AU558707B2 - Water soluble rifamycin derivatives - Google Patents
Water soluble rifamycin derivativesInfo
- Publication number
- AU558707B2 AU558707B2 AU29411/84A AU2941184A AU558707B2 AU 558707 B2 AU558707 B2 AU 558707B2 AU 29411/84 A AU29411/84 A AU 29411/84A AU 2941184 A AU2941184 A AU 2941184A AU 558707 B2 AU558707 B2 AU 558707B2
- Authority
- AU
- Australia
- Prior art keywords
- water soluble
- derivatives
- rifamycin derivatives
- rifampicin
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 title abstract 2
- HJYYPODYNSCCOU-ODRIEIDWSA-N rifamycin SV Chemical class OC1=C(C(O)=C2C)C3=C(O)C=C1NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@H](C)[C@@H](OC)\C=C\O[C@@]1(C)OC2=C3C1=O HJYYPODYNSCCOU-ODRIEIDWSA-N 0.000 title 1
- JQXXHWHPUNPDRT-WLSIYKJHSA-N rifampicin Chemical class O([C@](C1=O)(C)O/C=C/[C@@H]([C@H]([C@@H](OC(C)=O)[C@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@@H](C)\C=C\C=C(C)/C(=O)NC=2C(O)=C3C([O-])=C4C)C)OC)C4=C1C3=C(O)C=2\C=N\N1CC[NH+](C)CC1 JQXXHWHPUNPDRT-WLSIYKJHSA-N 0.000 abstract 2
- 125000005041 acyloxyalkyl group Chemical group 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000007864 aqueous solution Substances 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 238000007911 parenteral administration Methods 0.000 abstract 1
- 229960001225 rifampicin Drugs 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Cephalosporin Compounds (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838318072A GB8318072D0 (en) | 1983-07-04 | 1983-07-04 | Water-soluble rifampicin derivatives |
| GB8318072 | 1983-07-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2941184A AU2941184A (en) | 1985-01-10 |
| AU558707B2 true AU558707B2 (en) | 1987-02-05 |
Family
ID=10545208
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU29411/84A Ceased AU558707B2 (en) | 1983-07-04 | 1984-06-15 | Water soluble rifamycin derivatives |
Country Status (17)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU571956B2 (en) * | 1984-04-06 | 1988-04-28 | Dobfar S.P.A. | 3-azinomethyl rifamycins |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR890701591A (ko) * | 1987-09-25 | 1989-12-21 | 베르너 발데그 | 4-(트리알킬벤질)-피페라지닐 화합물의 디아실 유도체 |
| US5180718A (en) * | 1989-03-02 | 1993-01-19 | Ciba-Geigy Corporation | Acyl derivatives of oxazolorifamycins |
| US6143740A (en) * | 1996-11-19 | 2000-11-07 | Georgetown University | Heregulin antagonists and methods for their use |
| CA2465846A1 (en) * | 2001-11-21 | 2003-06-05 | Activbiotics, Inc. | Targeted therapeutics and uses thereof |
| US7137963B2 (en) * | 2002-08-26 | 2006-11-21 | Flowcardia, Inc. | Ultrasound catheter for disrupting blood vessel obstructions |
| US7820652B2 (en) * | 2003-09-24 | 2010-10-26 | Activbiotics Pharma, Llc | Regimen for the administration of rifamycin-class antibiotics |
| WO2015157512A1 (en) * | 2014-04-11 | 2015-10-15 | Drexel University | Novel methods and kits for detecting a rifamycin, or derivative or analogue thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR208F (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1964-07-31 | |||
| GB1159267A (en) * | 1966-11-03 | 1969-07-23 | Lepetit Spa | Rifamycin Derivatives |
| NL145554B (nl) * | 1967-06-07 | 1975-04-15 | Lepetit Spa | Werkwijze voor het bereiden van een 3-formylrifamycine sv-derivaat |
| AR207763A1 (es) * | 1973-07-25 | 1976-10-29 | Archifar Ind Chim Trentino | Metodo para la preparacion de 1,3-oxacino(5,6-c)rifamicinas |
| GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
| US4298692A (en) * | 1979-01-25 | 1981-11-03 | Ciba-Geigy Corporation | Fermentation process for producing a rifamycin derivative |
| US4411896A (en) * | 1981-06-03 | 1983-10-25 | Ciba-Geigy Corporation | Rifamycins, their compositions and use as antibiotics |
-
1983
- 1983-07-04 GB GB838318072A patent/GB8318072D0/en active Pending
-
1984
- 1984-06-15 AU AU29411/84A patent/AU558707B2/en not_active Ceased
- 1984-06-17 EP EP84106938A patent/EP0133887B1/en not_active Expired
- 1984-06-17 AT AT84106938T patent/ATE29136T1/de not_active IP Right Cessation
- 1984-06-17 DE DE8484106938T patent/DE3465597D1/de not_active Expired
- 1984-06-20 ZA ZA844661A patent/ZA844661B/xx unknown
- 1984-06-26 DK DK311484A patent/DK157875C/da active
- 1984-06-27 IL IL72234A patent/IL72234A/xx unknown
- 1984-06-27 PH PH30892A patent/PH20342A/en unknown
- 1984-06-29 US US06/626,358 patent/US4585589A/en not_active Expired - Fee Related
- 1984-07-02 JP JP59135371A patent/JPS6036490A/ja active Granted
- 1984-07-03 ES ES533957A patent/ES533957A0/es active Granted
- 1984-07-03 IE IE1693/84A patent/IE57930B1/en not_active IP Right Cessation
- 1984-07-03 NZ NZ208757A patent/NZ208757A/en unknown
- 1984-07-03 KR KR1019840003836A patent/KR910005847B1/ko not_active Expired
- 1984-07-03 HU HU842575A patent/HU190576B/hu not_active IP Right Cessation
- 1984-07-03 CA CA000457960A patent/CA1212670A/en not_active Expired
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU571956B2 (en) * | 1984-04-06 | 1988-04-28 | Dobfar S.P.A. | 3-azinomethyl rifamycins |
Also Published As
| Publication number | Publication date |
|---|---|
| CA1212670A (en) | 1986-10-14 |
| NZ208757A (en) | 1987-08-31 |
| JPS6036490A (ja) | 1985-02-25 |
| HU190576B (en) | 1986-09-29 |
| EP0133887A1 (en) | 1985-03-13 |
| GB8318072D0 (en) | 1983-08-03 |
| AU2941184A (en) | 1985-01-10 |
| DK311484D0 (da) | 1984-06-26 |
| IE57930B1 (en) | 1993-05-19 |
| ATE29136T1 (de) | 1987-09-15 |
| ES8601949A1 (es) | 1985-11-01 |
| ES533957A0 (es) | 1985-11-01 |
| DK157875C (da) | 1990-08-20 |
| KR910005847B1 (ko) | 1991-08-05 |
| PH20342A (en) | 1986-12-04 |
| DK157875B (da) | 1990-02-26 |
| DE3465597D1 (en) | 1987-10-01 |
| IL72234A0 (en) | 1984-10-31 |
| HUT36128A (en) | 1985-08-28 |
| IE841693L (en) | 1985-01-04 |
| KR850001207A (ko) | 1985-03-16 |
| US4585589A (en) | 1986-04-29 |
| EP0133887B1 (en) | 1987-08-26 |
| IL72234A (en) | 1987-09-16 |
| JPH0544467B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1993-07-06 |
| DK311484A (da) | 1985-01-05 |
| ZA844661B (en) | 1985-04-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU7162487A (en) | Cephalosporin derivatives | |
| IE782546L (en) | Amino-thiazolyl cephalosporins | |
| AU558707B2 (en) | Water soluble rifamycin derivatives | |
| NZ211594A (en) | The preparation of certain cephalosporin derivatives | |
| GR860382B (en) | Process for the preparation of heterocyclic derivatives | |
| UA8042A1 (uk) | Спосіб отримання поліциклічного ефірного антибіотика або його фармацевтично прийнятної катіонної солі | |
| AU566944B2 (en) | Preparation of 3-cephem derivatives | |
| AU8163287A (en) | Cephalosporin derivatives | |
| HUT41053A (en) | Process for preparing ester derivatives of l 17046 antibiotic | |
| AU1313488A (en) | Process for the preparation of nitroethene derivatives | |
| PH24371A (en) | An intermediate compound of cephalosporin derivatives | |
| AU3760489A (en) | Derivatives of cyclic amp as treatment for cancer | |
| CS8000660A2 (en) | Method of penicillin's or cephalosporin's derivatives preparation | |
| AU1271488A (en) | 27-halo derivatives of LL-F28249 compounds | |
| AU1271188A (en) | Mono- and diepoxide derivatives of ll-f28249 compounds | |
| AU6423386A (en) | Process for the preparation of sodium amoxycillin | |
| AU6485986A (en) | Derivatives of quinuclidine | |
| NO851488L (no) | Fremgangsmaate for fremstilling av cefalosporin-derivater | |
| EP0242551A3 (en) | Process for the preparation of diaziridines and their derivatives | |
| AU585973B2 (en) | Process for the preparation of eburnamenine derivatives | |
| ZA89130B (en) | Preparation of 5,8,13,14-tetrahydrobenz(5,6)isoindolo(2,1-b)isoquinolin-8,13-dione derivatives | |
| AU8412682A (en) | Preparation of pyrazine derivatives | |
| AU1271588A (en) | Mono- and diepoxide derivatives of 23-deoxy-LL-F28249 compounds | |
| IE862910L (en) | Crystalline cephalosporin monohydrate | |
| PT83111B (en) | Process for the preparation of heterocyclic derivatives of dihydroquinoline |