilyl) methyl-1H-1,2,4-triazole, strobilurines such as methyl-E-methoxyimino- (a

- (o-tolyoxy) -o-tolyl) acetate, methyl E-2- (2- (6- (2-cyanophenoxy) pyrimidin-4-yloxy) phenyl) -3-methoxyacrylate, methyl E -methoxyimino- (α- (2-phenoxyphenyl) acetamide, methyl-E-methoximino- (α- (2,5-dimethylphenoxy) -o-tolyl) acemide, anilinopyrimidines such as N- (4,6-dimethylpyrimidin-2-yl) .) aniline, N- (4-methyl-6- (1-propynyl) pyrimidin-2-yl) aniline,

N- (4-methyl-6-cyclopropyl-pyrimidin-2-yl) aniline;

4- (2,2-difluoro-1,3-benzodioxiox-4-yl) pyrrole-3-carbonitrile,

cinnamic acid amides Acrylic 3- (4-chlorophenyl) -3- (3,4-dimethoxyphenyl) morpholide as acids

~ 3V (2RS,

3SR) -1- (3- (2-chlorophenyl) -2- (4-fluorophenyl) oxiran-2-ylmethyl) -1H -1,2,4-triazole.

The compounds of formula I are furthermore suitable for the effective control of insect, spider and mite pests. They can be used for plant protection as well as in the field of hygiene, preventive protection and veterinary use as effective means of pest control.

To the harmful insects count from the order of the butterfly (Lepidptera) to. examples of Agrtis ypsilon, Agrotis segetum, Alabama argillacea, Anticarsia gemmatalis, Argyresthia conjugella, Autographa garrana, Baupalus piniarius, Cacoecia mu.r.inana, Capua reticulana, Cheimatobia brumata, Chistoryura f um isera na, Choristone ur. C irphisunipuncta, Cydia pomonella, Dendrolimus plni, Diaphani a. Nitidal is, Diatraea grandiosella, Earias insulana, Ε1 asmopa .1pus lignosellus, Eupoecilia. ambiguella, Evetria bouliana, Feltia subterranea, Galleria mellonella, Grapholitha funebrana, Grapholitha molesta, Heliothis armigera, Heliothis virescens, Heliothis zea, Hibernia defoliaria, Hyphantria cunea, Hypoptera maleacellus, Keifeae, Malvella, Keifeae, Maldica, Keifeae. cóffeella, Leucoptera scitella, Lithocolletis blancardella, Lobesia botrana, Loxostege sticticalis,

Lymantria dispar

Lyonetia clerkella,

Malacosoma neustria,

Mamestra brassicae,

Orgyia pseudotsugata, Ostrinia nubilalis

Panolis flammea,

Pectinophora gossypiella; Peridroma saucia; Phalera bucephala

Phthorimaea brassicae,

Pseudoplusia absoluta,

Spodoptera litura,

Trichoplusia ni. Zeraphera canadensis.

Phy11o c ni sti scabra, Plutella xylostella,

S c r o b i p a 1 p u 1 a pilleriana,

Spodoptera viridana, opercuiella

Plathypena incens, Rhyacionía f rustrana,

Sitotroga cerea Fly, frugiperda,

Taumatopoea citrella, Pieris

Spařganothis

Spodoptera iittoralis pityocampa

Tortrix

From the order of the beetles (Colepotera), for example, Agrilus sinuatus, Agriotes lineatus, Agriotes obscurus, Amphimallus solstitialis, Anisandrus dispar, Anthonomus grandis,

Anthonomus pomorum, Atomaria linearis

Blastophagus piniperda, Blitophaga undata, Bruchus rufimanus, Bruchus pisorum, Bruchus lenti.s, Byctiscus betulae, Cassida nebulosa, C e r e t h e r t c t t, C e t h o r r t h e s s i s i i s i i s.

Ceutthorrhynchus napi, Chaetocnema. tibialis, Conoderus vespertinus, Crioceris asparagi, Diabrotice longicornis, Diabrotica 12-punctata, Diabrotica virgifera, Epilachna varivestis, Epitrix hirtipennis, Eutinobothrus brasiliensis,

Hylobius abietis, Hypera brunneipennis, Hypera Postica, Ips typographus,

Lema bilineata, Lema melanopus

Leptinotarsa decemli neat

Limonius californicus,

Lissorhoptrus oryzophilus,

Melanotus communis,

Meligethes aeneus,

Melolontha hippocastani,

Melolontha melolontha,

Oulema oryzae, Ortiorrhynchus sulcatus,

Ortiorrhynchus ovatus,

Phaedon cochleariae, Phyllotreta chrasocephala, Phyllophaga sp., Phyllbpertha horticola, Phyllotreta nemorum, Phylotreta striolata, Popillia japonica, Sitona lineatus, Sitophilus granaria.

9 this • it • it • it • it • it • it • it

From the order of diptera (Diptera) then for example

Aedes vexans, Anast repha! .. udens

Anopheles macuJipennis,

Ceratitis capitata,

Chry> arable of the elderly,

Chrysomya top ni vor ax, Chrysomya mace 1 i a ria,

Contarinia sorghicola,

Cordylobia anthropophaga, Cul.ex pipiens, Dacus cucurbitae

Dacus oleae, Dasineura brassicae

Fanniai canicularis,

Ga s t e r o p h i u s i n t e s t 1 n i,

Glossin plague s i t a n s, Ha ema t ob i a.

H a p 1 o d i p 1 o s, s equestris, platura,

Hypoderma 1ineata, Liriomyza sativae, Liriomyza trifoli,

Lucilia caprina, Lucilia scurf, Lucilia sericata, Lycoria pectoralis, Mayetiola destructor. Musea domestica. Muscina stabulans, Oestrus ovis, Oscinella frit, Pegomya hysocyami, Phorbia antiqua, Phorbia brassicae, Phorbia coarctata, Rhagoletis cerasi, Rhagoletis pomonella, Tabanus bovi mis, T i p u J and o]. e r a cea, T i puI and pa dii d axis.

From the order of Thripse (Thysanoptera), for example, Frank! Iniellm f usca, Frankli niealla occi denta1is, Frank! inie l la frosting, Scirtothrips citrins, Thrips oryzae, Thrips palmi, Thrips tabaci.

From the order of Hymenoptera, for example, Atha.1 ia rosae, Atta. cephalotes, Atta sexdens, Atta. texana, Hoplocampa minute, Hoplocampa testudinea, Monomorium pharaonsis, Solenopsis geminata, Solenopsis invicta.

From the order of the Heteroptera, for example, Acrosternum hilare, Blissus leucopterus, Crtopeltis notatus, Dysdercus cingulatus, Dysdercus intermedius, Eurygaster intergriceps,

Euschistus impictiventris, Leptoglossus phyllopus, Lygus

l..i neolaris, Lygus pratensis, Nezara Viola, Piesma quadrata, Solubea. insularis, Zhyanta. perdotor.

From the order of the Homoptera, for example, Acyrthosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphis fabae, Aphis pomi, Aphis sambuci, Brachycaudus cardui, Brevicorne brasicae, Cerosipha gossypii, Dreyfusia nordmanysaphase, Dicosusolae, Freyfola, Freyfola , Macrosiphum. euphorbiae, Macrosiphon rosae, Megoura viciae, Metopolophium dirhodum, Myzod. persicae, Myzus cerasi, Nilaparvata lugens, Pemphigus bursarius, Prkinsie11 and saccharicida, Phorodon humuli, Dogs 1.1 and young, Psylla. piri., Rhopalomy zus ascalonicus, Rhopalosiphum maidis, Appaphis maia, Sappaphis small, Schl,.-oplii with grams, Schizon.eu.ra lanug i nosa, Tri and I eu rod es va.po.rar i. o rum, Viteus viti fol ii.

From the order of the termites (Izoptera), for example, Calotermes f. 1 a v i c 11, s, Le c c t e r m s 11, v v t p r s, Re t cul t t r m s, u t c t f g, Termes natalensis.

For example, from the order of the Orthoptera (Orthoptera), for example by Achet, it is possible to carry out ca, Blat ta orientalis, Blat tel la germanica, Forficula a u r i c u 1 a r i a, G r y.1.1. o t a .1. p <i g r o 11 y t a 1 p a, L o c u s t a. m i g r a t o r i a,

Melanoplus bivittatus,

Me1aη op1us femu r-r ub r um

Melanoplus mexinacus,

Melanoplus sanguinipes,

Mela η o p1u s s pretus,

Nomadacris whisper! Asciata,

Per i p e a n e e a t e r a c e n a, s t o c t e r a a n r e, a c t i e t a r e a r e r i n a, S t a. U r o t s maroccanus, Tach.ycin.es asynamorus.

From the class of Arachnoidea then for example spiders (Acarina) as

Amblyomma Americanum, Amblyomma variegatum, Argas persicus,

Boophilus annulatus, Boopki lus decoloratus

m icr op1us, Brevobi pusenis c 1 s, B ryobi and the third axis, Dermacentor silvarum, Eotetranýchus carpini, Eriophyes sheldoni, Hyalomma truncatum, Ixodes ricinus, Ixodes rubicundus, Ornithodorus moubini, Detrususus moubchus, Otobius megnchus, Otobius megnchus, gallinae, Phyllocoptruta oleivora, Polyphagotarsonemus latus, Psoroptes Ovis, Rhipicephalus appendiculatus, Rhipicephalus evertsi,

Sarcoptes scabiai, Tetranychus cinnabarinus, Tetranychus kanzawai, Tetranychus pacificus, Tetranychus telarius, Tetraychus telarius.

From the mite class, for example

Meloidogyne incognita,

Meloidogyne j avanica, mites at a and d G.1bod era ro s t oc ί i en s i s,

B e 1 o η o 1 a i m u s I. o n g i c a u d a t u s, D i t y I e n c u s d e s i r r u c t o r,

Ditylenchus dipsaci, Hel i. Vinegars lenchus mul.tle i nctus,

L ong 1 doruse 1 ongatas, Ra d oph o I. ussi m. I 1. is, Ro ty 1. enc ί iusr ob ustus, T richo do ruspr im itivus, Ty 1 enchorchynchusc 1 ay toni, Tylenchorhynchus dubius, Pratylenchus neglectus Pratylenchus penetrans, Prtylnchus curvitatus, Pratylenchus goodeyi.

The active compounds may be applied as such in the form of the selected formulation or in the selected application forms, for example in the form of spray solutions, powders, suspensions or dispersions, emulsions, oil dispersions, pastes, dusts, sprays, granulates. or toppings. Application forms always depend on the purpose, use. In any case, however, they should ensure the finest possible distribution of the active substances.

• · • ·

However, the concentration of the active ingredients in the ready-to-use preparations may vary considerably.

In general, the application rate is from 0.0001 to 10%, most preferably from 0.01 to 1%.

The active compounds can also be successfully applied in the low-volume process (ULV), whereby formulations with more than 95% by weight of the active compound can be applied, even the active compound can be applied without any additives.

The application rate of the active ingredient required for pest control. under field conditions 0.1 to 2.0 kg, preferably 0.2 to 1.0 kg / ha.

For the production of directly applicable solutions, emulsions, pastes or oily dispersions, suitable are the medium and high boiling mineral oil fractions, and coal tar oils of animal origin, aliphatic, for example benzol, alkylated ethanol, propanol, butanol, cyclic oils. ohexa η o 1, cyclo ohexa η o η, polar solvents, dimethylsulfoxide, N-methylpyrrolidone, applications can be prepared from as kerosene or naphtha, as well as vegetable oils or hydrocarbons, three rahydronaphthal η, derivatives, methanol., tetrac Hydrocarbon, isophorone, strongly dimethylformamide Aqueous forms of cyclic aromatic toluene, xylene, paraffin, naphthalines or their chloroform, chlorobenzol, for example water.

for emulsion concentrates, pastes or wettable powders (spray powders, oil dispersions) by the addition of water.

By preparing emulsions, pastes or oil dispersions, the substances can be used as such or dissolved in an oily solvent and then dispersed homogeneously in water by means of a suitable wetting, dispersing adhesive or emulsifying agent. However, concentrates suitable for dilution with water can also be prepared on the basis of the active ingredient, wetting agents, adhesives, dispersing agents or emulsifying agents and, optionally, solvents or oils.

Surfactants include, but are not limited to, salt, alkaline earth and ammonium salts of ignino sulfonium, naphthalene, sulfonic acid, dihydroxybenzoate, and naphthalene. alkyl sulfonates, as well as their sulfated considerations, alkali salts of sulfonic acid condensation glycol ether

1 kγ 1 ary 1 su 11 onates, akyl cyanides, sulfates of fatty alcohols and fatty acids, alkali salts and. alkaline earth salts, fatty acids, .1., naphthaline products; and. naphthalene derivatives with resp. acid with formaldehyde; f e η o 1, f o r ma i d e h y dem, products n a. f t a 1 i n s u .1. Phenoxyphenol polyoxyethylenoctylphenol ether, ethoxylated octylphenol, nonylphenol, alkylphenylpolyglycolether, tributylphenylpolyglycolether, alkylarylpolyether alcohols, isotridecylene alcohol condensates. fatty alcohols, ethoxylated castor oil, polyoxyethylene alkyl ether, ethoxylated oil, lauryl alcohol polyglycol ether acetal, sorbitester, glycerol and stroke 1. ó z a.

Powdered, dusting and spreading agents can be made by mixing or grinding the active ingredients with a solid carrier.

• · ········· · · · · · · · · · · · · ·

The unitary formulations generally contain from 0.01 to 95% by weight, preferably from 0.1 to 90% by weight of the active ingredient. The active substances are applied in a purity of from 90% to 100%, preferably from 95% to 100% (according to

NMR spectra).

DETAILED DESCRIPTION OF THE INVENTION

I. 5 parts by weight of a compound according to the invention are mixed with 95 parts by weight of fine kaolin. A dusting composition containing 5% by weight of the active ingredient is obtained.

II. 30 parts by weight of a compound of the invention are mixed with a mixture consisting of 92 parts by weight of powdery silica gel and a five-part paraffin oil and spray-coated onto the surface of the silica gel. An active substance treatment having a good adhesion is obtained (active substance content 23% by weight).

III. 10 parts by weight of a compound of the invention are dissolved in a mixture consisting of 90 parts by weight of xylene, 6 parts by weight of an adduct of from 8 to 10 moles of ethylene oxide per 1 mol of N-monoethanolamide oleic acid, 2 parts by weight of calcium dodecylbenzenesulfonate. 40 mole of ethylene oxide per mole of castor oil (active ingredient content 9% by weight).

• · • *

- Αοβ -

IV. 20 parts by weight of a compound of the invention are dissolved in a mixture consisting of 60 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 5 parts by weight of an adduct of 7 moles of ethylene oxide per mole of isooctylphenol and 5 parts by weight of an adduct. 40 moles of ethylene oxide per mole of castor oil (active ingredient content 16% by weight).

V. 80 parts by weight of a compound of the invention are mixed with 3 parts by weight of diisobutylnaphthalinalphasifonic acid sodium salt, 10 parts by weight of ligninsulphonic acid sodium salt of suifite lye and 7 parts by weight of powdery silica gel, all in a seroele hammer (80% active substance content) ).

VI. 90 parts by weight of a compound of the invention are mixed with 10 parts by weight of N-methyl-alpha-pyrrolidone to obtain. solution suitable for application in the form of tiny droplets (active substance content 90% by weight).

VII. 20 parts by weight of a compound of the invention are dissolved in a mixture consisting of 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight, of an addition product of 7 moles of ethylene oxide per. 1 mole of isooctylphenol and 10 parts by weight of the addition product of 40 mole of ethylene oxide per mole of castor oil. By mixing the solution with 100,000 wt. parts of water gave an aqueous dispersion containing 0.02% by weight of the active ingredient.

• · · · ·

VITI. 20 parts by weight of a compound according to the invention are mixed with three parts by weight of a sodium salt of diesel oil. 11 parts, 17 parts by weight of sodium salt of Lignin sulphonic acid from sulphate lye and 60 parts by weight of powdered silica gel are then ground in a hammer mill. Mixing the resulting mixture with 20,000 parts by weight of water gives a spray mixture containing 0.1% by weight of active ingredient.

Granules, for example, coating, impregnating and homogeneous, can be prepared by binding the active ingredients to solid carriers.

These are, for example, mineral soils such as silica gel, silicic acid, silicates, talc, kaolin, ataclay, limestone, chalk, bolus, loess, clay, dolomite, diatomaceous earth, calcium and magnesium sulphate, magnesium oxide, ground plastics, fertilizers,

for example ammonium sulfate, ammonium phosphate, ammonium nitrate, urea and products of plant origin such as cereal flour, flour of tree bark, wood and walnut shells,

cellulose powder and other solid carriers.

Effective. The compounds may optionally be mixed with oils of various types, herbicides, fungicides and other pest control agents, bactericides, just prior to application. These compositions may be admixed with the compositions of the invention in a weight ratio of 1:10 to 10: 1.

• 9 9 9 999

9 99

9 9 · ··· »·· ♦ ·

9 99 »999

99 99

99

Φ · ··

The advantages of synthesis

The regulations mentioned in the subsequent examples of the synthesis of y and y are utilized by appropriate treatment of the starting compounds to obtain further compounds I. The compounds thus obtained are listed in the following tables together with physical data.

Example 1

Obtaining E-2-Methoxyimino-2 - (2'-1-phthalinoxymethyl) -phenyl) methyl ester. of acetic acid.

To a solution of 1.50 g (0.52 mol) of E-2-methoxymino-2- (2'-bromomethyl) phenyl) methyl acetate and 85 g (0.52 mol) of N-hydroxyphthalimide in 350 ml of N- of methylpyurolone is added dropwise to 59 g (0.58 mol) of triethylamine and the mixture is stirred at room temperature for 2 hours. at 70 ° C. Resulting reaction. the mixture is poured into 2.1. ice water, the crystals formed are filtered off with suction and made methylene chloride. After washing the organic phase with water, drying over sodium sulphate and removing the solvent, 168 g (88% yield) are obtained.

E-2-Methoxyxyimino-2 - ((2'-phthalimidoxymethyl) phenyl) methyl ester. acetic acid in the form of a light gray powder, m.p. 152-153 ° C.

1 H-NMR (CDCl ₃ ): δ = 3.81 (s, 3H), 3.95 (S, 3H), 5.05 (s, 2H), 7.1.2-7.81 (m, 8H) ppm .

· ·)))))))))))))))))))))))))))))))))) · · · · · · · · · · · · · ·

- -íoq

Example 2

Obtain (E, E) -2-methoxy-amino-2- (2 '- ((1-methyl-1,1'-hydroxycarbonyl) -iminooxymethyl) -phenyl) -acetate

To a solution of 100 g (0.27 mol) of the compound of Example 1 in 1000 ml of methanol was added 14 g (0.28 mol) of hydrazine hydrate and stirred thoroughly for one hour at room temperature. Subsequently, 30 g of molecular sieves (3 Ά) and 24 g (0.27 moles) of pyrosulphonic acid are added and mixed thoroughly for 1 hour. The reaction mixture was filtered and the filtrate was concentrated. The residue was then treated with a saturated Na.HCO ₃ solution and extracted with methylene chloride. After acidification of the aqueous phase with 2M hydrochloric acid, everything is again extracted with methylene chloride, the organic phase is washed with water, dried over sodium sulphate and concentrated. This gave 71 g (86% yield) of the title compound.

1 H-NMR (CDC1 _3): δ = 2.20 (s, 311), 3.87 (s, 3H), 4.04 (s, 3H), 5.13 (s, 2H), 7.15 - 7.46 (m, 4H); 8.80 (s, br.

1H) ppm

Example 3

Obtaining acetic acid (E, E) -2-methoxyimino-2- (2 '- (1-methyl, 1'-methoxyaminocarbonyl) -iminooxymethyl) -phenyl) methyl ester

To a solution of 71 g (0.23 mL) of the compound of Example 2 in 1000 mL of tetrahydrofuran was added 37 g (0.23 mol) of carbonyldiimidazole. 38g is added after gas evolution is complete.

-440 (0.46 mol) of methoxyaminohydrochloride a) was stirred vigorously for 16 hours at room temperature. The mixture is then concentrated, the residue is taken up in methylene chloride and the organic phase is extracted with a saturated NaHCO ₃ solution. After washing the organic phase with 2 M hydrochloric acid and water, it is dried over sodium sulphate and then concentrated. This afforded 72.5 g (94% yield) of the title compound as a white powder, mp 105-108 ° C.

1 H-NMR (CDCl 3: δ-2.00 (s, 3H), 3.77 (s, 3H), 3.88 (s, 31 '), 4.03 (s, 3H), 5.00 (s (2H), 7.13-7.42 (m, 4.H), 9.19 (s, 1H) ppm.

Example 4

Obtaining (Z, E, E) -2-methoxyimino-2- (2 '- ((1-methyl, 1- (1'-bromo, 1' '-methoxyiminomethyl)) -iminooxymethyl)) -phenyl Acetic acid methyl ester

A mixture consisting of 50 g (0.15 mol) and 117 g (0.45 mol) of triphenylphosphine was enriched with 148 g (0.45 mol) of the compound of Example 3 in 1000 ml of acetone nitrile tetrabrom et al. hours and then

5 ° C). The filtrate reaction mixture was under gentle conditions and the residue thus obtained was chromatographed (purified by purification). For further purification, the product recrystallized was refluxed for 100 minutes and then cooled to room temperature (freed from solids). substances.

Then, using a tert-butyl methyl ether / hexane column, the thus obtained (methylene chloride / hexane) was obtained.

• • •

34 g (58%) of the title compound were obtained as a colorless powder (Fp.: 103-105 ° C).

1 H-NMR (δ in ppm, CDCl ₃ ): 2.10 (s, 3H), 3.86 (s, 3H),

4.05 (s, 3H), 4.10 (s, 3H), 5.16 (s, 2H), 7.16-7.51 (m, 4H)

Example 5

Obtaining (Z, Ε, E) -2-methoxyimino-2- (2 '- ((1-methyl, 1- (1'-bromo, 1'-methoxyiminomethyl)) - iminooxymethyl) phenyl) -N-methylamide Acetic acid

A solution of 8 g (20 nmol) of the compound of Example 4 in 200 ml of tetrahydrofuran was enriched with 50 ml of methylamine (40% solution in water). After 20 minutes at room temperature (ca. 25 ° C), the reaction mixture was poured into cooled 2N hydrochloric acid. The product was then extracted from the mixture with tert-butyl methyl ether. 7.7 g (96%) of the title compound were obtained from the ether phase after washing with water, drying and removal of solvent as a colorless powder (Fp: 135-137 ° C).

1 H-NMR (δ in ppm, CDCl ₃ ): 2.09 (s, 3H), 2.88 (d, 3H), 3.94 (s, 3H), 4.08 (s, 3H), 5.15 (s, 2H), 6.74 (s) (br, 1H)

7.15 - 7.51 (m, 4H)

Example 6

Obtain (Z, E, R ') -2-methoxyimino-2- (2' - ((1-methyl, 1 (1 (1'-pyrazolyl), 1'-methoxyiminomethyl))) -iminooxymethyl) -phenyl -N-methylamide of acetic acid (Example I. 011)

A mixture of 1 g (40 nmol) of sodium hydride and 100 ml was enriched dropwise with a solution of 2.7 g (40 50 ml of dimethylformamide). After 30 minutes at ca. The reaction mixture was allowed to stand at 100 DEG C. After cooling, the mixture of tert-butyl methyl ether was obtained and the ether was washed with dilute acid to remove the solvent (5.7 g) in the colorless oil.

dimethylformamide du runo 1) pyrazole at room temperature with a solution of 7.7 g 5 in 100 ml of dimethylformamide.

stored at water temperature for one hour. The product was eluted with the aid of a cannula with water, after drying and the compounds in the night.

(7 6

%) ¹ rh I other

1 H-NMR (δ in ppm, CDCl ₃ ):

(s, 3H), 4.02 (s, 3H),

2.04

5.05

2.87

6.38 (d, 3H), (t, 1H);

3.91

7.01

IH), 7.20

7.40

Example

Obtaining (Z, E, E) -2-methoxyimino-2- (2 '- ((1-methyl, 1- (1''-piperidinyl), 1'-methoxyiminoethyl)) -iminooxymethyl) -phenyl - acetic acid methyl ester (Example I. 002) (1)

Mixture 1.0 g (7 nmol) Hydrocarbon, dr 100 ml Dimethylformamide by J. a Mixed not going e with 2.0 g (5 nmol) s 4 and then se 4.3 g (50 nmol)

piperidine. After 60 hours at room temperature (ca. 25 ° C), the reaction was poured into cooled, dilute hydrochloric acid. The product was extracted from the mixture so obtained with tert-butyl methyl ether. 0.8 g (40%) of the title compound was obtained as a colorless oil from the ether phase after washing with water, drying and solvent removal.

1 H-NMR (δ in ppm, CDCl ₃ ): 1.45-1.60 (m, 6H), 1.94 (s, 3H), 3.04-3.11 (m, 4H), 3.66 (s, 3H), 3.86 (s, 311) 4.04 (s, 3H), 5.06 (s, 2H), 7.17-7.50 (m, 4H);

Example 8

Obtaining (Z, E, E) -2-methoxyimino-2- (2 '- ((1-methyl), 1 (1' (1'-piperidinyl)),

1'-methoxyiminomethyl) -imidinooxymethyl) -phenyl) -N-methylamide acetic acid (Example I. 007)

A solution of 0.8 g (2 nmol) of the compound of Example 7 in 1.00 ml of tetrahydrofuran was mixed with 10 ml of a methylamine solution (40% in water). After 60 hours at room temperature (ca. 25 ° C), the reaction mixture was poured in water. The product was. extracted from the mixture thus obtained with tert-butyl methyl ether. The ether phase was obtained after washing with water, drying and solvent removal. 0.7 g (87%) of the title compound as a colorless oil.

• • •

1 H-NMR (δ in ppm, CDCl ₃ ): 1.41 - 1.62 (m, 6H), 1.93 (s, 3H),

2.88 (d, 3H), 2.98-3.06 (m, 4H), 3.65 (s, 3H), 3.94 (s,

3H), 5.05 (s, 2H), 6.80 (s, br, 1H), 7.17-7.46 (m, 4H)

Example 9

Obtaining E-2-benzyloxyimino, -N-methoxy-propionamide

To a solution of 65 g (337 nmol) of (E) -2-benzyloxyiminopropionic acid (J. Org. Chem. 46 (1981), 3346-8) in 500 ml of tetrahydrofuran was added 55 g (337 nmol) of carbonyl diimidazole. After gas evolution was complete, the solution was mixed with 43 g (510 nmol) of methoxyamine hydrochloride and stirred for 2 hours at room temperature. The resulting pellet was aspirated and the filtrate was poured onto 2 M hydrochloric acid. Extraction with tert-butyl methyl ether, washing the organic phase with water, drying over sodium sulfate and removing the solvent gave 53.5 g (72% yield) of the title compound as a white powder, mp 59-62 ° C.

1 H-NMR (δ in ppm, CDCl ₃ ): 2.05 (s, 3H), 3.78 (s, 3H), 5.17 (s, 2H), 7.25-7.40 (m, 5H) ), 9.17 (s, 1H)

Example 10

Obtaining E-2-benzyloxyimino, (Z) -N-methoxy-propane-imidoyl bromide

A mixture of 53.5 g (240 nmol) of the compound of Example 9 and 189 g (720 nmol) of triphenylphosphine in 1000 ml of acetonitrile was mixed with

240 g (720 nmol) of tetrabromomethane.

• ·

The mixture thus obtained was heated for 7 hours and then cooled to room temperature (ca. 25 ° C). The reaction mixture was then freed from all solids. The solvent was distilled off under gentle pressure, and the residue was purified by column chromatography (silica gel, tert-butyl 1-methyl ether / cyclohexane). . This gave 59 g (87% yield) of the title compound as a colorless oil.

1 H-NMR. (6 ppm, CDC1 _3): 2,1.5 (s, 311), 4.08 (. ;, · 3H), 5,2o (s, 2H), 7.26 - 7.45 (m, 5H)

Example. 11

Detection of 1. - ((E) - 2.benzyloxymethyl, (Z) -N-methoxyethoxy-propanimidoyl) -4-methylpyrazole

To a suspension of 4.8 g (200 nmol) of sodium hydride in 200 ml of dimethylformamide was added 16.4 g (200 nmol) of 4-methyl. pyrazole. After 30 minutes at room temperature (ca. 25 ° C), the mixture thus obtained was mixed with a solution of 20 g (70 nmol) of the compound of Example 10 in 100 ml of DMF and the reaction mixture was then stirred at room temperature for 16 hours. . The reaction mixture was then poured onto. 2 M hydrochloric acid and extracted with tert-butyl methyl ether. After washing with hydrochloric acid (2 M) and water, drying and removal of the solvent, 11 g (55% yield) of the title compound were obtained as a light brown oil from the ethanol phase.

-4461H - NMR (δ ppm, CDCl _i): 2.08 (s, 3H), 2.10 (s, 3H), 4.00 (s, 3H), 5.18 (s, 2H) 7.25 - 7.40 (m, 5H); 7.47 (s, 1H);

7.80 (s, 1H).

Example 12

Obtaining

1 - ((E) -2-hydroxyimino), (Z) -N-methoxy-propanimidoyl) -4-methylpyrazole

11.0 g (38.6 nmol) of the compound of Example 11 was dissolved with 250 ml of ethanol and, under nitrogen, hay was mixed with 5 g of palladium on activated carbon (10%). After purging the reaction apparatus with hydrogen. The mixture was stirred at 60 ° C until no more hydrogen was detected. After rinsing the parathy, the catalyst was flattened, the filtrate was concentrated. the residue is taken up in 10% sodium hydroxide solution. After extraction with tert-butyl methyl ether, the aqueous phase was acidified with hydrochloric acid (2 M) and extracted with tert-butyl methyl ether. The organic phase was washed with water to give 2.5 g (29% yield) of the title compound as a pale yellow oil.

1 H-NMR (δ in ppm, CDCl ₃ ): 2.11 (s, 6H), 3.99 (s, 3H), 7.48 (s, 1H), 7.73 (s, 1H)

Example 13

Obtaining (Z, E, E) -2- (2 '- ((1-methyl, 1- (1 '- 4-lpy ra ra; <o l y 1.), 1 ’´´-methoxyiminomethyl)) -iminooxymethy

1) -phenyl.) - Crotonic acid methyl ester (Example I. 002

Κ 0.1.2 g (4 nmol) of sodium hydride (80%) in 10 ml

d. Imam 11 mM amide was added 0.8 g (3.6 nmol) of the compound of Example 12 dissolved in 1.0 mL of dimethylformamide. After stirring for 30 minutes, 0.97 g of (E) -3-methyl-2- ((2'-bromomethyl) phenyl) methyl acrylate was added and again stirred for 16 hours at room temperature. Reaction. The mixture was poured onto water and extracted with tert-butyl methyl ether. The organic phase was washed with sodium hydroxide solution. (10%) a. Water, dried and concentrated. After column chromatography on silica gel (tert-butyl methyl ether / n-hexane), 1.2 g (51% yield) of the title compound was obtained as a white oil.

1 H-NMR (δ in ppm, CDCl ₃ ) (s, 3H), 3.67 (s, 3H),

1.59 (d, 311);

4.01 (s, .311),

2.05 (s, 3H), 2.11

2.H)

7.02 - 7.51 (m, 6H), 7.80 (S, 1H)

Example 14

Obtaining (Z, Ε, E) -3-methoxy-2- (2 '- ((1-methyl., 1' - (1- (1'-4-methylparyzoyl), 1'-methoxyiminomethyl)) - iminooxymethyl) Acrylic acid methyl ester (Example I. 023)

To 0.12 g (4 nmol) of sodium hydride (80%) in 10 ml of dimethylformamide was added 0.8 g (3.6 nmol) of the compound of Example 12 dissolved in 10 ml of dimethylformamide. After stirring for 30 minutes, 1.0 g (3.6 nmol) of (E) -3-methoxy-2 - ((2'-bromomethyl) phenyl) methyl acrylate was added and stirred for 1.6 hours at room temperature.

• · ·

• · ·

The reaction mixture was then added to 1 L of La. to water and extracted with tert-butyl methyl ether. The organic phase was washed with sodium hydroxide solution (1.0%) and water, dried and concentrated. Po pillar c h r om a t og r a. Fi .i. The title compound (tert-butyl methyl ether / n-hexane) gave 1.0 g (65% yield) of the title compound as a colorless oil.

1 H-NMR (δ in ppm, CDCl ₃ ): 2.06 (s, 3H), 2.11 (s, 3H), 3.66 (s, 3H), 3.79 (s, 3H), 4, O 2 (s, 3H), 5.14 (s, 2H), 7.10 7.55 (m 6H), 7.83 (s, 1H)

- 449 _

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-623 Examples of effects against harmful fungi and fungi:

The efficacy of the compounds of Formula 1 'was demonstrated by the following experiments:

The active ingredients were formulated as a 20% emulsion in a mixture of 70% by weight of cycklohexane, 20% by weight of Nekanii LN (Lutensol AP6, a wetting agent with emulsifying and dispersing effect based on ethoxylated alkylphenols) and 10% by weight of Emulpho.ru EL (Emulan EL, emulsifier based on ethoxylated fatty alcohols) and diluted with water to the required concentration.

The known active substances A (according to WO-A 95/21, 154, X-NOCH, YR ¹ = NHCH 3, R ² m-H,

R ³ = R ⁴ = Cii., Z'- 1-CH _? -pyrazol-3-yl), B (p o d 1 e W-A 95/21, 154, X = NCH ,, NHCIL YR ¹ = ^R; ζ = H, R ³ - IV - - CH ₃ , 7, - pyrimidi n-2-y.l) and C (according to WO-A 95/21, 158 X = NOCH ,, YR ^: = 00! E, C = h, R ³ R ⁴ == == CH ,, Z = pyramid n- -3-yl)

Effect against Erysiphe graminis var. tritici (wheat powdery mildew)

Wheat germination leaves (Fruehgold variety) were first treated with an aqueous solution of the active ingredients (application rate: 63 ppm). After 24 hours, the plants were dusted with spores of wheat mildew (Erysiphie graminis var. Tritici). The treated plants were then incubated for 7 days at 20-22 ° C and 75-80% relative humidity. The extent of mold development was then determined.

-Wl-

In this test, plants treated with the compounds of the invention Nos. 1.007, 1.011, 1.012, 1.014 and 1.016 showed an attack rate of 1.5% or less, while plants treated with known active substances A and B showed an attack rate of 40%. Untreated (control) plants were infected with 70%.

Effect against Puccinia recondita (brown rust wheat)

The leaves of germinating wheat plants (Kanzler variety) were dusted with spores of wheat rust (Puccinia recondita). The plants so treated were then incubated for 24 hours at 20-22 ° C and 90-95% relative humidity and then treated with aqueous orzotec of active ingredients (application rate: 63 ppm). After an additional 8 days at temperature

20-22 ° C and at a relative humidity of 65 - 70% air, the extent of mold development was then determined. Viatus evaluation was performed visually.

In this test, plants treated with the compounds of the invention Nos. 1.007, 1.01.1, 1.013 to 1.017 and 1.019 showed an attack of 25% or less, whereas plants treated with known active substances A, B and C as well as untreated (control) plants were attacked 75%.

Examples of efficacy against animal pests

The efficacy of the compounds of formula I against animal pests has been demonstrated by the following experiments:

The active substances were treated as

-asr-

(a) 0, 1% -ηi r ο z k u in acet onu r or e

b) 10% emulsion in a mixture of 70 weight percent cyclohexane, 20 weight percent Non-LN (Lutensol. AP6, ethoxylated alkylphenol surfactant wetting agent) and 10 weight percent Emulphor EL (Emulan EL, emulsifier based ethoxylated fatty alcohols) and were diluted with acetone according to the desired concentration; water in case b).

At the end of the experiments, the lowest concentration at which the compounds used in comparison with the control experiments (without treatment of plants) were still found still ensured an 80-100% reduction in development and / or control. mortality (efficiency threshold or minimum concentration) of fungal spores.

Claims (12)

Ρ A 1 Ε Ν Τ Ο V É R R R Υ A compound of formula I wherein the substituents and the index have the following meanings: X NCH ₃ , CHOCH ₃ , CHCH ₃ and CHCH ₂ CH ₃ , Y O and NR And R is hydrogen of C ₁ -C ₄ -alkyl, From 1-aziridinyl, 1-diaziridinyl, 1-azetidinyl, 1 - pyrrolidine 1, 2 - i from oxa z 1 i diene 1, 2 - i z o 3 i z z 1 i diene 1, 1 -pyr z z 1 i diy 1, 3-oxado 1 i di. nyl. z ol i di nyl, 1-imidazolidinyl, 1,2,4-oxadiazolidin-2-yl, 1,2,4-oxadiazolidin-4-yl, 1,2,4-thiadiazolidin-2-yl, 1,2,4-thiadiazolidin-4- yl, 1-triazolidinyl, 1,3,4-oxadiazolidin-3-yl, 1,3,4-thiadiazolidin-3-yl, 2,3-dihydropyrrol-1-yl., 2,5-dihydropyrrol-1-yl, 2,3-dihydroisoxazol-2-yl, -29- 2,5-dihydroxy-1-y-2-yl, 2,3-dihydroxy-1-2-y-1, 2,5-dihydroisazolazol-2-yl 1,2,3-dihydropyrazol-1-yl; 2,3-dihydropyrazol-2-yl-4,5,5-dihydropyrazol-1-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydro-thiazol-3-yl, 2,3-dihydro-imidazol-1-yl, 4,5-dihydro-imidazol-1-yl, 2,5-dihydroimidazol-1-yl, 1-piperidinyl, 4-morpholinyl, 1-piperazinyl, 1-hexahydropyridinyl, 1-hexahydropyridinyl 1,2,3-dihydroindol-1-yl, 4-thiomorpholinyl; 1,2,4-hexahydrotriazin-1-yl, 2,3-dihydroisoindol-2-yl, 1-pyrrolyl, 1-imidazolyl, 1-pyrazolyl, 1-triazolyl, 1-tetrazolyl, 2-tetrazolyl, 1-indole. yl, 1-indazolyl, benzimidazol-1-yl, pyrimidine-1-yl, pyrrolidinyl-1-yl, pyrrolidinyl, -1-y-1, py rro 1. pyrimidin-1-yl, pyrrolo pyrazin-1, pyrrolotriazin-1-yl, imidazopyridin-1-yl, imidazy opi ri da zi-1-y 1-mi from opyrazin-1-yl, idaz-opyrazin-1-yl, pyrazolopyridin-1-yl, pyrazolopyridazin-1-yl, pyrazolopyrimidin-1-yl, pyrazolopyrazin-1-yl and pyrazolotriazine -1-yl, wherein the above radicals may be partially or fully halogenated and / or may carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl 1, and i. C 1 -C ₆ -alkyl, C 1 -C ₆ -haloalkyl, C 1 -C 6 -alkylcarbonyl, C 1 -C ₆ -alkyl. su .1 foeny 1., C. - C ₆ - and 1 kyl. are 1-oxy .1 f., C ₁ -C ₆ -al.koxy, _C-C6 - haloalkoxy, _Cj-C6 alkoxy carbonyl -al, C, -Cg-alkyl and 1 1 i. io, Ci-C ₆ -alkylamino, C 1 -C 8 -alkylamino, C 1 -C 8 -alkylamino. arons 1., Di - C, - C ₆ - and 1 am 1. i. nocarbones 1, C ₆ -C ₆ -alkyl 1. thiocarbonyl, Di-C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkenyloxy or C (= NOR ^a ) -A 1 R ¹³ , 9 9 9 9 9 9 9 9 9 9 · ···· · 999 9 9 9 9 99 99 99999 9 9 9 9 9 99 9 99 9 9 99 9 99 9 ~ 9i <P- C ₃ -Cg-cycloalkyl, C ₃ -C ₆ cycloalkyl- 1oa one alkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, and rvioxy, arylthio, hetaryl, and hetatvIoxy hetarylthio, wherein the cyclic groups may be partially or fully halogenated or may carry one to three of the following: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C ₃ -C ₆ -alkyl, C ₃ - C ₆ -haloalkyl, C ^ Cg-alkylsulfonyl, C -C ₆ -alkylsulfoxyl, _C-C6 alkoxy, Cg-Cy-haloalkoxy, C ^ -Cg alkoxycarbonyl, Cj-Cg-alkylthio, (Y-Cg- alkylamino, di-C-C ₆ -alkylamino, Cp-Cg-alkylaminocarbonyl, di-C - C ₆ --alkyl.aminokarbonyl C, -CY -alkylaminothiocarbonyl D i - C - C ₆ - a. 1 ky 1 Amine 1 ot about 1 carbonyl, _Ci-C6-al keny 1 C, -Cg al-alkenyloxy, C (= -nor ^u) -A _n -R ^b or substituted by customary groups, benzyl, benzyloxy, aryl, aryloxy , arylthio, hetaryl, hetaryloxy and hetaryltio, and / or wherein these residues may be linked to one another by one of the following: C ₁ -C ₅ -alkylene, oxy-C ₁ -C ₄ -alkylene, and oxy-C ₁ -C ₄ -alkenyloxy, wherein the alkylene chains may be partially or fully halogenated and / or may carry one to three C ₁ -C ₃ -alkyl groups. R ^{1 is} hydrogen and C 1 -C ₄ -alkyl, R ^{2 is} cyano, nitro, trifluoromethyl, halogen, C ₁ -C ₄ -alkyl and C ₁ -C ₄ -alkoxy, m 0, 1 or 2, wherein the radicals R ² may be different when m is 2; · ·· · · · · · · R ^{3 is} hydrogen, cyano, nitro, hydroxy, amino, cyclopropyl, halogen, C ₁ -C ₄ -alkyl, C ₁ -C ₄ -haloogen, C ₁ -C ₄ -a. ko xy, C, - C ₄ - haloalkyloxy, C _x - C 1 - thio, C _x - C ... - a 1 cy 1 am i 11 oa i) -C 1 -C ₄ -alkylamino; R ^{4 is} hydrogen C _x -C _xo -alkyl, C ₂ -C ₁₀ -alkenyl, C ₂ --C ₁₀ -A to 1: 1 ins, TY-C ^ -alkylcarbonyl, C ₂ -C ₁₀ -alkenylkarbony 1, C ₂ -C _10- alkynylcarbonyl. or C ₁ -C ₃₀ -alkylsulfonyl, these radicals may be partially or fully halogenated or carry one to three of the following groups: - cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, - halogen, C _x -C ₆ -ha logenalkyl C _x -C ₆ -al sulfates onyl, C 1 -C ₆ -alkyloxycarbonyl, C ₁ -C ₆ -alkyloxy, C ₁ -C ₆ -haloalkyloxy, C 1 -C ₆ -alkoxycarbonyl, C 1 -C ₆ -alkyloxy _{x 6} -C io -alkylt C _x -C ₆ -al alkylamino, di-C-Cg-alkylamino, Cy-Cy-alkyl and 1 1aminokarbony 1 D i - C _x - C ₆ - alkyl and 1 1 amino they nokarb 1 C _x - C ₆ - alkyl and 1 .1 1 am Inotia carbonyl, di-C _x -C ₆ -al ky.1 aminothiocarbonyl, _{C2 phi} -C alkenyloxy, "C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -cykioalkoxy, heterocyclyl, heterocyclyloxy, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy and hetaryltio, wherein the cyclic groups may be partially or fully halogenated or they may carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, at least one of the following groups: · Aminocarbonyl, aminothiocarbonyl, halogen, C 1 -, -, - - - - - - - - - - - - - - - - - - - - C ₆ -C ₇ - C 1 -C ₆ -cycloalkyl 1, C ₆ -C ₆ -haloalkenyl, C ₆ -C ₆ -alkylene 1 C ₁ - Cg-alkyl and I L. sulfoxy1, C-C _(-A 1 alkoxy, C 1 -C ₆ -ha1ogena alkoxy, Cj-C ₆ -alkoxycarbonyl, C, -Cg-alkyl, and even thio, C-C ₆ - alkyl, amino, C 1 -C ₆ -alkylamino, C 1 -C ₆ -alkyl minokarbonyl, di-C-Cg-alkylaminocarbonyl, C ₆ -C -alkylaminotiokarbonyl, di-C -alkylaminothiocarbonyl, C ₂ -C ₆ -alkenyl, C ₆ -C -al.kenyloxy, benzyl, benzyloxy, aryl, aryloxy , arylthio, hetaryl, hetaryloxy, hetaryltio and C (NOR ¹ ) -A _n -i \ ^b C ₃ -C ₆ -cycloalkyl, aryl, arylcarbonyl !, arylsulfonyl, hetaryl, hetarylcarbonyl and hetarylsulfonyl, where these radicals may be partially or fully halogenated or may carry one to three of the following moieties are: - cyano, nitro, hydroxy, mercapto, amino, carboxyl, and amino acid, 1, am. i η o I i. o k a r b o ny 1, - halogen, C ₁ -C ₆ alkyl, _C-C6 haloalkyl., C 1 -C ₆ -alkylcarbonyl, C 1 -C ₆ -alkylsulfonyl, Cj-Cg alkyl-Al sulfoxyl, _C3 "C cyk.l.oalkyl, C ~ C ~ _f I and alkoxy, C ₁ -C ₆ -haloalkyloxy, C ₁ -C ₆ -alkyloxycarbonyl 1, C 1 -C 6 -alkylthio, C 1 -C ₆ -alkylene, Di-C 1 -C ₆ -al alkyl amino, Cj-Cg-alkylaminocarbonyl, di-C-Cg al alkylaminocarbonyl, _Cj-C6 alkyl -al aminothiocarbonyl, di-C ₃ -C ₆ -alkylaminotiokarbony .1 ..., C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkyenyloxy, benzyl, beznyloxy, aryl, aryloxy, hetaryl, hetaryloxy and C (= NOR ^a ) -A n -R ^b , wherein: Λ denotes oxygen, sulfur and nitrogen wherein d denotes hydrogen or C 6 -C 7 -alkyl, n denotes 0 or 1 and R ^a , R ^b are each hydrogen or C 1 -C 8 -alkyl. and salts thereof. Compounds of formula I according to claim 1, wherein m is 0. Compounds of formula I according to claim 1, wherein R ¹ is methyl. A process for the preparation of compounds of formula I according to claim 1, wherein R ^{3 is} not halogen, characterized in that the benzyl derivative of formula I 1, II, wherein L ¹ represents a nuclonephile exchange group, is reacted in a manner known per se with the hydroxyimine of the formula III NOR ⁴ H0N = CR ³ III · * * * · · · «« « .. Process for producing compounds of formula I according to claim 1, wherein R ^J is other than halogen, which is characterized in that the benzyl · der.i.vát formula II according to claim 4 indicating per se known manner with a dihydroxyimine of the formula IIIa is reacted NOH and converted to the compound of formula IVa 0 = ^C-YR1 The NOH and IVa are then converted to a compound of formula V wherein Ib is a nucleophilically replaceable depletion group with nu. A process for the preparation of compounds of formula I according to claim 1, wherein R ^{3 is} not halogen, characterized in that the benzyl derivative of formula II according to claim 4 is reacted with a carbonyl hydroxylamine of formula 11Ib and converted to. HON - CR ³ IIIb is a compound of formula VIa ₃ from ° CH ₂ ON = CR ^{3 -} cf via a Via is then converted with thiosulfate into VI VIb and VIb are then either a.) first with hydroxylamine or its ammonium salt and then with a compound of formula V (R ⁴ -L ^a) according to claim 5 or b) with hydroxylamine or an ammonium salt thereof, of formula VIIa, respectively; VIIb R ⁴ -ONH ₂ R ⁴ -ONH · Q Vila VIIb where Q ~ represents an acid anion, converts to I. «· V ·· ·· ···· 9 9 9 9 9 9 99 999 99,999 9,999 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 9 99 99 9 · 9 99 99 9999 Ί. A product suitable for controlling pests of animal origin or harmful hulle? or a fungus comprising a solid or liquid carrier and a compound of formula I according to claim 1. A process for combating harmful fungi and fungi, characterized in that fungi or fungi or material, soil, seed or plants which need to be protected from fungi and fungi are treated with an effective amount of a compound of formula 1 according to claim 1. 9. A method of controlling animal pests, characterized in that pests or material. A compound which is a compound of formula (1) as defined in claim 1 is treated with an effective amount of a compound of formula (1). Use of the compounds I according to claim 1 for the manufacture of a composition suitable for controlling animal pests or harmful fungi and fungi. Use of the compounds of formula I according to claim 1 for controlling animal pests or harmful fungi and fungi. Compounds of formula Vha according to claim 6. Compounds of formula VIb according to claim 1. 6. Compounds of formula III (R ⁴ AH) according to claim 4.