BR112012020951A2 - compounds as bradykinin-b1 antagonists - Google Patents
compounds as bradykinin-b1 antagonistsInfo
- Publication number
- BR112012020951A2 BR112012020951A2 BR112012020951A BR112012020951A BR112012020951A2 BR 112012020951 A2 BR112012020951 A2 BR 112012020951A2 BR 112012020951 A BR112012020951 A BR 112012020951A BR 112012020951 A BR112012020951 A BR 112012020951A BR 112012020951 A2 BR112012020951 A2 BR 112012020951A2
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- bradykinin
- antagonists
- production
- salts
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
compostos como antagonistas de bradiquinina-b1. a presente invenção refere-se a compostos da fórmula geral i, em que n,r1,r2,r3,r4,r5,r6,r7,r8,r9,r10,r11 e x são cada um definidos tal como descrito a seguir, seus enantiômetros, seus diastereômetros, suas misturas e seus sais, especialmente seus sais fisiologicamente compatíves com ácidos ou bases orgâniicos ou inorgânicos, os quais apresentam valiosas propriedades, sua produção, os fármacos contendo os compsotos farmacologicamnete eficazes, sua produção e seu uso.compounds as bradykinin-b1 antagonists. The present invention relates to compounds of the general formula I, wherein n, r 1, r 2, r 3, r 4, r 5, r 6, r 7, r 8, r 9, r 10, r 11 and n are each defined as described below. enantiometers, their diastereometers, their mixtures and their salts, especially their physiologically compatible salts with organic or inorganic acids or bases, which have valuable properties, their production, drugs containing the pharmacologically effective compounds, their production and their use.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2010/052232 WO2010097372A1 (en) | 2009-02-26 | 2010-02-23 | Compounds as bradykinin b1 antagonists |
| PCT/EP2011/052512 WO2011104203A1 (en) | 2010-02-23 | 2011-02-21 | Compounds as bradykinin b1 antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012020951A2 true BR112012020951A2 (en) | 2016-04-26 |
Family
ID=55859312
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012020951A BR112012020951A2 (en) | 2010-02-23 | 2011-02-21 | compounds as bradykinin-b1 antagonists |
Country Status (1)
| Country | Link |
|---|---|
| BR (1) | BR112012020951A2 (en) |
-
2011
- 2011-02-21 BR BR112012020951A patent/BR112012020951A2/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
| B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
| B11E | Dismissal acc. art. 34 of ipl - requirements for examination incomplete | ||
| B11T | Dismissal of application maintained [chapter 11.20 patent gazette] |