CU20090035A7 - BENZOXAZOLES AND OXAZOLOPIRIDINS THAT ARE USEFUL AS INHIBITORS OF JANUS KINASES - Google Patents
BENZOXAZOLES AND OXAZOLOPIRIDINS THAT ARE USEFUL AS INHIBITORS OF JANUS KINASESInfo
- Publication number
- CU20090035A7 CU20090035A7 CU20090035A CU20090035A CU20090035A7 CU 20090035 A7 CU20090035 A7 CU 20090035A7 CU 20090035 A CU20090035 A CU 20090035A CU 20090035 A CU20090035 A CU 20090035A CU 20090035 A7 CU20090035 A7 CU 20090035A7
- Authority
- CU
- Cuba
- Prior art keywords
- treatment
- disease
- compounds
- formula
- oxazolopiridins
- Prior art date
Links
Abstract
La invención se refiere a compuestos de benzoxazol 2,7-disustituido y oxazolo-[5,4-c]-piridina 2,4-disustituida de la fórmula I que se da más adelante, así como a sales de los mismos, a procesos para su preparación, a la aplicación de los mismos en un proceso para el tratamiento del cuerpo humano o animal, estos compuestos para utilizarse en el tratamiento (incluyendo profilaxis) del cuerpo del animal, en especial humano (especialmente con respecto a una enfermedad proliferativa), el uso de los mismos- solos o en combinación con uno o más compuestos farmacéuticamente activos diferentes- para el tratamiento en especial de una enfermedad mediada por la cinasa de proteína tirosina (tal como una enfermedad tumoral) o para la fabricación de una preparación farmacéutica para utilizarse en el tratamiento de esta enfermedad, un método para el tratamiento de esta enfermedad y una preparación farmacéutica para el tratamiento de una enfermedad como se menciona. Los compuestos son de la fórmula I: ESPACIO PARA FÓRMULA en donde los símbolos son como se definen en la descripción. Los compuestos inhiben, por ejemplo, JAK2 y JAK3.The invention relates to 2,7-disubstituted benzoxazole and 2,4-disubstituted oxazolo- [5,4-c] -pyridine compounds of the formula I given below, as well as salts thereof, to processes for their preparation, to the application thereof in a process for the treatment of the human or animal body, these compounds for use in the treatment (including prophylaxis) of the animal's body, especially human (especially with respect to a proliferative disease) , the use thereof - alone or in combination with one or more other pharmaceutically active compounds - for the treatment in particular of a tyrosine protein kinase mediated disease (such as a tumor disease) or for the manufacture of a pharmaceutical preparation to be used in the treatment of this disease, a method for the treatment of this disease and a pharmaceutical preparation for the treatment of a disease as mentioned. The compounds are of the formula I: FORMULA SPACE where the symbols are as defined in the description. The compounds inhibit, for example, JAK2 and JAK3.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CU20090035A CU20090035A7 (en) | 2009-03-11 | 2009-03-11 | BENZOXAZOLES AND OXAZOLOPIRIDINS THAT ARE USEFUL AS INHIBITORS OF JANUS KINASES |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CU20090035A CU20090035A7 (en) | 2009-03-11 | 2009-03-11 | BENZOXAZOLES AND OXAZOLOPIRIDINS THAT ARE USEFUL AS INHIBITORS OF JANUS KINASES |
Publications (1)
Publication Number | Publication Date |
---|---|
CU20090035A7 true CU20090035A7 (en) | 2011-03-21 |
Family
ID=44280884
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CU20090035A CU20090035A7 (en) | 2009-03-11 | 2009-03-11 | BENZOXAZOLES AND OXAZOLOPIRIDINS THAT ARE USEFUL AS INHIBITORS OF JANUS KINASES |
Country Status (1)
Country | Link |
---|---|
CU (1) | CU20090035A7 (en) |
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2009
- 2009-03-11 CU CU20090035A patent/CU20090035A7/en unknown
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