CA1271744A - Prepartion d'aminoglycosides - Google Patents
Prepartion d'aminoglycosidesInfo
- Publication number
- CA1271744A CA1271744A CA000297395A CA297395A CA1271744A CA 1271744 A CA1271744 A CA 1271744A CA 000297395 A CA000297395 A CA 000297395A CA 297395 A CA297395 A CA 297395A CA 1271744 A CA1271744 A CA 1271744A
- Authority
- CA
- Canada
- Prior art keywords
- kanamycin
- benzyloxycarbonyl
- aminoglycoside
- acylating reagent
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA000297395A CA1271744A (fr) | 1978-02-21 | 1978-02-21 | Prepartion d'aminoglycosides |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA000297395A CA1271744A (fr) | 1978-02-21 | 1978-02-21 | Prepartion d'aminoglycosides |
Publications (2)
Publication Number | Publication Date |
---|---|
CA1271744C CA1271744C (fr) | 1990-07-17 |
CA1271744A true CA1271744A (fr) | 1990-07-17 |
Family
ID=4110829
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA000297395A Expired CA1271744A (fr) | 1978-02-21 | 1978-02-21 | Prepartion d'aminoglycosides |
Country Status (1)
Country | Link |
---|---|
CA (1) | CA1271744A (fr) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7893039B2 (en) | 2005-12-02 | 2011-02-22 | Isis Pharmaceuticals, Inc. | Antibacterial 4,5-substituted aminoglycoside analogs having multiple substituents |
US8318685B2 (en) | 2010-11-17 | 2012-11-27 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8367625B2 (en) | 2008-10-09 | 2013-02-05 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8372813B2 (en) | 2008-10-09 | 2013-02-12 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8377896B2 (en) | 2008-09-10 | 2013-02-19 | Isis Pharmaceuticals, Inc | Antibacterial 4,6-substituted 6′, 6″ and 1 modified aminoglycoside analogs |
US8399419B2 (en) | 2008-09-10 | 2013-03-19 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8481502B2 (en) | 2009-10-09 | 2013-07-09 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
-
1978
- 1978-02-21 CA CA000297395A patent/CA1271744A/fr not_active Expired
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7893039B2 (en) | 2005-12-02 | 2011-02-22 | Isis Pharmaceuticals, Inc. | Antibacterial 4,5-substituted aminoglycoside analogs having multiple substituents |
US8114856B2 (en) | 2005-12-02 | 2012-02-14 | Isis Pharmaceuticals, Inc. | Antibacterial 4,5-substituted aminoglycoside analogs having multiple substituents |
US8569264B2 (en) | 2005-12-02 | 2013-10-29 | Isis Pharmaceuticals, Inc. | Antibacterial 4,5-substituted aminoglycoside analogs having multiple substituents |
US8377896B2 (en) | 2008-09-10 | 2013-02-19 | Isis Pharmaceuticals, Inc | Antibacterial 4,6-substituted 6′, 6″ and 1 modified aminoglycoside analogs |
US8399419B2 (en) | 2008-09-10 | 2013-03-19 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8742078B2 (en) | 2008-09-10 | 2014-06-03 | Isis Pharmaceuticals, Inc. | Antibacterial 4,6-substituted 6′, 6″ and 1 modified aminoglycoside analogs |
US8367625B2 (en) | 2008-10-09 | 2013-02-05 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8372813B2 (en) | 2008-10-09 | 2013-02-12 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8481502B2 (en) | 2009-10-09 | 2013-07-09 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8318685B2 (en) | 2010-11-17 | 2012-11-27 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
US8653041B2 (en) | 2010-11-17 | 2014-02-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
Also Published As
Publication number | Publication date |
---|---|
CA1271744C (fr) | 1990-07-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MKEX | Expiry | ||
MKEX | Expiry |
Effective date: 20070717 |