CR11776A - BACE INHIBITORS - Google Patents

BACE INHIBITORS

Info

Publication number
CR11776A
CR11776A CR11776A CR11776A CR11776A CR 11776 A CR11776 A CR 11776A CR 11776 A CR11776 A CR 11776A CR 11776 A CR11776 A CR 11776A CR 11776 A CR11776 A CR 11776A
Authority
CR
Costa Rica
Prior art keywords
bace inhibitors
methods
bace
inhibitors
intermediates
Prior art date
Application number
CR11776A
Other languages
Spanish (es)
Inventor
Edmund Audia James
James Mergott Dustin
Martin Sheehan Scott
Morgan Watson Brian
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40839645&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR11776(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CR11776A publication Critical patent/CR11776A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C07D279/06—1,3-Thiazines; Hydrogenated 1,3-thiazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

La presente invención se refiere a inhibidores de BACE de Fórmula I métodos para su uso, e intermediarios y métodos para su preparación.The present invention relates to BACE inhibitors of Formula I methods for their use, and intermediates and methods for their preparation.

CR11776A 2008-05-02 2010-11-02 BACE INHIBITORS CR11776A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4988108P 2008-05-02 2008-05-02

Publications (1)

Publication Number Publication Date
CR11776A true CR11776A (en) 2011-01-28

Family

ID=40839645

Family Applications (1)

Application Number Title Priority Date Filing Date
CR11776A CR11776A (en) 2008-05-02 2010-11-02 BACE INHIBITORS

Country Status (32)

Country Link
US (1) US7648983B2 (en)
EP (1) EP2297120B1 (en)
JP (3) JP5658139B2 (en)
KR (1) KR101253835B1 (en)
CN (1) CN102015667B (en)
AR (1) AR071187A1 (en)
AU (1) AU2009241515B2 (en)
CA (1) CA2723207C (en)
CL (1) CL2009000860A1 (en)
CO (1) CO6311079A2 (en)
CR (1) CR11776A (en)
DK (1) DK2297120T3 (en)
DO (1) DOP2010000328A (en)
EA (1) EA016955B1 (en)
EC (1) ECSP10010582A (en)
ES (1) ES2549087T3 (en)
HR (1) HRP20150941T1 (en)
HU (1) HUE025520T2 (en)
IL (1) IL208350A (en)
MA (1) MA32351B1 (en)
MX (1) MX2010011972A (en)
NZ (1) NZ588300A (en)
PE (1) PE20091816A1 (en)
PL (1) PL2297120T3 (en)
PT (1) PT2297120E (en)
RS (1) RS54260B1 (en)
SI (1) SI2297120T1 (en)
SV (1) SV2010003718A (en)
TW (1) TWI431004B (en)
UA (1) UA102251C2 (en)
WO (1) WO2009134617A1 (en)
ZA (1) ZA201006868B (en)

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Also Published As

Publication number Publication date
AU2009241515B2 (en) 2012-04-19
CL2009000860A1 (en) 2010-05-07
CA2723207A1 (en) 2009-11-05
HRP20150941T1 (en) 2015-10-09
EP2297120B1 (en) 2015-08-19
WO2009134617A1 (en) 2009-11-05
TW200946522A (en) 2009-11-16
JP2011519854A (en) 2011-07-14
RS54260B1 (en) 2016-02-29
JP5658139B2 (en) 2015-01-21
PT2297120E (en) 2015-10-26
EA016955B1 (en) 2012-08-30
CA2723207C (en) 2016-07-12
PL2297120T3 (en) 2016-01-29
IL208350A (en) 2014-05-28
PE20091816A1 (en) 2009-11-25
US20090275566A1 (en) 2009-11-05
IL208350A0 (en) 2010-12-30
US7648983B2 (en) 2010-01-19
EP2297120A1 (en) 2011-03-23
AR071187A1 (en) 2010-06-02
SI2297120T1 (en) 2015-11-30
UA102251C2 (en) 2013-06-25
SV2010003718A (en) 2011-02-14
ECSP10010582A (en) 2010-11-30
DOP2010000328A (en) 2010-11-15
AU2009241515A1 (en) 2009-11-05
KR101253835B1 (en) 2013-04-15
HUE025520T2 (en) 2016-02-29
CN102015667B (en) 2013-06-12
DK2297120T3 (en) 2015-10-12
MX2010011972A (en) 2010-11-25
JP2017048212A (en) 2017-03-09
ZA201006868B (en) 2012-03-28
JP2015051980A (en) 2015-03-19
CO6311079A2 (en) 2011-08-22
MA32351B1 (en) 2011-06-01
KR20100125475A (en) 2010-11-30
TWI431004B (en) 2014-03-21
CN102015667A (en) 2011-04-13
EA201071264A1 (en) 2011-04-29
NZ588300A (en) 2012-07-27
ES2549087T3 (en) 2015-10-22

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