BE851052A - Nouvelles compositions anti-hypertensives contenant des derives d'alanine - Google Patents
Nouvelles compositions anti-hypertensives contenant des derives d'alanineInfo
- Publication number
- BE851052A BE851052A BE174630A BE174630A BE851052A BE 851052 A BE851052 A BE 851052A BE 174630 A BE174630 A BE 174630A BE 174630 A BE174630 A BE 174630A BE 851052 A BE851052 A BE 851052A
- Authority
- BE
- Belgium
- Prior art keywords
- compositions containing
- new anti
- alanine derivatives
- containing alanine
- hypertensive compositions
- Prior art date
Links
- 150000001294 alanine derivatives Chemical class 0.000 title 1
- 230000003276 anti-hypertensive effect Effects 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/657,824 US4051251A (en) | 1976-02-13 | 1976-02-13 | Novel anti-hypertensive compositions |
Publications (1)
Publication Number | Publication Date |
---|---|
BE851052A true BE851052A (fr) | 1977-08-03 |
Family
ID=24638794
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE174630A BE851052A (fr) | 1976-02-13 | 1977-02-03 | Nouvelles compositions anti-hypertensives contenant des derives d'alanine |
Country Status (10)
Country | Link |
---|---|
US (2) | US4051251A (fr) |
JP (1) | JPS5299225A (fr) |
AU (1) | AU513541B2 (fr) |
BE (1) | BE851052A (fr) |
DE (1) | DE2705883A1 (fr) |
FR (1) | FR2340732A1 (fr) |
GB (1) | GB1526172A (fr) |
NL (1) | NL7700944A (fr) |
NZ (1) | NZ183226A (fr) |
ZA (1) | ZA77814B (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4070478A (en) * | 1977-02-17 | 1978-01-24 | Merck & Co., Inc. | Benzimidazole substituted alanines |
US4401676A (en) * | 1977-06-01 | 1983-08-30 | Merck & Co., Inc. | Novel α-amino acids |
AU2003293423A1 (en) * | 2002-12-06 | 2004-06-30 | Xenoport, Inc. | Carbidopa prodrugs and uses thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3462536A (en) * | 1960-07-22 | 1969-08-19 | Merck & Co Inc | Method of inhibiting decarboxylase |
US3839585A (en) * | 1970-08-05 | 1974-10-01 | Merck & Co Inc | Method of treating hypertension |
AU464903B2 (en) * | 1970-11-12 | 1975-09-11 | Merck & Co., Inc | Treatment of hypertension |
-
1976
- 1976-02-13 US US05/657,824 patent/US4051251A/en not_active Expired - Lifetime
-
1977
- 1977-01-28 NL NL7700944A patent/NL7700944A/xx not_active Application Discontinuation
- 1977-02-01 NZ NZ183226A patent/NZ183226A/xx unknown
- 1977-02-03 AU AU21919/77A patent/AU513541B2/en not_active Expired
- 1977-02-03 BE BE174630A patent/BE851052A/fr unknown
- 1977-02-08 US US05/766,636 patent/US4069333A/en not_active Expired - Lifetime
- 1977-02-10 JP JP1308077A patent/JPS5299225A/ja active Pending
- 1977-02-10 GB GB5518/77A patent/GB1526172A/en not_active Expired
- 1977-02-11 FR FR7703909A patent/FR2340732A1/fr active Granted
- 1977-02-11 ZA ZA00770814A patent/ZA77814B/xx unknown
- 1977-02-11 DE DE19772705883 patent/DE2705883A1/de not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
FR2340732B1 (fr) | 1979-08-24 |
NZ183226A (en) | 1980-03-05 |
US4051251A (en) | 1977-09-27 |
JPS5299225A (en) | 1977-08-19 |
DE2705883A1 (de) | 1977-08-18 |
ZA77814B (en) | 1978-09-27 |
NL7700944A (nl) | 1977-08-16 |
AU513541B2 (en) | 1980-12-11 |
FR2340732A1 (fr) | 1977-09-09 |
US4069333A (en) | 1978-01-17 |
AU2191977A (en) | 1978-08-10 |
GB1526172A (en) | 1978-09-27 |
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