AU2004208842B2 - Antiglucocorticoids for the treatment of postpartum psychosis - Google Patents
Antiglucocorticoids for the treatment of postpartum psychosis Download PDFInfo
- Publication number
- AU2004208842B2 AU2004208842B2 AU2004208842A AU2004208842A AU2004208842B2 AU 2004208842 B2 AU2004208842 B2 AU 2004208842B2 AU 2004208842 A AU2004208842 A AU 2004208842A AU 2004208842 A AU2004208842 A AU 2004208842A AU 2004208842 B2 AU2004208842 B2 AU 2004208842B2
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- Australia
- Prior art keywords
- glucocorticoid receptor
- psychosis
- receptor antagonist
- postpartum
- psychotic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- ZUOUZKKEUPVFJK-UHFFFAOYSA-N phenylbenzene Natural products C1=CC=CC=C1C1=CC=CC=C1 ZUOUZKKEUPVFJK-UHFFFAOYSA-N 0.000 description 1
- 230000004962 physiological condition Effects 0.000 description 1
- 229920001223 polyethylene glycol Polymers 0.000 description 1
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- YGSDEFSMJLZEOE-UHFFFAOYSA-M salicylate Chemical compound OC1=CC=CC=C1C([O-])=O YGSDEFSMJLZEOE-UHFFFAOYSA-M 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44528403P | 2003-02-04 | 2003-02-04 | |
| US60/445,284 | 2003-02-04 | ||
| PCT/US2004/003183 WO2004069202A2 (en) | 2003-02-04 | 2004-02-04 | Antiglucocorticoids for the treatment of postpartum psychosis |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2004208842A1 AU2004208842A1 (en) | 2004-08-19 |
| AU2004208842B2 true AU2004208842B2 (en) | 2009-05-28 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2004208842A Ceased AU2004208842B2 (en) | 2003-02-04 | 2004-02-04 | Antiglucocorticoids for the treatment of postpartum psychosis |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20040229855A1 (enExample) |
| EP (1) | EP1599208A4 (enExample) |
| JP (1) | JP2006516651A (enExample) |
| AU (1) | AU2004208842B2 (enExample) |
| CA (1) | CA2514966A1 (enExample) |
| WO (1) | WO2004069202A2 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2676670C (en) | 2007-02-02 | 2012-03-13 | Pfizer Products Inc. | Tricyclic compounds, compositions, and methods |
| EP2306830A4 (en) * | 2008-07-01 | 2012-06-06 | Corcept Therapeutics Inc | USE OF MIFEPRISTONE FOR THE TREATMENT OF AMYOTROPHER LATERAL SCLEROSIS |
| US10500216B2 (en) | 2011-11-18 | 2019-12-10 | Corcept Therapeutics, Inc. | Optimizing mifepristone absorption |
| US12226412B2 (en) | 2012-05-25 | 2025-02-18 | Corcept Therapeutics, Inc. | Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators |
| US8859774B2 (en) | 2012-05-25 | 2014-10-14 | Corcept Therapeutics, Inc. | Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators |
| US9943526B2 (en) | 2015-04-21 | 2018-04-17 | Corcept Therapeutics, Inc. | Optimizing mifepristone levels for cushing's patients |
| SG11202105770YA (en) | 2018-12-19 | 2021-07-29 | Corcept Therapeutics Inc | Pharmaceutical formulations containing relacorilant, a heteroaryl-ketone fused azadecalin compound |
| WO2022134033A1 (en) | 2020-12-25 | 2022-06-30 | Corcept Therapeutics Incorporated | Methods of preparing heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators |
| CN119997939A (zh) | 2022-10-06 | 2025-05-13 | 科赛普特治疗公司 | 糖皮质激素受体调节剂的制剂 |
| CN120202004A (zh) | 2022-10-28 | 2025-06-24 | 科赛普特治疗学股份有限公司 | 使用达祖可兰治疗肌萎缩侧索硬化症 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6150349A (en) * | 1997-10-06 | 2000-11-21 | The Board Of Trustees Of The Leland Stanford Junior University | Methods for treating psychosis associated with glucocorticoid related dysfunction |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5468741A (en) * | 1993-05-28 | 1995-11-21 | The Regents Of The University Of California | Use of low levels of mifepristone to treat leiomyomata |
| IL118974A (en) * | 1995-08-17 | 2001-09-13 | Akzo Nobel Nv | History 11 - (Transformed Phenyl) - Astra - 4, 9 - Diane, their preparation and pharmaceutical preparations containing them |
-
2004
- 2004-02-04 CA CA002514966A patent/CA2514966A1/en not_active Abandoned
- 2004-02-04 WO PCT/US2004/003183 patent/WO2004069202A2/en not_active Ceased
- 2004-02-04 AU AU2004208842A patent/AU2004208842B2/en not_active Ceased
- 2004-02-04 JP JP2006503313A patent/JP2006516651A/ja active Pending
- 2004-02-04 US US10/772,919 patent/US20040229855A1/en not_active Abandoned
- 2004-02-04 EP EP04708184A patent/EP1599208A4/en not_active Withdrawn
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6150349A (en) * | 1997-10-06 | 2000-11-21 | The Board Of Trustees Of The Leland Stanford Junior University | Methods for treating psychosis associated with glucocorticoid related dysfunction |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004069202A2 (en) | 2004-08-19 |
| EP1599208A4 (en) | 2007-09-12 |
| US20040229855A1 (en) | 2004-11-18 |
| JP2006516651A (ja) | 2006-07-06 |
| CA2514966A1 (en) | 2004-08-19 |
| WO2004069202A3 (en) | 2005-01-06 |
| EP1599208A2 (en) | 2005-11-30 |
| AU2004208842A1 (en) | 2004-08-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FGA | Letters patent sealed or granted (standard patent) | ||
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |