AU2844800A - Process for preparing a stable non-hygroscopic crystalline n-(n-(n- piperdin- 4-yl)butanoyl)- n.ethylglycyl)- (l)-aspartyl) -ss-cyclohexylalanine amide - Google Patents

Process for preparing a stable non-hygroscopic crystalline n-(n-(n- piperdin- 4-yl)butanoyl)- n.ethylglycyl)- (l)-aspartyl) -ss-cyclohexylalanine amide

Info

Publication number
AU2844800A
AU2844800A AU28448/00A AU2844800A AU2844800A AU 2844800 A AU2844800 A AU 2844800A AU 28448/00 A AU28448/00 A AU 28448/00A AU 2844800 A AU2844800 A AU 2844800A AU 2844800 A AU2844800 A AU 2844800A
Authority
AU
Australia
Prior art keywords
ethylglycyl
piperdin
butanoyl
aspartyl
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU28448/00A
Inventor
Jean-Rene Authelin
Pierre Bailly
Fabrice Mangin
Alain Thouzery
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Aventis Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharmaceuticals Inc filed Critical Aventis Pharmaceuticals Inc
Publication of AU2844800A publication Critical patent/AU2844800A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
AU28448/00A 1998-12-30 1999-12-15 Process for preparing a stable non-hygroscopic crystalline n-(n-(n- piperdin- 4-yl)butanoyl)- n.ethylglycyl)- (l)-aspartyl) -ss-cyclohexylalanine amide Abandoned AU2844800A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11428998P 1998-12-30 1998-12-30
US60114289 1998-12-30
PCT/US1999/029969 WO2000040601A1 (en) 1998-12-30 1999-12-15 Process for preparing a stable non-hygroscopic crystalline n-[n-[n- piperdin- 4-yl)butanoyl)- n.ethylglycyl]- (l)-aspartyl] -ss-cyclohexylalanine amide

Publications (1)

Publication Number Publication Date
AU2844800A true AU2844800A (en) 2000-07-24

Family

ID=22354353

Family Applications (1)

Application Number Title Priority Date Filing Date
AU28448/00A Abandoned AU2844800A (en) 1998-12-30 1999-12-15 Process for preparing a stable non-hygroscopic crystalline n-(n-(n- piperdin- 4-yl)butanoyl)- n.ethylglycyl)- (l)-aspartyl) -ss-cyclohexylalanine amide

Country Status (3)

Country Link
EP (1) EP1155033A1 (en)
AU (1) AU2844800A (en)
WO (1) WO2000040601A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2982668A3 (en) 2002-12-03 2016-04-13 Pharmacyclics LLC 2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors for the treatment of thromboembolic disorders

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2890881B2 (en) * 1990-06-27 1999-05-17 味の素株式会社 Crystallization of amino acids or nucleic acids
RU2134695C1 (en) * 1993-10-15 1999-08-20 Рон-Пуленк Рорер Фармасьютикалз Инк. Antithrombotic azacycloalkylakanoyl peptides
US5780590A (en) * 1993-10-15 1998-07-14 Rhone-Poulenc Rorer Pharmaceuticals Inc. Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
CA2263647C (en) * 1996-08-21 2011-02-15 Zofia J. Chrzan Stable non-hygroscopic crystalline form of n-[n-n-(4-(piperidin-4-yl)butanoyl)-n-ethylglycyl] compounds
DE69711514T2 (en) * 1996-08-27 2002-10-24 Showa Denko K.K., Tokio/Tokyo Non-hygroscopic crystals of p-aminomethylbenzoic acid and process for their preparation

Also Published As

Publication number Publication date
WO2000040601A1 (en) 2000-07-13
EP1155033A1 (en) 2001-11-21

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase