CY1117600T1 - DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES - Google Patents

DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES

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Publication number
CY1117600T1
CY1117600T1 CY20161100492T CY161100492T CY1117600T1 CY 1117600 T1 CY1117600 T1 CY 1117600T1 CY 20161100492 T CY20161100492 T CY 20161100492T CY 161100492 T CY161100492 T CY 161100492T CY 1117600 T1 CY1117600 T1 CY 1117600T1
Authority
CY
Cyprus
Prior art keywords
diazorazoli
producers
methods
cellular
connectors
Prior art date
Application number
CY20161100492T
Other languages
Greek (el)
Inventor
Eckhard Günther
Olaf Schaefer
Michael Teifel
Klaus Paulini
Original Assignee
Aeterna Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP06018750A external-priority patent/EP1900742A1/en
Application filed by Aeterna Zentaris Gmbh filed Critical Aeterna Zentaris Gmbh
Publication of CY1117600T1 publication Critical patent/CY1117600T1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει συζυγή διζοραζολίων και τα παράγωγα τους με μόρια κυτταρικής σύνδεσης, όπως πεπτίδια, πρωτεΐνες, ορμόνες, πρωτεΐνες αίματος και αντισώματα. Η παρούσα εφεύρεση παρέχει περαιτέρω νέα παράγωγα διζοραζολίου και μεθόδους παραγωγής τέτοιων συζυγών και παραγώγων διζοραζολίου. Αυτές οι ενώσεις μπορούν να χρησιμοποιηθούν ως φάρμακα για τη θεραπεία φυσιολογικών και/ή παθοφυσιολογικών καταστάσεων σε θηλαστικά, συγκεκριμένα για τη θεραπεία ποικίλων όγκων.The present invention provides a conjugate of diazorazoles and their derivatives with cellular binding molecules, such as peptides, proteins, hormones, blood proteins and antibodies. The present invention further provides novel diisorazole derivatives and methods of producing such conjugates and diisorazole derivatives. These compounds can be used as medicaments for the treatment of physiological and / or pathophysiological conditions in mammals, in particular for the treatment of various tumors.

CY20161100492T 2006-09-06 2016-06-03 DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES CY1117600T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US84235706A 2006-09-06 2006-09-06
EP06018750A EP1900742A1 (en) 2006-09-07 2006-09-07 Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof
EP07803270.3A EP2066679B1 (en) 2006-09-06 2007-09-06 Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof

Publications (1)

Publication Number Publication Date
CY1117600T1 true CY1117600T1 (en) 2017-04-26

Family

ID=58606644

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20161100492T CY1117600T1 (en) 2006-09-06 2016-06-03 DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES

Country Status (1)

Country Link
CY (1) CY1117600T1 (en)

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