CY1113762T1 - TOSSULIC SALT OF A THERAPEUTIC UNION AND ITS PHARMACEUTICAL COMPOSITIONS - Google Patents

TOSSULIC SALT OF A THERAPEUTIC UNION AND ITS PHARMACEUTICAL COMPOSITIONS

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Publication number
CY1113762T1
CY1113762T1 CY20121101105T CY121101105T CY1113762T1 CY 1113762 T1 CY1113762 T1 CY 1113762T1 CY 20121101105 T CY20121101105 T CY 20121101105T CY 121101105 T CY121101105 T CY 121101105T CY 1113762 T1 CY1113762 T1 CY 1113762T1
Authority
CY
Cyprus
Prior art keywords
disorders
congestion
pharmaceutical compositions
allergies
fluoro
Prior art date
Application number
CY20121101105T
Other languages
Greek (el)
Inventor
Travis T Wager
Todd William Butler
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP08702250A external-priority patent/EP2124933B1/en
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of CY1113762T1 publication Critical patent/CY1113762T1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση αφορά στο τοσυλικό άλας του trans-Ν-αιθυλ-3-φθορο-3-[3-φθορο-4-(πυρρολιδιν-1-υλμεθυλ)-φαινυλ]-κυκλοβουτανοκαρβοξαμιδίου (1): σε επιδιαλυτωμένα άλατα (π.χ. υδρίτες) αυτού, σε πολύμορφα αυτού, σε φαρμακευτικές συνθέσεις αυτού και σε μια μέθοδο θεραπείας της κατάθλιψης, διαταραχών της διάθεσης, σχιζοφρένειας, διαταραχών άγχους, νοητικών διαταραχών, της νόσου του Alzheimer, της διαταραχής ελλειμματικής προσοχής (ADD), του ελλείμματος προσοχής υπερκινητικότητας (ADHD) , ψυχωτικών διαταραχών, διαταραχών του ύπνου, παχυσαρκίας, ζάλης, επιληψίας, ναυτίας, αναπνευστικών ασθενειών, αλλεργίας, αποκρίσεις των αεραγωγών που προκαλούνται από αλλεργίες, αλλεργικής ρινίτιδας, ρινικής συμφόρησης, αλλεργικής συμφόρησης, συμφόρησης, υπότασης, καρδιαγγειακής νόσου, ασθενειών του γαστρεντερικού σωλήνα, υπερ- και υπο-κινητικότητας και όξινης έκκρισης του γαστρεντερικού σωλήνα, η οποία περιλαμβάνει την χορήγηση μιας θεραπευτικά αποτελεσματικής ποσότητας αυτών.The present invention relates to the tosylate of trans-N-ethyl-3-fluoro-3- [3-fluoro-4- (pyrrolidin-1-ylmethyl) -phenyl] -cyclobutanecarboxamide (1): in solvates (e.g. hydrates), polymorphs, pharmaceutical compositions, and a method of treating depression, mood disorders, schizophrenia, anxiety disorders, mental disorders, Alzheimer's disease, Attention Deficit Disorder (ADD), Attention Deficit Hyperactivity Disorder (ADHD), psychotic disorders, sleep disorders, obesity, dizziness, epilepsy, n cause, respiratory diseases, allergies, airway responses caused by allergies, allergic rhinitis, nasal congestion, allergic congestion, congestion, hypotension, cardiovascular disease, gastrointestinal tract diseases, hypertriglyceridemia and hypoxicemia which comprises administering a therapeutically effective amount thereof.

CY20121101105T 2007-01-22 2012-11-16 TOSSULIC SALT OF A THERAPEUTIC UNION AND ITS PHARMACEUTICAL COMPOSITIONS CY1113762T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88593107A 2007-01-22 2007-01-22
EP08702250A EP2124933B1 (en) 2007-01-22 2008-01-10 Tosylate salt of a therapeutic compound and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
CY1113762T1 true CY1113762T1 (en) 2016-07-27

Family

ID=57102335

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121101105T CY1113762T1 (en) 2007-01-22 2012-11-16 TOSSULIC SALT OF A THERAPEUTIC UNION AND ITS PHARMACEUTICAL COMPOSITIONS

Country Status (1)

Country Link
CY (1) CY1113762T1 (en)

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