CY1117573T1 - BARONIC AS ARGINATION Suspensions - Google Patents

BARONIC AS ARGINATION Suspensions

Info

Publication number
CY1117573T1
CY1117573T1 CY20161100317T CY161100317T CY1117573T1 CY 1117573 T1 CY1117573 T1 CY 1117573T1 CY 20161100317 T CY20161100317 T CY 20161100317T CY 161100317 T CY161100317 T CY 161100317T CY 1117573 T1 CY1117573 T1 CY 1117573T1
Authority
CY
Cyprus
Prior art keywords
argination
baronic
suspensions
arginase
activity
Prior art date
Application number
CY20161100317T
Other languages
Greek (el)
Inventor
Zandt Michael Van
Jr Gunnar Erik Jagdmann
Original Assignee
Mars Incorporated
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP11779904.9A external-priority patent/EP2632927B1/en
Application filed by Mars Incorporated filed Critical Mars Incorporated
Publication of CY1117573T1 publication Critical patent/CY1117573T1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Οι χημικές ενώσεις σύμφωνα με τον Χημικό Τύπο I είναι δυνατοί αναστολείς της δραστηριότητας της αργινάσης I και II, όπου τα R1, R2, R3, R4, D, W, Χ, Υ και Ζ ορίζονται στις προδιαγραφές. Η εφεύρεση παρέχει ακόμη φαρμακευτικές συνθέσεις των χημικών ενώσεων και μεθόδους για τη χρήση τους κατά την αντιμετώπιση ή πρόληψη ασθενειών ή παθήσεων σχετικών με τη δραστηριότητα της αργινάσης.The compounds according to Formula I are potent inhibitors of arginase I and II activity, wherein R1, R2, R3, R4, D, W, X, Y and Z are specified in the specification. The invention further provides pharmaceutical compositions of the compounds and methods for their use in the treatment or prevention of diseases or conditions related to arginase activity.

CY20161100317T 2010-10-26 2016-04-18 BARONIC AS ARGINATION Suspensions CY1117573T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40676010A 2010-10-26 2010-10-26
EP11779904.9A EP2632927B1 (en) 2010-10-26 2011-10-19 Boronates as arginase inhibitors

Publications (1)

Publication Number Publication Date
CY1117573T1 true CY1117573T1 (en) 2017-04-26

Family

ID=58606649

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20161100317T CY1117573T1 (en) 2010-10-26 2016-04-18 BARONIC AS ARGINATION Suspensions

Country Status (1)

Country Link
CY (1) CY1117573T1 (en)

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