CA2821433C - Agonistes et antagonistes du recepteur lpa et methodes d'utilisation - Google Patents

Agonistes et antagonistes du recepteur lpa et methodes d'utilisation Download PDF

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Publication number
CA2821433C
CA2821433C CA2821433A CA2821433A CA2821433C CA 2821433 C CA2821433 C CA 2821433C CA 2821433 A CA2821433 A CA 2821433A CA 2821433 A CA2821433 A CA 2821433A CA 2821433 C CA2821433 C CA 2821433C
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Canada
Prior art keywords
lpa
receptor
leu
cells
ser
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2821433A
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English (en)
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CA2821433A1 (fr
Inventor
Duane D. Miller
Gabor Tigyi
Gangadhar G. Durgam
Tamas Virag
Michelle D. Walker
Ryoko Tsukahara
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University of Tennessee Research Foundation
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University of Tennessee Research Foundation
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Publication date
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Priority claimed from CA2540809A external-priority patent/CA2540809C/fr
Publication of CA2821433A1 publication Critical patent/CA2821433A1/fr
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Publication of CA2821433C publication Critical patent/CA2821433C/fr
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Abstract

La présente invention concerne des composés de formule (I) ainsi que des compositions pharmaceutiques contenant ces mêmes composés. Ladite invention a également trait à des procédés dutilisation de ces composés qui présentent une activité en tant quagonistes ou quantagonistes des récepteurs de lacide lysophosphatidique (LPA); ces procédés comprenant linhibition de lactivité LPA sur un récepteur LPA, la modulation de lactivité du récepteur LPA, le traitement du cancer, lactivation de la prolifération cellulaire, le traitement dune blessure, le traitement de lapoptose ou la préservation ou la restauration de la fonction dans une cellule, un tissu ou un organe, la culture cellulaire, la préservation de la fonction dun organe ou dun tissu et le traitement dun état dermatologique (voir la formule I).
CA2821433A 2003-10-09 2004-10-12 Agonistes et antagonistes du recepteur lpa et methodes d'utilisation Active CA2821433C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US50997103P 2003-10-09 2003-10-09
US60/509,971 2003-10-09
CA2540809A CA2540809C (fr) 2003-10-09 2004-10-12 Agonistes et antagonistes du recepteur lpa et methodes d'utilisation

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA2540809A Division CA2540809C (fr) 2003-10-09 2004-10-12 Agonistes et antagonistes du recepteur lpa et methodes d'utilisation

Publications (2)

Publication Number Publication Date
CA2821433A1 CA2821433A1 (fr) 2005-04-14
CA2821433C true CA2821433C (fr) 2015-06-16

Family

ID=49118031

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2821433A Active CA2821433C (fr) 2003-10-09 2004-10-12 Agonistes et antagonistes du recepteur lpa et methodes d'utilisation

Country Status (1)

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CA (1) CA2821433C (fr)

Also Published As

Publication number Publication date
CA2821433A1 (fr) 2005-04-14

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