CR7729A - DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV - Google Patents
DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIVInfo
- Publication number
- CR7729A CR7729A CR7729A CR7729A CR7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A
- Authority
- CR
- Costa Rica
- Prior art keywords
- hiv
- modulators
- derivatives
- treatment
- dicianophenoxi
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Esta invencion se refiere a los derivados del pirazol de formula (I) y sal, solvato o derivados farmaceuticamente aceptables del mismo, a su uso en medicina , a composiciones que los contienen, a procedimientos para su preparacion y a intermedios usados en tales procedmientos.Los compuestos de la invencion se unen a la enzima transcriptasa inversa y son moduladores, en especial inhibidores, de la misma. La transcriptsa inversa esta involucrada en el ciclo vital infeccioso del Virus de la Inmunodeficiencia Humana (VIH). Los compuestos que afectan a la funcion de esta enzima han mostrado su utilidad en el tratamientop de afecciones ptrdocuiodas por el VIH y retrovirus geneticamente relacionados, tales como el Sindrome de Inmunodeficienia Adquirida (SIDA).This invention relates to pyrazole derivatives of formula (I) and salt, solvate or pharmaceutically acceptable derivatives thereof, their use in medicine, compositions containing them, processes for their preparation and intermediates used in such processes. Compounds of the invention bind to the enzyme reverse transcriptase and are modulators, especially inhibitors, thereof. Reverse transcripting is involved in the infectious life cycle of Human Immunodeficiency Virus (HIV). Compounds that affect the function of this enzyme have shown their usefulness in the treatment of HIV-related conditions and genetically related retroviruses, such as Acquired Immune Deficiency Syndrome (AIDS).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0221477.3A GB0221477D0 (en) | 2002-09-16 | 2002-09-16 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
CR7729A true CR7729A (en) | 2005-06-15 |
Family
ID=44839280
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR7729A CR7729A (en) | 2002-09-16 | 2005-03-10 | DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV |
Country Status (1)
Country | Link |
---|---|
CR (1) | CR7729A (en) |
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2005
- 2005-03-10 CR CR7729A patent/CR7729A/en not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
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FA | Abandonment or withdrawal (granting procedure) |