CY1116277T1 - METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS - Google Patents
METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPASInfo
- Publication number
- CY1116277T1 CY1116277T1 CY20151100244T CY151100244T CY1116277T1 CY 1116277 T1 CY1116277 T1 CY 1116277T1 CY 20151100244 T CY20151100244 T CY 20151100244T CY 151100244 T CY151100244 T CY 151100244T CY 1116277 T1 CY1116277 T1 CY 1116277T1
- Authority
- CY
- Cyprus
- Prior art keywords
- preparation
- kaspas
- aspalo
- asparatic
- intermediates
- Prior art date
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Η εφεύρεση αφορά σε μεθόδους όπως αυτές που δείχνονται στο σχήμα και ενώσεις χρήσιμες για παρασκευή τροποποιημένων παραγώγων ασπαρτικού οξέος, όπως χαρακτηριστικών ομάδων αλδεϋδης ασπαρτικού οξέος. Παράγωγα ασπαρτικού οξέος είναι χρήσιμα για παρασκευή αναστολέων κασπάσης ή/και προφαρμάκων αυτών.The invention relates to methods such as those shown in the figure and compounds useful for the preparation of modified aspartic acid derivatives, such as aldehyde aspartic acid moieties. Aspartic acid derivatives are useful for the preparation of caspase inhibitors and / or prodrugs thereof.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US55248004A | 2004-03-12 | 2004-03-12 | |
EP11178126.6A EP2399915B1 (en) | 2004-03-12 | 2005-03-11 | Process and intermediates for the preparation of aspartic acetal caspase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1116277T1 true CY1116277T1 (en) | 2017-02-08 |
Family
ID=58457916
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20151100232T CY1116276T1 (en) | 2004-03-12 | 2015-03-06 | METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS |
CY20151100244T CY1116277T1 (en) | 2004-03-12 | 2015-03-12 | METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS |
CY20151100245T CY1116278T1 (en) | 2004-03-12 | 2015-03-12 | METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20151100232T CY1116276T1 (en) | 2004-03-12 | 2015-03-06 | METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20151100245T CY1116278T1 (en) | 2004-03-12 | 2015-03-12 | METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS |
Country Status (1)
Country | Link |
---|---|
CY (3) | CY1116276T1 (en) |
-
2015
- 2015-03-06 CY CY20151100232T patent/CY1116276T1/en unknown
- 2015-03-12 CY CY20151100244T patent/CY1116277T1/en unknown
- 2015-03-12 CY CY20151100245T patent/CY1116278T1/en unknown
Also Published As
Publication number | Publication date |
---|---|
CY1116276T1 (en) | 2017-02-08 |
CY1116278T1 (en) | 2017-02-08 |
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