CR9962A - ENZYMATIC INHIBITION COMPOUNDS - Google Patents
ENZYMATIC INHIBITION COMPOUNDSInfo
- Publication number
- CR9962A CR9962A CR9962A CR9962A CR9962A CR 9962 A CR9962 A CR 9962A CR 9962 A CR9962 A CR 9962A CR 9962 A CR9962 A CR 9962A CR 9962 A CR9962 A CR 9962A
- Authority
- CR
- Costa Rica
- Prior art keywords
- peptide
- based compounds
- enzymatic inhibition
- inhibition compounds
- ntn
- Prior art date
Links
Abstract
Compuestos basados en peptidos, incluyendo anillos de tres miembros que contienen heteroatomos, inhiben eficiente y selectivamente las actividades especificas de las hidrolasas de nucleofilos N-terminales (Ntn) asociadas al proteosoma. Los compuestos basados en peptidos incluyen un epoxido o aziridina y funcionalizacion en el extremo N. Entre otras utilidades terapeuticas, se espera que los compuestos basados en peptidos exhiban propiedades antiflamatorias e inhibicion de la proliferacion celular.Peptide-based compounds, including three-membered rings containing heteroatoms, efficiently and selectively inhibit the specific activities of N-terminal nucleophilic hydrolases (Ntn) associated with the proteasome. Peptide-based compounds include an epoxide or aziridine and functionalization at the N-terminus. Among other therapeutic utilities, peptide-based compounds are expected to exhibit anti-inflammatory properties and inhibition of cell proliferation.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US84258205P | 2005-09-05 | 2005-09-05 | |
US37611805P | 2005-11-09 | 2005-11-09 | |
CR20130545A CR20130545A (en) | 2005-09-05 | 2013-10-24 | COMPOUNDS FOR ENZYMATIC INHIBITION (PATENT DIVISIONAL 9962) |
Publications (1)
Publication Number | Publication Date |
---|---|
CR9962A true CR9962A (en) | 2008-10-17 |
Family
ID=44839428
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR9962A CR9962A (en) | 2005-09-05 | 2008-05-08 | ENZYMATIC INHIBITION COMPOUNDS |
CR20130545A CR20130545A (en) | 2005-09-05 | 2013-10-24 | COMPOUNDS FOR ENZYMATIC INHIBITION (PATENT DIVISIONAL 9962) |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR20130545A CR20130545A (en) | 2005-09-05 | 2013-10-24 | COMPOUNDS FOR ENZYMATIC INHIBITION (PATENT DIVISIONAL 9962) |
Country Status (1)
Country | Link |
---|---|
CR (2) | CR9962A (en) |
-
2008
- 2008-05-08 CR CR9962A patent/CR9962A/en unknown
-
2013
- 2013-10-24 CR CR20130545A patent/CR20130545A/en unknown
Also Published As
Publication number | Publication date |
---|---|
CR20130545A (en) | 2013-11-29 |
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