CY1117600T1 - DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES - Google Patents
DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USESInfo
- Publication number
- CY1117600T1 CY1117600T1 CY20161100492T CY161100492T CY1117600T1 CY 1117600 T1 CY1117600 T1 CY 1117600T1 CY 20161100492 T CY20161100492 T CY 20161100492T CY 161100492 T CY161100492 T CY 161100492T CY 1117600 T1 CY1117600 T1 CY 1117600T1
- Authority
- CY
- Cyprus
- Prior art keywords
- diazorazoli
- producers
- methods
- cellular
- connectors
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Η παρούσα εφεύρεση παρέχει συζυγή διζοραζολίων και τα παράγωγα τους με μόρια κυτταρικής σύνδεσης, όπως πεπτίδια, πρωτεΐνες, ορμόνες, πρωτεΐνες αίματος και αντισώματα. Η παρούσα εφεύρεση παρέχει περαιτέρω νέα παράγωγα διζοραζολίου και μεθόδους παραγωγής τέτοιων συζυγών και παραγώγων διζοραζολίου. Αυτές οι ενώσεις μπορούν να χρησιμοποιηθούν ως φάρμακα για τη θεραπεία φυσιολογικών και/ή παθοφυσιολογικών καταστάσεων σε θηλαστικά, συγκεκριμένα για τη θεραπεία ποικίλων όγκων.The present invention provides a conjugate of diazorazoles and their derivatives with cellular binding molecules, such as peptides, proteins, hormones, blood proteins and antibodies. The present invention further provides novel diisorazole derivatives and methods of producing such conjugates and diisorazole derivatives. These compounds can be used as medicaments for the treatment of physiological and / or pathophysiological conditions in mammals, in particular for the treatment of various tumors.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US84235706A | 2006-09-06 | 2006-09-06 | |
EP06018750A EP1900742A1 (en) | 2006-09-07 | 2006-09-07 | Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof |
EP07803270.3A EP2066679B1 (en) | 2006-09-06 | 2007-09-06 | Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1117600T1 true CY1117600T1 (en) | 2017-04-26 |
Family
ID=58606644
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20161100492T CY1117600T1 (en) | 2006-09-06 | 2016-06-03 | DIAZORAZOLI CODES AND ITS PRODUCERS WITH CELLULAR CONNECTORS, NEW DIAZORAZOLI PRODUCERS, METHODS OF PRODUCTION, AND THEIR USES |
Country Status (1)
Country | Link |
---|---|
CY (1) | CY1117600T1 (en) |
-
2016
- 2016-06-03 CY CY20161100492T patent/CY1117600T1/en unknown
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