CH518940A - Verfahren zur Herstellung von Isochinuclidin-Derivaten - Google Patents

Verfahren zur Herstellung von Isochinuclidin-Derivaten

Info

Publication number
CH518940A
CH518940A CH633271A CH633271A CH518940A CH 518940 A CH518940 A CH 518940A CH 633271 A CH633271 A CH 633271A CH 633271 A CH633271 A CH 633271A CH 518940 A CH518940 A CH 518940A
Authority
CH
Switzerland
Prior art keywords
preparation
isoquinuclidine
derivatives
isoquinuclidine derivatives
Prior art date
Application number
CH633271A
Other languages
English (en)
Inventor
Nagata Wataru
Hirai Shoichi
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of CH518940A publication Critical patent/CH518940A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH633271A 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuclidin-Derivaten CH518940A (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP3564767 1967-06-03
JP762068 1968-02-07

Publications (1)

Publication Number Publication Date
CH518940A true CH518940A (de) 1972-02-15

Family

ID=26341953

Family Applications (3)

Application Number Title Priority Date Filing Date
CH633171A CH511233A (de) 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuklidin-Derivaten
CH633271A CH518940A (de) 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuclidin-Derivaten
CH821368A CH510669A (de) 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuclidin-Derivaten

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH633171A CH511233A (de) 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuklidin-Derivaten

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH821368A CH510669A (de) 1967-06-03 1968-06-04 Verfahren zur Herstellung von Isochinuclidin-Derivaten

Country Status (6)

Country Link
US (2) US3639408A (de)
CH (3) CH511233A (de)
DE (1) DE1770561A1 (de)
FR (1) FR1572766A (de)
GB (1) GB1236488A (de)
NL (1) NL6807826A (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4003905A (en) * 1974-12-11 1977-01-18 E. R. Squibb & Sons, Inc. Diels-alder adducts of benzdiazepines
US4022790A (en) * 1975-04-15 1977-05-10 E. R. Squibb & Sons, Inc. Hydrogenated diels-alder adducts of benzdiazepines
US3984418A (en) * 1975-04-15 1976-10-05 E. R. Squibb & Sons, Inc. Hydrogenated diels-alder adducts of benzdiazepines
HU188022B (en) * 1983-06-29 1986-03-28 Richter Gedeon Vegyeszeti Gyar Rt,Hu Process for production of derivatives of indolo /2,3-g/cyylopent /a/ indolizin
EP2246058A1 (de) 1997-09-04 2010-11-03 Novoneuron, Inc. Noribogain zur Behandlung von Schmerzen und Drogenabhängigheit
US7220737B1 (en) 1997-09-04 2007-05-22 Novoneuron, Inc Noribogaine in the treatment of pain and drug addiction
US9394294B2 (en) 2010-05-11 2016-07-19 Demerx, Inc. Methods and compositions for preparing and purifying noribogaine
US8362007B1 (en) 2010-05-11 2013-01-29 Demerx, Inc. Substituted noribogaine
US8765737B1 (en) 2010-05-11 2014-07-01 Demerx, Inc. Methods and compositions for preparing and purifying noribogaine
US9586954B2 (en) 2010-06-22 2017-03-07 Demerx, Inc. N-substituted noribogaine prodrugs
US8802832B2 (en) 2010-06-22 2014-08-12 Demerx, Inc. Compositions comprising noribogaine and an excipient to facilitate transport across the blood brain barrier
US8637648B1 (en) 2010-06-22 2014-01-28 Demerx, Inc. Compositions comprising noribogaine and an excipient to facilitate transport across the blood brain barrier
US8741891B1 (en) 2010-06-22 2014-06-03 Demerx, Inc. N-substituted noribogaine prodrugs
MX2013000733A (es) 2010-07-23 2013-05-30 Demerx Inc Composiciones de noribogaina.
EP2481740B1 (de) 2011-01-26 2015-11-04 DemeRx, Inc. Verfahren und Zusammensetzungen zur Herstellung von Noribogain aus Voacangin
WO2013028999A1 (en) * 2011-08-24 2013-02-28 The Trustees Of Columbia University In The City Of New York Small molecule inducers of gdnf as potential new therapeutics for neuropsychiatric disorders
US9617274B1 (en) 2011-08-26 2017-04-11 Demerx, Inc. Synthetic noribogaine
CA3122767C (en) 2011-12-08 2023-03-28 Demerx, Inc. Stereoselective total synthesis of noribogaine
CA2855994A1 (en) 2011-12-09 2013-06-13 Demerx, Inc. Phosphate esters of noribogaine
US9150584B2 (en) 2012-01-25 2015-10-06 Demerx, Inc. Indole and benzofuran fused isoquinuclidene derivatives and processes for preparing them
AU2013212139A1 (en) 2012-01-25 2014-06-26 Demerx, Inc. Synthetic voacangine
US8940728B2 (en) 2012-12-20 2015-01-27 Demerx, Inc. Substituted noribogaine
WO2014098877A1 (en) 2012-12-20 2014-06-26 Demerx, Inc. Substituted noribogaine
US9045481B2 (en) 2012-12-20 2015-06-02 Demerx, Inc. Substituted noribogaine
US9550789B2 (en) 2014-06-18 2017-01-24 Demerx, Inc. Halogenated indole and benzofuran derivatives of isoquinuclidene and processes for preparing them
EP3224261B1 (de) 2014-11-26 2024-09-18 The Trustees of Columbia University in the City of New York Opioid-rezeptor-modulatoren
US12564597B2 (en) 2020-03-05 2026-03-03 The Trustees Of Columbia University In The Of New York Ibogaine analogs as therapeutics for neurological and psychiatric disorders
EP4185578A4 (de) * 2020-07-20 2025-03-12 The Trustees Of Columbia University In The City Of New York Ibogain-analoga als therapeutika für neurologische und psychiatrische erkrankungen

Also Published As

Publication number Publication date
GB1236488A (en) 1971-06-23
CH511233A (de) 1971-08-15
DE1770561A1 (de) 1971-11-04
US3639408A (en) 1972-02-01
NL6807826A (de) 1968-12-04
US3716528A (en) 1973-02-13
FR1572766A (de) 1969-06-27
CH510669A (de) 1971-07-31

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Legal Events

Date Code Title Description
PL Patent ceased