CY1115616T1 - PREPARATION AND THERAPEUTIC APPLICATIONS OF (2S, 3R) N-2 ((3-PYDYNYL) Methyl) -1-Azadicyclo [2.2.2] OCT-3-Yl) -3,5-difluorobenzuamide - Google Patents

PREPARATION AND THERAPEUTIC APPLICATIONS OF (2S, 3R) N-2 ((3-PYDYNYL) Methyl) -1-Azadicyclo [2.2.2] OCT-3-Yl) -3,5-difluorobenzuamide

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Publication number
CY1115616T1
CY1115616T1 CY20141100590T CY141100590T CY1115616T1 CY 1115616 T1 CY1115616 T1 CY 1115616T1 CY 20141100590 T CY20141100590 T CY 20141100590T CY 141100590 T CY141100590 T CY 141100590T CY 1115616 T1 CY1115616 T1 CY 1115616T1
Authority
CY
Cyprus
Prior art keywords
preparation
compounds
pydynyl
difluorobenzuamide
azadicyclo
Prior art date
Application number
CY20141100590T
Other languages
Greek (el)
Inventor
Merouane Bencherif
Nikolai Fedorov
Terry Hauser
Kristen Jordan
Sharon Rae Letchworth
Anatoly Mazurov
Julio A Munoz
Jason Speake
Daniel Yohannes
Original Assignee
Targacept, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP20100701307 external-priority patent/EP2389378B1/en
Application filed by Targacept, Inc. filed Critical Targacept, Inc.
Publication of CY1115616T1 publication Critical patent/CY1115616T1/en

Links

Abstract

Η παρούσα εφεύρεση σχετίζεται με ενώσεις που δεσμεύονται και τροποποιούν την δραστηριότητα των νευρωνικών νικοτινικών υποδοχέων ακετυλχολίνης, με διεργασίες για την παρασκευή αυτών των ενώσεων, με φαρμακευτικές συνθέσεις περιέχοντας αυτές τις ενώσεις και με μεθόδους χρήσης αυτών των ενώσεων για την αγωγή μιας ευρείας ποικιλίας καταστάσεων και διαταραχών, συμπεριλαμβάνοντας εκείνες που συσχετίζονται με δυσλειτουργία του κεντρικού νευρικού συστήματος (ΚΝΣ).The present invention relates to compounds that bind and modify the activity of neuronal nicotinic acetylcholine receptors, processes for the preparation of these compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds for the treatment of a wide variety of conditions and conditions. , including those associated with central nervous system (CNS) dysfunction.

CY20141100590T 2009-01-26 2014-08-04 PREPARATION AND THERAPEUTIC APPLICATIONS OF (2S, 3R) N-2 ((3-PYDYNYL) Methyl) -1-Azadicyclo [2.2.2] OCT-3-Yl) -3,5-difluorobenzuamide CY1115616T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14726009A 2009-01-26 2009-01-26
EP20100701307 EP2389378B1 (en) 2009-01-26 2010-01-25 Preparation and therapeutic applications of (2s,3r)-n-2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)-3,5-difluorobenzamide

Publications (1)

Publication Number Publication Date
CY1115616T1 true CY1115616T1 (en) 2017-01-04

Family

ID=58461587

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20141100590T CY1115616T1 (en) 2009-01-26 2014-08-04 PREPARATION AND THERAPEUTIC APPLICATIONS OF (2S, 3R) N-2 ((3-PYDYNYL) Methyl) -1-Azadicyclo [2.2.2] OCT-3-Yl) -3,5-difluorobenzuamide

Country Status (1)

Country Link
CY (1) CY1115616T1 (en)

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