BE751029A - 5'-esters d'ara-cytidine et leur preparation - Google Patents

5'-esters d'ara-cytidine et leur preparation

Info

Publication number
BE751029A
BE751029A BE751029DA BE751029A BE 751029 A BE751029 A BE 751029A BE 751029D A BE751029D A BE 751029DA BE 751029 A BE751029 A BE 751029A
Authority
BE
Belgium
Prior art keywords
cytidine
ara
esters
preparation
Prior art date
Application number
Other languages
English (en)
Inventor
Der C Kelly
W J Wechter
D T Gish
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BE751029A publication Critical patent/BE751029A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE751029D 1969-05-27 1970-05-27 5'-esters d'ara-cytidine et leur preparation BE751029A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US82838069A 1969-05-27 1969-05-27
US00011826A US3847898A (en) 1969-05-27 1970-02-16 N4-trihaloethoxy carbonyl arabino-furanosyl cytosine 5'-esters

Publications (1)

Publication Number Publication Date
BE751029A true BE751029A (fr) 1970-11-27

Family

ID=26682835

Family Applications (1)

Application Number Title Priority Date Filing Date
BE751029D BE751029A (fr) 1969-05-27 1970-05-27 5'-esters d'ara-cytidine et leur preparation

Country Status (11)

Country Link
US (1) US3847898A (fr)
JP (1) JPS5035077B1 (fr)
BE (1) BE751029A (fr)
CA (1) CA928290A (fr)
CH (1) CH586234A5 (fr)
DE (1) DE2025624C2 (fr)
FR (1) FR2051563B1 (fr)
GB (1) GB1263408A (fr)
IL (1) IL34400A (fr)
NL (1) NL7007505A (fr)
PH (1) PH10225A (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5159880A (en) * 1974-11-22 1976-05-25 Asahi Chemical Ind N44 ashirunukureoshidojikarubonsanesuteruno seiho
FR2306701A1 (fr) * 1975-04-08 1976-11-05 Asahi Chemical Ind Derives de nucleotides
US4118484A (en) * 1976-03-29 1978-10-03 The Upjohn Company Method of treating rheumatoid arthritis
US4816570A (en) * 1982-11-30 1989-03-28 The Board Of Regents Of The University Of Texas System Biologically reversible phosphate and phosphonate protective groups
FR2556726B1 (fr) * 1983-12-20 1987-02-20 California Inst Of Techn Compositions a base d'oligonucleotides monocatenaires et procede pour leur preparation
DE3689223T2 (de) * 1985-05-15 1994-03-03 Amoco Corp Cytidinanaloga.
EP0216357A3 (fr) * 1985-09-25 1988-08-31 Nippon Zeon Co., Ltd. Composés phosphoramidites et leur procédé de préparation
ATE243039T1 (de) * 1987-10-28 2003-07-15 Wellstat Therapeutics Corp Acyldeoxyribonukleosid-derivate und verwendungen davon
US5470838A (en) 1987-10-28 1995-11-28 Pro-Neuron, Inc. Method of delivering exogenous uridine or cytidine using acylated uridine or cytidine
US6743782B1 (en) 1987-10-28 2004-06-01 Wellstat Therapeutics Corporation Acyl deoxyribonucleoside derivatives and uses thereof
DE3883374T2 (de) * 1987-10-28 1993-12-09 Pro Neuron Inc Acylatiertes uridin und cytidin und deren verwendungen.
KR100334695B1 (ko) * 1991-08-05 2002-04-27 리차아드제이마세이 표적화된 촉매 단백질에 의해 활성화되는 선구 약제

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3407191A (en) * 1966-08-29 1968-10-22 Lilly Co Eli Adamantoate esters of nucleosides

Also Published As

Publication number Publication date
GB1263408A (en) 1972-02-09
PH10225A (en) 1976-10-04
CA928290A (en) 1973-06-12
JPS5035077B1 (fr) 1975-11-13
FR2051563A1 (fr) 1971-04-09
IL34400A (en) 1974-05-16
DE2025624C2 (de) 1984-01-12
DE2025624A1 (de) 1970-12-03
NL7007505A (fr) 1970-12-01
US3847898A (en) 1974-11-12
CH586234A5 (fr) 1977-03-31
FR2051563B1 (fr) 1974-04-12
IL34400A0 (en) 1970-06-17

Similar Documents

Publication Publication Date Title
BE764179A (fr) " 5-azapyrimidine-nucleosides et leur procede de preparation
BE753635A (fr) " o-acyl-lysergols et leur preparation
BE772940A (fr) Azetidinones-(2) et leur preparation
BE751029A (fr) 5'-esters d'ara-cytidine et leur preparation
BE792906A (fr) Aryl-cetones et leur preparation
BE772990A (fr) Azetidinones-(2) et leur preparation
FR2009960A1 (fr) Nouveaux 1,3,4-oxazaborinides et leur preparation
BE783272A (fr) Triazolobenzodiazepines et leur preparation
BE787759A (fr) Thioloesters d'acides guanidine-organiques et leur preparation
BE758969A (fr) Alcoyl-adamantanes et leur preparation
BE785375A (fr) Thiolincosaminides et leur preparation
BE761438A (fr) Alpha-halo-phenylacetamides et leur preparation
BE769877A (fr) Composes de sulfinyl- et sulfonylpyridine et leur preparation
BE763671A (fr) Azidosulfonylcarbanilates et leur preparation
BE764456A (fr) Amino-3-cardenolides et leur preparation
BE767180A (fr) Composes anthraquinoniques et leur preparation
BE782846A (fr) Triazolobenzodiazepines substituees et leur preparation
BE750627A (fr) Thiocarboxylates d'organoetain et leur preparation
BE771463A (fr) Preparation d'halogeno-hydroxy-6-pyridone-2, et leur utilisation
BE762366A (fr) Quinobenzazepines basiques et leur preparation
BE772454A (fr) Pigments disazoiques et leur preparation
BE782851A (fr) Pyrimidines 2,5-bis-substituees et leur preparation
BE754021A (fr) Derives d'hydroxyisoquinuclidine et leur preparation
BE746442A (fr) Derives d'organo-etains et leur utilisation
BE756792A (fr) Poly-organosiloxanes modifies et leur preparation

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19860531