CO5780122A1 - BECIMIDAZOL-, BENZTRIAZOL-, AND BENCIMIDAZOLONA-O-GUCOSIDOS REPLACED - Google Patents
BECIMIDAZOL-, BENZTRIAZOL-, AND BENCIMIDAZOLONA-O-GUCOSIDOS REPLACEDInfo
- Publication number
- CO5780122A1 CO5780122A1 CO06062524A CO06062524A CO5780122A1 CO 5780122 A1 CO5780122 A1 CO 5780122A1 CO 06062524 A CO06062524 A CO 06062524A CO 06062524 A CO06062524 A CO 06062524A CO 5780122 A1 CO5780122 A1 CO 5780122A1
- Authority
- CO
- Colombia
- Prior art keywords
- independently selected
- heteroatoms independently
- fused
- gucosidos
- bencimidazolona
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
? Un compuesto de formula (III): <EMI FILE="06062524_1" ID="1" IMF=JPEG HE=50 WI=50 >en donde: X es CH, N, o C=O; R1 es H o está ausente; R2 es H, F, CI, OCH3, OCH2CH3, alquilo de C1-4, CF3, SCH3, fenilo sustituido o no sustituido y NR3R4; R3 y R4 son H, alquilo de C1-6, o se toman junto con el átomo de nitrógeno al cual están unidos para formar un anillo heterocíclico de 5-6 miembros con opcionalmente 1-2 heteroátomos adicionales independientemente seleccionados a partir de O, S, y N; Q es -(CH2)n- en donde n es 1 ó 2; P es H, acilo de C2-7, o alcoxicarbonilo (de C1-6); y Z está sustituido o no sustituido, y se selecciona a partir de cicloalquilo de C3-7, fenilo, heteroarilo de 5 ó 6 miembros que tiene 1 ó 2 heteroátomos independientemente seleccionados a partir de N, O, y S, un biarilo, y un biciclilo fusionado o heterobiciclilo fusionado de 9 ó 10 miembros, en donde dicho heterobiciclilo fusionado tiene entre 1 y 4 heteroátomos independientemente seleccionados a partir de N, O, y S; o una sal farmacéuticamente aceptable, de los mismos.? A compound of formula (III): <EMI FILE = "06062524_1" ID = "1" MFI = JPEG HE = 50 WI = 50> where: X is CH, N, or C = O; R1 is H or is absent; R2 is H, F, CI, OCH3, OCH2CH3, C1-4 alkyl, CF3, SCH3, substituted or unsubstituted phenyl and NR3R4; R3 and R4 are H, C1-6 alkyl, or are taken together with the nitrogen atom to which they are attached to form a 5-6 membered heterocyclic ring with optionally 1-2 additional heteroatoms independently selected from O, S , and N; Q is - (CH2) n- where n is 1 or 2; P is H, C2-7 acyl, or (C1-6) alkoxycarbonyl; and Z is substituted or unsubstituted, and is selected from C 3-7 cycloalkyl, phenyl, 5- or 6-membered heteroaryl having 1 or 2 heteroatoms independently selected from N, O, and S, a biaryl, and a fused bicyclyl or fused 9 or 10 membered heterobicyclyl, wherein said fused heterobicyclyl has between 1 and 4 heteroatoms independently selected from N, O, and S; or a pharmaceutically acceptable salt thereof.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CO06062524A CO5780122A1 (en) | 2006-06-28 | 2006-06-28 | BECIMIDAZOL-, BENZTRIAZOL-, AND BENCIMIDAZOLONA-O-GUCOSIDOS REPLACED |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CO06062524A CO5780122A1 (en) | 2006-06-28 | 2006-06-28 | BECIMIDAZOL-, BENZTRIAZOL-, AND BENCIMIDAZOLONA-O-GUCOSIDOS REPLACED |
Publications (1)
Publication Number | Publication Date |
---|---|
CO5780122A1 true CO5780122A1 (en) | 2007-07-31 |
Family
ID=40973994
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO06062524A CO5780122A1 (en) | 2006-06-28 | 2006-06-28 | BECIMIDAZOL-, BENZTRIAZOL-, AND BENCIMIDAZOLONA-O-GUCOSIDOS REPLACED |
Country Status (1)
Country | Link |
---|---|
CO (1) | CO5780122A1 (en) |
-
2006
- 2006-06-28 CO CO06062524A patent/CO5780122A1/en not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC | Application refused |