AU3952593A - Amides having inhibiting activity on phospholipase A2, a process for the preparation thereof and pharmaceutical compositions containing them - Google Patents
Amides having inhibiting activity on phospholipase A2, a process for the preparation thereof and pharmaceutical compositions containing themInfo
- Publication number
- AU3952593A AU3952593A AU39525/93A AU3952593A AU3952593A AU 3952593 A AU3952593 A AU 3952593A AU 39525/93 A AU39525/93 A AU 39525/93A AU 3952593 A AU3952593 A AU 3952593A AU 3952593 A AU3952593 A AU 3952593A
- Authority
- AU
- Australia
- Prior art keywords
- phospholipase
- amides
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/0606—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing heteroatoms not provided for by C07K5/06086 - C07K5/06139, e.g. Ser, Met, Cys, Thr
- C07K5/06069—Ser-amino acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES09200809A ES2044781B1 (en) | 1992-04-14 | 1992-04-14 | PROCEDURE FOR THE PREPARATION OF NEW AMIDES WITH PHOSPHOLIPASE A2 INHIBITING ACTION |
ES9200809 | 1992-04-14 |
Publications (1)
Publication Number | Publication Date |
---|---|
AU3952593A true AU3952593A (en) | 1993-11-18 |
Family
ID=8276745
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU39525/93A Abandoned AU3952593A (en) | 1992-04-14 | 1993-04-07 | Amides having inhibiting activity on phospholipase A2, a process for the preparation thereof and pharmaceutical compositions containing them |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU3952593A (en) |
ES (1) | ES2044781B1 (en) |
WO (1) | WO1993021211A1 (en) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU708306B2 (en) * | 1995-07-24 | 1999-07-29 | Fujisawa Pharmaceutical Co., Ltd. | Esters and amides as PLA2 inhibitors |
CA2227466A1 (en) * | 1995-07-24 | 1997-02-06 | Fujisawa Pharmaceutical Co., Ltd. | Esters and amides as pla2 inhibitors |
US7893226B2 (en) | 2004-09-29 | 2011-02-22 | Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. | Use of lipid conjugates in the treatment of diseases |
US9040078B2 (en) | 2000-01-10 | 2015-05-26 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Use of lipid conjugates in the treatment of diseases of the nervous system |
US7608598B2 (en) | 2000-01-10 | 2009-10-27 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Use of lipid conjugates in the treatment of conjunctivitis |
US8916539B2 (en) | 2000-01-10 | 2014-12-23 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Use of lipid conjugates in the treatment of disease |
US7772196B2 (en) | 2000-01-10 | 2010-08-10 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Use of lipid conjugates in the treatment of diseases |
US8883761B2 (en) | 2001-01-10 | 2014-11-11 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Use of lipid conjugates in the treatment of diseases associated with vasculature |
ATE343375T1 (en) | 2001-03-27 | 2006-11-15 | Biomira Inc | VACCINE FOR MODULATION BETWEEN T1 AND T2 IMMUNE RESPONSES |
US20060069238A1 (en) * | 2002-04-15 | 2006-03-30 | Biomira, Inc. | Synthetic glyco-lipo-peptides as vaccines |
TW201204410A (en) | 2004-04-01 | 2012-02-01 | Oncothyreon Inc | Mucinous glycoprotein (MUC-1) vaccine |
EA012138B1 (en) * | 2004-11-17 | 2009-08-28 | Йиссум Рисерч Дивелопмент Компани Оф Дзе Хебрю Юниверсити Оф Иерусалим | Use of lipid conjugates in the treatment of diseases |
DK2366400T3 (en) | 2005-06-28 | 2016-01-11 | Oncothyreon Inc | A method for the treatment of patients with mucinous glycoprotein (MUC-1) vaccine |
WO2012116225A2 (en) | 2011-02-24 | 2012-08-30 | Oncothyreon Inc. | Muc1 based glycolipopeptide vaccine with adjuvant |
CN105152986B (en) * | 2015-09-09 | 2017-08-25 | 武汉华纳联合药业有限公司 | Cysteine Homotaurine dipeptides and its derivative and its medical usage |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1964798A1 (en) * | 1969-01-07 | 1970-07-16 | Ciba Geigy | New pharmaceutical preparations |
NL175293C (en) * | 1972-02-08 | 1984-10-16 | Akzo Nv | METHOD FOR PREPARING OR MANUFACTURING A PHARMACEUTICAL PREPARATION WITH A PSYCHOPHARMACOLOGICAL ACTION, AND A METHOD FOR PREPARING A VASOPRESSIN DERIVED PEPTIDE. |
US4111924A (en) * | 1976-01-05 | 1978-09-05 | Takeda Chemical Industries, Ltd. | Method for removal of thiol-protecting groups |
IL84252A (en) * | 1987-10-23 | 1994-02-27 | Yissum Res Dev Co | Phospholipase inhibiting compositions |
-
1992
- 1992-04-14 ES ES09200809A patent/ES2044781B1/en not_active Expired - Fee Related
-
1993
- 1993-04-07 WO PCT/EP1993/000866 patent/WO1993021211A1/en active Application Filing
- 1993-04-07 AU AU39525/93A patent/AU3952593A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
ES2044781A1 (en) | 1994-01-01 |
WO1993021211A1 (en) | 1993-10-28 |
ES2044781B1 (en) | 1994-10-01 |
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