AU7856194A - N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists - Google Patents

N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists

Info

Publication number
AU7856194A
AU7856194A AU78561/94A AU7856194A AU7856194A AU 7856194 A AU7856194 A AU 7856194A AU 78561/94 A AU78561/94 A AU 78561/94A AU 7856194 A AU7856194 A AU 7856194A AU 7856194 A AU7856194 A AU 7856194A
Authority
AU
Australia
Prior art keywords
thio
oxy
benzoyl
substance
receptor antagonists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU78561/94A
Inventor
Silvio Dr. Ofner
Silvio Roggo
Walter Schilling
Siem J Dr. Veenstra
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU7856194A publication Critical patent/AU7856194A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/54—Sulfur atoms
AU78561/94A 1993-10-26 1994-10-14 N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists Abandoned AU7856194A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH322393 1993-10-26
CH3223/93 1993-10-26
PCT/EP1994/003394 WO1995011895A1 (en) 1993-10-26 1994-10-14 N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists

Publications (1)

Publication Number Publication Date
AU7856194A true AU7856194A (en) 1995-05-22

Family

ID=4251310

Family Applications (1)

Application Number Title Priority Date Filing Date
AU78561/94A Abandoned AU7856194A (en) 1993-10-26 1994-10-14 N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists

Country Status (2)

Country Link
AU (1) AU7856194A (en)
WO (1) WO1995011895A1 (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0783490T3 (en) * 1994-09-30 2002-05-13 Novartis Ag 1-Acyl-4-aliphatic aminopiperidine compounds
RU2156250C2 (en) * 1995-04-24 2000-09-20 Новартис Аг Derivatives of chromone, method of their synthesis and pharmaceutical composition
NZ321575A (en) * 1995-10-30 1999-05-28 Janssen Pharmaceutica Nv 1-(1,2-disubstituted piperidinyl)-4- substituted piperazine derivatives
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
EP1858896B1 (en) 2005-03-08 2010-08-18 Janssen Pharmaceutica NV Diaza-spiro-[4.4]-nonane derivatives as neurokinin (nk1) antagonists
UA105182C2 (en) 2008-07-03 2014-04-25 Ньюрексон, Інк. Benzoxazines, benzothiazines, and related compounds having nos inhibitory activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8804104D0 (en) * 1988-02-23 1988-03-23 Glaxo Group Ltd Chemical compounds
DE69210029T2 (en) * 1991-08-20 1997-01-09 Merck Sharp & Dohme AZACYCLIC COMPOUNDS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM

Also Published As

Publication number Publication date
WO1995011895A1 (en) 1995-05-04

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