BR6348675D0 - Processo para estabilizar solucoes aquosas de esteres 21-fosfatos de 21-hidroxi-esteroides - Google Patents

Processo para estabilizar solucoes aquosas de esteres 21-fosfatos de 21-hidroxi-esteroides

Info

Publication number
BR6348675D0
BR6348675D0 BR148675/63A BR14867563A BR6348675D0 BR 6348675 D0 BR6348675 D0 BR 6348675D0 BR 148675/63 A BR148675/63 A BR 148675/63A BR 14867563 A BR14867563 A BR 14867563A BR 6348675 D0 BR6348675 D0 BR 6348675D0
Authority
BR
Brazil
Prior art keywords
steroids
phosphates
hydroxy
esters
aqueous solutions
Prior art date
Application number
BR148675/63A
Other languages
English (en)
Inventor
D Marcus
C Riffkin
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of BR6348675D0 publication Critical patent/BR6348675D0/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
BR148675/63A 1962-05-01 1963-04-25 Processo para estabilizar solucoes aquosas de esteres 21-fosfatos de 21-hidroxi-esteroides BR6348675D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US191424A US3138528A (en) 1962-05-01 1962-05-01 Stable, aqueous solutions of 21-phosphate esters of 21-hydroxy steroids

Publications (1)

Publication Number Publication Date
BR6348675D0 true BR6348675D0 (pt) 1973-07-03

Family

ID=22705453

Family Applications (1)

Application Number Title Priority Date Filing Date
BR148675/63A BR6348675D0 (pt) 1962-05-01 1963-04-25 Processo para estabilizar solucoes aquosas de esteres 21-fosfatos de 21-hidroxi-esteroides

Country Status (4)

Country Link
US (1) US3138528A (pt)
BR (1) BR6348675D0 (pt)
FR (1) FR2734M (pt)
GB (1) GB1036907A (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3898330A (en) * 1973-08-01 1975-08-05 Squibb & Sons Inc Corticosteroid phosphate salts/neomycin sulfate ophthalmic
US4931473A (en) * 1989-02-15 1990-06-05 Richardson-Vicks Inc. Anesthetic oral compositions
CA2605138A1 (en) * 2005-04-15 2006-10-26 Lyotropic Therapeutics, Inc. Formulations of quaternary ammonium neuromuscular blocking agents
US20150164882A1 (en) 2013-07-22 2015-06-18 Imprimis Pharmaceuticals, Inc. Pharmaceutical compositions for intraocular administration and methods for fabricating thereof
US20160279055A1 (en) 2013-07-22 2016-09-29 Imprimis Pharmaceuticals, Inc. Pharmaceutical ophthalmic compositions for intraocular administration and methods for fabricating thereof
US20160101118A1 (en) * 2014-08-15 2016-04-14 Imprimis Pharmaceuticals, Inc. Pharmaceutical compositions for intraocular administration and methods for fabricating thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2686145A (en) * 1951-04-19 1954-08-10 Lloyd Brothers Inc Water solution of khellin
US2870177A (en) * 1954-08-04 1959-01-20 Merck & Co Inc delta4-11-oxygenated-pregnene-17alpha, 21-diol-3, 20-dione 21-phosphate and salts thereof
US2779775A (en) * 1954-09-30 1957-01-29 Merck & Co Inc Phosphate derivatives of 9alpha-fluorosteroids
US2950298A (en) * 1957-11-19 1960-08-23 Glaxo Lab Ltd Steroid secondary 21-phosphate esters
US2990401A (en) * 1958-06-18 1961-06-27 American Cyanamid Co 11-substituted 16alpha, 17alpha-substituted methylenedioxy steroids
US2970944A (en) * 1958-04-04 1961-02-07 Merck & Co Inc Parenteral solutions of steroid phosphates stabilized with creatinines
US3073743A (en) * 1959-07-30 1963-01-15 Upjohn Co Antiinflammatory steroid acetonide compositions and therapy
US3053834A (en) * 1961-01-26 1962-09-11 Olin Mathieson 21-phosphates of steroid acetals and ketals

Also Published As

Publication number Publication date
FR2734M (fr) 1964-08-17
GB1036907A (en) 1966-07-20
US3138528A (en) 1964-06-23

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