AU2002335231A1 - Activator for peroxisome proliferator-activated receptor delta - Google Patents
Activator for peroxisome proliferator-activated receptor deltaInfo
- Publication number
- AU2002335231A1 AU2002335231A1 AU2002335231A AU2002335231A AU2002335231A1 AU 2002335231 A1 AU2002335231 A1 AU 2002335231A1 AU 2002335231 A AU2002335231 A AU 2002335231A AU 2002335231 A AU2002335231 A AU 2002335231A AU 2002335231 A1 AU2002335231 A1 AU 2002335231A1
- Authority
- AU
- Australia
- Prior art keywords
- activator
- activated receptor
- peroxisome proliferator
- receptor delta
- delta
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 108010015181 PPAR delta Proteins 0.000 title 1
- 102100003648 PPARD Human genes 0.000 title 1
- 239000012190 activator Substances 0.000 title 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001-315694 | 2001-10-12 | ||
| JP2001315694 | 2001-10-12 | ||
| PCT/JP2002/010472 WO2003033493A1 (en) | 2001-10-12 | 2002-10-09 | ACTIVATOR FOR PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR δ |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2002335231A1 true AU2002335231A1 (en) | 2003-07-03 |
| AU2002335231B2 AU2002335231B2 (en) | 2008-05-08 |
Family
ID=19133818
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002335231A Ceased AU2002335231B2 (en) | 2001-10-12 | 2002-10-09 | Activator for peroxisome proliferator-activated receptor delta |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7119104B2 (en) |
| EP (1) | EP1445258B1 (en) |
| JP (1) | JP4276074B2 (en) |
| KR (1) | KR100933652B1 (en) |
| CN (1) | CN1293076C (en) |
| AT (1) | ATE434616T1 (en) |
| AU (1) | AU2002335231B2 (en) |
| BR (1) | BRPI0213243B8 (en) |
| CA (1) | CA2463569C (en) |
| CY (1) | CY1110355T1 (en) |
| DE (1) | DE60232739D1 (en) |
| DK (1) | DK1445258T3 (en) |
| ES (1) | ES2326411T3 (en) |
| IL (2) | IL161351A0 (en) |
| MX (1) | MXPA04003398A (en) |
| PT (1) | PT1445258E (en) |
| WO (1) | WO2003033493A1 (en) |
Families Citing this family (45)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60232739D1 (en) * | 2001-10-12 | 2009-08-06 | Nippon Chemiphar Co | ACTIVATOR OF THE PEROXISOMPROLIFERATOR-ACTIVATED RECEPTOR DELTA |
| EP1637161A4 (en) * | 2003-04-22 | 2007-06-27 | Astellas Pharma Inc | REMEDY FOR CEREBRAL NEURODEGENERATIVE DISEASES USING PPAR [delta] AGONIST |
| AU2004285849B2 (en) | 2003-09-19 | 2011-04-28 | Janssen Pharmaceutica, N.V. | 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs |
| US20050203151A1 (en) * | 2003-12-19 | 2005-09-15 | Kalypsys, Inc. | Novel compounds, compositions and uses thereof for treatment of metabolic disorders and related conditions |
| WO2005097127A2 (en) | 2004-04-02 | 2005-10-20 | Merck & Co., Inc. | Method of treating men with metabolic and anthropometric disorders |
| JP2007536343A (en) | 2004-05-05 | 2007-12-13 | ノボ ノルディスク アクティーゼルスカブ | Phenoxyacetic acid derivatives as PPAR agonists |
| EP1745014B1 (en) | 2004-05-05 | 2011-07-06 | High Point Pharmaceuticals, LLC | Novel compounds, their preparation and use |
| KR20070053243A (en) | 2004-09-11 | 2007-05-23 | 사노피-아벤티스 도이칠란트 게엠베하 | 7-azaindoles and their use as ppar agonists |
| US7833513B2 (en) * | 2004-12-03 | 2010-11-16 | Rhode Island Hospital | Treatment of Alzheimer's Disease |
| ATE529404T1 (en) | 2005-06-30 | 2011-11-15 | High Point Pharmaceuticals Llc | PHENOXYACETIC ACIDS AS PPAR-DELTA ACTIVATORS |
| ZA200800892B (en) * | 2005-07-06 | 2009-04-29 | Nippon Chemiphar Co | Activator of peroxisome proliferator activated receptor δ |
| CA2621275A1 (en) * | 2005-09-07 | 2007-03-15 | Plexxikon, Inc. | 1 , 4 and 1 , 5-disubstituted indole derivatives for use as ppar active compounds |
| JO3006B1 (en) | 2005-09-14 | 2016-09-05 | Janssen Pharmaceutica Nv | Novel Lysine Salts of 4-((Phenoxy Alkyl)Thio)-Phenoxy Acetic Acid Derivatives |
| EA015717B1 (en) | 2005-12-22 | 2011-10-31 | ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи | Phenoxy acetic acids as ppar delta activators |
| EP1999098A2 (en) | 2006-03-09 | 2008-12-10 | High Point Pharmaceuticals, LLC | Compounds that modulate ppar activity, their preparation and use |
| UY30288A1 (en) * | 2006-04-18 | 2007-08-31 | Janssen Pharmaceutica Nv | DERIVATIVES OF BENZOAZEPIN-OXI-ACETIC ACID AS PPAR-DELTA AGONISTS USED TO INCREASE HDL-C. REDUCE LDL-C AND REDUCE CHOLESTEROL |
| CN101466687B (en) * | 2006-04-18 | 2012-04-11 | 日本化学医药株式会社 | Activating agent for peroxisome proliferator activated receptor delta |
| WO2008016175A1 (en) * | 2006-08-03 | 2008-02-07 | Nippon Chemiphar Co., Ltd. | Activator for peroxisome proliferator activated receptor |
| BRPI0811612A2 (en) | 2007-05-21 | 2014-11-11 | Senju Pharma Co | PHARMACEUTICAL COMPOSITIONS CONTAINING PPARDELON AGONIST |
| WO2008154023A1 (en) * | 2007-06-11 | 2008-12-18 | Cerenis Therapeutics S.A. | Novel uses of ppar delta agonists |
| CA2721339C (en) | 2008-04-15 | 2017-01-24 | Nippon Chemiphar Co., Ltd. | Activating agent for peroxisome proliferator activated receptor |
| WO2010047982A1 (en) | 2008-10-22 | 2010-04-29 | Merck Sharp & Dohme Corp. | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
| CA2741672A1 (en) | 2008-10-31 | 2010-05-06 | Merck Sharp & Dohme Corp. | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
| WO2011020001A2 (en) | 2009-08-14 | 2011-02-17 | Cerenis Therapeutics S.A. | Use of ppar delta ligands for the treatment or prevention of inflammation or energy metabolism/production related diseases |
| CA2774999A1 (en) | 2009-09-30 | 2011-04-07 | President And Fellows Of Harvard College | Methods for modulation of autophagy through the modulation of autophagy-enhancing gene products |
| JP2013006769A (en) * | 2009-10-08 | 2013-01-10 | Nippon Chemiphar Co Ltd | Activator for peroxisome proliferator activating receptor |
| AU2011218830B2 (en) | 2010-02-25 | 2014-07-24 | Merck Sharp & Dohme Corp. | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
| US20130156720A1 (en) | 2010-08-27 | 2013-06-20 | Ironwood Pharmaceuticals, Inc. | Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders |
| EP3243385B1 (en) | 2011-02-25 | 2021-01-13 | Merck Sharp & Dohme Corp. | Novel cyclic azabenzimidazole derivatives useful as anti-diabetic agents |
| JP2015525782A (en) | 2012-08-02 | 2015-09-07 | メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． | Antidiabetic tricyclic compounds |
| MX365408B (en) | 2013-01-31 | 2019-05-31 | Senju Pharma Co | Stable aqueous solution. |
| CN105025896B (en) | 2013-01-31 | 2017-11-14 | 千寿制药株式会社 | The aqueous liquid preparation of clarification |
| CN104994848A (en) | 2013-02-22 | 2015-10-21 | 默沙东公司 | Antidiabetic bicyclic compounds |
| WO2014139388A1 (en) | 2013-03-14 | 2014-09-18 | Merck Sharp & Dohme Corp. | Novel indole derivatives useful as anti-diabetic agents |
| US9487493B2 (en) | 2013-09-09 | 2016-11-08 | Vtv Therapeutics Llc | Use of a PPAR-delta agonist for treating muscle atrophy |
| WO2015051496A1 (en) | 2013-10-08 | 2015-04-16 | Merck Sharp & Dohme Corp. | Antidiabetic tricyclic compounds |
| JPWO2017195875A1 (en) * | 2016-05-12 | 2019-03-22 | 日本ケミファ株式会社 | Wound healing agent |
| US11072602B2 (en) | 2016-12-06 | 2021-07-27 | Merck Sharp & Dohme Corp. | Antidiabetic heterocyclic compounds |
| US10968232B2 (en) | 2016-12-20 | 2021-04-06 | Merck Sharp & Dohme Corp. | Antidiabetic spirochroman compounds |
| KR102495798B1 (en) * | 2016-12-30 | 2023-02-03 | 뉴스케일 파워, 엘엘씨 | Control rod drive mechanism (CRDM) with remote disconnect mechanism |
| US11634387B2 (en) | 2019-09-26 | 2023-04-25 | Abionyx Pharma Sa | Compounds useful for treating liver diseases |
| CN113912547B (en) | 2020-07-10 | 2024-04-30 | 成都凡诺西生物医药科技有限公司 | Substituted benzene imidazole derivative and application thereof |
| WO2022189856A1 (en) * | 2021-03-08 | 2022-09-15 | Abionyx Pharma Sa | Compounds useful for treating liver diseases |
| WO2023147309A1 (en) | 2022-01-25 | 2023-08-03 | Reneo Pharmaceuticals, Inc. | Use of ppar-delta agonists in the treatment of disease |
| CN115215856A (en) * | 2022-08-19 | 2022-10-21 | 沈阳药科大学 | Preparation method of PPAR delta agonist finadepa and intermediate thereof |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5089514A (en) | 1990-06-14 | 1992-02-18 | Pfizer Inc. | 3-coxazolyl [phenyl, chromanyl or benzofuranyl]-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents |
| US5089541A (en) * | 1990-11-23 | 1992-02-18 | Shell Oil Company | Removal of hydrogenation catalyst from polymer solutions by contact with activated carbon |
| GB9027023D0 (en) | 1990-12-12 | 1991-01-30 | Wellcome Found | Anti-atherosclerotic aryl compounds |
| HUT64023A (en) | 1991-03-22 | 1993-11-29 | Sandoz Ag | Process for producing aminoguanidine derivatives and pharmaceutical compositions comprising such compounds |
| GB9426448D0 (en) | 1994-12-30 | 1995-03-01 | Wellcome Found | Process |
| KR100436812B1 (en) * | 1995-01-06 | 2004-08-31 | 도레이 가부시끼가이샤 | Benzene condensed heterocyclic derivatives and pharmaceutical compositions containing the derivatives as active ingredients |
| CA2171702A1 (en) | 1995-03-14 | 1996-09-15 | Takashi Sohda | Benzofuran compounds and their use |
| WO1996035688A1 (en) | 1995-05-08 | 1996-11-14 | Nippon Chemiphar Co., Ltd. | 2,4-thiazolidinedione or oxazolidinedione derivatives and hypoglycemic agent |
| KR19990076788A (en) | 1996-01-22 | 1999-10-15 | 후지야마 아키라 | Thiazolylbenzofuran derivatives and pharmaceutical compositions containing the same |
| WO1997028115A1 (en) | 1996-02-02 | 1997-08-07 | Merck & Co., Inc. | Antidiabetic agents |
| US20020032330A1 (en) | 1996-12-24 | 2002-03-14 | Yutaka Nomura | Propionic acid derivatives |
| ATE421336T1 (en) | 1997-07-24 | 2009-02-15 | Astellas Pharma Inc | MEDICINAL COMPOSITIONS HAVING A CHOLESTEROL-LOWERING EFFECT |
| US6589969B1 (en) | 1998-10-16 | 2003-07-08 | Ono Pharmaceutical Co., Ltd. | Carboxylic acid derivatives and drugs containing the same as the active ingredient |
| JP2001354671A (en) | 2000-04-14 | 2001-12-25 | Nippon Chemiphar Co Ltd | ACTIVATOR FOR PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR delta |
| JP2004506722A (en) * | 2000-08-23 | 2004-03-04 | イーライ・リリー・アンド・カンパニー | Methods of modulating peroxisome proliferator-activated receptors |
| AU2002233271A1 (en) * | 2000-12-20 | 2002-07-01 | Glaxo Group Limited | Substitued oxazoles and thiazoles as hppar alpha agonists |
| US7105551B2 (en) * | 2000-12-20 | 2006-09-12 | Smithkline Beecham Corporation | Thiazole derivatives for treating PPAR related disorders |
| GB0031109D0 (en) * | 2000-12-20 | 2001-01-31 | Glaxo Group Ltd | Chemical compounds |
| GB0113231D0 (en) * | 2001-05-31 | 2001-07-25 | Glaxo Group Ltd | Chemical compounds |
| PT1424330E (en) * | 2001-08-10 | 2011-12-22 | Nippon Chemiphar Co | Activator for peroxisome proliferator-responsive receptor delta |
| DE60232739D1 (en) * | 2001-10-12 | 2009-08-06 | Nippon Chemiphar Co | ACTIVATOR OF THE PEROXISOMPROLIFERATOR-ACTIVATED RECEPTOR DELTA |
| US6867224B2 (en) * | 2002-03-07 | 2005-03-15 | Warner-Lambert Company | Compounds that modulate PPAR activity and methods of preparation |
-
2002
- 2002-10-09 DE DE60232739T patent/DE60232739D1/en not_active Expired - Lifetime
- 2002-10-09 JP JP2003536232A patent/JP4276074B2/en not_active Expired - Fee Related
- 2002-10-09 MX MXPA04003398A patent/MXPA04003398A/en active IP Right Grant
- 2002-10-09 CA CA2463569A patent/CA2463569C/en not_active Expired - Lifetime
- 2002-10-09 AU AU2002335231A patent/AU2002335231B2/en not_active Ceased
- 2002-10-09 KR KR1020047005398A patent/KR100933652B1/en active IP Right Grant
- 2002-10-09 EP EP02801515A patent/EP1445258B1/en not_active Expired - Lifetime
- 2002-10-09 WO PCT/JP2002/010472 patent/WO2003033493A1/en active Application Filing
- 2002-10-09 PT PT02801515T patent/PT1445258E/en unknown
- 2002-10-09 BR BRPI0213243A patent/BRPI0213243B8/en not_active IP Right Cessation
- 2002-10-09 AT AT02801515T patent/ATE434616T1/en active
- 2002-10-09 US US10/491,935 patent/US7119104B2/en not_active Expired - Lifetime
- 2002-10-09 CN CNB028202422A patent/CN1293076C/en not_active Expired - Fee Related
- 2002-10-09 IL IL16135102A patent/IL161351A0/en unknown
- 2002-10-09 DK DK02801515T patent/DK1445258T3/en active
- 2002-10-09 ES ES02801515T patent/ES2326411T3/en not_active Expired - Lifetime
-
2004
- 2004-04-13 IL IL161351A patent/IL161351A/en active IP Right Grant
-
2006
- 2006-10-06 US US11/544,505 patent/US7402597B2/en active Active
-
2009
- 2009-08-06 CY CY20091100833T patent/CY1110355T1/en unknown
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