AU4540096A - Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics - Google Patents
Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibioticsInfo
- Publication number
- AU4540096A AU4540096A AU45400/96A AU4540096A AU4540096A AU 4540096 A AU4540096 A AU 4540096A AU 45400/96 A AU45400/96 A AU 45400/96A AU 4540096 A AU4540096 A AU 4540096A AU 4540096 A AU4540096 A AU 4540096A
- Authority
- AU
- Australia
- Prior art keywords
- pct
- amide derivatives
- antibiotics
- sec
- oxazoline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
PCT No. PCT/EP96/00425 Sec. 371 Date Jul. 31, 1997 Sec. 102(e) Date Jul. 31, 1997 PCT Filed Feb. 1, 1996 PCT Pub. No. WO96/24608 PCT Pub. Date Aug. 15, 1996The present invention refers to basic oxazoline-amide derivatives of GE 2270 and GE 2270-like antibiotics of general formula (I), wherein the group GE represents the antibiotic core molecule. The amide derivatives of antibiotic GE 2270 of formula (I) are antimicrobial agents mainly active against gram positive bacteria. <IMAGE> (I)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP95101596 | 1995-02-07 | ||
EP95101596 | 1995-02-07 | ||
PCT/EP1996/000425 WO1996024608A1 (en) | 1995-02-07 | 1996-02-01 | Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics |
Publications (2)
Publication Number | Publication Date |
---|---|
AU4540096A true AU4540096A (en) | 1996-08-27 |
AU693989B2 AU693989B2 (en) | 1998-07-09 |
Family
ID=8218960
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU45400/96A Ceased AU693989B2 (en) | 1995-02-07 | 1996-02-01 | Basic oxazoline-amide derivatives of GE 2270 and GE 2270-like antibiotics |
Country Status (13)
Country | Link |
---|---|
US (1) | US5891869A (en) |
EP (1) | EP0808326B1 (en) |
JP (1) | JP3518606B2 (en) |
KR (1) | KR100394930B1 (en) |
AT (1) | ATE205505T1 (en) |
AU (1) | AU693989B2 (en) |
CA (1) | CA2212437A1 (en) |
DE (1) | DE69615155T2 (en) |
DK (1) | DK0808326T3 (en) |
ES (1) | ES2161344T3 (en) |
PT (1) | PT808326E (en) |
SI (1) | SI0808326T1 (en) |
WO (1) | WO1996024608A1 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU714958B2 (en) * | 1996-02-14 | 2000-01-13 | Vicuron Pharmaceuticals Inc. | Derivatives of antibiotic GE2270 factors C2a D2 and E |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0801655T3 (en) * | 1995-02-07 | 1999-02-08 | Biosearch Italia Spa | Basic prolinamide derivatives of GE 2270 and GE 2270-like antibiotics |
CA2404273A1 (en) * | 2000-04-11 | 2001-10-18 | Bristol-Myers Squibb Pharma Company | Substituted lactams as inhibitors of a.beta. protein production |
MXPA05005338A (en) | 2002-11-18 | 2005-12-14 | Vicuron Pharm Inc | Methods of administering dalbavancin for treatment of bacterial infections. |
US20060074014A1 (en) * | 2002-11-18 | 2006-04-06 | Vicuron Pharmaceuticals Inc. | Dalbavancin compositions for treatment of bacterial infections |
US7119061B2 (en) * | 2002-11-18 | 2006-10-10 | Vicuron Pharmaceuticals, Inc. | Dalbavancin compositions for treatment of bacterial infections |
US7035113B2 (en) * | 2003-01-30 | 2006-04-25 | Endicott Interconnect Technologies, Inc. | Multi-chip electronic package having laminate carrier and method of making same |
CA2455024A1 (en) * | 2003-01-30 | 2004-07-30 | Endicott Interconnect Technologies, Inc. | Stacked chip electronic package having laminate carrier and method of making same |
US7023707B2 (en) * | 2003-01-30 | 2006-04-04 | Endicott Interconnect Technologies, Inc. | Information handling system |
US6828514B2 (en) * | 2003-01-30 | 2004-12-07 | Endicott Interconnect Technologies, Inc. | High speed circuit board and method for fabrication |
PE20121011A1 (en) * | 2006-05-31 | 2012-08-25 | Novartis Ag | AMINOTIZOLES AS MODULATORS OF THE ELONGATION FACTOR EF-Tu |
EP2097423B1 (en) * | 2006-12-20 | 2011-03-02 | Novartis AG | Aminothiazole macrocycles, their use as antibacterial compounds and processes for their production |
JP5286366B2 (en) | 2007-12-12 | 2013-09-11 | ノバルティス アーゲー | Aminothiazoles and uses thereof |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5202241A (en) * | 1988-09-09 | 1993-04-13 | Gruppo Lepetit S.P.A. | Antibiotic GE 2270 |
DE69016284T2 (en) | 1989-07-04 | 1995-05-24 | Lepetit Spa | Antibiotic GE 22270, factors A1, A2, A3 and H. |
DE69108972T2 (en) * | 1990-03-08 | 1995-10-19 | Lepetit Spa | Antibiotics GE 2270 factors B1, B2, C1, D1, D2, E and T. |
IL100572A (en) * | 1991-01-03 | 1997-01-10 | Lepetit Spa | Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them |
DE69224497T2 (en) * | 1991-08-30 | 1998-07-02 | Biosearch Italia Spa | Factor C2a of the antibiotic CE 2270 |
DK0801655T3 (en) * | 1995-02-07 | 1999-02-08 | Biosearch Italia Spa | Basic prolinamide derivatives of GE 2270 and GE 2270-like antibiotics |
EP0880541B1 (en) * | 1996-02-14 | 2003-01-15 | Biosearch Italia S.p.A. | Derivatives of antibiotic ge2270 factors |
-
1996
- 1996-02-01 JP JP52395596A patent/JP3518606B2/en not_active Expired - Fee Related
- 1996-02-01 ES ES96901344T patent/ES2161344T3/en not_active Expired - Lifetime
- 1996-02-01 AT AT96901344T patent/ATE205505T1/en not_active IP Right Cessation
- 1996-02-01 WO PCT/EP1996/000425 patent/WO1996024608A1/en active IP Right Grant
- 1996-02-01 KR KR1019970705392A patent/KR100394930B1/en not_active IP Right Cessation
- 1996-02-01 US US08/875,715 patent/US5891869A/en not_active Expired - Fee Related
- 1996-02-01 CA CA002212437A patent/CA2212437A1/en not_active Abandoned
- 1996-02-01 DE DE69615155T patent/DE69615155T2/en not_active Expired - Fee Related
- 1996-02-01 AU AU45400/96A patent/AU693989B2/en not_active Ceased
- 1996-02-01 PT PT96901344T patent/PT808326E/en unknown
- 1996-02-01 SI SI9630306T patent/SI0808326T1/en unknown
- 1996-02-01 DK DK96901344T patent/DK0808326T3/en active
- 1996-02-01 EP EP96901344A patent/EP0808326B1/en not_active Expired - Lifetime
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU714958B2 (en) * | 1996-02-14 | 2000-01-13 | Vicuron Pharmaceuticals Inc. | Derivatives of antibiotic GE2270 factors C2a D2 and E |
Also Published As
Publication number | Publication date |
---|---|
SI0808326T1 (en) | 2001-12-31 |
ES2161344T3 (en) | 2001-12-01 |
KR100394930B1 (en) | 2003-12-18 |
JP3518606B2 (en) | 2004-04-12 |
KR19980701995A (en) | 1998-06-25 |
AU693989B2 (en) | 1998-07-09 |
EP0808326B1 (en) | 2001-09-12 |
CA2212437A1 (en) | 1996-08-15 |
DE69615155D1 (en) | 2001-10-18 |
WO1996024608A1 (en) | 1996-08-15 |
EP0808326A1 (en) | 1997-11-26 |
US5891869A (en) | 1999-04-06 |
DE69615155T2 (en) | 2002-01-17 |
JPH10513461A (en) | 1998-12-22 |
PT808326E (en) | 2002-02-28 |
DK0808326T3 (en) | 2001-10-01 |
ATE205505T1 (en) | 2001-09-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Assignment registered |
Owner name: VERSICOR INC Free format text: FORMER OWNER WAS: BIOSEARCH ITALIA S.P.A. |
|
HB | Alteration of name in register |
Owner name: VICURON PHARMACEUTICALS INC. Free format text: FORMER NAME WAS: VERSICOR INC |