CY1117389T1 - HYDROSYL-SUBSTITUTED PYROLID [2,3-b] PYRIDINES AND PYROLID [2,3-b] PYRAMIDINES AS JANUS MOVEMENTS - Google Patents
HYDROSYL-SUBSTITUTED PYROLID [2,3-b] PYRIDINES AND PYROLID [2,3-b] PYRAMIDINES AS JANUS MOVEMENTSInfo
- Publication number
- CY1117389T1 CY1117389T1 CY20161100097T CY161100097T CY1117389T1 CY 1117389 T1 CY1117389 T1 CY 1117389T1 CY 20161100097 T CY20161100097 T CY 20161100097T CY 161100097 T CY161100097 T CY 161100097T CY 1117389 T1 CY1117389 T1 CY 1117389T1
- Authority
- CY
- Cyprus
- Prior art keywords
- pyrolid
- janus
- pyridines
- pyramidines
- hydrosyl
- Prior art date
Links
Abstract
Η παρούσα εφεύρεση παρέχει ετεροαρυλο υποκατεστημένες πυρρολο[2,3-b]πυριδίνες (I) και ετεροαρυλο υποκατεστημένες πυρρολο[2,3-b]πυριμιδίνες που διαμορφώνουν τη δραστικότητα κινασών Janus και είναι χρήσιμες στη θεραπευτική αγωγή νόσων που σχετίζονται με τη δραστικότητα κινασών Janus συμπεριλαμβανομένων, για παράδειγμα, ανοσοσχετιζόμενων νόσων, δερματικών διαταραχών, μυελοειδών βλαστικών διαταραχών, καρκίνου, και άλλων νόσων.The present invention provides heteroaryl substituted pyrrolo [2,3-b] pyridines (I) and heteroaryl substituted pyrrolo [2,3-b] pyrimidines that modulate Janus kinase activity and are useful in the treatment of Janus activity-related diseases including, for example, immunosuppressive diseases, skin disorders, myeloid stem cells, cancer, and other diseases.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US74990505A | 2005-12-13 | 2005-12-13 | |
US81023106A | 2006-06-02 | 2006-06-02 | |
US85062506A | 2006-10-10 | 2006-10-10 | |
US85687206A | 2006-11-03 | 2006-11-03 | |
US85940406A | 2006-11-16 | 2006-11-16 | |
EP11152677.8A EP2343299B9 (en) | 2005-12-13 | 2006-12-12 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1117389T1 true CY1117389T1 (en) | 2017-04-26 |
Family
ID=58606651
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20161100097T CY1117389T1 (en) | 2005-12-13 | 2016-02-03 | HYDROSYL-SUBSTITUTED PYROLID [2,3-b] PYRIDINES AND PYROLID [2,3-b] PYRAMIDINES AS JANUS MOVEMENTS |
Country Status (2)
Country | Link |
---|---|
CY (1) | CY1117389T1 (en) |
HK (1) | HK1168090A1 (en) |
-
2012
- 2012-09-06 HK HK12108719.9A patent/HK1168090A1/en unknown
-
2016
- 2016-02-03 CY CY20161100097T patent/CY1117389T1/en unknown
Also Published As
Publication number | Publication date |
---|---|
HK1168090A1 (en) | 2012-12-21 |
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