CY1117573T1 - BARONIC AS ARGINATION Suspensions - Google Patents
BARONIC AS ARGINATION SuspensionsInfo
- Publication number
- CY1117573T1 CY1117573T1 CY20161100317T CY161100317T CY1117573T1 CY 1117573 T1 CY1117573 T1 CY 1117573T1 CY 20161100317 T CY20161100317 T CY 20161100317T CY 161100317 T CY161100317 T CY 161100317T CY 1117573 T1 CY1117573 T1 CY 1117573T1
- Authority
- CY
- Cyprus
- Prior art keywords
- argination
- baronic
- suspensions
- arginase
- activity
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Οι χημικές ενώσεις σύμφωνα με τον Χημικό Τύπο I είναι δυνατοί αναστολείς της δραστηριότητας της αργινάσης I και II, όπου τα R1, R2, R3, R4, D, W, Χ, Υ και Ζ ορίζονται στις προδιαγραφές. Η εφεύρεση παρέχει ακόμη φαρμακευτικές συνθέσεις των χημικών ενώσεων και μεθόδους για τη χρήση τους κατά την αντιμετώπιση ή πρόληψη ασθενειών ή παθήσεων σχετικών με τη δραστηριότητα της αργινάσης.The compounds according to Formula I are potent inhibitors of arginase I and II activity, wherein R1, R2, R3, R4, D, W, X, Y and Z are specified in the specification. The invention further provides pharmaceutical compositions of the compounds and methods for their use in the treatment or prevention of diseases or conditions related to arginase activity.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US40676010A | 2010-10-26 | 2010-10-26 | |
EP11779904.9A EP2632927B1 (en) | 2010-10-26 | 2011-10-19 | Boronates as arginase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1117573T1 true CY1117573T1 (en) | 2017-04-26 |
Family
ID=58606649
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20161100317T CY1117573T1 (en) | 2010-10-26 | 2016-04-18 | BARONIC AS ARGINATION Suspensions |
Country Status (1)
Country | Link |
---|---|
CY (1) | CY1117573T1 (en) |
-
2016
- 2016-04-18 CY CY20161100317T patent/CY1117573T1/en unknown
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