AU2022413551A1 - Stable formulations of shr0302 - Google Patents
Stable formulations of shr0302 Download PDFInfo
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- AU2022413551A1 AU2022413551A1 AU2022413551A AU2022413551A AU2022413551A1 AU 2022413551 A1 AU2022413551 A1 AU 2022413551A1 AU 2022413551 A AU2022413551 A AU 2022413551A AU 2022413551 A AU2022413551 A AU 2022413551A AU 2022413551 A1 AU2022413551 A1 AU 2022413551A1
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- shr0302
- topical pharmaceutical
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
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| US202163289780P | 2021-12-15 | 2021-12-15 | |
| US63/289,780 | 2021-12-15 | ||
| US202263370740P | 2022-08-08 | 2022-08-08 | |
| US63/370,740 | 2022-08-08 | ||
| PCT/US2022/081535 WO2023114832A1 (en) | 2021-12-15 | 2022-12-14 | Stable formulations of shr0302 |
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| US3711602A (en) * | 1970-10-30 | 1973-01-16 | Crown Zellerbach Corp | Compositions for topical application for enhancing tissue penetration of physiologically active agents with dmso |
| US3934013A (en) | 1975-02-21 | 1976-01-20 | Syntex (U.S.A.) Inc. | Pharmaceutical composition |
| JP5732471B2 (ja) | 2009-12-22 | 2015-06-10 | レオ ファーマ アクティーゼルスカブ | 溶媒混合物およびビタミンｄ誘導体から成る医薬品組成物または類似体 |
| PT2796460T (pt) * | 2011-12-21 | 2018-11-05 | Shanghai hengrui pharmaceutical co ltd | Derivado pirrole de anel heteroarilo de seis membros, método de preparação do mesmo e suas utilizações médicas |
| PT3006445T (pt) | 2013-06-07 | 2018-01-09 | Jiangsu Hengrui Medicine Co | Bissulfato de inibidor de janus quinase (jak) e método de preparação para o mesmo |
| CN105566327A (zh) | 2014-10-09 | 2016-05-11 | 江苏恒瑞医药股份有限公司 | 一种jak激酶抑制剂的硫酸氢盐的i型结晶及其制备方法 |
| WO2016070697A1 (zh) | 2014-11-05 | 2016-05-12 | 江苏恒瑞医药股份有限公司 | 一种jak激酶抑制剂的硫酸氢盐的结晶形式及其制备方法 |
| CA3014090A1 (en) | 2016-02-19 | 2017-08-24 | Jiangsu Hengrui Medicine Co., Ltd. | Pharmaceutical composition containing jak kinase inhibitor or pharmaceutically acceptable salt thereof |
| US20190060311A1 (en) | 2017-08-24 | 2019-02-28 | Aclaris Therapeutics, Inc. | Compositions and methods for treatment of vitiligo |
| SG11202001706RA (en) | 2017-10-27 | 2020-03-30 | Theravance Biopharma R&D Ip Llc | Pyrimidine compound as jak kinase inhibitor |
| WO2019096303A1 (zh) * | 2017-11-20 | 2019-05-23 | 江苏恒瑞医药股份有限公司 | 一种局部给药的药物组合物及其制备方法 |
| JP7268132B2 (ja) | 2018-07-31 | 2023-05-02 | エムシー２・セラピューティクス・リミテッド | 局所用組成物 |
| WO2020136650A1 (en) | 2018-12-25 | 2020-07-02 | Sol-Gel Technologies Ltd. | Treatment of skin disorders with compositions comprising an egfr inhibitor |
| WO2020236950A1 (en) | 2019-05-21 | 2020-11-26 | Dauntless 1, Inc. | Therapeutic microsphere formulations containing charged polymers |
| WO2022027041A1 (en) * | 2020-07-28 | 2022-02-03 | Arcutis Biotherapeutics, Inc. | Topical formulation containing jak inhibitor and laureth-4 |
| EP4237080A1 (en) | 2020-10-29 | 2023-09-06 | Arcutis Biotherapeutics, Inc. | Methods for treating vitiligo lesions having improved efficacy |
| MX2023005763A (es) * | 2020-11-17 | 2023-05-29 | Arcutis Biotherapeutics Inc | Composiciones y metodos para la administracion dermica profunda de farmacos. |
| CN114907353A (zh) * | 2021-02-09 | 2022-08-16 | 明慧医药（杭州）有限公司 | 一种前药化合物及其制备方法和用途 |
| CN114870016B (zh) | 2022-04-21 | 2023-05-26 | 上海博悦生物科技有限公司 | 一种jak抑制剂的微乳泡沫剂及其应用 |
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