AU2003279550A1 - Scaffolds useful to the synthesis of compounds with biological activity - Google Patents

Scaffolds useful to the synthesis of compounds with biological activity

Info

Publication number
AU2003279550A1
AU2003279550A1 AU2003279550A AU2003279550A AU2003279550A1 AU 2003279550 A1 AU2003279550 A1 AU 2003279550A1 AU 2003279550 A AU2003279550 A AU 2003279550A AU 2003279550 A AU2003279550 A AU 2003279550A AU 2003279550 A1 AU2003279550 A1 AU 2003279550A1
Authority
AU
Australia
Prior art keywords
synthesis
compounds
biological activity
scaffolds useful
scaffolds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003279550A
Inventor
Giuseppe Giannini
Leonardo Manzoni
Carlo Scolastico
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sigma Tau Industrie Farmaceutiche Riunite SpA
Original Assignee
Sigma Tau Industrie Farmaceutiche Riunite SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma Tau Industrie Farmaceutiche Riunite SpA filed Critical Sigma Tau Industrie Farmaceutiche Riunite SpA
Publication of AU2003279550A1 publication Critical patent/AU2003279550A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
AU2003279550A 2002-11-19 2003-10-14 Scaffolds useful to the synthesis of compounds with biological activity Abandoned AU2003279550A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0227007.2 2002-11-19
GB0227007A GB2395480A (en) 2002-11-19 2002-11-19 Pyrrolo[1,2-a]pyridine & pyrrolo[1,2-a]azepine scaffolds useful for the synthesis of compounds with biological activity
PCT/IT2003/000625 WO2004046173A1 (en) 2002-11-19 2003-10-14 Scaffolds useful to the synthesis of compounds with biological activity

Publications (1)

Publication Number Publication Date
AU2003279550A1 true AU2003279550A1 (en) 2004-06-15

Family

ID=9948141

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003279550A Abandoned AU2003279550A1 (en) 2002-11-19 2003-10-14 Scaffolds useful to the synthesis of compounds with biological activity

Country Status (3)

Country Link
AU (1) AU2003279550A1 (en)
GB (1) GB2395480A (en)
WO (1) WO2004046173A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20032102A1 (en) * 2003-10-30 2005-04-30 Univ Degli Studi Milano PEPTIDOMYMETIC COMPOUNDS, STEREOUSELECTIVE PROCEDURE FOR THEIR PREPARATION, THEIR USE AS INTERMEDIATES OF SYNTHESIS OF BIOLOGICALLY ACTIVE DERIVATIVES.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6235877B1 (en) * 1999-08-04 2001-05-22 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors

Also Published As

Publication number Publication date
GB2395480A (en) 2004-05-26
WO2004046173A1 (en) 2004-06-03
GB0227007D0 (en) 2002-12-24

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase