CA2318298A1 - 7-alkoxycoumarines en tant que substrats de cytochrome p450 - Google Patents

7-alkoxycoumarines en tant que substrats de cytochrome p450 Download PDF

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Publication number
CA2318298A1
CA2318298A1 CA 2318298 CA2318298A CA2318298A1 CA 2318298 A1 CA2318298 A1 CA 2318298A1 CA 2318298 CA2318298 CA 2318298 CA 2318298 A CA2318298 A CA 2318298A CA 2318298 A1 CA2318298 A1 CA 2318298A1
Authority
CA
Canada
Prior art keywords
compound
formula
enzyme
cyp2d6
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA 2318298
Other languages
English (en)
Inventor
Stephen Edward Clarke
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Priority to CA 2318298 priority Critical patent/CA2318298A1/fr
Publication of CA2318298A1 publication Critical patent/CA2318298A1/fr
Abandoned legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/06Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2
    • C07D311/08Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2 not hydrogenated in the hetero ring
    • C07D311/16Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2 not hydrogenated in the hetero ring substituted in position 7
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12QMEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
    • C12Q1/00Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions
    • C12Q1/26Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving oxidoreductase

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Microbiology (AREA)
  • Molecular Biology (AREA)
  • Analytical Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA 2318298 2000-09-01 2000-09-01 7-alkoxycoumarines en tant que substrats de cytochrome p450 Abandoned CA2318298A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA 2318298 CA2318298A1 (fr) 2000-09-01 2000-09-01 7-alkoxycoumarines en tant que substrats de cytochrome p450

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CA 2318298 CA2318298A1 (fr) 2000-09-01 2000-09-01 7-alkoxycoumarines en tant que substrats de cytochrome p450

Publications (1)

Publication Number Publication Date
CA2318298A1 true CA2318298A1 (fr) 2002-03-01

Family

ID=41651480

Family Applications (1)

Application Number Title Priority Date Filing Date
CA 2318298 Abandoned CA2318298A1 (fr) 2000-09-01 2000-09-01 7-alkoxycoumarines en tant que substrats de cytochrome p450

Country Status (1)

Country Link
CA (1) CA2318298A1 (fr)

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