BR9915900A - Compound, pharmaceutical composition, and process for treating or inhibiting disorders associated with smooth muscle contraction. - Google Patents
Compound, pharmaceutical composition, and process for treating or inhibiting disorders associated with smooth muscle contraction.Info
- Publication number
- BR9915900A BR9915900A BR9915900-7A BR9915900A BR9915900A BR 9915900 A BR9915900 A BR 9915900A BR 9915900 A BR9915900 A BR 9915900A BR 9915900 A BR9915900 A BR 9915900A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- pharmaceutical composition
- smooth muscle
- disorders associated
- muscle contraction
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/58—[b]- or [c]-condensed
- C07D209/70—[b]- or [c]-condensed containing carbocyclic rings other than six-membered
Abstract
"COMPOSTO, COMPOSIçãO FARMACêUTICA, E, PROCESSO PARA TRATAR OU INIBIR DISTúRBIOS ASSOCIADOS COM CONTRAçãO DA MUSCULATURA LISA" Compostos de Fórmulas (I) e (II): onde R~ 1~, R~ 2~, R~ 3~, X, Y e Z são como definidos na especificação compostos estes úteis no tratamento de distúrbios associados com contração de musculatura lisa via modulação por canal de potássio."COMPOUND, PHARMACEUTICAL COMPOSITION, AND, PROCESS TO TREAT OR INHIBIT DISTURBANCES ASSOCIATED WITH SMOOTH MUSCULATURE CONTRACTION" Compounds of Formulas (I) and (II): where R ~ 1 ~, R ~ 2 ~, R ~ 3 ~, X, Y and Z are as defined in the specification compounds which are useful in the treatment of disorders associated with smooth muscle contraction via potassium channel modulation.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US20577098A | 1998-12-04 | 1998-12-04 | |
PCT/US1999/028619 WO2000034285A2 (en) | 1998-12-04 | 1999-12-03 | Substituted benzofuranoindoles and indenoindoles as novel potassium channel openers |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9915900A true BR9915900A (en) | 2001-08-21 |
Family
ID=22763580
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9915900-7A BR9915900A (en) | 1998-12-04 | 1999-12-03 | Compound, pharmaceutical composition, and process for treating or inhibiting disorders associated with smooth muscle contraction. |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1135393A2 (en) |
JP (1) | JP2002531569A (en) |
CN (1) | CN1333774A (en) |
AU (1) | AU2163600A (en) |
BR (1) | BR9915900A (en) |
CA (1) | CA2350590A1 (en) |
WO (1) | WO2000034285A2 (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101072780B (en) * | 2004-09-20 | 2010-06-23 | 詹森药业有限公司 | Novel tetracyclic derivative containing heteroatoms useful as sex steroid hormone receptor modulators |
KR100659498B1 (en) * | 2005-03-10 | 2006-12-20 | 애니젠 주식회사 | Potassium channel opener having benzofuroindole skeleton |
AU2006267077A1 (en) | 2005-07-14 | 2007-01-18 | Irm Llc | Heterotetracyclic compounds as TPO mimetics |
JP6091445B2 (en) * | 2013-02-07 | 2017-03-08 | 富士フイルム株式会社 | Organic thin film transistor, organic semiconductor thin film and organic semiconductor material |
PL3292116T3 (en) | 2015-02-02 | 2022-02-21 | Valo Health, Inc. | 3-aryl-4-amido-bicyclic [4,5,0]hydroxamic acids as hdac inhibitors |
TW201636329A (en) | 2015-02-02 | 2016-10-16 | 佛瑪治療公司 | Bicyclic [4,6,0] hydroxamic acids as HDAC inhibitors |
WO2017218950A1 (en) | 2016-06-17 | 2017-12-21 | Forma Therapeutics, Inc. | 2-spiro-5- and 6-hydroxamic acid indanes as hdac inhibitors |
CN106632360A (en) * | 2016-09-27 | 2017-05-10 | 上海道亦化工科技有限公司 | Compound based on benzofuroindole and organic electroluminescent device thereof |
CN109942545A (en) * | 2019-04-15 | 2019-06-28 | 中国药科大学 | Competitive sour retarding agent of potassium ion containing indole structure and preparation method thereof and purposes |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE8902273D0 (en) * | 1989-06-22 | 1989-06-22 | Univ Cincinnati | INDENOINDOLE COMPOUNDS I |
SE8902274D0 (en) * | 1989-06-22 | 1989-06-22 | Univ Cincinnati | INDENOIDOLE COMPOUNDS II |
MC2251A1 (en) * | 1990-03-20 | 1993-03-25 | Wellcome Found | BIOCIDAL HETEROCYCLIC COMPOUNDS, THEIR SYNTHESIS AND THEIR INTERIORS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN MEDICINE |
-
1999
- 1999-12-03 CN CN99815495A patent/CN1333774A/en active Pending
- 1999-12-03 BR BR9915900-7A patent/BR9915900A/en not_active Application Discontinuation
- 1999-12-03 EP EP99965977A patent/EP1135393A2/en not_active Withdrawn
- 1999-12-03 WO PCT/US1999/028619 patent/WO2000034285A2/en not_active Application Discontinuation
- 1999-12-03 JP JP2000586730A patent/JP2002531569A/en active Pending
- 1999-12-03 CA CA002350590A patent/CA2350590A1/en not_active Abandoned
- 1999-12-03 AU AU21636/00A patent/AU2163600A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU2163600A (en) | 2000-06-26 |
WO2000034285A2 (en) | 2000-06-15 |
CN1333774A (en) | 2002-01-30 |
WO2000034285A3 (en) | 2000-11-16 |
CA2350590A1 (en) | 2000-06-15 |
JP2002531569A (en) | 2002-09-24 |
EP1135393A2 (en) | 2001-09-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |