AU2013205607A1 - Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase - Google Patents

Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase

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Publication number
AU2013205607A1
AU2013205607A1 AU2013205607A AU2013205607A AU2013205607A1 AU 2013205607 A1 AU2013205607 A1 AU 2013205607A1 AU 2013205607 A AU2013205607 A AU 2013205607A AU 2013205607 A AU2013205607 A AU 2013205607A AU 2013205607 A1 AU2013205607 A1 AU 2013205607A1
Authority
AU
Australia
Prior art keywords
yloxy
phenyl
thiazolopyrazin
thiazolopyridin
modulators
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2013205607A
Other versions
AU2013205607B2 (en
Inventor
Genesis M. Bacani
Diego Broggini
Eugene Y. Cheung
Christa C. Chrovian
Xiaohu Deng
Anne M. Fourine
Laurent Gomez
Cheryl A. Grice
Aaron M. Kearney
Adrienne M. Landry-Bayle
Alice Lee-Dutra
Jimmy T. Liang
Susanne Lochner
Neelakandha S. Mani
Alejandro Santillan
Kathleen C. Sappey
Kia Sepassi
Virginia M. Tanis
Alvah T. Wickboldt
John J.M. Wiener
Hartmut Zinser
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2009234140A external-priority patent/AU2009234140B2/en
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Priority to AU2013205607A priority Critical patent/AU2013205607B2/en
Publication of AU2013205607A1 publication Critical patent/AU2013205607A1/en
Application granted granted Critical
Publication of AU2013205607B2 publication Critical patent/AU2013205607B2/en
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

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  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amine compounds are described, which are useful as LTA4 hydrolase (LTA4H) modulators. Such compounds may be used in pharmaceutical compositions and methods for modulation of LTA4H and for the treatment of disease states, disorders, and conditions mediated by LTA4 hydrolase activity.
AU2013205607A 2008-04-11 2013-05-01 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase Ceased AU2013205607B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2013205607A AU2013205607B2 (en) 2008-04-11 2013-05-01 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US61/044,349 2008-04-11
US61/149,129 2009-02-02
AU2009234140A AU2009234140B2 (en) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase
AU2013205607A AU2013205607B2 (en) 2008-04-11 2013-05-01 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
AU2009234140A Division AU2009234140B2 (en) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase

Publications (2)

Publication Number Publication Date
AU2013205607A1 true AU2013205607A1 (en) 2013-05-30
AU2013205607B2 AU2013205607B2 (en) 2016-04-21

Family

ID=48483539

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2013205607A Ceased AU2013205607B2 (en) 2008-04-11 2013-05-01 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase

Country Status (1)

Country Link
AU (1) AU2013205607B2 (en)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5220063A (en) * 1991-05-10 1993-06-15 Hoechst Celanese Corporation Method for the preparation of arylalkanolacylamides

Also Published As

Publication number Publication date
AU2013205607B2 (en) 2016-04-21

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Legal Events

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FGA Letters patent sealed or granted (standard patent)
MK14 Patent ceased section 143(a) (annual fees not paid) or expired