CO5590920A2 - DERIVATIVES OF 4-AMINOPIRIMIDINA-5-ONA - Google Patents
DERIVATIVES OF 4-AMINOPIRIMIDINA-5-ONAInfo
- Publication number
- CO5590920A2 CO5590920A2 CO05070756A CO05070756A CO5590920A2 CO 5590920 A2 CO5590920 A2 CO 5590920A2 CO 05070756 A CO05070756 A CO 05070756A CO 05070756 A CO05070756 A CO 05070756A CO 5590920 A2 CO5590920 A2 CO 5590920A2
- Authority
- CO
- Colombia
- Prior art keywords
- lower alkyl
- substituted
- nr5r6
- heterocycle
- co2r12
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
1.- Un compuesto de la fórmula En dondeR1 se selecciona del grupo constituido porheterociclo y alquilo inferior-heterociclo, en donde la fracción heterociclo en ambos casos opcionalmente puedeestar sustituida por hasta cuatro sustituyentes independientemente seleccionados deH,alquilo inferior,alquilo inferior sustituido mediante oxo, OR12, CO2R12, NR5R6, S(O)nR15 o C(O)NR5R6, CO2R7,COR12,COR11,C(O)NR13R14,S(O)nR15,oxo,OR12, oNR5R6;arilo;arilo sustituido porH,-S(O)n-R15, NR5R6,carbonilo, carbonilo sustituido por alquilo inferior, OR12 ó NR5R6, alquilo inferior, alquilo inferior sustituido mediante OR10 ó NR5R6, OR", ohalógeno;cicloalquilo;cicloalquilo sustituido por OR7, NR5R6 ó S(O)nR15;alquilo inferior; yalquilo inferior sustituido por NR5R6,NR11SO2R15, CO2R10,S(O)nR15,heterociclo,heterociclo sustituido poralquilo inferior,CO2R12 óSO2R15,heteroarilo, ...1. A compound of the formula Where R 1 is selected from the group consisting of heterocycle and lower alkyl heterocycle, in which the heterocycle fraction in both cases may optionally be substituted by up to four substituents independently selected from H, lower alkyl, lower alkyl substituted by oxo, OR12, CO2R12, NR5R6, S (O) nR15 or C (O) NR5R6, CO2R7, COR12, COR11, C (O) NR13R14, S (O) nR15, oxo, OR12, oNR5R6; aryl; aryl substituted by H, -S (O) n-R15, NR5R6, carbonyl, carbonyl substituted by lower alkyl, OR12 or NR5R6, lower alkyl, lower alkyl substituted by OR10 or NR5R6, OR ", halogen; cycloalkyl; cycloalkyl substituted by OR7, NR5R6 or S (O) nR15; lower alkyl; lower alkyl substituted by NR5R6, NR11SO2R15, CO2R10, S (O) nR15, heterocycle, substituted heterocycle lower poralkyl, CO2R12 or SO2R15, heteroaryl, ...
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44627303P | 2003-02-10 | 2003-02-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO5590920A2 true CO5590920A2 (en) | 2005-12-30 |
Family
ID=38808947
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO05070756A CO5590920A2 (en) | 2003-02-10 | 2005-07-18 | DERIVATIVES OF 4-AMINOPIRIMIDINA-5-ONA |
Country Status (3)
| Country | Link |
|---|---|
| CN (1) | CN101044121A (en) |
| CO (1) | CO5590920A2 (en) |
| ZA (1) | ZA200505564B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104053442B (en) * | 2011-08-26 | 2017-06-23 | 润新生物公司 | Some chemical entities, composition and method |
| CN108299312B (en) * | 2018-03-29 | 2020-10-30 | 郑州大学第一附属医院 | Pyrimidine derivatives and application thereof in preparation of antitumor drugs |
| JP2024506039A (en) * | 2021-02-05 | 2024-02-08 | シャンハイ チールー ファーマシューティカル リサーチ アンド ディベロップメント センター リミテッド | CDK inhibitor |
-
2004
- 2004-02-03 CN CN 200480003929 patent/CN101044121A/en active Pending
-
2005
- 2005-07-11 ZA ZA200505564A patent/ZA200505564B/en unknown
- 2005-07-18 CO CO05070756A patent/CO5590920A2/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200505564B (en) | 2007-01-31 |
| CN101044121A (en) | 2007-09-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Application refused |