CU23596A3 - DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION - Google Patents

DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION

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Publication number
CU23596A3
CU23596A3 CU20050228A CU20050228A CU23596A3 CU 23596 A3 CU23596 A3 CU 23596A3 CU 20050228 A CU20050228 A CU 20050228A CU 20050228 A CU20050228 A CU 20050228A CU 23596 A3 CU23596 A3 CU 23596A3
Authority
CU
Cuba
Prior art keywords
preparation
derivatives
quinazolina
pirazol
depirazolo
Prior art date
Application number
CU20050228A
Other languages
Spanish (es)
Inventor
Gabriella Traquandi
Daniele Fancelli
Paola Vianello
Ron Ferguson
Francesca Quartieri
Achille Panzeri
Fulvia Roletto
Paolo Polucci
Roberto D'alessio
Paolo Pevarello
Anna Vulpetti
Maria Gabriella Brasca
Original Assignee
Pharmacia Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Italia Spa filed Critical Pharmacia Italia Spa
Priority to CU20050228A priority Critical patent/CU23596A3/en
Publication of CU23596A3 publication Critical patent/CU23596A3/en

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Abstract

Se revelan derivados depirazolo-quinazolina de fórmula (Ia) o (Ib) como se definen en la memoria y sales farmacéuticamente aceptables de los mismos, un procedimiento para su preparación y composiciones farmacéuticas que los comprenden; los compuestos de la invención pueden ser útiles, en terapéutica, en el tratamiento de enfermedades asociadas con una actividad desregulada de la proteína quinasa, como cáncer.Depirazolo-quinazoline derivatives of formula (Ia) or (Ib) are disclosed as defined herein and pharmaceutically acceptable salts thereof, a process for their preparation and pharmaceutical compositions comprising them; The compounds of the invention may be useful, in therapeutics, in the treatment of diseases associated with a deregulated protein kinase activity, such as cancer.

CU20050228A 2005-11-21 2005-11-21 DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION CU23596A3 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20050228A CU23596A3 (en) 2005-11-21 2005-11-21 DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20050228A CU23596A3 (en) 2005-11-21 2005-11-21 DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION

Publications (1)

Publication Number Publication Date
CU23596A3 true CU23596A3 (en) 2010-11-11

Family

ID=43302733

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20050228A CU23596A3 (en) 2005-11-21 2005-11-21 DERIVATIVES OF PIRAZOL-QUINAZOLINA AND PROCESS FOR PREPARATION

Country Status (1)

Country Link
CU (1) CU23596A3 (en)

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