CY1115143T1 - CRYSTALS CONTAINING APPROPRIATE SALT OF N- [2- (DIETHYLAMINE) SAME] -5 - [(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-indol-3-indol-3-indol) DIMETHYL-1H-PYRROLO-3-CARBOXAMIDE, PREPARATION PROCEDURES FOR THESE AND THEIR COMPOSITIONS - Google Patents

CRYSTALS CONTAINING APPROPRIATE SALT OF N- [2- (DIETHYLAMINE) SAME] -5 - [(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-indol-3-indol-3-indol) DIMETHYL-1H-PYRROLO-3-CARBOXAMIDE, PREPARATION PROCEDURES FOR THESE AND THEIR COMPOSITIONS

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Publication number
CY1115143T1
CY1115143T1 CY20141100219T CY141100219T CY1115143T1 CY 1115143 T1 CY1115143 T1 CY 1115143T1 CY 20141100219 T CY20141100219 T CY 20141100219T CY 141100219 T CY141100219 T CY 141100219T CY 1115143 T1 CY1115143 T1 CY 1115143T1
Authority
CY
Cyprus
Prior art keywords
indol
pyrrolo
carboxamide
dihydro
oxo
Prior art date
Application number
CY20141100219T
Other languages
Greek (el)
Inventor
Michael Hawley
Thomas J Fleck
Stephen P Prescott
Mark T Maloney
Original Assignee
Pharmacia & Upjohn Company Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP02759342.5A external-priority patent/EP1419151B1/en
Application filed by Pharmacia & Upjohn Company Llc filed Critical Pharmacia & Upjohn Company Llc
Publication of CY1115143T1 publication Critical patent/CY1115143T1/en

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  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει κρυστάλλους, και συνθέσεις αυτών, όπου οι κρύσταλλοι περιλαμβάνουν ένα μηλικό άλας του Ν-[2-(διαιθυλαμινο)αιθυλο]-5-[(5-φθορο-1,2-διϋδρο-2-οξο-3Η-ινδολ-3-ιλιδενο)μεθυλο]-2,4-διμεθυλο-1Η-πυρρολο-3-καρβοξαμιδιου. Επίσης φέρονται στο προσκήνιο μέθοδοι παρασκευής τέτοιων κρυστάλλων.The present invention provides crystals, and compositions thereof, wherein the crystals comprise a maleic salt of N- [2- (diethylamino) ethyl] -5 - [(5-fluoro-1,2-dihydro-2-oxo-3H-indole) -3-ilideno) methyl] -2,4-dimethyl-1H-pyrrolo-3-carboxamide. Methods for preparing such crystals are also brought to the fore.

CY20141100219T 2001-08-15 2014-03-21 CRYSTALS CONTAINING APPROPRIATE SALT OF N- [2- (DIETHYLAMINE) SAME] -5 - [(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-indol-3-indol-3-indol) DIMETHYL-1H-PYRROLO-3-CARBOXAMIDE, PREPARATION PROCEDURES FOR THESE AND THEIR COMPOSITIONS CY1115143T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31235301A 2001-08-15 2001-08-15
EP02759342.5A EP1419151B1 (en) 2001-08-15 2002-08-13 Chrystals including a malic acid salt of n-[2-(diethylamino)ethyl] -5-[(5-fluoro-1,2-dihydro-2-oxo-3h-indole-3-ylidene)methyl] -2,4-dimethyl-1h-pyrrole-3-carboxamide, processes for its preparation and compositions thereof

Publications (1)

Publication Number Publication Date
CY1115143T1 true CY1115143T1 (en) 2016-12-14

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CY20141100219T CY1115143T1 (en) 2001-08-15 2014-03-21 CRYSTALS CONTAINING APPROPRIATE SALT OF N- [2- (DIETHYLAMINE) SAME] -5 - [(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-indol-3-indol-3-indol) DIMETHYL-1H-PYRROLO-3-CARBOXAMIDE, PREPARATION PROCEDURES FOR THESE AND THEIR COMPOSITIONS

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CY (1) CY1115143T1 (en)

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