AU6382701A - 2-hydroxy-mutilin carbamate derivatives for antibacterial use - Google Patents
2-hydroxy-mutilin carbamate derivatives for antibacterial useInfo
- Publication number
- AU6382701A AU6382701A AU6382701A AU6382701A AU6382701A AU 6382701 A AU6382701 A AU 6382701A AU 6382701 A AU6382701 A AU 6382701A AU 6382701 A AU6382701 A AU 6382701A AU 6382701 A AU6382701 A AU 6382701A
- Authority
- AU
- Australia
- Prior art keywords
- hydroxy
- carbamate derivatives
- antibacterial use
- mutilin carbamate
- mutilin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0008260.2A GB0008260D0 (en) | 2000-04-04 | 2000-04-04 | Novel compounds |
| GB0027182A GB0027182D0 (en) | 2000-11-04 | 2000-11-04 | Novel comounds |
| PCT/EP2001/003594 WO2001074788A1 (en) | 2000-04-04 | 2001-03-29 | 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU6382701A true AU6382701A (en) | 2001-10-15 |
Family
ID=26244040
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU6382701A Withdrawn AU6382701A (en) | 2000-04-04 | 2001-03-29 | 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
| AU2001263827A Ceased AU2001263827B2 (en) | 2000-04-04 | 2001-03-29 | 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001263827A Ceased AU2001263827B2 (en) | 2000-04-04 | 2001-03-29 | 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US6972297B2 (en) |
| EP (1) | EP1268443B1 (en) |
| JP (1) | JP2003529593A (en) |
| KR (1) | KR100758441B1 (en) |
| CN (1) | CN1210267C (en) |
| AR (1) | AR030203A1 (en) |
| AT (1) | ATE437860T1 (en) |
| AU (2) | AU6382701A (en) |
| BR (1) | BR0109809A (en) |
| CA (1) | CA2405132A1 (en) |
| CO (1) | CO5280223A1 (en) |
| CZ (1) | CZ20023290A3 (en) |
| DE (1) | DE60139382D1 (en) |
| ES (1) | ES2328109T3 (en) |
| HU (1) | HUP0300370A3 (en) |
| IL (1) | IL151887A0 (en) |
| MX (1) | MXPA02009816A (en) |
| NO (1) | NO324229B1 (en) |
| NZ (1) | NZ521536A (en) |
| PL (1) | PL358666A1 (en) |
| WO (1) | WO2001074788A1 (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0024811D0 (en) | 2000-10-10 | 2000-11-22 | Smithkline Beecham Plc | Novel compounds |
| US7176310B1 (en) | 2002-04-09 | 2007-02-13 | Ucb Sa | Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents |
| GB0209262D0 (en) * | 2002-04-23 | 2002-06-05 | Biochemie Gmbh | Organic compounds |
| AU2003257493A1 (en) * | 2002-07-24 | 2004-02-16 | Sandoz Ag | Pleuromutilin derivatives as antimicrobbials |
| GB0218578D0 (en) | 2002-08-09 | 2002-09-18 | Glaxo Group Ltd | Novel method |
| GB0308114D0 (en) * | 2003-04-08 | 2003-05-14 | Glaxo Group Ltd | Novel compounds |
| FR2856685B1 (en) * | 2003-06-25 | 2005-09-23 | Merck Sante Sas | THIAZOLYLPIPERIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| US20090291987A1 (en) * | 2004-12-13 | 2009-11-26 | Glaxo Group Limited | Novel polymorph of (5-amino-6-methoxy-3-pyridincarbonyl) carbamic acid 2-(s)-hydroxymutilin 14-ester |
| CA2591898A1 (en) * | 2004-12-27 | 2006-07-06 | Kyorin Pharmaceutical Co., Ltd. | Mutilin-derivative substituted at position 12 |
| WO2006099196A1 (en) * | 2005-03-10 | 2006-09-21 | Smithkline Beecham Corporation | Novel method |
| TW200738701A (en) | 2005-07-26 | 2007-10-16 | Du Pont | Fungicidal carboxamides |
| KR100695541B1 (en) * | 2005-10-31 | 2007-03-16 | 한국단자공업 주식회사 | Connecting terminal |
| WO2007079173A2 (en) * | 2005-12-30 | 2007-07-12 | Emergent Biosolutions Inc. | Novel 2-heteroaryloxy-phenol derivatives as antibacterial agents |
| JP5322927B2 (en) | 2007-05-24 | 2013-10-23 | 杏林製薬株式会社 | A mutilin derivative having a heteroaromatic carboxylic acid structure at the 14-position substituent. |
| EP2014640A1 (en) * | 2007-07-13 | 2009-01-14 | Nabriva Therapeutics AG | Pleuromutilin derivatives |
| JP2010100582A (en) * | 2008-10-24 | 2010-05-06 | Kyorin Pharmaceut Co Ltd | Mutilin derivative containing heteroaromatic ring carboxylic acid structure at 14-position substituent |
| EP2184273A1 (en) | 2008-11-05 | 2010-05-12 | Bayer CropScience AG | Halogen substituted compounds as pesticides |
| EP2253617A1 (en) | 2009-05-20 | 2010-11-24 | Bayer CropScience AG | Halogenated compounds as pesticides |
| MX2017015812A (en) * | 2015-06-17 | 2018-07-06 | Nabriva Therapeutics GmbH | Injectable pharmaceutical formulations of lefamulin. |
| KR20210131341A (en) * | 2019-02-27 | 2021-11-02 | 오티카라 인코포레이티드 | Methods of treating nasal, sinus, and nasopharyngeal tissue infections and/or inflammations |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL327737A1 (en) | 1996-01-03 | 1998-12-21 | Smithkline Beecham Plc | Carbamoyloxylic derivatives of mutiline and their application as bactericides |
| HUP0001741A3 (en) | 1996-08-02 | 2000-11-28 | Smithkline Beecham Plc | Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use, process for preparing them, pharmaceuticals contg. them and their use |
| UY25225A1 (en) | 1997-10-29 | 2000-12-29 | Smithkline Beecham Plc | PLEUROMUTILINE DERIVATIVES USEFUL AS ANTIMICROBIAL AGENTS |
| FR2771008B1 (en) | 1997-11-17 | 2000-04-28 | Hoechst Marion Roussel Inc | USE OF KETOLIDES FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS FOR PREVENTING ARTERIAL THROMBOTIC COMPLICATIONS LINKED TO ATHEROSCLEROSIS |
| GB9817029D0 (en) * | 1998-08-05 | 1998-09-30 | Smithkline Beecham Plc | Novel compounds |
-
2001
- 2001-03-29 JP JP2001572483A patent/JP2003529593A/en active Pending
- 2001-03-29 WO PCT/EP2001/003594 patent/WO2001074788A1/en active IP Right Grant
- 2001-03-29 AU AU6382701A patent/AU6382701A/en not_active Withdrawn
- 2001-03-29 CN CNB018091989A patent/CN1210267C/en not_active Expired - Fee Related
- 2001-03-29 NZ NZ521536A patent/NZ521536A/en unknown
- 2001-03-29 EP EP01938069A patent/EP1268443B1/en not_active Expired - Lifetime
- 2001-03-29 HU HU0300370A patent/HUP0300370A3/en unknown
- 2001-03-29 PL PL01358666A patent/PL358666A1/en not_active Application Discontinuation
- 2001-03-29 CA CA002405132A patent/CA2405132A1/en not_active Abandoned
- 2001-03-29 IL IL15188701A patent/IL151887A0/en unknown
- 2001-03-29 AU AU2001263827A patent/AU2001263827B2/en not_active Ceased
- 2001-03-29 BR BR0109809-8A patent/BR0109809A/en not_active Application Discontinuation
- 2001-03-29 AT AT01938069T patent/ATE437860T1/en not_active IP Right Cessation
- 2001-03-29 ES ES01938069T patent/ES2328109T3/en not_active Expired - Lifetime
- 2001-03-29 US US10/240,908 patent/US6972297B2/en not_active Expired - Fee Related
- 2001-03-29 MX MXPA02009816A patent/MXPA02009816A/en active IP Right Grant
- 2001-03-29 DE DE60139382T patent/DE60139382D1/en not_active Expired - Lifetime
- 2001-03-29 KR KR1020027013202A patent/KR100758441B1/en not_active IP Right Cessation
- 2001-03-29 CZ CZ20023290A patent/CZ20023290A3/en unknown
- 2001-03-30 CO CO01025487A patent/CO5280223A1/en not_active Application Discontinuation
- 2001-03-30 AR ARP010101559A patent/AR030203A1/en not_active Application Discontinuation
-
2002
- 2002-10-02 NO NO20024745A patent/NO324229B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE60139382D1 (en) | 2009-09-10 |
| BR0109809A (en) | 2003-01-21 |
| KR20030011815A (en) | 2003-02-11 |
| JP2003529593A (en) | 2003-10-07 |
| EP1268443B1 (en) | 2009-07-29 |
| ATE437860T1 (en) | 2009-08-15 |
| NZ521536A (en) | 2004-05-28 |
| CO5280223A1 (en) | 2003-05-30 |
| CN1210267C (en) | 2005-07-13 |
| ES2328109T3 (en) | 2009-11-10 |
| EP1268443A1 (en) | 2003-01-02 |
| IL151887A0 (en) | 2003-04-10 |
| NO20024745L (en) | 2002-11-19 |
| CA2405132A1 (en) | 2001-10-11 |
| AR030203A1 (en) | 2003-08-13 |
| US6972297B2 (en) | 2005-12-06 |
| PL358666A1 (en) | 2004-08-09 |
| NO324229B1 (en) | 2007-09-10 |
| KR100758441B1 (en) | 2007-09-14 |
| AU2001263827B2 (en) | 2004-06-17 |
| NO20024745D0 (en) | 2002-10-02 |
| MXPA02009816A (en) | 2003-03-27 |
| WO2001074788A1 (en) | 2001-10-11 |
| CN1427827A (en) | 2003-07-02 |
| US20030114674A1 (en) | 2003-06-19 |
| HUP0300370A3 (en) | 2005-07-28 |
| HUP0300370A2 (en) | 2003-06-28 |
| CZ20023290A3 (en) | 2003-03-12 |
| WO2001074788A8 (en) | 2001-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase | ||
| TH | Corrigenda |
Free format text: IN VOL 16, NO 10, PAGE(S) 2150-2167 UNDER THE HEADING APPLICATIONS LAPSED, REFUSED OR WITHDRAWN PLEASE DELETE ALL REFERENCE TO APPLICATION NO. 39411/01, 46763/01, 46764/01, 46785/01, 60038/01, 63827/01, 67264/01 AND 73786/01 |