CA2195759A1 - Tetrahydropyridinylmethyl derivatives of pyrrolo[2,3-b]pyridine - Google Patents

Tetrahydropyridinylmethyl derivatives of pyrrolo[2,3-b]pyridine

Info

Publication number
CA2195759A1
CA2195759A1 CA002195759A CA2195759A CA2195759A1 CA 2195759 A1 CA2195759 A1 CA 2195759A1 CA 002195759 A CA002195759 A CA 002195759A CA 2195759 A CA2195759 A CA 2195759A CA 2195759 A1 CA2195759 A1 CA 2195759A1
Authority
CA
Canada
Prior art keywords
pyrrolo
pyridine
derivatives
tetrahydropyridinylmethyl
dopamine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002195759A
Other languages
French (fr)
Other versions
CA2195759C (en
Inventor
Neil Roy Curtis
Janusz Jozef Kulagowski
Paul David Leeson
Mark Peter Ridgill
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Organon Pharma UK Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9416160A external-priority patent/GB9416160D0/en
Priority claimed from GB9416161A external-priority patent/GB9416161D0/en
Priority claimed from GBGB9505888.9A external-priority patent/GB9505888D0/en
Application filed by Individual filed Critical Individual
Priority claimed from PCT/GB1995/001820 external-priority patent/WO1996005200A1/en
Publication of CA2195759A1 publication Critical patent/CA2195759A1/en
Application granted granted Critical
Publication of CA2195759C publication Critical patent/CA2195759C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Abstract

A class of pyrrolo[2,3-b]pyridine derivatives of formula (I), wherein Q
represents a moiety of formula Qa or Qb, are ligands for dopamine receptor subtypes within the body, in particular the dopamine D4 receptor subtype and are therefore useful in the treatment and/or prevention of disorders of the dopamine system, including schizophrenia.
CA002195759A 1994-08-10 1995-08-01 Tetrahydropyridinylmethyl derivatives of pyrrolo[2,3-b]pyridine Expired - Fee Related CA2195759C (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB9416160A GB9416160D0 (en) 1994-08-10 1994-08-10 Therapeutic agents
GB9416161A GB9416161D0 (en) 1994-08-10 1994-08-10 Therapeutic agents
GB9505888.9 1995-03-23
GBGB9505888.9A GB9505888D0 (en) 1995-03-23 1995-03-23 Therapeutic agents
GB9416161.9 1995-03-23
GB9416160.1 1995-03-23
PCT/GB1995/001820 WO1996005200A1 (en) 1994-08-10 1995-08-01 TETRAHYDROPYRIDINYLMETHYL DERIVATIVES OF PYRROLO[2,3-b]PYRIDINE

Publications (2)

Publication Number Publication Date
CA2195759A1 true CA2195759A1 (en) 1996-02-22
CA2195759C CA2195759C (en) 2006-04-11

Family

ID=36178102

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002195759A Expired - Fee Related CA2195759C (en) 1994-08-10 1995-08-01 Tetrahydropyridinylmethyl derivatives of pyrrolo[2,3-b]pyridine

Country Status (1)

Country Link
CA (1) CA2195759C (en)

Also Published As

Publication number Publication date
CA2195759C (en) 2006-04-11

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