CU20100110A7 - NEW AGONISTS OF GLUCOCORTICOID RECEPTORS - Google Patents

NEW AGONISTS OF GLUCOCORTICOID RECEPTORS

Info

Publication number
CU20100110A7
CU20100110A7 CU20100110A CU20100110A CU20100110A7 CU 20100110 A7 CU20100110 A7 CU 20100110A7 CU 20100110 A CU20100110 A CU 20100110A CU 20100110 A CU20100110 A CU 20100110A CU 20100110 A7 CU20100110 A7 CU 20100110A7
Authority
CU
Cuba
Prior art keywords
glucocorticoid receptors
new agonists
formula
relates
present
Prior art date
Application number
CU20100110A
Other languages
Spanish (es)
Inventor
David Simon Millan
Paul Alan Glossop
David Anthony Price
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Priority to CU20100110A priority Critical patent/CU20100110A7/en
Publication of CU20100110A7 publication Critical patent/CU20100110A7/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a agonistas novedosos del receptor de glucocorticoides de la fórmula (I): ESPACIO PARA LA FÓRMULA y a procedimientos e intermedios para su preparación. La presente invención también se refiere a composiciones farmacéuticas que contienen estos compuestos, a su combinación con otro u otros agentes terapéuticos, así como a su uso para el tratamiento de un número de enfermedades, trastornos y afecciones inflamatorias y alérgicos.The present invention relates to novel glucocorticoid receptor agonists of the formula (I): SPACE FOR FORMULA and procedures and intermediates for its preparation. The present invention also relates to pharmaceutical compositions containing these compounds, their combination with another or other therapeutic agents, as well as their use for the treatment of a number of inflammatory and allergic diseases, disorders and conditions.

CU20100110A 2010-05-28 2010-05-28 NEW AGONISTS OF GLUCOCORTICOID RECEPTORS CU20100110A7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20100110A CU20100110A7 (en) 2010-05-28 2010-05-28 NEW AGONISTS OF GLUCOCORTICOID RECEPTORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20100110A CU20100110A7 (en) 2010-05-28 2010-05-28 NEW AGONISTS OF GLUCOCORTICOID RECEPTORS

Publications (1)

Publication Number Publication Date
CU20100110A7 true CU20100110A7 (en) 2011-10-14

Family

ID=45000093

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20100110A CU20100110A7 (en) 2010-05-28 2010-05-28 NEW AGONISTS OF GLUCOCORTICOID RECEPTORS

Country Status (1)

Country Link
CU (1) CU20100110A7 (en)

Similar Documents

Publication Publication Date Title
ECSP10010209A (en) NEW AGONISTS OF GLUCOCORTICOID RECEPTORS
CU20170144A7 (en) TETRAHYDROQUINOLINONE SUBSTITUTED COMPOUNDS AS GAMMA ROR MODULATORS
UY35177A (en) NEWS DERIVED FROM BENCIMIDAZOL AS ANTAGONISTS OF EP4
GT201200201A (en) POSITIVE ALOSTERIC MODULATORS OF M1 QUINOLINE RECEPTORS
SV2011003802A (en) USEFUL TRIAZOL DERIVATIVES FOR THE TREATMENT OF DISEASES
ECSP11011517A (en) ANTIVIRAL COMPOUNDS
UY32675A (en) NEW GLUCOCORTICOID RECEPTOR AGONISTS
CR10489A (en) PHENYL-PIRAZOL DERIVATIVES AS LEGANDS OF NON-STEROID GLUCOCORTICOID RECEPTORS
CO6640327A2 (en) Pyrazole compounds as sigma receptor inhibitors
UY30572A1 (en) N- (1-FTALAZIN-1-IL-PIPERIDIN-4-IL) -AMIDAS AS MODULATORS OF THE EP2 RECEIVER
UY33238A (en) "Compounds as bradykinin-b1 antagonists"
UY32167A (en) NEW DERIVATIVES OF 2-AMIDOTIADIAZOL
UY35906A (en) NEWS DERIVED FROM BENCIMIDAZOL AS LIGANDOS OF EP4
ECSP13012600A (en) CO-crystals and salts of CCR3 inhibitors
ECSP14002542A (en) NOVEL 2HINDAZOLES AS EP2 RECEPTOR ANTAGONISTS
CU20200067A7 (en) IMIDAZOLIDIN-2-ONA DERIVATIVES REPLACED AS PRMT5 INHIBITORS
UY32744A (en) DERIVATIVES OF 2-CARBOXAMIDA-7-PIPERAZINIL-BENZOFURANO 774
UY33230A (en) AMINOTIAZOLONAS AS MODULATORS OF THE ALFA RECEIVER RELATED TO ESTROGEN
CO2021001174A2 (en) Ckd8 / 19 inhibitors
CU20100110A7 (en) NEW AGONISTS OF GLUCOCORTICOID RECEPTORS
UY32718A (en) COMPOUNDS DERIVED FROM 1, 3, 4-TIADIAZOL, USEFUL AS ASPHONOSINE RECEPTOR AGONISTS 1-PHOSPHATE
UA95861C2 (en) Glucocorticoid receptor agonists
CU20080116A7 (en) 3-AMINOCICLOPENTANOCARBOXAMIDS AS MUDULATORS OF CHEMIOKIN RECEPTORS
CU23564A3 (en) CARBOXAMIDE DERIVATIVES AS ANTAGONISTS OF THE MUSCARINIC RECEIVER
CU20110002A7 (en) USEFUL TRIAZOL DERIVATIVES FOR THE TREATMENT OF DISEASES