AU4607497A - Synthesis of aromatic compounds by diels-alder reaction on solid support - Google Patents

Synthesis of aromatic compounds by diels-alder reaction on solid support

Info

Publication number
AU4607497A
AU4607497A AU46074/97A AU4607497A AU4607497A AU 4607497 A AU4607497 A AU 4607497A AU 46074/97 A AU46074/97 A AU 46074/97A AU 4607497 A AU4607497 A AU 4607497A AU 4607497 A AU4607497 A AU 4607497A
Authority
AU
Australia
Prior art keywords
diels
synthesis
solid support
aromatic compounds
alder reaction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU46074/97A
Inventor
James S. Panek
Bin Zhu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boston University
Original Assignee
Boston University
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boston University filed Critical Boston University
Publication of AU4607497A publication Critical patent/AU4607497A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU46074/97A 1996-10-02 1997-10-01 Synthesis of aromatic compounds by diels-alder reaction on solid support Abandoned AU4607497A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US2724696P 1996-10-02 1996-10-02
US60027246 1996-10-02
US2998496P 1996-11-04 1996-11-04
US60029984 1996-11-04
PCT/US1997/017940 WO1998016508A2 (en) 1996-10-02 1997-10-01 Synthesis of aromatic compounds by diels-alder reaction on solid support

Publications (1)

Publication Number Publication Date
AU4607497A true AU4607497A (en) 1998-05-11

Family

ID=26702235

Family Applications (1)

Application Number Title Priority Date Filing Date
AU46074/97A Abandoned AU4607497A (en) 1996-10-02 1997-10-01 Synthesis of aromatic compounds by diels-alder reaction on solid support

Country Status (2)

Country Link
AU (1) AU4607497A (en)
WO (1) WO1998016508A2 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458789B1 (en) * 1999-09-29 2002-10-01 Lion Bioscience Ag 2-aminopyridine derivatives and combinatorial libraries thereof
US7172905B2 (en) 2001-08-07 2007-02-06 The University Of Chicago Polypeptide immobilization
WO2003032903A2 (en) 2001-10-12 2003-04-24 New York University Trisubstituted triazines compounds with antitubulin activity
KR101238525B1 (en) * 2004-12-31 2013-02-28 레디 유에스 테라퓨틱스 인코포레이티드 Novel benzylamine derivatives as cetp inhibitors
US7592451B2 (en) 2005-06-23 2009-09-22 New York University Treatment for diabetes and obesity as well as method of screening compounds useful for such treatments
EP1867638A1 (en) * 2006-06-16 2007-12-19 Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts Procedure for the Conection of two Molecules via Diels-Alder Reactions with Inverse Electron Demand
US20220371973A1 (en) * 2019-07-05 2022-11-24 Medimmune, Llc Method and Molecules
CN110563663A (en) * 2019-10-28 2019-12-13 南京红杉生物科技有限公司 valdecoxib and synthetic method thereof

Also Published As

Publication number Publication date
WO1998016508A2 (en) 1998-04-23

Similar Documents

Publication Publication Date Title
AU8589698A (en) Selective synthesis of organodiphosphite compounds
AU4583997A (en) Apparatus for the chemical synthesis of molecular arrays
AU2594697A (en) Nitroxyl containing compounds
AU4705697A (en) Systems and methods for the synthesis of organic compounds
AU6049396A (en) Novel urea- and thiourea-type compounds
AU1430499A (en) Production of catalysts for olefin conversion
AU6811298A (en) System and methods for parallel synthesis of organic compounds
AU4754893A (en) Activation of hydrocarbon synthesis catalyst
AU5147498A (en) Synthesis of large crystal zeolites
AU3224497A (en) Processes for the synthesis of sialyl lewisx compounds
AU8056898A (en) Synthesis of intermediates useful in preparing bromo-substituted tricyclic compounds
AU7287598A (en) Process for the conversion of hydrocarbons
AU2280697A (en) Support for the synthesis of modular polymers
AU5372598A (en) Tfpx synthesis
AU4233096A (en) Azepine synthesis via a diels-alder reaction
AU9025898A (en) Solid phase synthesis of 2,3-disubstituted indole compounds
AU4607497A (en) Synthesis of aromatic compounds by diels-alder reaction on solid support
AU6944798A (en) Solid phase synthesis of immunosuppressive agents
AU5521498A (en) An improved synthesis of cyclopropylacetylene
AU2217797A (en) Synthesis of indolylmaleimides
AU2609997A (en) Plate for reaction system
AU4157097A (en) Synthesis of bisindolylmalimides
AU4945697A (en) Solid phase synthesis of heterocyclic compounds
AU5135796A (en) Novel intermediates for the synthesis of trifluoromethylated organic compounds
AU2429097A (en) Fixed bed conversion of methoxy compounds to olefins