BRPI0907504A2 - crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1 - Google Patents
crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1Info
- Publication number
- BRPI0907504A2 BRPI0907504A2 BRPI0907504A BRPI0907504A BRPI0907504A2 BR PI0907504 A2 BRPI0907504 A2 BR PI0907504A2 BR PI0907504 A BRPI0907504 A BR PI0907504A BR PI0907504 A BRPI0907504 A BR PI0907504A BR PI0907504 A2 BRPI0907504 A2 BR PI0907504A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- producing
- pharmaceutical composition
- inhibitory effect
- crystalline form
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
forma cristalina de um composto, composição farmacêutica, uso de um composto, e, método para produzir um efeito inibidor de l lbhsd l. novas formas cristalinas do ácido 4-[4-(2- adamantilcarbamoil)-5-terc-butil-pirazol-1-il]benzóico; seu uso na inibição de 11 ~hsd 1, processos para fabricá-las e composições farmacêuticas que as compreendam também são descritas.crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 1 lbhsd l. new crystalline forms of 4- [4- (2-adamantylcarbamoyl) -5-tert-butyl-pyrazol-1-yl] benzoic acid; Their use in inhibiting 11 hsd 1, processes for making them and pharmaceutical compositions comprising them are also described.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PK10808 | 2008-02-04 | ||
PCT/GB2008/000454 WO2008099145A1 (en) | 2007-02-12 | 2008-02-11 | Pyrazole derivatives as 11-beta-hsd1 inhibitors |
US8229308P | 2008-07-21 | 2008-07-21 | |
PCT/GB2009/050096 WO2009098501A1 (en) | 2008-02-04 | 2009-02-03 | Novel crystalline forms of 4- [4- (2-adamantylcarbam0yl) -5-tert-butyl-pyrazol-1-yl] benzoic acid |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0907504A2 true BRPI0907504A2 (en) | 2019-02-26 |
Family
ID=65686632
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0907504A BRPI0907504A2 (en) | 2008-02-04 | 2009-02-03 | crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1 |
Country Status (2)
Country | Link |
---|---|
BR (1) | BRPI0907504A2 (en) |
CL (1) | CL2009000237A1 (en) |
-
2009
- 2009-02-03 CL CL2009000237A patent/CL2009000237A1/en unknown
- 2009-02-03 BR BRPI0907504A patent/BRPI0907504A2/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CL2009000237A1 (en) | 2010-02-19 |
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Legal Events
Date | Code | Title | Description |
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B08F | Application fees: application dismissed [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 6A, 7A, 8A, 9A E 10A ANUIDADES. |
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B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2513 DE 06-03-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |
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B350 | Update of information on the portal [chapter 15.35 patent gazette] |