CO5180595A1 - TIAZOL POLICE SYSTEMS, PROCEDURE FOR THE PREPARATION AND MEDICINAL PRODUCT CONTAINING THESE COMPOUNDS - Google Patents

TIAZOL POLICE SYSTEMS, PROCEDURE FOR THE PREPARATION AND MEDICINAL PRODUCT CONTAINING THESE COMPOUNDS

Info

Publication number
CO5180595A1
CO5180595A1 CO00011822A CO00011822A CO5180595A1 CO 5180595 A1 CO5180595 A1 CO 5180595A1 CO 00011822 A CO00011822 A CO 00011822A CO 00011822 A CO00011822 A CO 00011822A CO 5180595 A1 CO5180595 A1 CO 5180595A1
Authority
CO
Colombia
Prior art keywords
compounds
preparation
tiazol
procedure
product containing
Prior art date
Application number
CO00011822A
Other languages
Spanish (es)
Inventor
Gerhard Jahne
Karl Geisen
Hans-Jochen Lang
Martin Bickel
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of CO5180595A1 publication Critical patent/CO5180595A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/84—Naphthothiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

The invention relates to polycyclic thiazole systems and their physiologically tolerated salts and physiologically functional derivatives.Compounds of the formula I,in which the radicals have the stated meanings, and their physiologically tolerated salts and processes for their preparation are described. The compounds are suitable, for example, as anorectics.
CO00011822A 1999-02-26 2000-02-21 TIAZOL POLICE SYSTEMS, PROCEDURE FOR THE PREPARATION AND MEDICINAL PRODUCT CONTAINING THESE COMPOUNDS CO5180595A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19908533A DE19908533A1 (en) 1999-02-26 1999-02-26 Polycyclic thiazole systems, processes for their preparation and medicaments containing these compounds

Publications (1)

Publication Number Publication Date
CO5180595A1 true CO5180595A1 (en) 2002-07-30

Family

ID=7899078

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00011822A CO5180595A1 (en) 1999-02-26 2000-02-21 TIAZOL POLICE SYSTEMS, PROCEDURE FOR THE PREPARATION AND MEDICINAL PRODUCT CONTAINING THESE COMPOUNDS

Country Status (18)

Country Link
US (1) US6187801B1 (en)
EP (1) EP1183247B1 (en)
JP (1) JP4728485B2 (en)
KR (1) KR20020000545A (en)
CN (1) CN1149205C (en)
AT (1) ATE296295T1 (en)
AU (1) AU762802B2 (en)
BR (1) BR0008511A (en)
CA (1) CA2364903A1 (en)
CO (1) CO5180595A1 (en)
DE (2) DE19908533A1 (en)
DK (1) DK1183247T3 (en)
ES (1) ES2241574T3 (en)
HK (1) HK1042300B (en)
PT (1) PT1183247E (en)
TW (1) TW593294B (en)
WO (1) WO2000051997A1 (en)
ZA (1) ZA200106440B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19908535A1 (en) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Use of polycyclic thiazole systems for the preparation of medicaments for the prophylaxis or treatment of obesity
AU4413601A (en) * 2000-02-26 2001-09-03 Aventis Pharma Gmbh 8,8a-dihydro-indeno(1,2-d)thiazole derivatives with a sulphonamido or sulphono substituent in the 2 position, a method for production thereof and use thereof as a medicament
DE10142663B4 (en) 2001-08-31 2004-08-19 Aventis Pharma Deutschland Gmbh C2-Disubstituted indan-1-ol systems
KR100712171B1 (en) * 2004-09-17 2007-05-02 김진우 Jointable pipeblock using abandoned tire
PL2276767T3 (en) 2008-03-31 2014-09-30 Genentech Inc Benzopyran and benzoxepin pi3k inhibitor compounds and methods of use
US8242104B2 (en) 2009-09-28 2012-08-14 F. Hoffman-La Roche Ag Benzoxazepin P13K inhibitor compounds and methods of use
AU2010299820A1 (en) * 2009-09-28 2012-04-19 F. Hoffmann-La Roche Ag Benzoxepin PI3K inhibitor compounds and methods of use
WO2012126901A1 (en) 2011-03-21 2012-09-27 F. Hoffmann-La Roche Ag Benzoxazepin compounds selective for pi3k p110 delta and methods of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2640358A1 (en) * 1976-09-08 1978-03-16 Hoechst Ag THIAZOLIDE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
US5834499A (en) * 1994-03-11 1998-11-10 Yamanouchi Pharmaceutical Co., Ltd. 5-HT3 receptor agonist, novel thiazole derivative and intermediate thereof
JPH1179993A (en) * 1997-09-05 1999-03-23 Sumitomo Pharmaceut Co Ltd Immunosuppressant
DE19831878C2 (en) * 1998-07-17 2001-05-17 Aventis Pharma Gmbh Polycyclic thiazolidin-2-ylidene amines, process for their preparation and their use as medicaments
DE19908535A1 (en) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Use of polycyclic thiazole systems for the preparation of medicaments for the prophylaxis or treatment of obesity

Also Published As

Publication number Publication date
ES2241574T3 (en) 2005-11-01
HK1042300A1 (en) 2002-08-09
CN1341108A (en) 2002-03-20
PT1183247E (en) 2005-07-29
EP1183247B1 (en) 2005-05-25
DK1183247T3 (en) 2005-09-19
EP1183247A1 (en) 2002-03-06
WO2000051997A1 (en) 2000-09-08
CA2364903A1 (en) 2000-09-08
HK1042300B (en) 2004-12-10
KR20020000545A (en) 2002-01-05
AU762802B2 (en) 2003-07-03
TW593294B (en) 2004-06-21
DE50010403D1 (en) 2005-06-30
ATE296295T1 (en) 2005-06-15
JP4728485B2 (en) 2011-07-20
ZA200106440B (en) 2002-03-06
US6187801B1 (en) 2001-02-13
JP2002538150A (en) 2002-11-12
AU2441600A (en) 2000-09-21
BR0008511A (en) 2002-04-02
CN1149205C (en) 2004-05-12
DE19908533A1 (en) 2000-08-31

Similar Documents

Publication Publication Date Title
AR021844A1 (en) ARIL-SUBSTITUTED PROPANOLAMINE DERIVATIVES, PROCEDURES FOR PREPARATION, MEDICATIONS CONTAINING THESE COMPOUNDS AND THEIR USE
JO2353B1 (en) Novel heterocyclic fluoroglycoside derivatives, medicaments containing these compounds, and the use thereof
BR0312513A (en) Thiophene glycoside derivatives, processes for their production, medicines containing these compounds and their use
BR0208338A (en) Pyridine Derivatives
UY27417A1 (en) AROMATIC BICYCLIC COMPOUNDS REPLACED WITH AMINO-RENT, PROCEDURE FOR PREPARATION AND USE AS A MEDICINAL PRODUCT
HRP20050531B1 (en) Novel aromatic fluoroglycoside derivatives, pharmaceutical products containing said compounds and the use thereof
AR029175A1 (en) 2-AMINO-PHENYLPURINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM, AND THE USE OF THEM FOR THE PREPARATION OF A MEDICINAL PRODUCT
SE9904505D0 (en) Novel compounds
CR9182A (en) DERIVATIVE OF QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT
AR021843A1 (en) DERIVATIVES OF PROPANOLAMINE SUBSTITUTED WITH HETEROCICLES, PROCEDURE FOR THEIR PREPARATION, AND ITS USE.
BR0109483A (en) Imidazopyridine Derivative Prodrugs
CO5180595A1 (en) TIAZOL POLICE SYSTEMS, PROCEDURE FOR THE PREPARATION AND MEDICINAL PRODUCT CONTAINING THESE COMPOUNDS
ID29025A (en) FENILALKENOILGUANIDINA-SUBSTITUTED EMPEDUIC ACID, PROCESSES FOR MAKING IT, USE IT AS A DRUG OR ANNNOSTIC AND DRUGS CONTAINING IT
BR0008510A (en) Polycyclic 2-amino-thiazole systems, process for their preparation and medicine containing these compounds
DK1173176T3 (en) Use of polycyclic 2-aminothiazole systems for the manufacture of drugs for the prevention or treatment of obesity
PT1156805E (en) USE OF TIAZOLE PILICLIC SYSTEMS FOR THE MANUFACTURE OF MEDICINES FOR PROPHYLAXIS OR THE TREATMENT OF OBESITY
MX9400165A (en) DERIVATIVES OF TER-BUTYLERGOLINE, PROCESS FOR ITS PRODUCTION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM.
UY26517A1 (en) PIRAZOLO (4,3-E) NOVEL SUBSTITUTED DIAZEPINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, THEIR USE AS MEDICINAL PRODUCTS AND PROCESSES TO PREPARE THEM
MXPA04001855A (en) Derivatives of c2-substituted indan-1-ol systems, methods for the production thereof and their use as medicaments.
ES2164454T3 (en) NEW COMPOUNDS DERIVED FROM ALQUILENDIAMINE DI OR TRI-ACETIC ACID, ITS PREPARATION PROCEDURE, ITS USE IN COSMETIC AND PHARMACEUTICAL COMPOSITIONS AND COMPOSITIONS THAT CONTAIN THEM.
AR022735A1 (en) 2-AMINO-DIHYDROTIAZOL POLICE SYSTEMS, PROCEDURE FOR PREPARATION OF THE MEDICINAL PRODUCT AND ITS EMPLOYMENT AS A MEDICINAL PRODUCT
AR029303A1 (en) INHIBITORS OF THE SOLUBLE HUMAN CD-23 FORMATION, A PROCEDURE FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM, AND THE USE OF THE SAME FOR THE PRODUCTION OF MEDICINES
NO20020914D0 (en) Alkoxy-substituted benzimidazole compounds, preparations containing them and their applications
TR200003451T2 (en) Pyrimidine-Aminomethyl-Pyridine Derivatives, Their Preparation and Their Use in the Control of Helicobacter Bacteria
AR022736A1 (en) POLYCLY SYSTEMS OF TIAZOL, MEDICINAL CONTAINING THESE COMPOUNDS, AND PROCEDURE FOR THE PREPARATION OF THE MEDICINAL PRODUCT

Legal Events

Date Code Title Description
FC Application refused