AU8873591A - Use of 2h-1,2,4-benzothiadiazine-3(4h)-thion-1,1-dioxides as antiviral medicaments - Google Patents

Use of 2h-1,2,4-benzothiadiazine-3(4h)-thion-1,1-dioxides as antiviral medicaments

Info

Publication number
AU8873591A
AU8873591A AU88735/91A AU8873591A AU8873591A AU 8873591 A AU8873591 A AU 8873591A AU 88735/91 A AU88735/91 A AU 88735/91A AU 8873591 A AU8873591 A AU 8873591A AU 8873591 A AU8873591 A AU 8873591A
Authority
AU
Australia
Prior art keywords
alkyl
benzothiadiazine
thion
dioxides
radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU88735/91A
Inventor
Bernhard Konig
Herbert Leinert
Ulrike Leser
Alfred Mertens
Hans Seidel
Harald Zilch
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roche Diagnostics GmbH
Original Assignee
Boehringer Mannheim GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim GmbH filed Critical Boehringer Mannheim GmbH
Publication of AU8873591A publication Critical patent/AU8873591A/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/15—Six-membered rings
    • C07D285/16—Thiadiazines; Hydrogenated thiadiazines
    • C07D285/18—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines
    • C07D285/20—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems
    • C07D285/22—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D285/24—1,2,4-Thiadiazines; Hydrogenated 1,2,4-thiadiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with oxygen atoms directly attached to the ring sulfur atom

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention relates to the novel use of compounds of formula (I) in which R1? is a hydrogen atom, a C1?-C6? alkyl radical or a phenyl radical optionally substituted by C1?-C6? alkyl; R2?-R4? are the same or different and may independently be a hydrogen or halogen atom, a C1?-C6? alkyl, a C1?-C6? alkoxy, a trifluoromethyl or aminosulphonyl radical; R is a hydrogen atom, a C1?-C6? alkyl or a phenyl-C1?-C6?-alkyl group, or their tautomers, for the production of medicaments for the treatment of viral or retroviral infections.
AU88735/91A 1990-11-16 1991-11-14 Use of 2h-1,2,4-benzothiadiazine-3(4h)-thion-1,1-dioxides as antiviral medicaments Abandoned AU8873591A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4036571A DE4036571A1 (en) 1990-11-16 1990-11-16 USE OF 2H-1,2,4-BENZOTHIADIAZIN-3 (4H) -THION-1,1-DIOXIDES AS ANTIVIRAL MEDICAMENTS
DE4036571 1990-11-16

Publications (1)

Publication Number Publication Date
AU8873591A true AU8873591A (en) 1992-06-11

Family

ID=6418404

Family Applications (1)

Application Number Title Priority Date Filing Date
AU88735/91A Abandoned AU8873591A (en) 1990-11-16 1991-11-14 Use of 2h-1,2,4-benzothiadiazine-3(4h)-thion-1,1-dioxides as antiviral medicaments

Country Status (7)

Country Link
EP (1) EP0557336B1 (en)
JP (1) JPH06502172A (en)
AT (1) ATE121937T1 (en)
AU (1) AU8873591A (en)
CA (1) CA2096239A1 (en)
DE (2) DE4036571A1 (en)
WO (1) WO1992008462A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4135479A1 (en) * 1991-10-28 1993-04-29 Goedecke Ag MEDICINES FOR TREATING AIDS

Also Published As

Publication number Publication date
DE59105404D1 (en) 1995-06-08
EP0557336B1 (en) 1995-05-03
JPH06502172A (en) 1994-03-10
ATE121937T1 (en) 1995-05-15
CA2096239A1 (en) 1992-05-17
EP0557336A1 (en) 1993-09-01
WO1992008462A1 (en) 1992-05-29
DE4036571A1 (en) 1992-05-21

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