AU6734598A - Thiazolobenzoheterocycles, preparation and medicines containing same - Google Patents
Thiazolobenzoheterocycles, preparation and medicines containing sameInfo
- Publication number
- AU6734598A AU6734598A AU67345/98A AU6734598A AU6734598A AU 6734598 A AU6734598 A AU 6734598A AU 67345/98 A AU67345/98 A AU 67345/98A AU 6734598 A AU6734598 A AU 6734598A AU 6734598 A AU6734598 A AU 6734598A
- Authority
- AU
- Australia
- Prior art keywords
- alkyl
- alk
- ch2oh
- preparation
- nr11r12
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Saccharide Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
The invention concerns compounds of formula (I) in which R1 represents a sulphur or selenium atom, R2 represents hydrogen or alkyl, -R3-R4-R5- represents a chain of formula -CH2-CH2-CH2-, -CH(R7)-CH2-CH2-, -CH2-CH2-CH(R8)-, -CH2-CH(R9)-CH2-, -CH2-CH2-S-, -CH2-CH2-SO-, -CH2-CH2-SO2-, -CH2-CH2-Se-, -CH2-CH2-O-, -CH2-CH2-CO-, -CH2-CH2-N(R10)-, -CH2-CO-N(R10)-, -CH2-CF2-CH2-, -CH2-CF2-CH(OH)-, -CH2-CH(R13)-S-, -CH2-CH(R13)-SO-, or -CH2-CH(R13)-SO2-, R6 represents a polyfluoroalkyl, polyfluoroalcoxy or polyfluoroalkylthio radical, R7 represents alkyl, -CH2OH, -CH2-SO2-alk or -CH2-NR11R12, R8 represents alkyl, hydroxy, -CH2OH, -NR11R12, -CH2-NR11R12, -S-alk, -SO-alk, -SO2-alk, thienyl, furyl, phenyl, or phenyl substituted, R9 represents alkyl or -CH2OH, R10 represents hydrogen or alkyl, R11 represents hydrogen or alkyl, -CO-alk or -CO-CF3, R12 represents hydrogen or alkyl, or R11 and R12 form with the nitrogen atom to which they are bound a heterocyclic compound, R13 represents alkyl or -CH2OH, their salts, their methods of preparation, medicines containing them and the intermediates.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9702436A FR2760237B1 (en) | 1997-02-28 | 1997-02-28 | THIAZOLOBENZOHETEROCYCLES, THEIR PREPARATION AND THE MEDICINES CONTAINING THEM |
| FR9702436 | 1997-02-28 | ||
| PCT/FR1998/000376 WO1998038194A1 (en) | 1997-02-28 | 1998-02-26 | Thiazolobenzoheterocycles, preparation and medicines containing same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU6734598A true AU6734598A (en) | 1998-09-18 |
Family
ID=9504307
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU67345/98A Abandoned AU6734598A (en) | 1997-02-28 | 1998-02-26 | Thiazolobenzoheterocycles, preparation and medicines containing same |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP0966473B1 (en) |
| JP (1) | JP4436460B2 (en) |
| AT (1) | ATE221075T1 (en) |
| AU (1) | AU6734598A (en) |
| DE (1) | DE69806734T2 (en) |
| DK (1) | DK0966473T3 (en) |
| ES (1) | ES2180156T3 (en) |
| FR (1) | FR2760237B1 (en) |
| PT (1) | PT966473E (en) |
| WO (1) | WO1998038194A1 (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA90269C2 (en) * | 2004-04-02 | 2010-04-26 | Мицубиси Танабе Фарма Корпорейшн | Tetrahydroquinoline derivatives and a process for preparing the same |
| DE102005027168A1 (en) * | 2005-06-13 | 2006-12-14 | Merck Patent Gmbh | Tetrahydroquinolines |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3992378A (en) * | 1973-12-26 | 1976-11-16 | Eli Lilly And Company | Fluoralkyl quinoxadinediones |
| JPS55111406A (en) * | 1979-02-19 | 1980-08-28 | Takeda Chem Ind Ltd | Agent for controlling plant disease |
| DK160941C (en) * | 1988-06-28 | 1991-10-21 | Novo Nordisk As | CONDENSED 2,3-DIHYDROXYPYRAZINES, THEIR PROCEDURES FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THE COMPOUNDS |
| DE69016430T2 (en) * | 1989-06-09 | 1995-06-01 | Upjohn Co | HETEROCYCLIC AMINES WITH CNS EFFECTIVENESS. |
| ES2164639T3 (en) * | 1991-04-15 | 2002-03-01 | Aventis Pharma Gmbh | QUINOXALINAS, PROCEDURE FOR PREPARATION AND EMPLOYMENT. |
| EP0705835A1 (en) * | 1994-09-01 | 1996-04-10 | Ciba-Geigy Ag | Quinoxalic-2,3-diones with an oxa or thiaheterocyclic fused ring |
-
1997
- 1997-02-28 FR FR9702436A patent/FR2760237B1/en not_active Expired - Fee Related
-
1998
- 1998-02-26 ES ES98912552T patent/ES2180156T3/en not_active Expired - Lifetime
- 1998-02-26 AU AU67345/98A patent/AU6734598A/en not_active Abandoned
- 1998-02-26 DK DK98912552T patent/DK0966473T3/en active
- 1998-02-26 AT AT98912552T patent/ATE221075T1/en active
- 1998-02-26 WO PCT/FR1998/000376 patent/WO1998038194A1/en active IP Right Grant
- 1998-02-26 DE DE69806734T patent/DE69806734T2/en not_active Expired - Lifetime
- 1998-02-26 EP EP98912552A patent/EP0966473B1/en not_active Expired - Lifetime
- 1998-02-26 JP JP53738098A patent/JP4436460B2/en not_active Expired - Fee Related
- 1998-02-26 PT PT98912552T patent/PT966473E/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0966473B1 (en) | 2002-07-24 |
| PT966473E (en) | 2002-12-31 |
| FR2760237A1 (en) | 1998-09-04 |
| FR2760237B1 (en) | 1999-04-16 |
| ES2180156T3 (en) | 2003-02-01 |
| JP4436460B2 (en) | 2010-03-24 |
| ATE221075T1 (en) | 2002-08-15 |
| EP0966473A1 (en) | 1999-12-29 |
| DE69806734T2 (en) | 2002-12-05 |
| DE69806734D1 (en) | 2002-08-29 |
| WO1998038194A1 (en) | 1998-09-03 |
| JP2001517214A (en) | 2001-10-02 |
| DK0966473T3 (en) | 2002-11-18 |
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