CA1189503A - Omt ester derivatives - Google Patents

Omt ester derivatives

Info

Publication number
CA1189503A
CA1189503A CA000417149A CA417149A CA1189503A CA 1189503 A CA1189503 A CA 1189503A CA 000417149 A CA000417149 A CA 000417149A CA 417149 A CA417149 A CA 417149A CA 1189503 A CA1189503 A CA 1189503A
Authority
CA
Canada
Prior art keywords
omt
acetyl
methyl
ethyl
solution
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000417149A
Other languages
English (en)
French (fr)
Inventor
Herbert A. Kirst
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of CA1189503A publication Critical patent/CA1189503A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA000417149A 1981-12-14 1982-12-07 Omt ester derivatives Expired CA1189503A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US330,341 1981-12-14
US06/330,341 US4401660A (en) 1981-12-14 1981-12-14 Ester derivatives of 5-O-mycaminosyl tylonolide and method of using same

Publications (1)

Publication Number Publication Date
CA1189503A true CA1189503A (en) 1985-06-25

Family

ID=23289335

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000417149A Expired CA1189503A (en) 1981-12-14 1982-12-07 Omt ester derivatives

Country Status (12)

Country Link
US (1) US4401660A (cg-RX-API-DMAC7.html)
EP (1) EP0082003B1 (cg-RX-API-DMAC7.html)
JP (1) JPS58110598A (cg-RX-API-DMAC7.html)
KR (1) KR850000978B1 (cg-RX-API-DMAC7.html)
CA (1) CA1189503A (cg-RX-API-DMAC7.html)
DE (1) DE3268461D1 (cg-RX-API-DMAC7.html)
DK (2) DK153794C (cg-RX-API-DMAC7.html)
GB (1) GB2111497B (cg-RX-API-DMAC7.html)
GR (1) GR77094B (cg-RX-API-DMAC7.html)
HU (1) HU194268B (cg-RX-API-DMAC7.html)
IE (1) IE54283B1 (cg-RX-API-DMAC7.html)
IL (1) IL67452A (cg-RX-API-DMAC7.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
CA1196915A (en) * 1982-01-22 1985-11-19 Hideo Sakakibara 23-0-acyl-23-demycinosyldesmycosin
US4443436A (en) 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
GB8333624D0 (en) * 1983-12-16 1984-01-25 Lepetit Spa Antibiotics l 17054 and l 17392
US4576931A (en) * 1985-04-03 1986-03-18 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai (Microbial Chemistry Research Foundation) 23-C-Substituted mycaminosyl tylonolide, pharmaceutical compositions and method of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE667952A (cg-RX-API-DMAC7.html) * 1964-08-05
CH619267A5 (cg-RX-API-DMAC7.html) * 1975-08-01 1980-09-15 Sanraku Ocean Co
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
US4438109A (en) * 1980-07-25 1984-03-20 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Tylosin derivatives
US4299953A (en) * 1980-07-29 1981-11-10 Eli Lilly And Company Mycarosyltylactone

Also Published As

Publication number Publication date
IE822952L (en) 1983-06-14
DK553982A (da) 1983-06-15
GB2111497B (en) 1985-10-30
GR77094B (cg-RX-API-DMAC7.html) 1984-09-06
EP0082003A1 (en) 1983-06-22
DK153794B (da) 1988-09-05
DK623786D0 (da) 1986-12-22
DK153794C (da) 1989-02-20
DE3268461D1 (de) 1986-02-20
US4401660A (en) 1983-08-30
DK623786A (da) 1986-12-22
IL67452A (en) 1985-12-31
IL67452A0 (en) 1983-05-15
IE54283B1 (en) 1989-08-16
JPS58110598A (ja) 1983-07-01
KR850000978B1 (ko) 1985-07-05
HU194268B (en) 1988-01-28
GB2111497A (en) 1983-07-06
EP0082003B1 (en) 1986-01-08
KR840002855A (ko) 1984-07-21

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Legal Events

Date Code Title Description
MKEC Expiry (correction)
MKEX Expiry