AU7679987A - New (benzofuran-2-yl) imidazoles having pharmaceutical activity, their salts and relevant production processes - Google Patents

New (benzofuran-2-yl) imidazoles having pharmaceutical activity, their salts and relevant production processes

Info

Publication number
AU7679987A
AU7679987A AU76799/87A AU7679987A AU7679987A AU 7679987 A AU7679987 A AU 7679987A AU 76799/87 A AU76799/87 A AU 76799/87A AU 7679987 A AU7679987 A AU 7679987A AU 7679987 A AU7679987 A AU 7679987A
Authority
AU
Australia
Prior art keywords
benzofuran
imidazoles
salts
new
production processes
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU76799/87A
Other versions
AU604042B2 (en
Inventor
Adriano Barzanti
Rossella Ciappi
Mario Ghelardoni
Danilo Giannotti
Alessandro Giolitti
Carlo Ortolani
Vittorio Pestillini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Menarini SAS
Original Assignee
Menarini SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini SAS filed Critical Menarini SAS
Publication of AU7679987A publication Critical patent/AU7679987A/en
Application granted granted Critical
Publication of AU604042B2 publication Critical patent/AU604042B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU76799/87A 1986-08-13 1987-08-12 New (benzofuran-2-yl) imidazoles having pharmaceutical activity, their salts and relevant production processes Ceased AU604042B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT8609461A IT1216256B (en) 1986-08-13 1986-08-13 (BENZOFURAN-2-IL) IMIDAZOLI, WITH PHARMACOLOGICAL ACTIVITY, THEIR SALTS AND RELATED MANUFACTURING PROCEDURES.
IT9461/86 1986-08-13

Publications (2)

Publication Number Publication Date
AU7679987A true AU7679987A (en) 1988-02-18
AU604042B2 AU604042B2 (en) 1990-12-06

Family

ID=11130481

Family Applications (1)

Application Number Title Priority Date Filing Date
AU76799/87A Ceased AU604042B2 (en) 1986-08-13 1987-08-12 New (benzofuran-2-yl) imidazoles having pharmaceutical activity, their salts and relevant production processes

Country Status (23)

Country Link
US (1) US4800208A (en)
EP (1) EP0257171B1 (en)
JP (1) JPS6372687A (en)
AR (1) AR243181A1 (en)
AT (1) ATE56008T1 (en)
AU (1) AU604042B2 (en)
CA (1) CA1325212C (en)
CS (1) CS272226B2 (en)
DD (1) DD270305A5 (en)
DE (1) DE3673822D1 (en)
DK (1) DK166917B1 (en)
ES (1) ES2037011T3 (en)
GR (1) GR3000903T3 (en)
HU (1) HU202864B (en)
IE (1) IE61019B1 (en)
IT (1) IT1216256B (en)
MX (1) MX7723A (en)
NO (1) NO170085C (en)
PL (1) PL149009B1 (en)
PT (1) PT85491B (en)
SU (1) SU1600630A3 (en)
YU (1) YU46222B (en)
ZA (1) ZA875908B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9212833D0 (en) * 1992-06-17 1992-07-29 Glaxo Group Ltd Chemical compounds
EP0574992A1 (en) * 1992-06-17 1993-12-22 Glaxo Group Limited 5-(1,2,4-Triazol-1-ylmethyl)-3H-isobenzofuran-1-one derivatives, their preparation and use as aromatase inhibitors
US5426196A (en) * 1993-12-22 1995-06-20 Glaxo Inc. Synthesis of diaryl methanes
IT1286866B1 (en) * 1996-10-28 1998-07-17 Menarini Farma Ind FURANO-HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS
US6503935B1 (en) 1998-08-07 2003-01-07 Abbott Laboratories Imidazoles and related compounds as α1A agonists
GB0223915D0 (en) * 2002-10-15 2002-11-20 Univ Cardiff Benzofuran derivatives formulations and uses thereof
CA2652280C (en) 2006-05-15 2014-01-28 Massachusetts Institute Of Technology Polymers for functional particles
MX350501B (en) 2007-10-12 2017-09-07 Massachusetts Inst Technology Vaccine nanotechnology.
US7762049B2 (en) 2008-12-31 2010-07-27 Black & Decker Inc. Electric mower having two-motion activation system
CN112063532B (en) * 2020-08-11 2022-05-24 浙江工业大学 Geotrichum linum and application thereof in preparation of (S) -1- (2-trifluoromethylphenyl) ethanol

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR6915465D0 (en) * 1969-03-07 1973-01-04 Bayer Ag PROCESS TO PREPARE SUBSTITUTED N-BENZIMIDAZOLES IN THE ALPHA POSITION BY PENTA-MEMBER HETEROCYCLES WITH ANTIMYCOTIC ACTIVITY
DE2009020C3 (en) * 1970-02-26 1979-09-13 Bayer Ag, 5090 Leverkusen Process for the preparation of N- (l, l, l-trisubstituted) -methylazoles
US3928348A (en) * 1970-03-23 1975-12-23 Bayer Ag N-methyl-imidazole derivatives and their production
IT1154888B (en) * 1980-11-12 1987-01-21 Menarini Sas 2-SUBSTITUTED BENZOFURAN DERIVATIVES AND RELATED METHODS OF PREPARATION
DE3049542A1 (en) * 1980-12-31 1982-07-29 Basf Ag, 6700 Ludwigshafen AZOLYLALKYL-2,3-DIHYDROBENZOFURANE, FUNGICIDES CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF
ZA825413B (en) * 1981-08-26 1983-06-29 Pfizer Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them
FI842502A (en) * 1983-06-27 1984-12-28 Ciba Geigy Ag FRAMEWORK FOR FRAMSTAELLNING AV NYA 2-SUBSTITUERADE BENSOFURAN DERIVAT.
DE3413363A1 (en) * 1984-04-09 1985-10-17 Merz + Co GmbH & Co, 6000 Frankfurt Benzofuran-2-ylethylimidazole derivatives, process for their preparation, and pharmaceuticals

Also Published As

Publication number Publication date
HUT46910A (en) 1988-12-28
MX7723A (en) 1993-12-01
ES2037011T3 (en) 1993-06-16
PL267298A1 (en) 1988-12-08
YU150787A (en) 1988-10-31
IT1216256B (en) 1990-02-22
DK166917B1 (en) 1993-08-02
CS272226B2 (en) 1991-01-15
ZA875908B (en) 1988-02-12
HU202864B (en) 1991-04-29
GR3000903T3 (en) 1991-12-10
NO170085C (en) 1992-09-09
NO873383L (en) 1988-02-15
DK418187A (en) 1988-02-14
PT85491B (en) 1990-06-29
JPS6372687A (en) 1988-04-02
PT85491A (en) 1987-09-01
EP0257171B1 (en) 1990-08-29
US4800208A (en) 1989-01-24
CS597887A2 (en) 1990-03-14
CA1325212C (en) 1993-12-14
IT8609461A0 (en) 1986-08-13
ATE56008T1 (en) 1990-09-15
PL149009B1 (en) 1989-12-30
DE3673822D1 (en) 1990-10-04
NO873383D0 (en) 1987-08-12
EP0257171A1 (en) 1988-03-02
IE61019B1 (en) 1994-09-07
NO170085B (en) 1992-06-01
YU46222B (en) 1993-05-28
IE872153L (en) 1988-02-13
DK418187D0 (en) 1987-08-11
DD270305A5 (en) 1989-07-26
AR243181A1 (en) 1993-07-30
AU604042B2 (en) 1990-12-06
SU1600630A3 (en) 1990-10-15

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