CR7729A - DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV - Google Patents

DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV

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Publication number
CR7729A
CR7729A CR7729A CR7729A CR7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A CR 7729 A CR7729 A CR 7729A
Authority
CR
Costa Rica
Prior art keywords
hiv
modulators
derivatives
treatment
dicianophenoxi
Prior art date
Application number
CR7729A
Other languages
Spanish (es)
Inventor
Eric Mowbray Charles
Anthony Price David
Duncan Selby Matthew
Anthony Stupple Paul
Original Assignee
Pfizer
Prestwick Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0221477.3A external-priority patent/GB0221477D0/en
Application filed by Pfizer, Prestwick Pharmaceuticals Inc filed Critical Pfizer
Publication of CR7729A publication Critical patent/CR7729A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Esta invencion se refiere a los derivados del pirazol de formula (I) y sal, solvato o derivados farmaceuticamente aceptables del mismo, a su uso en medicina , a composiciones que los contienen, a procedimientos para su preparacion y a intermedios usados en tales procedmientos.Los compuestos de la invencion se unen a la enzima transcriptasa inversa y son moduladores, en especial inhibidores, de la misma. La transcriptsa inversa esta involucrada en el ciclo vital infeccioso del Virus de la Inmunodeficiencia Humana (VIH). Los compuestos que afectan a la funcion de esta enzima han mostrado su utilidad en el tratamientop de afecciones ptrdocuiodas por el VIH y retrovirus geneticamente relacionados, tales como el Sindrome de Inmunodeficienia Adquirida (SIDA).This invention relates to pyrazole derivatives of formula (I) and salt, solvate or pharmaceutically acceptable derivatives thereof, their use in medicine, compositions containing them, processes for their preparation and intermediates used in such processes. Compounds of the invention bind to the enzyme reverse transcriptase and are modulators, especially inhibitors, thereof. Reverse transcripting is involved in the infectious life cycle of Human Immunodeficiency Virus (HIV). Compounds that affect the function of this enzyme have shown their usefulness in the treatment of HIV-related conditions and genetically related retroviruses, such as Acquired Immune Deficiency Syndrome (AIDS).

CR7729A 2002-09-16 2005-03-10 DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV CR7729A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0221477.3A GB0221477D0 (en) 2002-09-16 2002-09-16 Chemical compounds

Publications (1)

Publication Number Publication Date
CR7729A true CR7729A (en) 2005-06-15

Family

ID=44839280

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7729A CR7729A (en) 2002-09-16 2005-03-10 DERIVATIVES OF 4- (3,5-DICIANOPHENOXI) PIRAZOL FOR USE AS TRANSCRIPT MODULATORS IN THE TREATMENT, AMONG OTHERS, OF HIV

Country Status (1)

Country Link
CR (1) CR7729A (en)
  • 2005

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)