AU568575B2 - Avermectin epoxide derivatives - Google Patents

Avermectin epoxide derivatives

Info

Publication number
AU568575B2
AU568575B2 AU33772/84A AU3377284A AU568575B2 AU 568575 B2 AU568575 B2 AU 568575B2 AU 33772/84 A AU33772/84 A AU 33772/84A AU 3377284 A AU3377284 A AU 3377284A AU 568575 B2 AU568575 B2 AU 568575B2
Authority
AU
Australia
Prior art keywords
avermectin
epoxide derivatives
epoxide
derivatives
avermectin epoxide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU33772/84A
Other versions
AU3377284A (en
Inventor
Helmut H. Mrozik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU3377284A publication Critical patent/AU3377284A/en
Application granted granted Critical
Publication of AU568575B2 publication Critical patent/AU568575B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/195—Antibiotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
AU33772/84A 1983-10-03 1984-10-02 Avermectin epoxide derivatives Ceased AU568575B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US538612 1983-10-03
US06/538,612 US4530921A (en) 1983-10-03 1983-10-03 Avermectin epoxide derivatives and method of use

Publications (2)

Publication Number Publication Date
AU3377284A AU3377284A (en) 1985-04-18
AU568575B2 true AU568575B2 (en) 1988-01-07

Family

ID=24147656

Family Applications (1)

Application Number Title Priority Date Filing Date
AU33772/84A Ceased AU568575B2 (en) 1983-10-03 1984-10-02 Avermectin epoxide derivatives

Country Status (7)

Country Link
US (1) US4530921A (en)
EP (1) EP0136892B1 (en)
JP (1) JPS6094983A (en)
AU (1) AU568575B2 (en)
DE (1) DE3468216D1 (en)
NZ (1) NZ209652A (en)
ZA (1) ZA847732B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK614084A (en) * 1983-12-30 1985-07-01 Ciba Geigy Ag MILBEMYCIM DERIVATIVES AND THEIR PREPARATION AND USE
US4666937A (en) * 1985-03-04 1987-05-19 Merck & Co., Inc. Avermectin bioconversion products
JPH0678342B2 (en) * 1986-01-07 1994-10-05 三共株式会社 New macrolide compound
GB8606108D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Chemical compounds
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4876272A (en) * 1987-03-06 1989-10-24 American Cyanamid Company Mono- and diepoxide derivatives of LL-F28249 compounds
US4886829A (en) * 1987-03-06 1989-12-12 American Cyanamid Company 23-Oxo (keto) and 23-imino derivatives of mono- and diepoxy LL-F28249 compounds
US4851428A (en) * 1987-03-06 1989-07-25 American Cyanamid Company Mono- and diepoxide derivatives of Δ22-LL-F28249 compounds
US4956479A (en) * 1987-03-06 1990-09-11 American Cyanamid Company 23-deoxy-27-chloro derivatives of LL-F28249 compounds
US4886830A (en) * 1987-03-06 1989-12-12 American Cyanamid Company Mono- and diepoxide derivatives of 23-deoxyl-LL-F28249 compounds
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives
NZ233792A (en) * 1989-06-02 1992-06-25 Merck & Co Inc Avermectin 3,4-epoxide derivatives; pesticidal compositions
US5140042A (en) * 1990-09-12 1992-08-18 Merck & Co., Inc. 28-hydroxy ivermectin aglycone
CA2105251C (en) * 1992-09-01 2004-12-07 Mitsugi Shibano Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4310519A (en) * 1976-04-19 1982-01-12 Merck & Co., Inc. Novel substances and process for their production

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4056616A (en) * 1976-03-05 1977-11-01 Schering Corporation Rosamicin derivatives and method of using same
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
NZ201681A (en) * 1981-09-03 1985-11-08 Merck & Co Inc Avermectin derivatives and parasiticidal compositions
US4454314A (en) * 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4310519A (en) * 1976-04-19 1982-01-12 Merck & Co., Inc. Novel substances and process for their production
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076

Also Published As

Publication number Publication date
JPS6094983A (en) 1985-05-28
DE3468216D1 (en) 1988-02-04
NZ209652A (en) 1988-04-29
JPH0461876B2 (en) 1992-10-02
EP0136892A2 (en) 1985-04-10
AU3377284A (en) 1985-04-18
ZA847732B (en) 1986-05-28
EP0136892B1 (en) 1987-12-23
EP0136892A3 (en) 1985-05-08
US4530921A (en) 1985-07-23

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