CR6999A - BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa - Google Patents

BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa

Info

Publication number
CR6999A
CR6999A CR6999A CR6999A CR6999A CR 6999 A CR6999 A CR 6999A CR 6999 A CR6999 A CR 6999A CR 6999 A CR6999 A CR 6999A CR 6999 A CR6999 A CR 6999A
Authority
CR
Costa Rica
Prior art keywords
compounds
cns
gabaa
piridilimidazol
ligandos
Prior art date
Application number
CR6999A
Other languages
Spanish (es)
Inventor
Li Guiying
M Peterson John
Albaugh Pamela
S Curie Kevin
M Gustavson Linda
Lee Kyungae
Hutchison Alan
Singh Vinod
D Maynard George
Yuan Jun
Xie Linghong
Ghosh Manuka
Liu Nian
P Luke George
Mitchell Scott
Patrick Allen Martin
Liras Spiros
Original Assignee
Neurogen Corp
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogen Corp, Pfizer filed Critical Neurogen Corp
Priority to CR6999A priority Critical patent/CR6999A/en
Publication of CR6999A publication Critical patent/CR6999A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La invencion esta particularmente relacionada con los compuestos que se adhieren con alta selectividad y alta afinidad al sitio benzodiazepina de los receptores GABAa. Esta invencion se refiere tambien a las composiciones farmaceuticas que comprenden dichos compuestos y al uso de dichos compuestos para el tratamiento de ciertas enfermedades del sistema nervioso central (CNS). Se describen nuevos procedimientos para preparar los compuestos de la Formula I. Se refiere tambien al uso de bencimidazoles, piridilimidazoles y compuestos heteroarilo biciclicos relacionados de la Formula I en combinacion con uno o mas de otros agentes del CNS para potenciar los efectos de los otros agentes CNS.The invention is particularly related to compounds that adhere with high selectivity and high affinity to the benzodiazepine site of GABAa receptors. This invention also relates to pharmaceutical compositions comprising said compounds and the use of said compounds for the treatment of certain diseases of the central nervous system (CNS). New methods are described for preparing the compounds of Formula I. It also refers to the use of benzimidazoles, pyridylimidazoles and related bicyclic heteroaryl compounds of Formula I in combination with one or more other CNS agents to enhance the effects of the other agents. CNS

CR6999A 2003-06-17 2003-06-17 BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa CR6999A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CR6999A CR6999A (en) 2003-06-17 2003-06-17 BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CR6999A CR6999A (en) 2003-06-17 2003-06-17 BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa

Publications (1)

Publication Number Publication Date
CR6999A true CR6999A (en) 2004-06-25

Family

ID=44839108

Family Applications (1)

Application Number Title Priority Date Filing Date
CR6999A CR6999A (en) 2003-06-17 2003-06-17 BENZIMIDAZOL AND PIRIDILIMIDAZOL DERIVATIVES AS LIGANDOS FOR GABAa

Country Status (1)

Country Link
CR (1) CR6999A (en)
  • 2003

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)