AU2002359923A1 - 6-fluorobicyclo[3.1.0]hexane derivatives - Google Patents
6-fluorobicyclo[3.1.0]hexane derivativesInfo
- Publication number
- AU2002359923A1 AU2002359923A1 AU2002359923A AU2002359923A AU2002359923A1 AU 2002359923 A1 AU2002359923 A1 AU 2002359923A1 AU 2002359923 A AU2002359923 A AU 2002359923A AU 2002359923 A AU2002359923 A AU 2002359923A AU 2002359923 A1 AU2002359923 A1 AU 2002359923A1
- Authority
- AU
- Australia
- Prior art keywords
- fluorobicyclo
- hexane derivatives
- hexane
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- CGRSIAQTWWBUEJ-UHFFFAOYSA-N 6-fluorobicyclo[3.1.0]hexane Chemical class C1CCC2C(F)C21 CGRSIAQTWWBUEJ-UHFFFAOYSA-N 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2001-395797 | 2001-12-27 | ||
JP2001395797 | 2001-12-27 | ||
PCT/JP2002/013693 WO2003061698A1 (en) | 2001-12-27 | 2002-12-26 | 6-fluorobicyclo[3.1.0]hexane derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002359923A1 true AU2002359923A1 (en) | 2003-09-18 |
AU2002359923B2 AU2002359923B2 (en) | 2007-12-20 |
Family
ID=27602080
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002359923A Ceased AU2002359923B2 (en) | 2001-12-27 | 2002-12-26 | 6-fluorobicyclo[3.1.0]hexane derivatives |
Country Status (24)
Country | Link |
---|---|
US (1) | US7157594B2 (en) |
EP (1) | EP1459765B1 (en) |
JP (1) | JP4230919B2 (en) |
KR (2) | KR20090031962A (en) |
CN (1) | CN1281274C (en) |
AT (1) | ATE405289T1 (en) |
AU (1) | AU2002359923B2 (en) |
BR (1) | BR0215462A (en) |
CA (1) | CA2471642C (en) |
CY (1) | CY1108380T1 (en) |
DE (1) | DE60228491D1 (en) |
DK (1) | DK1459765T3 (en) |
ES (1) | ES2311642T3 (en) |
HK (1) | HK1073258A1 (en) |
HU (1) | HU228436B1 (en) |
MX (1) | MXPA04006322A (en) |
NO (1) | NO328844B1 (en) |
NZ (1) | NZ533699A (en) |
PL (1) | PL208123B1 (en) |
PT (1) | PT1459765E (en) |
RU (1) | RU2315622C2 (en) |
SI (1) | SI1459765T1 (en) |
WO (1) | WO2003061698A1 (en) |
ZA (2) | ZA200404795B (en) |
Families Citing this family (47)
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NZ560966A (en) * | 2000-10-27 | 2010-06-25 | Novartis Vaccines & Diagnostic | Nucleic acids and proteins from streptococcus groups A & B |
BR0311558A (en) | 2002-06-11 | 2007-04-27 | Lilly Co Eli | pharmaceutically acceptable compound or salt thereof, process for preparing same, methods for affecting camp-linked metabotropic glutamate receptors, for administering an effective amount of a compound and for treating a neurological and psychiatric disorder in a patient, and, pharmaceutical formulation |
US7109383B2 (en) | 2002-09-27 | 2006-09-19 | Central Glass Company, Limited | Fluorine-containing allyl ether compounds, their copolymers, and resist compositions and anti-reflection film materials using such copolymers |
WO2005000791A1 (en) | 2003-06-26 | 2005-01-06 | Taisho Pharmaceutical Co., Ltd. | 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic ester derivative |
JP5485492B2 (en) * | 2004-12-15 | 2014-05-07 | 大正製薬株式会社 | Drugs for the prevention and treatment of depression |
EP2258359A3 (en) | 2005-08-26 | 2011-04-06 | Braincells, Inc. | Neurogenesis by muscarinic receptor modulation with sabcomelin |
US7678363B2 (en) | 2005-08-26 | 2010-03-16 | Braincells Inc | Methods of treating psychiatric conditions comprising administration of muscarinic agents in combination with SSRIs |
EP1940389A2 (en) | 2005-10-21 | 2008-07-09 | Braincells, Inc. | Modulation of neurogenesis by pde inhibition |
US20070112017A1 (en) | 2005-10-31 | 2007-05-17 | Braincells, Inc. | Gaba receptor mediated modulation of neurogenesis |
US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
TWI417095B (en) | 2006-03-15 | 2013-12-01 | Janssen Pharmaceuticals Inc | 1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of mglur2-receptors |
MX2008014320A (en) | 2006-05-09 | 2009-03-25 | Braincells Inc | 5 ht receptor mediated neurogenesis. |
EP2021000A2 (en) | 2006-05-09 | 2009-02-11 | Braincells, Inc. | Neurogenesis by modulating angiotensin |
EP2068872A1 (en) | 2006-09-08 | 2009-06-17 | Braincells, Inc. | Combinations containing a 4-acylaminopyridine derivative |
US20100184806A1 (en) | 2006-09-19 | 2010-07-22 | Braincells, Inc. | Modulation of neurogenesis by ppar agents |
TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
CN101801930B (en) | 2007-09-14 | 2013-01-30 | 奥梅-杨森制药有限公司 | 1,3-disubstituted-4-phenyl-1 h-pyridin-2-ones |
JP5366269B2 (en) | 2007-09-14 | 2013-12-11 | ジャンセン ファーマシューティカルズ, インコーポレイテッド. | 1,3-disubstituted 4- (allyl-X-phenyl) -1H-pyridin-2-one |
US9114138B2 (en) | 2007-09-14 | 2015-08-25 | Janssen Pharmaceuticals, Inc. | 1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones |
US8785486B2 (en) | 2007-11-14 | 2014-07-22 | Janssen Pharmaceuticals, Inc. | Imidazo[1,2-A]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors |
WO2010025890A1 (en) | 2008-09-02 | 2010-03-11 | Ortho-Mcneil-Janssen Pharmaceuticals, Inc | 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors |
WO2010043396A1 (en) | 2008-10-16 | 2010-04-22 | Ortho-Mcneil-Janssen Pharmaceuticals, Inc. | Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors |
WO2010060589A1 (en) | 2008-11-28 | 2010-06-03 | Ortho-Mcneil-Janssen Pharmaceuticals, Inc. | Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors |
US20100216805A1 (en) | 2009-02-25 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis using d-cycloserine combinations |
SG10201402250TA (en) | 2009-05-12 | 2014-07-30 | Janssen Pharmaceuticals Inc | 1,2,4-triazolo [4,3-a] pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders |
MX2011011962A (en) | 2009-05-12 | 2012-02-28 | Janssen Pharmaceuticals Inc | 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors. |
MY153913A (en) | 2009-05-12 | 2015-04-15 | Janssen Pharmaceuticals Inc | 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
TW201129700A (en) | 2009-11-18 | 2011-09-01 | Taisho Pharmaceutical Co Ltd | Method for producing optically active bicyclo [310] hexane derivative using oxygen |
US8642777B2 (en) | 2009-11-19 | 2014-02-04 | Taisho Pharmaceutical Co., Ltd | Process for producing 3-alkoxy-2-amino-6-fluorobicyclo [3.1.0] hexane-2,6-dicarboxylic acid derivative and intermediate thereof |
WO2012062750A1 (en) | 2010-11-08 | 2012-05-18 | Janssen Pharmaceuticals, Inc. | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
ES2552879T3 (en) | 2010-11-08 | 2015-12-02 | Janssen Pharmaceuticals, Inc. | 1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors |
EP2643320B1 (en) | 2010-11-08 | 2015-03-04 | Janssen Pharmaceuticals, Inc. | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
TWI520935B (en) | 2010-11-18 | 2016-02-11 | 美國禮來大藥廠 | 4-substituted-3-phenylsulfanylmethyl-bicyclo(3.1.0)hexane compounds as mglur 2/3 antagonists |
BR112013012384A2 (en) | 2010-11-18 | 2019-09-24 | Lilly Co Eli | 4-substituted 3-benzyloxy-bicyclo [3.1.0] hexane compounds as receptor antagonists of mglu2 and mglu3 |
EA023553B1 (en) | 2011-06-17 | 2016-06-30 | Эли Лилли Энд Компани | mGlu2 RECEPTOR AGONISTS |
WO2013062680A1 (en) * | 2011-10-25 | 2013-05-02 | Braincells, Inc. | Novel compounds and compositions thereof for treating nervous system disorders |
RU2496495C2 (en) * | 2011-12-05 | 2013-10-27 | Учреждение Российской академии медицинских наук Научно-исследовательский институт нормальной физиологии имени П.К. Анохина РАМН | USING SELECTIVE ANTAGONIST OF GLUAMATE RECEPTOR Ro-256981 FOR TARGETED EFFECT ON COGNITIVE FUNCTIONS |
CN104334524B (en) * | 2012-06-01 | 2016-10-12 | 大正制药株式会社 | The prodrug of fluorinated amino acids |
JO3368B1 (en) | 2013-06-04 | 2019-03-13 | Janssen Pharmaceutica Nv | 6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
JO3367B1 (en) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
HUE053734T2 (en) | 2014-01-21 | 2021-07-28 | Janssen Pharmaceutica Nv | Combinations comprising positive allosteric modulators of metabotropic glutamatergic receptor subtype 2 and their use |
EA201891617A3 (en) | 2014-01-21 | 2019-04-30 | Янссен Фармацевтика Нв | COMBINATIONS CONTAINING POSITIVE ALLOSTERIC MODULATORS OR ORTHOSTERIC AGONISTS OF METABOTROPIC GLUTAMATERGIC RECEPTOR 2 SUBTIPES AND THEIR APPLICATION |
CA3019097C (en) | 2016-04-18 | 2023-08-29 | Taisho Pharmaceutical Co., Ltd. | Prodrug of amino acid derivative |
JP7314494B2 (en) * | 2017-10-17 | 2023-07-26 | 大正製薬株式会社 | Pharmaceuticals containing prodrugs of amino acid derivatives |
KR20220062838A (en) | 2020-11-09 | 2022-05-17 | 대우조선해양 주식회사 | Full spade rudder and ship having the same |
JP2024004505A (en) * | 2020-11-26 | 2024-01-17 | 大正製薬株式会社 | Method for producing amino acid derivative |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU703093B2 (en) | 1995-11-16 | 1999-03-18 | Eli Lilly And Company | Excitatory amino acid receptor antagonists |
ZA969485B (en) * | 1995-11-16 | 1998-05-12 | Lilly Co Eli | Excitatory amino acid receptor antagonists. |
ZA983930B (en) * | 1997-05-14 | 1999-11-08 | Lilly Co Eli | Excitatory amino acid receptor modulators. |
JP4194715B2 (en) | 1998-08-31 | 2008-12-10 | 大正製薬株式会社 | 6-Fluorobicyclo [3.1.0] hexane derivative |
CA2341865C (en) * | 1998-08-31 | 2006-01-17 | Taisho Pharmaceutical Co., Ltd. | 6-fluorobicyclo[3.1.0]hexane derivatives |
CH694053A5 (en) | 1998-09-03 | 2004-06-30 | Hoffmann La Roche | Ver method for the production of 2-amino-bicyclo [3.1.0] hexane-2,6-dicarboxylic acid derivatives. |
US7034055B1 (en) * | 1999-06-30 | 2006-04-25 | Prescient Neuropharma Inc. | 2-aminoindane analogs |
NZ522674A (en) * | 2000-05-11 | 2004-10-29 | Kenneth Curry | Novel spiro[2.4]heptane amino carboxy compounds and derivatives thereof |
US6770676B2 (en) | 2000-06-28 | 2004-08-03 | Taisho Pharmaceutical Co., Ltd. | Dicarboxylic acid derivatives |
CA2442557C (en) * | 2001-04-12 | 2008-12-23 | F. Hoffmann-La Roche Ag | Dihydro-benzo¬b|¬1,4|diazepin-2-one derivatives as mglur2 antagonists ii |
-
2002
- 2002-12-26 KR KR1020097005135A patent/KR20090031962A/en not_active Application Discontinuation
- 2002-12-26 NZ NZ533699A patent/NZ533699A/en not_active IP Right Cessation
- 2002-12-26 KR KR1020047010069A patent/KR100897970B1/en not_active IP Right Cessation
- 2002-12-26 PL PL371014A patent/PL208123B1/en unknown
- 2002-12-26 DK DK02793421T patent/DK1459765T3/en active
- 2002-12-26 CA CA2471642A patent/CA2471642C/en not_active Expired - Fee Related
- 2002-12-26 SI SI200230736T patent/SI1459765T1/en unknown
- 2002-12-26 PT PT02793421T patent/PT1459765E/en unknown
- 2002-12-26 EP EP02793421A patent/EP1459765B1/en not_active Expired - Lifetime
- 2002-12-26 HU HU0402649A patent/HU228436B1/en not_active IP Right Cessation
- 2002-12-26 ES ES02793421T patent/ES2311642T3/en not_active Expired - Lifetime
- 2002-12-26 MX MXPA04006322A patent/MXPA04006322A/en active IP Right Grant
- 2002-12-26 AT AT02793421T patent/ATE405289T1/en active
- 2002-12-26 US US10/500,101 patent/US7157594B2/en not_active Expired - Fee Related
- 2002-12-26 BR BR0215462-5A patent/BR0215462A/en not_active IP Right Cessation
- 2002-12-26 RU RU2004122916/15A patent/RU2315622C2/en not_active IP Right Cessation
- 2002-12-26 WO PCT/JP2002/013693 patent/WO2003061698A1/en active Application Filing
- 2002-12-26 DE DE60228491T patent/DE60228491D1/en not_active Expired - Lifetime
- 2002-12-26 CN CNB02826388XA patent/CN1281274C/en not_active Expired - Fee Related
- 2002-12-26 AU AU2002359923A patent/AU2002359923B2/en not_active Ceased
- 2002-12-26 JP JP2003561641A patent/JP4230919B2/en not_active Expired - Fee Related
-
2004
- 2004-06-16 NO NO20042530A patent/NO328844B1/en not_active IP Right Cessation
- 2004-06-17 ZA ZA2004/04795A patent/ZA200404795B/en unknown
-
2005
- 2005-03-11 ZA ZA2005/02085A patent/ZA200502085B/en unknown
- 2005-07-15 HK HK05106035A patent/HK1073258A1/en not_active IP Right Cessation
-
2008
- 2008-09-29 CY CY20081101068T patent/CY1108380T1/en unknown
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