AU2007267176A1 - Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use - Google Patents

Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use Download PDF

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Publication number
AU2007267176A1
AU2007267176A1 AU2007267176A AU2007267176A AU2007267176A1 AU 2007267176 A1 AU2007267176 A1 AU 2007267176A1 AU 2007267176 A AU2007267176 A AU 2007267176A AU 2007267176 A AU2007267176 A AU 2007267176A AU 2007267176 A1 AU2007267176 A1 AU 2007267176A1
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AU
Australia
Prior art keywords
diaza
bicyclo
alkyl
carbonyl
pyrimidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2007267176A
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English (en)
Inventor
Jeppe Kejser Christensen
Tino Dyhring
Henrik Bjork Hansen
Steven Charles Loechel
Jens Damsgaard Mikkelsen
Elsebet Ostergaard Nielsen
Gunnar M. Olsen
Dan Peters
John Paul Redrobe
Daniel B. Timmermann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
NTG Nordic Transport Group AS
Original Assignee
Neurosearch AS
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Filing date
Publication date
Application filed by Neurosearch AS filed Critical Neurosearch AS
Publication of AU2007267176A1 publication Critical patent/AU2007267176A1/en
Abandoned legal-status Critical Current

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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  • Pain & Pain Management (AREA)
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  • Reproductive Health (AREA)
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  • Diabetes (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Obesity (AREA)
  • Pregnancy & Childbirth (AREA)
  • Psychology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Urology & Nephrology (AREA)
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AU2007267176A 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use Abandoned AU2007267176A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US80902306P 2006-05-30 2006-05-30
DKPA200600730 2006-05-30
US60/809,023 2006-05-30
DKPA200600730 2006-05-30
PCT/EP2007/055170 WO2007138039A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use

Publications (1)

Publication Number Publication Date
AU2007267176A1 true AU2007267176A1 (en) 2007-12-06

Family

ID=38258823

Family Applications (3)

Application Number Title Priority Date Filing Date
AU2007267176A Abandoned AU2007267176A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use
AU2007267178A Abandoned AU2007267178A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use
AU2007267177A Abandoned AU2007267177A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use

Family Applications After (2)

Application Number Title Priority Date Filing Date
AU2007267178A Abandoned AU2007267178A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use
AU2007267177A Abandoned AU2007267177A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use

Country Status (7)

Country Link
US (3) US20090197872A1 (https=)
EP (3) EP2049538A1 (https=)
JP (3) JP2009538868A (https=)
AU (3) AU2007267176A1 (https=)
CA (3) CA2653371A1 (https=)
MX (3) MX2008014885A (https=)
WO (3) WO2007138040A1 (https=)

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WO2007138040A1 (en) * 2006-05-30 2007-12-06 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use
JP2010536726A (ja) 2007-08-17 2010-12-02 ノイロサーチ アクティーゼルスカブ ニコチン性アセチルコリン受容体リガンドとして有用な新規１，４−ジアザ−ビシクロ〔３．２．２〕ノニルヘテロアリール誘導体
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US20100305108A1 (en) * 2007-11-14 2010-12-02 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
US8343960B2 (en) * 2007-11-14 2013-01-01 Neurosearch A/S 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
WO2009062987A1 (en) * 2007-11-14 2009-05-22 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
WO2010026176A1 (en) * 2008-09-05 2010-03-11 Neurosearch A/S 1,4 -diaza- bicyclo [3.2.2]n0nyl pyrimidine derivatives as nicotinic and monoamine receptor modulators
WO2010026177A1 (en) * 2008-09-05 2010-03-11 Neurosearch A/S 1,4-diaza-bicyclo [3.2.2] nonyl pyridine derivatives as nicotinic and monoamine receptor modulators
WO2010040806A1 (en) * 2008-10-10 2010-04-15 Neurosearch A/S Novel diphenyl purine derivatives useful as modulators of nicotinic acetylcholine receptors
WO2010063784A1 (en) * 2008-12-04 2010-06-10 Neurosearch A/S Novel diaza-bicyclononyl-phenyl derivatives and their medical use
WO2010084120A1 (en) * 2009-01-21 2010-07-29 Neurosearch A/S N-oxides of 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine receptor ligands
US20120028967A1 (en) * 2009-01-21 2012-02-02 Neurosearch A/S Novel diaza-bicyclononyl-pyrimidinyl derivatives and their medical use
JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7

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US20100286128A1 (en) 2007-08-17 2010-11-11 Dan Peters 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine-receptor ligands
JP2010536726A (ja) 2007-08-17 2010-12-02 ノイロサーチ アクティーゼルスカブ ニコチン性アセチルコリン受容体リガンドとして有用な新規１，４−ジアザ−ビシクロ〔３．２．２〕ノニルヘテロアリール誘導体
WO2009062987A1 (en) * 2007-11-14 2009-05-22 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
US20100305108A1 (en) * 2007-11-14 2010-12-02 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use

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