BR0010449A - 14beta-h-sterols, pharmaceutical compositions comprising the same and use of these derivatives for the preparation of meiosis regulating drugs - Google Patents

14beta-h-sterols, pharmaceutical compositions comprising the same and use of these derivatives for the preparation of meiosis regulating drugs

Info

Publication number
BR0010449A
BR0010449A BR0010449-3A BR0010449A BR0010449A BR 0010449 A BR0010449 A BR 0010449A BR 0010449 A BR0010449 A BR 0010449A BR 0010449 A BR0010449 A BR 0010449A
Authority
BR
Brazil
Prior art keywords
14beta
sterols
preparation
pharmaceutical compositions
derivatives
Prior art date
Application number
BR0010449-3A
Other languages
Portuguese (pt)
Inventor
Peter Esperling
Joachim Kuhnke
Henry Laurent
Thorsten Blume
Christa Hegele-Hartung
Monika Lessl
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of BR0010449A publication Critical patent/BR0010449A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J15/00—Stereochemically pure steroids containing carbon, hydrogen, halogen or oxygen having a partially or totally inverted skeleton, e.g. retrosteroids, L-isomers

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: "14BETA-H-ESTERóIS, COMPOSIçõES FARMACêUTICAS QUE COMPREENDEM OS MESMOS E USO DESTES DERIVADOS PARA A PREPARAçãO DE MEDICAMENTOS REGULADORES DA MEIOSE". A presente invenção refere-se a 14beta-H-esteróis, farmaceuticamente ativos, a composições farmacêuticas que compreendem as mesmas e ao uso destes novos compostos para a preparação de medicamentos. Mais particularmente foi descoberto que os 14beta-H-esteróis da invenção podem ser usados para regular a meiose.Invention Patent: "14BETA-H-STEROLS, PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THE SAME AND USE OF THESE DERIVATIVES FOR THE PREPARATION OF MEIOSIS REGULATORY DRUGS". The present invention relates to 14beta-H-sterols, pharmaceutically active, to pharmaceutical compositions comprising them and to the use of these new compounds for the preparation of medicaments. More particularly it has been found that the 14beta-H-sterols of the invention can be used to regulate meiosis.

BR0010449-3A 1999-05-10 2000-05-05 14beta-h-sterols, pharmaceutical compositions comprising the same and use of these derivatives for the preparation of meiosis regulating drugs BR0010449A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99250153 1999-05-10
PCT/EP2000/004092 WO2000068245A1 (en) 1999-05-10 2000-05-05 14β-H-STEROLS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND USE OF THESE DERIVATIVES FOR THE PREPARATION OF MEIOSIS REGULATING MEDICAMENTS

Publications (1)

Publication Number Publication Date
BR0010449A true BR0010449A (en) 2002-02-13

Family

ID=8241145

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0010449-3A BR0010449A (en) 1999-05-10 2000-05-05 14beta-h-sterols, pharmaceutical compositions comprising the same and use of these derivatives for the preparation of meiosis regulating drugs

Country Status (18)

Country Link
EP (1) EP1177205A1 (en)
JP (1) JP2002544136A (en)
KR (1) KR20020013541A (en)
CN (1) CN1350543A (en)
AU (1) AU4756100A (en)
BG (1) BG106093A (en)
BR (1) BR0010449A (en)
CA (1) CA2373442A1 (en)
CZ (1) CZ20013981A3 (en)
EA (1) EA200101157A1 (en)
EE (1) EE200100592A (en)
HU (1) HUP0201098A2 (en)
IL (1) IL145373A0 (en)
NO (1) NO20015488L (en)
PL (1) PL352029A1 (en)
SK (1) SK16212001A3 (en)
WO (1) WO2000068245A1 (en)
ZA (1) ZA200110073B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012044817A2 (en) * 2010-10-01 2012-04-05 Indiana University Research And Technology Corporation Process for preparing delta-7,9(11) steroids from ganoderma lucidum and analogs thereof
WO2021046678A1 (en) * 2019-09-09 2021-03-18 邦泰生物工程(深圳)有限公司 Method for synthesising chenodeoxycholic acid and application therefor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4202891A (en) * 1977-05-16 1980-05-13 Kandutsch Andrew A 15-Oxygenated sterol compounds and the use of such compounds to inhibit the biosynthesis of sterols
PL322106A1 (en) * 1995-03-06 1998-01-05 Novo Nordisk As Meiosis stimulation
WO1999058549A1 (en) * 1998-05-13 1999-11-18 Novo Nordisk A/S Meiosis regulating compounds

Also Published As

Publication number Publication date
NO20015488L (en) 2002-01-09
HUP0201098A2 (en) 2002-08-28
EP1177205A1 (en) 2002-02-06
KR20020013541A (en) 2002-02-20
SK16212001A3 (en) 2002-02-05
WO2000068245A1 (en) 2000-11-16
CZ20013981A3 (en) 2002-02-13
AU4756100A (en) 2000-11-21
EA200101157A1 (en) 2002-06-27
ZA200110073B (en) 2003-03-06
CA2373442A1 (en) 2000-11-16
CN1350543A (en) 2002-05-22
IL145373A0 (en) 2002-06-30
PL352029A1 (en) 2003-07-28
BG106093A (en) 2002-05-31
EE200100592A (en) 2003-02-17
JP2002544136A (en) 2002-12-24
NO20015488D0 (en) 2001-11-09

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]