CY1116277T1 - METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS - Google Patents

METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS

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Publication number
CY1116277T1
CY1116277T1 CY20151100244T CY151100244T CY1116277T1 CY 1116277 T1 CY1116277 T1 CY 1116277T1 CY 20151100244 T CY20151100244 T CY 20151100244T CY 151100244 T CY151100244 T CY 151100244T CY 1116277 T1 CY1116277 T1 CY 1116277T1
Authority
CY
Cyprus
Prior art keywords
preparation
kaspas
aspalo
asparatic
intermediates
Prior art date
Application number
CY20151100244T
Other languages
Greek (el)
Inventor
Gerald J Tanoury
Minzhang Chen
Andrew D Jones
Philip L Nyce
Martin Trudeau
David J Guerin
John R Snoonian
Original Assignee
Vertex Pharmaceuticals Incorporated
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP11178126.6A external-priority patent/EP2399915B1/en
Application filed by Vertex Pharmaceuticals Incorporated filed Critical Vertex Pharmaceuticals Incorporated
Publication of CY1116277T1 publication Critical patent/CY1116277T1/en

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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Η εφεύρεση αφορά σε μεθόδους όπως αυτές που δείχνονται στο σχήμα και ενώσεις χρήσιμες για παρασκευή τροποποιημένων παραγώγων ασπαρτικού οξέος, όπως χαρακτηριστικών ομάδων αλδεϋδης ασπαρτικού οξέος. Παράγωγα ασπαρτικού οξέος είναι χρήσιμα για παρασκευή αναστολέων κασπάσης ή/και προφαρμάκων αυτών.The invention relates to methods such as those shown in the figure and compounds useful for the preparation of modified aspartic acid derivatives, such as aldehyde aspartic acid moieties. Aspartic acid derivatives are useful for the preparation of caspase inhibitors and / or prodrugs thereof.

CY20151100244T 2004-03-12 2015-03-12 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS CY1116277T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55248004A 2004-03-12 2004-03-12
EP11178126.6A EP2399915B1 (en) 2004-03-12 2005-03-11 Process and intermediates for the preparation of aspartic acetal caspase inhibitors

Publications (1)

Publication Number Publication Date
CY1116277T1 true CY1116277T1 (en) 2017-02-08

Family

ID=58457916

Family Applications (3)

Application Number Title Priority Date Filing Date
CY20151100232T CY1116276T1 (en) 2004-03-12 2015-03-06 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS
CY20151100244T CY1116277T1 (en) 2004-03-12 2015-03-12 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARATIC, ASPALO KASPAS
CY20151100245T CY1116278T1 (en) 2004-03-12 2015-03-12 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CY20151100232T CY1116276T1 (en) 2004-03-12 2015-03-06 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY20151100245T CY1116278T1 (en) 2004-03-12 2015-03-12 METHOD AND INTERMEDIATES FOR THE PREPARATION OF ACUTE ASPARTIC, CASPASE SUSPENSIONS

Country Status (1)

Country Link
CY (3) CY1116276T1 (en)

Also Published As

Publication number Publication date
CY1116276T1 (en) 2017-02-08
CY1116278T1 (en) 2017-02-08

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