BRPI0907504A2 - crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1 - Google Patents

crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1

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Publication number
BRPI0907504A2
BRPI0907504A2 BRPI0907504A BRPI0907504A BRPI0907504A2 BR PI0907504 A2 BRPI0907504 A2 BR PI0907504A2 BR PI0907504 A BRPI0907504 A BR PI0907504A BR PI0907504 A BRPI0907504 A BR PI0907504A BR PI0907504 A2 BRPI0907504 A2 BR PI0907504A2
Authority
BR
Brazil
Prior art keywords
compound
producing
pharmaceutical composition
inhibitory effect
crystalline form
Prior art date
Application number
BRPI0907504A
Other languages
Portuguese (pt)
Inventor
Stocker Andrew
Peter Tomkinson Gery
Stewart Scott James
Packer Martin
Robert Owen Whittamore Paul
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=65686632&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0907504(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from PCT/GB2008/000454 external-priority patent/WO2008099145A1/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority claimed from PCT/GB2009/050096 external-priority patent/WO2009098501A1/en
Publication of BRPI0907504A2 publication Critical patent/BRPI0907504A2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

forma cristalina de um composto, composição farmacêutica, uso de um composto, e, método para produzir um efeito inibidor de l lbhsd l. novas formas cristalinas do ácido 4-[4-(2- adamantilcarbamoil)-5-terc-butil-pirazol-1-il]benzóico; seu uso na inibição de 11 ~hsd 1, processos para fabricá-las e composições farmacêuticas que as compreendam também são descritas.crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 1 lbhsd l. new crystalline forms of 4- [4- (2-adamantylcarbamoyl) -5-tert-butyl-pyrazol-1-yl] benzoic acid; Their use in inhibiting 11 hsd 1, processes for making them and pharmaceutical compositions comprising them are also described.

BRPI0907504A 2008-02-04 2009-02-03 crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1 BRPI0907504A2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
PK10808 2008-02-04
PCT/GB2008/000454 WO2008099145A1 (en) 2007-02-12 2008-02-11 Pyrazole derivatives as 11-beta-hsd1 inhibitors
US8229308P 2008-07-21 2008-07-21
PCT/GB2009/050096 WO2009098501A1 (en) 2008-02-04 2009-02-03 Novel crystalline forms of 4- [4- (2-adamantylcarbam0yl) -5-tert-butyl-pyrazol-1-yl] benzoic acid

Publications (1)

Publication Number Publication Date
BRPI0907504A2 true BRPI0907504A2 (en) 2019-02-26

Family

ID=65686632

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0907504A BRPI0907504A2 (en) 2008-02-04 2009-02-03 crystalline form of a compound, pharmaceutical composition, use of a compound, and method for producing an inhibitory effect of 11bhsd1

Country Status (2)

Country Link
BR (1) BRPI0907504A2 (en)
CL (1) CL2009000237A1 (en)

Also Published As

Publication number Publication date
CL2009000237A1 (en) 2010-02-19

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Legal Events

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B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 6A, 7A, 8A, 9A E 10A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2513 DE 06-03-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

B350 Update of information on the portal [chapter 15.35 patent gazette]