AU3848297A - Process for preparing 16alpha-hydroxy-estra-1,3,5(10)-triene derivatives - Google Patents

Process for preparing 16alpha-hydroxy-estra-1,3,5(10)-triene derivatives

Info

Publication number
AU3848297A
AU3848297A AU38482/97A AU3848297A AU3848297A AU 3848297 A AU3848297 A AU 3848297A AU 38482/97 A AU38482/97 A AU 38482/97A AU 3848297 A AU3848297 A AU 3848297A AU 3848297 A AU3848297 A AU 3848297A
Authority
AU
Australia
Prior art keywords
16alpha
estra
hydroxy
preparing
triene derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU38482/97A
Inventor
Helmut Hauser
Michael Meyer
Manuel Morales
Daniel Ramirez
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Schering AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering AG filed Critical Schering AG
Publication of AU3848297A publication Critical patent/AU3848297A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/005—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
AU38482/97A 1996-07-25 1997-07-11 Process for preparing 16alpha-hydroxy-estra-1,3,5(10)-triene derivatives Abandoned AU3848297A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19631541 1996-07-25
DE1996131541 DE19631541C1 (en) 1996-07-25 1996-07-25 Simple production of oestriol from 1,3,5(10),16-oestratetraene derivative
PCT/EP1997/003708 WO1998004577A1 (en) 1996-07-25 1997-07-11 PROCESS FOR PREPARING 16α-HYDROXY-ESTRA-1,3,5(10)-TRIENE DERIVATIVES

Publications (1)

Publication Number Publication Date
AU3848297A true AU3848297A (en) 1998-02-20

Family

ID=7801803

Family Applications (1)

Application Number Title Priority Date Filing Date
AU38482/97A Abandoned AU3848297A (en) 1996-07-25 1997-07-11 Process for preparing 16alpha-hydroxy-estra-1,3,5(10)-triene derivatives

Country Status (6)

Country Link
EP (1) EP0915905A1 (en)
JP (1) JP2000515163A (en)
AU (1) AU3848297A (en)
CA (1) CA2260121A1 (en)
DE (1) DE19631541C1 (en)
WO (1) WO1998004577A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1149838A1 (en) * 2000-04-28 2001-10-31 AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.p.A. Estriol substantially free of 16alpha, 17alpha-estra-1,3,5(10)-triene-3,16,17-triol
WO2012032529A1 (en) 2010-09-08 2012-03-15 Reliance Life Sciences Pvt. Ltd Stereoselective reduction of alpha-hydroxyketone
CN108047295A (en) * 2017-12-29 2018-05-18 广西万德药业有限公司 The high-efficiency synthesis method of estriol

Also Published As

Publication number Publication date
WO1998004577A1 (en) 1998-02-05
EP0915905A1 (en) 1999-05-19
JP2000515163A (en) 2000-11-14
DE19631541C1 (en) 1997-09-18
CA2260121A1 (en) 1998-02-05

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